PhytoCAT-ID |
Phytochemical name or plant extracts |
Source of phytochemicals or plant Extracts |
Target gene or protein |
Cell line/ mice model |
PhytoCAT-0 |
Rocaglaol |
Aglaia crassinervia |
Bax, Bcl-xL, Caspase 9, Caspase 7, Cdc25c |
Lu1, LNCaP, HL-60, SMMC-7721, A-549, MCF-7, W480 |
PhytoCAT-1 |
Limonin |
Citrus limetta |
VEGF, VEGFR2, STAT3, MMP9, miR-216a-3p, ABCG2 |
MCF-7-Adr, MDA-MB-231, MCF-7 |
PhytoCAT-2 |
1'-acetoxychavicol acetate |
Alpinia galanga |
STAT-3, MMP2, MMP9 |
MCF-7, COR L23 |
PhytoCAT-3 |
25-O-acetylcimigenol-3-O-β-D-xylopyranoside |
Cimicifuga yunnanensis |
p53, Bax, Caspase 7 |
MCF-7 , R-MCF-7 |
PhytoCAT-4 |
23-O-acetylcimigenol-3-O-β-D-xylopyranoside |
Cimicifuga yunnanensis |
p53, Bax, Caspase 7 |
MCF-7, R-MCF-7 |
PhytoCAT-5 |
25-chlorodeoxycimigenol-3-O-β-D-xylopyranoside |
Cimicifuga yunnanensis |
p53, Bax, Caspase 7 |
MCF-7, R-MCF-7 |
PhytoCAT-6 |
25-O-acetylcimigenol-3-O-α-L-arabinopyranoside |
Cimicifuga yunnanensis |
p53, Bax, Caspase 7 |
MCF-7, R-MCF-7 |
PhytoCAT-7 |
Calotropis procera extract |
Calotropis procera |
Bcl-2 |
MCF-7, HCT-116, HepG-2, A-549 |
PhytoCAT-8 |
7′-methoxy-3′-O-demethyl-tanegool-9-O-β-d-glucopyranoside |
Calotropis procera |
NA |
MCF-7, HCT-116, HepG-2, A-549 |
PhytoCAT-9 |
Methyl ferulate |
Calotropis procera |
NA |
MCF-7, HCT-116, HepG-2, A-549, SK-LU-1, KB |
PhytoCAT-10 |
Methyl 4-β-d-glucopyranosyl-ferulate |
Calotropis procera |
NA |
MCF-7, HCT-116, HepG-2, A-549, SK-LU-1, KB |
PhytoCAT-11 |
Calotropagenin |
Calotropis procera |
NA |
MCF-7, HCT-116, HepG-2, A-549, SK-LU-1, KB |
PhytoCAT-12 |
Kaempferol 3-O-α-l-rhamnopyranosyl-(1→6)-β-d-glucopyranoside |
Calotropis procera |
NA |
MCF-7, HCT-116, HepG-2, A-549, SK-LU-1, KB |
PhytoCAT-13 |
Kudonol A |
Sophora alopecuroides |
NA |
HeLa, Hep3B, MCF-7, H1299 |
PhytoCAT-14 |
Kudonol B |
Sophora alopecuroides |
NA |
HeLa, Hep3B, MCF-7, H1299 |
PhytoCAT-15 |
Kudonol C |
Sophora alopecuroides |
NA |
HeLa, Hep3B, MCF-7, H1299 |
PhytoCAT-16 |
Kudolignan A |
Sophora alopecuroides |
NA |
HeLa, Hep3B, MCF-7, H1299 |
PhytoCAT-17 |
Kudolignan B |
Sophora alopecuroides |
NA |
HeLa, Hep3B, MCF-7, H1299 |
PhytoCAT-18 |
Stemophenanthrene A |
Stemona tuberosa |
NA |
KB, MCF7, SK-LU-1, HepG2 |
PhytoCAT-19 |
Stemophenanthrene B |
Stemona tuberosa |
NA |
KB, MCF7, SK-LU-1, HepG2 |
PhytoCAT-20 |
Stemophenanthrene C |
Stemona tuberosa |
NA |
KB, MCF7, SK-LU-1, HepG2 |
PhytoCAT-21 |
Isopinosylvin A |
Stemona tuberosa |
NA |
KB, MCF7, SK-LU-1, HepG2 |
PhytoCAT-22 |
Stemofuran X |
Stemona pierrei |
NA |
KB, MCF7, SK-LU-1, HepG2 |
PhytoCAT-23 |
Stemofuran Y |
Stemona tuberosa |
NA |
KB, MCF7, SK-LU-1, HepG2 |
PhytoCAT-24 |
Periploca hydaspidis Falc crude extract |
Periploca hydaspidis |
Survivin, Bcl-xL, XIAP, Myelocytomatosis, C-myc, MMP2, MMP9, Cyclin D1, Cyclin E, Bak, Bax, Caspase 3 , Caspase 7, Caspase 8, Caspase 9, PARPB |
MCF-7, MDA-MB-231, HCCLM3 |
PhytoCAT-25 |
Flavopereirine |
Geissospermum sericeum |
p-ERK, p38 MAPK siRNA, p-Akt, mTOR, LC3-II |
MCF-7, MDA-MB-231 |
PhytoCAT-26 |
Lippia citriodora essential oil |
Lippia citriodora |
Caspase 3, Survivin |
DA3 breast cancer model in mice |
PhytoCAT-27 |
D Rhamnose β-hederin (DRβ-H) |
Clematis ganpiniana |
Apaf-1, cyt-c, Caspase 3, Caspase 9, miR-16, miR-23a, miR-24, miR-26a, miR-27a |
MDA-MB-231, MCF-7/Doc, MCF-7/S |
PhytoCAT-28 |
Polyphenol mixtures of Euphorbia supina |
Euphorbia supina |
Snail1 , N-cadherin, MMP9, LOX, TNF-α-mediated VCAM-1 |
MDA-MB-231 |
PhytoCAT-29 |
Caudatin |
Cynanchum auriculatum |
DR5, CHOP, p38 MAPK, JNK |
MDA-MB-231, MCF-7/ nude mouse |
PhytoCAT-30 |
Rhodoeosein |
Fallopia convolvulus |
ERβ |
SKBR-3 |
PhytoCAT-31 |
Isotetrandrine |
Triclisia sacleuxii |
P-gp |
MCF-7/DOX, HeLa, Hep3B |
PhytoCAT-32 |
Magnoflorine |
Berberidaceae, Magnoliaceae, Menispermaceae, or Papaveraceae botanical families
Berberis cretica |
NA |
NCI-H1299, MDA-MB-468, T98G , TE671 |
PhytoCAT-33 |
Berberiside A |
Berberis tsarica |
NA |
A549, HepG2, MDA-MB-231 |
PhytoCAT-34 |
Berberiside D |
Berberis tsarica |
NA |
A549, HepG2, MDA-MB-231 |
PhytoCAT-35 |
Icariin |
Alseodaphne semecarpifolia |
ERK1/2 |
SKBR-3, MCF-7, MCF-7/TAM |
PhytoCAT-36 |
Sphagneticola trilobata extract |
Sphagneticola trilobata |
NA |
MCF-7 |
PhytoCAT-37 |
Pluchea dioscoridis essential oil |
Pluchea dioscoridis |
NA |
MCF-7, A-549 |
PhytoCAT-38 |
Taheebo |
Tabebuia avellandae |
Cyclin B1, PCNA, OKL38, Caspases, ESR1, CYP 1A1, CYP 1B1, Bcl-2 family, GADD-45 family |
MCF-7 |
PhytoCAT-39 |
Aronia melanocarpa extract |
Aronia melanocarpa |
NA |
NA |
PhytoCAT-40 |
5-hydroxy-skytanthine hydrochloride |
Tecoma stans |
NA |
Hep-G2, MCF-7 |
PhytoCAT-41 |
E/Z-acetoside |
Tecoma stans |
NA |
Hep-G2, MCF-7 |
PhytoCAT-42 |
Taxus chinensis extract |
Taxus chinensis |
NA |
MCF-7, Rat |
PhytoCAT-43 |
3ß-hydroxylup-20(29)-ene-27,28-dioic acid |
Ampelozizyphus amazonicus |
NA |
SKBR-3, C-8161 |
PhytoCAT-44 |
Cajanol |
Cajanus cajan |
Bcl-2, Bax, cyt-c, Caspase 3, caspase 9, PARP |
MCF-7 |
PhytoCAT-45 |
Taro-derived extracts (TEs) |
Colocasia esculenta |
NA |
Syngeneic Balb/c female mice, MDA-MD-231, MDA-MB-468, T47D, NCI-ADR RES-luc, OVCAR-3-luc |
PhytoCAT-46 |
Napabucasin |
Handroanthus impetiginosus |
STAT-3 |
K562, MDA-MB-231 |
PhytoCAT-47 |
β-lapachone |
Handroanthus impetiginosus |
NA |
K562, MDA-MB-231 |
PhytoCAT-48 |
Rhamnazin |
Retama sphaerocarpa |
VEGFR2 |
MDA-MB-231/xenograft, TK-10, MCF-7, UACC-62 |
PhytoCAT-49 |
Eclipta alba extract (CFEA) |
Eclipta alba |
Hsp60, XIAP |
MCF-7, MDA-MB-231, mouse breast cancer 4T1, MCF 10A |
PhytoCAT-50 |
Rhein |
Rheum palmatum |
PI3K, p-AKT, p-ERK, Hsp90α, NF-κB, COX-2, HER-2, HIF-1α, VEGF(165), EGF, TNF-α, IL-6, I-κB, Caspase 9, CHOP, , eIF2α, GRP78, FOXO, Akt |
MCF-7, MDA-MB-435, MCF-7/HER2, MCF-7/VEC, MDA-MB-231, HepG2, 4T1 breast cancer xenografts in mice |
PhytoCAT-51 |
5,3′-dihydroxy-6,7,8,4′-tetramethoxyflavanone (HLBT-100) |
Tillandsia recurvata |
Caspase 3, Caspase 7 |
U87 MG, MDA-MB-231, MV4-11, A375, IMR-32 |
PhytoCAT-52 |
Cimicifuga racemosa extract |
Cimicifuga racemosa |
Caspases, ER, p21, Cyclin D1, Progesterone receptor B1 |
MCF-7, MDA-MB-231, T47D, LNCaP |
PhytoCAT-53 |
Rich Lady peach extract |
Prunus persica |
NA |
MCF-7, MDA-MB-435, MCF-10A |
PhytoCAT-54 |
Kaempferide |
Azadirachta indica |
ER |
HL60, A549, AZ521, SKBR-3, MCF-7,PC-3, T-47D |
PhytoCAT-55 |
Isoazadironolide |
Azadirachta indica |
NA |
HL60, A549, AZ521, SKBR-3 |
PhytoCAT-56 |
4'-O-methyl-8-prenylnaringenin |
Azadirachta indica |
NA |
HL60, A549, AZ521, SKBR-3 |
PhytoCAT-57 |
Euchrestaflavanone A |
Azadirachta indica |
NA |
HL60, A549, AZ521, SKBR-3 |
PhytoCAT-58 |
9, and 3-methoxy-3'-prenylnaringenin |
Azadirachta indica |
NA |
HL60, A549, AZ521, SKBR-3 |
PhytoCAT-59 |
Gedunin |
Azadirachta indica |
Hsp90 |
MCF-7, SKBR-3 |
PhytoCAT-60 |
Nimbolide |
Azadirachta indica |
p21, Bax, Bad, Fas-L, TRAIL, FADDR, cyt-c, Bcl-2, Bcl-xL, Mcl-1, XIAP-1, pro-caspase 8, pro-caspase 3, integrin αV, integrin β3, ILK, FAK, PAK, DNMT-1, HDAC-6, miR-21, HOTAIR, H19, miR-148a/miR-152, PTEN, ABCB1/MDR1 mRNA, P-gp, HIF1α, FoxO1, MYC |
MDA-MB-231, HCC38, HEK293T, MCF-7, HL-60, SMMC7721, A549, SW-480 |
PhytoCAT-61 |
Bromelain proteinase (F9) |
Ananas comosus |
IL- 2, TNF-a |
MCF-7, SK-MEL-28 |
PhytoCAT-62 |
Jatropha curcas extract |
Jatropha curcas |
β1-integrin, FAK |
MCF-7 |
PhytoCAT-63 |
Pyrenacantha staudtii extract |
Pyrenacantha staudtii |
β1-integrin, FAK |
MCF-7 |
PhytoCAT-64 |
Jatropha gossypifolia extract |
Jatropha gossypifolia |
β1-integrin, FAK |
MCF-7 |
PhytoCAT-65 |
Styrylpyrone dehydrogoniothalamin |
Aniba heringeri |
NA |
PC-3, 786-0, HT-29, MCF-7, MDA-MB-231 |
PhytoCAT-66 |
Chimnitensin A |
Chimonanthus nitens Oliv |
NA |
MDA-MB-468, MDA-MB-231 |
PhytoCAT-67 |
Chimnitensin B |
Chimonanthus nitens |
NA |
MDA-MB-468, MDA-MB-231 |
PhytoCAT-68 |
Chimnitensin C |
Chimonanthus nitens |
NA |
MDA-MB-468, MDA-MB-231 |
PhytoCAT-69 |
Chimnitensin D |
Chimonanthus nitens |
NA |
MDA-MB-468, MDA-MB-231 |
PhytoCAT-70 |
Chimnitensin E |
Chimonanthus nitens |
NA |
MDA-MB-468, MDA-MB-231 |
PhytoCAT-71 |
Chimnitensin F |
Chimonanthus nitens |
NA |
MDA-MB-468, MDA-MB-231 |
PhytoCAT-72 |
Licania tomentosa extract |
Licania tomentosa |
NA |
MCF-7, Caco-2 |
PhytoCAT-73 |
Annona muricata extract |
Annona muricata |
AKT, MAPK, NF-κB,cyclin D1, Aromatase, EGFR |
MCF-7, MDA-MB-231, 4T1 |
PhytoCAT-74 |
Platycodin D (PD) |
Platycodon grandiflorus |
ASK1, PERK, eIF 2alpha, GRP78/Bip, CHOP/GADD153, Caspase 4 |
MDA-MB-231, MCF-7 |
PhytoCAT-75 |
18-hydroxydollabela-8(17)-ene |
Cleome droserifolia |
NA |
MCF-7, HCT116 |
PhytoCAT-76 |
Matricaria chamomilla extract |
Matricaria chamomilla |
NA |
MDA-MB-468, MCF-7 |
PhytoCAT-77 |
β-dihydroagarofuran-type sesquiterpene (MD-6) |
Maytenus disticha |
NA |
MCF-7, PC9, C4-2B |
PhytoCAT-78 |
(1α,2α,8β,9β)-1,8-bis(acetyloxy)-2,9-bis(benzoyloxy)-14-hydroxy-β-dihydroagarofuran |
Celastrus paniculatus |
AKT, NF-κB, p53, MAPK |
MCF-7 |
PhytoCAT-79 |
Demethylzeylasterone |
Kokoona zeylanica |
Topo II alpha |
MCF-7 |
PhytoCAT-80 |
Lapachol |
Plenckia populnea |
NA |
Breast cancer (4T1) tumor model, SKBR-3, MDA-MB-231, MCF-7 |
PhytoCAT-81 |
Mangiferin |
Mangifera indica |
MMP7, MMP9, Vimentin, E-cadherin, β-catenin, NF-κB, P-gp |
MDA-MB-231 xenograft mice, MCF-7 |
PhytoCAT-82 |
Triptolide |
Tripterygium wilfordii |
ADAM10, ATM, PARP-1, XRC1, RAD51, miR-146a, Bcl-2 family, RhoA, Rac1, PD-L1, CD206, Arginase 1, CD204, NF-κB, AP-1, MMP9, Notch-1, HES-1, HEY-1, DCLK1, ALDH1, CD133 |
MCF-7, BT-20,MKN-45, MKN-7, KATO-III, HL-60 , MDA-MB-231, BT-474 |
PhytoCAT-83 |
Triptonide |
Tripterygium wilfordii |
SNAI1 |
HCC1806, BT-549, MDA-MB-231 |
PhytoCAT-84 |
Montanoa guatemalensis essential oil |
Montanoa guatemalensis |
NA |
MDA-MB-231, Hs578T |
PhytoCAT-85 |
Betavulgarin |
Beta vulgaris |
NA |
MDA-MB-231, MCF-7 |
PhytoCAT-86 |
Coriolic acid |
Salicornia herbacea |
Nanog,Oct4, CD44, c-Myc |
MDA-MB-231, MCF-7 |
PhytoCAT-87 |
Lutein |
Spinacia oleracea |
HIF‑1α, Notch signaling, HES1, Bcl-2, Caspase 3, PARP, HO-1, SOD-1, Hsp-60 |
MDA‑MB‑157, MCF‑7, BALB/c mice |
PhytoCAT-88 |
Plectranthus amboinicus extract |
Plectranthus amboinicus |
Cyclin D1, Caspase 9, p53 |
T47D, MDA-MB-231, MCF-7 |
PhytoCAT-89 |
(-)-Cycloxanthochymol |
Garcinia celebica |
NA |
HeLa, MCF-7, A549, B16 |
PhytoCAT-90 |
Isoxanthochymol |
Garcinia celebica |
NA |
HeLa, MCF-7, A549, B16 |
PhytoCAT-91 |
Xanthochymol |
Garcinia celebica |
NA |
HeLa, MCF-7, A549, B16 |
PhytoCAT-92 |
Esculetin |
Dryopteris fragrans |
NA |
A549, MCF-7 , MDA-MB-435, MDA-MB-231, HepG2 |
PhytoCAT-93 |
Isoscopoletin |
Dryopteris fragrans |
NA |
A549, MCF-7, HepG2 |
PhytoCAT-94 |
Trans-3-(3,4-dimethoxyphenyl)-4-[(E)-3,4-dimethoxystyryl]cyclohex-1-ene |
Dryopteris fragrans |
NA |
A549, MCF-7, HepG2 |
PhytoCAT-95 |
Cis-3-(3,4-dimethoxyphenyl)-4-[(E)-3,4-dimethoxystyryl] cyclohex-1-ene |
Dryopteris fragrans |
NA |
A549, MCF-7, HepG2 |
PhytoCAT-96 |
Dryofracoumarin A |
Dryopteris fragrans |
NA |
A549, MCF-7, HepG2 |
PhytoCAT-97 |
Aspidinol |
Dryopteris fragrans |
NA |
A549, MCF-7, HepG2 |
PhytoCAT-98 |
Albicanol |
Dryopteris fragrans |
NA |
A549, MCF-7, HepG2 |
PhytoCAT-99 |
(E)-caffeic acid-9-O-β-d-xylpyranosyl-(1→2)-β-d-glucopyranosyl ester |
Dryopteris fragrans |
NA |
A549, MCF-7, SGC7901 , HUVEC |
PhytoCAT-100 |
Octyl gallate |
Terminalia bellirica |
Cyclin D1, Cyclin D3, CDK-4, CDK-6, p18 INK4, p21Waf-1, p27 KIP, MRP2 |
MCF-7, MDA-MB-231 |
PhytoCAT-101 |
Terminaloside Q |
Terminalia citrina |
NA |
MCF-7, T47D |
PhytoCAT-102 |
Terminaloside R |
Terminalia citrina |
NA |
MCF-7, T47D |
PhytoCAT-103 |
Terminaloside S |
Terminalia citrina |
NA |
MCF-7, T47D |
PhytoCAT-104 |
Terminaloside T |
Terminalia citrina |
NA |
MCF-7, T47D |
PhytoCAT-105 |
Terminaloside U |
Terminalia citrina |
NA |
MCF-7, T47D |
PhytoCAT-106 |
Terminaloside V |
Terminalia citrina |
NA |
MCF-7, T47D |
PhytoCAT-107 |
Terminaloside W |
Terminalia citrina |
NA |
MCF-7, T47D |
PhytoCAT-108 |
Thidiazuron |
Nymphaea alba |
uPAR, uPA, VEGF, MMP2, MMP9, TIMP-1/2 |
NA |
PhytoCAT-109 |
Ugonin J |
Helminthostachys zeylanica |
p53, NANOG |
MCF-7, MDA-MB-231 |
PhytoCAT-110 |
Orbignya speciosa extract |
Orbignya speciosa |
NA |
MCF-7, HL-60, K562, K562-Lucena 1, 3T3-L1 |
PhytoCAT-111 |
5,7-Dimethoxyflavone |
Anaphalis busua |
NA |
MDCK/Bcrp1 |
PhytoCAT-112 |
Capillarisin |
Artemisia capillaris |
MMP9 |
MCF-7 |
PhytoCAT-113 |
Artemisia ciniformis extract |
Artemisia ciniformis |
NA |
AGS, HeLa, HT-29, MCF-7 |
PhytoCAT-114 |
Artemisia diffusa extract |
Artemisia diffusa |
NA |
AGS, HeLa, HT-29, MCF-7 |
PhytoCAT-115 |
3R,8R-Dehydrofalcarindiol |
Artemisia monosperma |
NA |
MDA231, MCF-7, LS174T, SKCO1, COLO320DM, WIDR
|
PhytoCAT-116 |
Artemisia persica extract |
Artemisia persica |
NA |
AGS, HeLa, HT-29, MCF-7 |
PhytoCAT-117 |
Artemisia Capillaris extract (ACA) |
Artemisia Capillaris |
NA |
HS578T, T47D |
PhytoCAT-118 |
Shionone |
Aster poliothamnus |
Caspase 3, Caspase 9, Bcl-2, Bax |
SKBR-3, MB-157 |
PhytoCAT-119 |
Codonolactone |
Atractylodes lancea |
Runx2 |
MDA-MB-468, MDA-MB-231, Five-to 6-week-old female NOD/SCID mice |
PhytoCAT-120 |
Acacetin |
Calea urticifolia |
STAT-3, CYP1A1, CYP1B1 |
MDA-MB-231, MCF-7, T47D |
PhytoCAT-121 |
Calendula arvensis L. extract |
Calendula arvensis |
Bcl-2, Bax, Caspase 3, Caspase 7 |
MCF-7, MDA-MB-231 |
PhytoCAT-122 |
Carpesium abrotanoides extract |
Carpesium abrotanoides |
PKM2 |
MCF-7, MDA-MB-231 |
PhytoCAT-123 |
Centaurea aegyptiaca extract |
Centaurea aegyptiaca |
NA |
Hep-G2, MCF-7, HCT-116, HELA |
PhytoCAT-124 |
Centaurea bruguierana |
Centaurea bruguierana |
Bax, Bcl-2, Caspase 3, Caspase 9 |
MCF-7 |
PhytoCAT-125 |
13-O-acetylsolstitialin A |
Centaurea cyanus |
Bax, Bcl-2, Cyclin D1, CDK-4 |
MCF-7, MDA-MB-231 |
PhytoCAT-126 |
Perillic acid |
Perilla frutescens |
Cyclin D1 mRNA |
T47D, MCF-7, MDA-MB-231 |
PhytoCAT-127 |
Jaceosidin |
Centaurea diluta
Artemisia artica |
NA |
MCF-7 |
PhytoCAT-128 |
Pfaffia paniculata extract |
Pfaffia paniculata |
NA |
MCF-7 |
PhytoCAT-129 |
Brevilin A |
Centipeda minima |
AKT, mTOR, STAT-3 |
MDA-MB-231, MDA-MB-468, MCF-7 |
PhytoCAT-130 |
Cichorin D |
Cichorium intybus |
NA |
MDA-MB-468, MDA-MB-231, SK-N-MC, PC-3 |
PhytoCAT-131 |
Cichorin E |
Cichorium intybus |
NA |
MDA-MB-468, MDA-MB-231, SK-N-MC, PC-3 |
PhytoCAT-132 |
Cichorins F |
Cichorium intybus |
NA |
MDA-MB-468, MDA-MB-231, SK-N-MC, PC-3 |
PhytoCAT-133 |
Chicory's extract |
Cichorium Pumilum |
NA |
Female Sprague-Dawley rats |
PhytoCAT-134 |
Pectolinarigenin |
Cirsium chanroenicum |
MMP2, MMP9, TIMP-2, STAT-3 |
4T1, MDA-MB-231, MCF-7 |
PhytoCAT-135 |
Cirsimaritin |
Cirsium japonicum |
VEGF, AKT, ERK |
MDA-MB-231 |
PhytoCAT-136 |
Cirsium palustre essential oil |
Cirsium palustre |
NA |
MCF-7, MDA-MBA-231 |
PhytoCAT-137 |
Cirsium rivulare essential oil |
Cirsium rivulare |
NA |
MCF-7, MDA-MBA-231 |
PhytoCAT-138 |
Raddeanoside R13 |
Pulsatilla chinensis |
Cyclin D1, Cyclin A, Cyclin B1, PARP, Caspase 3 |
NA |
PhytoCAT-139 |
12-O-benzoyl-20-O-acetyl-3β,12β,14β,20β-tetrahydroxy-pregnan-3-ylO-β-D-glucopyranosyl-(1→4)-β-D-glucopyranosyl-(1 → 4)-3-methoxy-β-D-ribopyranoside |
Caralluma tuberculata |
PARP |
MCF-7, MDA-MB-468 |
PhytoCAT-140 |
7-O-acetyl-12-O-benzoyl-3β,7β,12β,14β-tetrahydroxy-17β-(3-methylbutyl-O-acetyl-1-yl)-androstan-3-ylO-β-D-glucopyranosyl-(1 → 4)-6-deoxy-β-D-allopyranosyl-(1 → 4)-β-D-cymaropyranosyl-(1 → 4)-β-D-cymapyranosyl-(1→ 4)-β-D-cymaropyranoside |
Caralluma tuberculata |
PARP |
MCF-7, MDA-MB-469 |
PhytoCAT-141 |
Cynara cardunculus extract |
Cynara cardunculus |
Caspase 9, Caspase 8, Bax, Bcl-2, p21(WAF1) |
MDA-MB-231 |
PhytoCAT-142 |
Hispidulin |
Dittrichia viscosa |
Vimentin , E-cadherin, occludin |
MCF-7, HCC38 |
PhytoCAT-143 |
Lupeol |
Elephantopus scaber |
Caspase 3, MMP9, MMP2, COX-2, NF-κB p65, Bcl-2, |
MDA-MB-231, MCF-7, K 562, SW620, KATO-III, A-549, Hep-G2, Hep3B |
PhytoCAT-144 |
Elephantopus scaber extract |
Elephantopus scaber |
ABCB1, ABCG2 |
HeLa, A549, MCF-7, Caco-2 |
PhytoCAT-145 |
Eupalinolide O |
Eupatorium lindleyanum |
Cyclin B1, cdc2 |
MDA-MB-468 |
PhytoCAT-146 |
Artemisia vulgaris extract |
Artemisia vulgaris |
NA |
NA |
PhytoCAT-147 |
Helenalin |
Psilostrophe cooperi |
Telomerase |
T47D |
PhytoCAT-148 |
Klugine |
Psychotria klugii |
HIF-1 |
T47D |
PhytoCAT-149 |
Isocephaeline |
Psychotria klugii |
HIF-1 |
T47D |
PhytoCAT-150 |
Emetine |
Psychotria klugii |
HIF-1 |
T47D |
PhytoCAT-151 |
Cyanidin-3-glucoside (Cy-3-gluc) |
Puya laxa |
ErbB2, Sirt1, KLF4, HER2, AKT, EMT |
MCF-7, BT-474, HCC1569, MDA-MB-453, 6–7-week-old female nude mice |
PhytoCAT-152 |
Black raspberry |
Rubus occidentalis |
NA |
KB, CAL-27, MCF-7, HT-29, HCT116, LNCaP |
PhytoCAT-153 |
Britannin |
Inula aucheriana |
Bcl-2, Bax, p53 |
MCF-7, MDA-MB-468 |
PhytoCAT-154 |
Nepetin |
Inula britannica |
NA |
MCF-7, Hep-2, Vero cell |
PhytoCAT-155 |
3,3'-di-O-methylquercetin |
Inula viscosa |
NA |
MCF-7, Hep-2, Vero cell |
PhytoCAT-156 |
3-O-methylquercetin |
Inula viscosa |
NA |
MCF-7, Hep-2, Vero cell |
PhytoCAT-157 |
Fischerisin A |
Ligularia fischeri |
NA |
MCF-7, KB |
PhytoCAT-158 |
fischerisin B |
Ligularia fischeri |
NA |
MCF-7, KB |
PhytoCAT-159 |
4beta,14-dihydro-3-dehydrozaluzanin C |
Onopordum acanthium |
NA |
HeLa, MCF-7 , A431 |
PhytoCAT-160 |
Pallenis spinosa essential oil |
Pallenis spinosa |
Bcl-2 , Bax , Cyclin D1, CDK4, p21 |
MCF-7, MDA-MB-231 |
PhytoCAT-161 |
Pulicaria undulata essential oil |
Pulicaria undulata |
VEGFR-2 |
MCF-7 |
PhytoCAT-162 |
Silymarin |
Silybum marianum |
P-gp, VEGF |
DU145, MCF-7, MDA-MB-468 |
PhytoCAT-163 |
Silibinin |
Silybum marianum |
p21, STAT-3, AKT, ERK, EGFR, CD44, MMP2, BRCA1, LRP6, BNIP3, p53, Bak, Bcl-xL, VEGF, MMP9, RAC1, BNIP3 |
HEK293, PC-3, DU-145, T-47D, MCF-7, MDA-MB-231, 4T1, MDA-MB-435/WT, MDA-MB-435/DOX, MCF-7/PAC |
PhytoCAT-164 |
Paclitaxel |
Taxus brevifolia |
EF1a ,FOXO3a, Bcl-2 |
MCF-7 |
PhytoCAT-165 |
Dandelion extract |
Taraxacum mongolicum |
pS2, PR |
MCF-7, immature rat uterotrophic assay |
PhytoCAT-166 |
Isorhamnetin |
Tephroseris kirilowii |
MMP2, MMP9, p38 MAPK, STAT-3 |
B16F10, MCF-7, MDA-MB-231 |
PhytoCAT-167 |
3,4-dihydroxy-phenylacetic acid (PAA) |
Tragopogon orientalis |
NA |
T47D |
PhytoCAT-168 |
7β-(3-Ethyl-cis-crotonoyloxy)-1α-(2-methylbutyryloxy)-3,14-dehydro-Z-notonipetranone (ECN) |
Tussilago farfara |
STAT-3 |
MDA-MB-231 |
PhytoCAT-169 |
Vernonia amygdalina (VA) extract |
Vernonia amygdalina |
ERα, AKT |
MCF-7, MDA-MB-231 |
PhytoCAT-170 |
Vernonia divaricata extract |
Vernonia divaricata |
NA |
HL-60, MCF-7, PC-3 |
PhytoCAT-171 |
Vernolactone |
Vernonia zeylanica |
Survivin, p53, Bax, Caspase 3, Caspase 7 |
MCF -7, MDA-MB-231, SKBR-3 |
PhytoCAT-172 |
Quercetin-3-methyl ether |
Wollastonia biflora |
Caspase 3, Caspase 7, PARP |
SKBR-3 |
PhytoCAT-173 |
Homoharringtonine |
Cephalotaxus harringtonia |
Bcl-x, Caspase 9 |
MCF-7, A549, UACC903 |
PhytoCAT-174 |
Blueberry extract |
Vaccinium corymbosum |
PTEN |
CT26, HCT-116, MDA-MB-231, PC-3, HeLa, SN12C, NCI-H125, MCF-7 |
PhytoCAT-175 |
Cranberry extract |
Vaccinium macrocarpon |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-176 |
2-hydroxy-6-tridecylbenzoic acid |
Ginkgo biloba |
E-cadherin, N-cadherin, Vimentin, Snail, MMP2, MMP9 |
MDA-MB-231, 4 T1 |
PhytoCAT-177 |
Hinokitiol |
Chamaecyparis obtusa |
EGFR |
AS-B244, MDA-MB-231 |
PhytoCAT-178 |
Erycibe elliptilimba extract |
Erycibe elliptilimba |
NA |
SKBR-3, MDA-MB-435 |
PhytoCAT-179 |
Pharbitis nil extract |
Pharbitis nil |
AKT, ERK, Cyclin D, HER2, AKT, ERK |
MCF-7 vec, MCF-7 HER2 |
PhytoCAT-180 |
Cornus mas extract |
Cornus mas |
NA |
SKOV3, MCF-7, PC-3, A549 |
PhytoCAT-181 |
Casearin G |
Casearia sylvestris |
NA |
PC-3, MCF-7 |
PhytoCAT-182 |
Eleutherine |
Cipura paludosa |
NA |
U251, MCF-7, NCI-ADR, 786-0, NCI-H460, HT29, K562, HaCat |
PhytoCAT-183 |
Cuphea aequipetala Extracts |
Cuphea aequipetala |
NA |
MCF-7, HepG2, B16F10, HCT-15, DU145 |
PhytoCAT-184 |
Camalexin |
Arabidopsis thaliana |
NA |
SKBR-3, PREC |
PhytoCAT-185 |
Sinigrin |
Armoracia rusticana |
COX-1 |
HCT-116, MCF-7, NCIH460, CNS, SF-268 |
PhytoCAT-186 |
Docosadienoic Acid (DDA) |
Brassica carinata |
IL-1β, IL-6, IFN-γ, MCP-1, TNF-α |
SKBR-3 and MDA-MB-231 |
PhytoCAT-187 |
Docosatrienoic acid (DTA) |
Brassica carinata |
IL-1β, IL-6, IFN-γ, MCP-1, TNF-α |
SKBR-3 and MDA-MB-231 |
PhytoCAT-188 |
Brassica oleracea juice |
Brassica oleracea |
CDK6, p27 |
MCF-7, BT-474, MDA-MB-231, BT-20 |
PhytoCAT-189 |
P-coumaric acid |
Carrichtera annua |
p53, p21, CDK4 |
SW 620, Hep G2, A549, T47D, HeLa, MCF-7 |
PhytoCAT-190 |
Carrichtera annua extract |
Carrichtera annua |
NA |
MCF-7, HepG2 |
PhytoCAT-191 |
LXY6090 - a novel manassantin A derivative |
Saururus cernuus |
HIF-1, VEGF, IGF-2 |
T47D, MCF-7 |
PhytoCAT-192 |
Semialarium mexicanum extract |
Semialarium mexicanum |
NA |
MDA-MB-231, MCF-7 |
PhytoCAT-193 |
Bryonia dioica extract |
Bryonia dioica Jacq |
NA |
MDA‑MB‑231 |
PhytoCAT-194 |
Bryonia multiflora extract |
Bryonia multiflora |
Bcl-2, p21 |
MCF-7, MDA-MB-231 |
PhytoCAT-195 |
Colocynth Extracts |
Citrullus lanatus |
Bcl-2, Bcl-xL, Bax, Caspase 3, keratin 19, Vimentin, N-cadherin, Zeb1, Zeb2, BMI-1, CD44 |
MCF-7, MDA-MB-231 |
PhytoCAT-196 |
Salix safsaf extract |
Salix safsaf |
Caspase 3, p53, Bcl-2, Bax |
MCF-7, HCT-116, HeLa, HepG2 |
PhytoCAT-197 |
Gypenoside 5 |
Gynostemma pentaphyllum |
Tyrosine phosphatase 1B |
MCF-7, MCF-7/ADR, MDA-MB-231 |
PhytoCAT-198 |
Gypenoside LI |
Gynostemma pentaphyllum |
ERCC6L |
MCF-7, MDA-MB-231 |
PhytoCAT-199 |
Momordica cochinchinensis extract |
Momordica cochinchinensis |
NA |
MCF-7, BT-474 |
PhytoCAT-200 |
Cucurbitacin B |
Trichosanthes cucumerina |
Cyclin D1, C-myc, β-catenin, F-actin, Vimentin, FAK, vinculin |
SKBR-3, MCF-7 |
PhytoCAT-201 |
Snakegourd root polysaccharide |
Trichosanthes cucumerina |
Caspase 3, Caspase 8 |
MCF-7 |
PhytoCAT-202 |
Bryonolic acid |
Trichosanthes cucumerina |
NA |
SKBR-3, MCF-7, T47D, MDA-MB-435, A549, SK-LU1, Caco-2 |
PhytoCAT-203 |
Coryllus avellana extract |
Corylus avellana |
NA |
HeLa, HepG2 and MCF-7 |
PhytoCAT-204 |
Quercus acutissima extract |
Quercus acutissima |
Caspase 3, Beclin-1, Atg5, Bcl-W |
SUM159, MCF-7, HeLa, Jurkat, HT-29 |
PhytoCAT-205 |
Artemisia absinthium extract |
Artemisia absinthium |
Caspase 7, Bad, Bcl-2 |
MDA-MB-231, MCF-7 |
PhytoCAT-206 |
Alisol A |
Alisma plantago-aquatica |
Cyclin D1, MMP2, MMP9 |
MDA-MB-231 |
PhytoCAT-207 |
Mentha arvensis extract |
Mentha arvensis |
PARP1, p53, P21, Bax, Bcl-2, Caspase 9 |
MDA-MB-231, A-549, COLO-205, HCT-116, MCF-7, NCI-H322, PC-3, THP-1, U-87MG |
PhytoCAT-208 |
American ginseng extract |
American ginseng |
pS2 RNA, RKIP, Cyclin A, Cyclin D1 |
MCF-7, T-47D, BT-20 |
PhytoCAT-209 |
Benzoiisovanillin |
Solanum nigrum |
NA |
MDA-MB-231, MCF-7 |
PhytoCAT-210 |
Mulberry leaf lectin |
Morus alba |
Caspase 3 |
MCF-7, HCT-15 |
PhytoCAT-211 |
Mulberry root bark extracts |
Morus alba |
Cyclin D1 |
MDA-MB-231, MCF-7, HCT116, SW480, LoVo |
PhytoCAT-212 |
Moracin O |
Morus alba |
BCL‑XL, Bcl‑2, p65 subunit of NF‑κB |
4T1 |
PhytoCAT-213 |
Moracin P |
Morus alba |
BCL‑XL, Bcl‑2, p65 subunit of NF‑κB |
4T1 |
PhytoCAT-214 |
Viscum album (VA) extract |
Viscum album |
p21, p53, p73, p38, Erk1/2, H2A histone family member X |
NCI-H460, DU-145, HCC1143, MV3, PA-TU-8902, SKBR-3, MCF-7, 4T1 tumor-bearing BALB/c mice |
PhytoCAT-215 |
Juniperus communis L. extract |
Juniperus communis |
ERK1/3 |
MCF-7/AZ |
PhytoCAT-216 |
Deoxypodophyllotoxin |
Juniperus communis |
NA |
MDA-MB-231 |
PhytoCAT-217 |
Dark sweet cherries |
Prunus avium |
Caspase 8, Bax, Bcl-2, PARP-1 |
MDA-MB-453 |
PhytoCAT-218 |
Strawberry extract |
Fragaria ananassa |
NA |
KB, CAL-27, MCF-7, HT-29, HCT116, LNCaP |
PhytoCAT-219 |
Citrus sphaerocarpa extract |
Citrus sphaerocarpa |
MMP9 |
MDA-MB-231 |
PhytoCAT-220 |
Chelidonine |
Chelidonium majus |
AKT, ERK1/2 |
MDA-MB-231 |
PhytoCAT-221 |
p-hydroxybenzoic acid-4-O-α-d-manopyranosyl-(1 → 3)-α-l-rhamnopyranoside |
Melilotus officinalis |
NA |
MCF-7 |
PhytoCAT-222 |
4-O-α-l-rhamnopyran-osyl-(1 → 6)-α-d-manopyranosyl-(1 → 3)-α-l-rhamnopyranoside |
Melilotus officinalis |
NA |
MCF-7 |
PhytoCAT-223 |
Artemisia annua extract |
Artemisia annua |
NA |
AGS, HeLa, HT-29, MCF-7 |
PhytoCAT-224 |
3β,13β-dihydroxy-12,13-dihydrooleanolic acid (1) |
Vitis vinifera |
NA |
MCF-7/DOX |
PhytoCAT-225 |
Resveratrol |
Juniperus polycarpos |
PTEN, STAT-3, VDR, BRCA1, EDA, miR-125b-5p, miR-200c-3p, miR-409-3p, miR-122-5p, miR-542-3p, PCNA, Rb, p53, Bcl-2, aromatase, IL-6, p53, HNRNPA1, Caspase 3, MMP9, AURKA, PLK1, PAK1, Bax, CYP19, p21, RAD51, Twist1, EMT , EGF, AHR, ERα, CYP1A1, CYP1B1, GREB1, cAMP |
MCF-7, HeLa, Seg-1, T47D, MDA-MB-231 , HCT116, PC12 , 4T1, ZR-75-1, MDA-MB-435, SKBR-3 |
PhytoCAT-226 |
3β,12β,13β-trihydroxy-12,13-dihydrooleanolic acid (2, TOA) |
Vitis vinifera |
NA |
MCF-7/DOX |
PhytoCAT-227 |
3β,13β-dihydroxy-12,13-dihydroursolic acid (7) |
Vitis vinifera |
NA |
MCF-7/DOX |
PhytoCAT-228 |
Artemisia biennis extract |
Artemisia biennis |
NA |
AGS, HeLa, HT-29, MCF-7 |
PhytoCAT-229 |
2-deacetoxytaxinine J (2-DAT-J) |
Taxus baccata |
NA |
MCF-7, MDA-MB-231 |
PhytoCAT-230 |
Papaverine |
Papaver rhoeas |
NA |
MCF-7, MDA-MB-231 |
PhytoCAT-231 |
Cannabidiolic acid |
Cannabis sativa |
COX-2 |
MDA-MB-231 |
PhytoCAT-232 |
Pomaces from Muscadinia rotundifolia |
Muscadinia rotundifolia |
Cyclin A, p21 |
MCF-7, MDA-MB-231 |
PhytoCAT-233 |
Muscadine grape extract (MGE) |
Vitis rotundifolia |
c-met, Cyclin D1 |
Mouse 4T1, MDA-MB-231, BT-549 |
PhytoCAT-234 |
Crataegus gracilior extract |
Crataegus gracilior |
NA |
NA |
PhytoCAT-235 |
Salidroside |
Rhodiola rosea |
NA |
MCF-7, Female BALB/c nude mice |
PhytoCAT-236 |
Fukinolic acid |
Actaea racemosa |
NA |
MCF-7 |
PhytoCAT-237 |
Black cohosh extract |
Black cohosh |
NA |
MDA-MB-453, MCF-7, MDA-MB-231 |
PhytoCAT-238 |
Cimiracemoside A |
Black cohosh |
NA |
MCF-7 |
PhytoCAT-239 |
Linalool |
Erythrina corallodendron |
NA |
MCF-7 |
PhytoCAT-240 |
Peonidin-3-glucoside |
Oryza sativa |
HER2, AKT |
BT-474, HCC1569, MDA-MB-453, 6–7-week-old female nude mice |
PhytoCAT-241 |
Vitexin |
Oryza sativa |
Bax, Caspase 7, Caspase 8, Caspase 9, p53, mdm2, Caspase 3 |
MCF-7 |
PhytoCAT-242 |
Orientin |
Oryza sativa |
MMP9, IL-8 |
MCF-7 |
PhytoCAT-243 |
Capsaicin |
Capsicum annuum |
NA |
MCF-7 |
PhytoCAT-244 |
Tomatine |
Solanum lycopersicum |
MMP2, MMP9, MMP9\NGAL |
MCF-7 |
PhytoCAT-245 |
Lycopene |
Solanum lycopersicum |
BRCA1, BRCA2 |
MDA-MB-231, MCF-7, HT-29, T84 |
PhytoCAT-246 |
3-O-α-L-arabinosyl oleanolic acid (3-O-L-AO) |
Schumacheria castaneifolia |
Bax, p53, Survivin, HIF-1α, HIF-2α |
NA |
PhytoCAT-247 |
Methyl protogracillin (NSC-698792) |
Dioscorea collettii |
NA |
MDA-MB-231 , MCF-7, NCI-ADR-RES, BT-549, MALME-3M, M14, KM12, SF-539, U251MDA-MB-435, |
PhytoCAT-248 |
Methyl protoneodioscin (NSC-698791) |
Dioscorea collettii |
NA |
A549, HCT-116, SF-539, SNB-75, M14, CAKI-1, DU-145, HS 578T, MDA-MB-435 |
PhytoCAT-249 |
Dioscorealide B |
Dioscorea membranacea |
Bax, Bak, Bcl-2, Caspase 8, Caspase 9, Caspase 7 |
NA |
PhytoCAT-250 |
Arachidin-1 |
Arachis hypogaea |
Caspase 9, PARP, Survivin |
MDA-MB-231, MDA-MB-435, MCF-10A |
PhytoCAT-251 |
Arachidin-3 |
Arachis hypogaea |
NA |
MDA-MB-231, MDA-MB-435, MCF-10A |
PhytoCAT-252 |
Ampelopsin E |
Dryobalanops rappa |
PDGF, MMP2, MMP9, MMP14 |
MDA-MB-231, MCF-7, HT-29, A-549, HeLa, 3T3, MCF10A |
PhytoCAT-253 |
Hibifolin |
Helicteres isora |
NA |
MCF-7 |
PhytoCAT-254 |
Chimaphilin |
Passiflora incarnata |
Bcl-2, Bad, Caspase 9, Caspase 3, PARP |
MCF-7 |
PhytoCAT-255 |
Safflower yellow (SY) |
Carthamus tinctorius |
MMP9, p-Src |
MBA-MD-231 |
PhytoCAT-256 |
Adiantum capillus veneris (ACV) extract |
Adiantum capillus |
Bcl-2, Cyclin D1 |
MCF-7, BT47 |
PhytoCAT-257 |
Hyperforin |
Hypericum undulatum |
ER1 |
A431 ,SB1 ,SB3 ,MV3 ,1F6 ,HT144 ,Jurkat ,MCF-7 ,MDA-MB-468 ,SK-OV-3 |
PhytoCAT-258 |
Persin |
Persea americana |
NA |
MCF-7, T-47D, MDA-MB-231 |
PhytoCAT-259 |
Lantana camara extract |
Lantana camara |
Bid, Bax, Bcl-2, Caspase 8, Caspase 9, PARP |
MCF-7 |
PhytoCAT-260 |
Berberis vulgaris extract |
Berberis vulgaris |
NA |
MCF10-A, MCF-7 |
PhytoCAT-261 |
Hancornia speciosa extract |
Hancornia speciosa |
NA |
MN, MCF-7 |
PhytoCAT-262 |
Gaillardin |
Gaillardia pulchella |
Bax, p53, Bcl-2 |
MCF-7, MDA-MB-468 |
PhytoCAT-263 |
Cyperus longus extract |
Cyperus longus |
NA |
PC3, MCF-7 |
PhytoCAT-264 |
Dracocephalum surmandinum essential oil |
Dracocephalum surmandinum |
NA |
MCF-7, K562 |
PhytoCAT-265 |
Flavonoid extract of wheat germ |
Triticum aestivum |
NA |
BCap-37 |
PhytoCAT-266 |
Cyclovirobuxine D (CVB-D) |
Buxus microphylla |
LC3-I, LC3-II, ATG5 |
MCF-7 |
PhytoCAT-267 |
Croton gratissimus extract |
Croton gratissimus |
Caspase 3, Caspase 7 |
MCF-7, Vero, A549, Caco-2, HeLa |
PhytoCAT-268 |
Kongensin D (6) |
Croton kongensis |
AKT, p21, Cyclin B1, CDK1, Bcl-2, Bax, Caspase 3, PARP, β-catenin, MMP2, MMP9 |
MDA-MB-231, MDA-MB-468, MCF-7, TNBC xenograft mouse model |
PhytoCAT-269 |
Euphoranginone D (3) |
Croton kongensis |
NA |
MDA-MB-231, MDA-MB-468, MCF-7 |
PhytoCAT-270 |
Ent-kaurane-3-oxo-16β,17-diol (4) |
Croton kongensis |
NA |
MDA-MB-231, MDA-MB-468, MCF-7 |
PhytoCAT-271 |
Ent-16β-H-3-oxokauran-17-ol (5) |
Croton kongensis |
NA |
MDA-MB-231, MDA-MB-468, MCF-7 |
PhytoCAT-272 |
Kongeniod B (7) |
Croton kongensis |
NA |
MDA-MB-231, MDA-MB-468, MCF-7 |
PhytoCAT-273 |
Kongensin A (8) |
Croton kongensis |
NA |
MDA-MB-231, MDA-MB-468, MCF-7 |
PhytoCAT-274 |
Kongensin F (9) |
Croton kongensis |
NA |
MDA-MB-231, MDA-MB-468, MCF-7 |
PhytoCAT-275 |
Crokongendin A (1) |
Croton kongensis |
NA |
MDA-MB-231, MDA-MB-468, MCF-7 |
PhytoCAT-276 |
Crokongendin B (2) |
Croton kongensis |
NA |
MDA-MB-231, MDA-MB-468, MCF-7 |
PhytoCAT-277 |
Laevifins A |
Croton oblongus |
NA |
MCF-7 |
PhytoCAT-278 |
Laevifins B |
Croton oblongus |
NA |
MCF-7 |
PhytoCAT-279 |
Laevifins G |
Croton oblongus |
NA |
MCF-7 |
PhytoCAT-280 |
Emblica officinalis extract |
Emblica officinalis |
ERα mRNA |
MCF-7, MDA-MB-231 |
PhytoCAT-281 |
Resiniferatoxin |
Euphorbia bicolor |
NA |
MDA-MB-231, MDA-MB-469 |
PhytoCAT-282 |
Ebracteolatain A |
Euphorbia ebracteolata |
NA |
NA |
PhytoCAT-283 |
Jolkinolide B |
Euphorbia fischeriana |
Cyclin D1, Cyclin E, mTOR, PI3K, AKT, PTEN, eIF4E, β1-integrin, FAK, U0126, ERK |
Female Balb/c nude mice, MCF-7, BT-474, MDA-MB-231 |
PhytoCAT-284 |
Euphorin C |
Euphorbia fischeriana |
NA |
MCF-7 |
PhytoCAT-285 |
Euphorin E |
Euphorbia fischeriana |
NA |
MCF-7 |
PhytoCAT-286 |
Euphorin H |
Euphorbia fischeriana |
NA |
MCF-7 |
PhytoCAT-287 |
Ebractenoid C |
Euphorbia fischeriana |
NA |
MCF-7 |
PhytoCAT-288 |
Ebractenoid F |
Euphorbia fischeriana |
NA |
MCF-7 |
PhytoCAT-289 |
Yuexiandajisu E |
Euphorbia fischeriana |
NA |
MCF-7 |
PhytoCAT-290 |
Ingenol-3-palmitate |
Euphorbia fischeriana |
NA |
MCF-7 |
PhytoCAT-291 |
Ingenol-3- myristinate |
Euphorbia fischeriana |
NA |
MCF-7 |
PhytoCAT-292 |
Ingenol-20-myristinate |
Euphorbia fischeriana |
NA |
MCF-7 |
PhytoCAT-293 |
Jolkinol A |
Euphorbia fischeriana |
NA |
MCF-7 |
PhytoCAT-294 |
Paratocarpin E |
Euphorbia humifusa |
NA |
MCF-7 |
PhytoCAT-295 |
Kopetdaghinane A |
Euphorbia kopetdaghi |
Bcl-2, Bax |
MCF-7, OVCAR-3 |
PhytoCAT-296 |
Euphorbia microsciadia extract |
Euphorbia microsciadia |
Let-7, miR-15, miR-16, miR-29, miR-34a |
MDA-MB-231 |
PhytoCAT-297 |
Euphopubescenol |
Euphorbia pubescens |
NA |
MCF-7, NCI-H460, SF-268 |
PhytoCAT-298 |
Euphopubescene |
Euphorbia pubescens |
NA |
MCF-7, NCI-H460, SF-268 |
PhytoCAT-299 |
Euphosorophane A |
Euphorbia sororia |
NA |
MCF-7/ADR |
PhytoCAT-300 |
Euphorbia tirucalli Extracts |
Euphorbia tirucalli |
p21, Bax, Caspase 8 |
MCF-7, MDA-MB 231 |
PhytoCAT-301 |
Rottlerin |
Mallotus philippinensis |
Atg12, Beclin-1, Bcl-2, Bcl-xL, XIAP, cIAP-1, LRP6 |
MDA-MB-231, T47D, PC-3, DU145, MCF-7 |
PhytoCAT-302 |
Terminamines K |
Pachysandra terminalis |
NA |
MDA-MB-231 |
PhytoCAT-303 |
Terminamines L |
Pachysandra terminalis |
NA |
MDA-MB-231 |
PhytoCAT-304 |
Terminamines M |
Pachysandra terminalis |
NA |
MDA-MB-231 |
PhytoCAT-305 |
Terminamines N |
Pachysandra terminalis |
NA |
MDA-MB-231 |
PhytoCAT-306 |
Terminamines O |
Pachysandra terminalis |
NA |
MDA-MB-231 |
PhytoCAT-307 |
Terminamines P |
Pachysandra terminalis |
NA |
MDA-MB-231 |
PhytoCAT-308 |
Terminamines Q |
Pachysandra terminalis |
NA |
MDA-MB-231 |
PhytoCAT-309 |
Terminamines R |
Pachysandra terminalis |
NA |
MDA-MB-231 |
PhytoCAT-310 |
Terminamines S |
Pachysandra terminalis |
NA |
MDA-MB-231 |
PhytoCAT-311 |
(+)-pachysandrine B |
Pachysandra terminalis |
NA |
MDA-MB-231 |
PhytoCAT-312 |
Epipachysandrine-A |
Pachysandra terminalis |
NA |
MDA-MB-231 |
PhytoCAT-313 |
3β-methylamino 16-oxo 5,17(20) cis-pregnadiene |
Pachysandra terminalis |
NA |
MDA-MB-231 |
PhytoCAT-314 |
Z-salignone |
Pachysandra terminalis |
NA |
MDA-MB-231 |
PhytoCAT-315 |
Terminamine H |
Pachysandra terminalis |
NA |
MDA-MB-231 |
PhytoCAT-316 |
3β-methylamino 16-oxo 5,17(20) trans-pregnadiene |
Pachysandra terminalis |
NA |
MDA-MB-231 |
PhytoCAT-317 |
E-salignone |
Pachysandra terminalis |
NA |
MDA-MB-231 |
PhytoCAT-318 |
(+)-spiropachysine |
Pachysandra terminalis |
NA |
MDA-MB-231 |
PhytoCAT-319 |
Terminamines A |
Pachysandra terminalis |
Epithelial growth factor, integrin β |
MDA-MB-231 |
PhytoCAT-320 |
Terminamines B |
Pachysandra terminalis |
Epithelial growth factor |
MDA-MB-231 |
PhytoCAT-321 |
Terminamines C |
Pachysandra terminalis |
Epithelial growth factor |
MDA-MB-231 |
PhytoCAT-322 |
Terminamines D |
Pachysandra terminalis |
Epithelial growth factor |
MDA-MB-231 |
PhytoCAT-323 |
Terminamines E |
Pachysandra terminalis |
Epithelial growth factor |
MDA-MB-231 |
PhytoCAT-324 |
Terminamines F |
Pachysandra terminalis |
NA |
MDA-MB-231 |
PhytoCAT-325 |
Terminamines G |
Pachysandra terminalis |
NA |
MDA-MB-231 |
PhytoCAT-326 |
Pachystermine B |
Pachysandra terminalis |
Epithelial growth factor |
MDA-MB-231 |
PhytoCAT-327 |
Pachystermine A |
Pachysandra terminalis |
Epithelial growth factor |
MDA-MB-231 |
PhytoCAT-328 |
Epipachysamine E |
Pachysandra terminalis |
Epithelial growth factor |
MDA-MB-231 |
PhytoCAT-329 |
Epipachysamine B |
Pachysandra terminalis |
Epithelial growth factor |
MDA-MB-231 |
PhytoCAT-330 |
Terminaline |
Pachysandra terminalis |
Epithelial growth factor |
MDA-MB-231 |
PhytoCAT-331 |
Terminamine I |
Pachysandra terminalis |
NA |
MDA-MB-231 |
PhytoCAT-332 |
Terminamine J |
Pachysandra terminalis |
NA |
MDA-MB-231 |
PhytoCAT-333 |
Secofriedelanophyllemblicine |
Phyllanthus emblica |
NA |
MCF-7 |
PhytoCAT-334 |
Putranjiva roxburghii Seed Extract |
Putranjiva roxburghii |
NA |
PANC-1, MDA-MB 231, HCT-116 |
PhytoCAT-335 |
9-O-demethyltrigonostemone |
Strophioblachia fimbricalyx |
NA |
NCI-H187, KB, MCF-7 |
PhytoCAT-336 |
Biebersteinia multifida extract |
Biebersteinia multifida |
NA |
MCF-7, A2780, HeLa |
PhytoCAT-337 |
2-methoxy-1, 4-naphthoquinone |
Impatiens balsamina |
GLUT1, AKT |
MDA-MB-231 |
PhytoCAT-338 |
Herbacetin |
Ephedra sinica |
TNF-α , IL-1β, JNK, NF-κB, c-met, AKT |
MDA-MB-231, HepG2, RAW 264.7 |
PhytoCAT-339 |
Bursera copallifera extract |
Bursera copallifera |
NA |
MCF-7, MDA-MB-231 |
PhytoCAT-340 |
Avenanthramide-C |
Avena sativa |
NA |
MDA-MB-231 |
PhytoCAT-341 |
Cymbopogon nervatus essential oil |
Cymbopogon nervatus |
NA |
MCF-7, HT29, HCT116 |
PhytoCAT-342 |
Cymbopogon schoenanthus essential oil |
Cymbopogon schoenanthus |
NA |
MCF-7, HT29, HCT116 |
PhytoCAT-343 |
Glyceryl 1-monopalmitate |
Phyllostachys heterocycla |
NA |
MCF-7 |
PhytoCAT-344 |
Corn silk extract |
Zea mays |
p53, Bax, Bcl-2, Caspase 3, Caspase 9 |
MCF-7 |
PhytoCAT-345 |
Calophyllum inophyllum extract |
Calophyllum inophyllum |
Bcl-2, Bax, Cyt-c, p53, Caspase 3 |
MCF-7 cells |
PhytoCAT-346 |
Neobractatin |
Garcinia bracteata |
MBNL2 |
MDA-MB-231 xenografts mouse model, A549, HepG2, T98, MCF-7 |
PhytoCAT-347 |
Naringenin |
Garcinia atroviridis |
Bax, Bcl-2, MAPK, PI3K, IL-6, Caspase 3, Caspase 9 |
T-47D, BT-474, MDA-MB-231, SKBR-3,A549, MDA-MB-435, HepG2 |
PhytoCAT-348 |
Epunctanone |
Garcinia epunctata |
NA |
MDA-MB-231, HCT116CEM/ADR5000, MDA-MB-231-BCRP,HCT116 (p53-/-),U87MG |
PhytoCAT-349 |
Gambogic acid |
Garcinia hanburyi |
Bid |
T47D |
PhytoCAT-350 |
Garcinia hombroniana extract |
Garcinia hombroniana |
NA |
MCF-7, DBTRG , PC-3, U2OS |
PhytoCAT-351 |
Garcinol |
Garcinia indica |
miR-200s, let-7s, NF-κB, E-cadherin, Vimentin, ZEB-1, ZEB-2, STAT-3 |
MDA-MB-231, BT-549/xenograft mouse model |
PhytoCAT-352 |
Garcinia mangostana extract |
Garcinia mangostana |
NA |
PC3, B16F10, MCF-7, U87 |
PhytoCAT-353 |
α-mangostin |
Garcinia mangostana |
MMP2, MMP9, MARK4 |
MCF-7, HepG2 |
PhytoCAT-354 |
5,7-dihydroxy-3-(3'-hydroxy-4',5'-dimethoxyphenyl)-6-methoxy-4H-chromen-4-one |
Garcinia nervosa |
NA |
MCF-7, MDA-MB 231 |
PhytoCAT-355 |
Friedelin |
Garcinia penangiana |
CDKN1a, pRb2, p53, Nrf2, Caspase 3, Bcl-2, mdm2, PCNA |
MCF-7 |
PhytoCAT-356 |
Garcinia quaesita extract |
Garcinia quaesita |
NA |
MDA-MB-231 |
PhytoCAT-357 |
Wightiic acid |
Garcinia wightii |
NA |
MCF-7, SKBR-3, A-375 |
PhytoCAT-358 |
Mammea F/BB |
Mammea americana |
VEGF, HIF-1 |
T47D, PC-3 |
PhytoCAT-359 |
Mammea F/BA |
Mammea americana |
NA |
T47D, PC-3 |
PhytoCAT-360 |
Mammea C/AA |
Mammea americana |
NA |
T47D, PC-3 |
PhytoCAT-361 |
Mammea C/AB |
Mammea americana |
NA |
T47D, PC-3 |
PhytoCAT-362 |
Mammea C/BB |
Mammea americana |
NA |
T47D, PC-3 |
PhytoCAT-363 |
Mammea B/AB |
Mammea americana |
NA |
T47D, PC-3 |
PhytoCAT-364 |
Mammea B/BB |
Mammea americana |
NA |
T47D, PC-3 |
PhytoCAT-365 |
Mammea A/AB |
Mammea americana |
NA |
T47D, PC-3 |
PhytoCAT-366 |
Mammea A/BB |
Mammea americana |
NA |
T47D, PC-3 |
PhytoCAT-367 |
Pristimerin |
Reissantia buchananii |
FASN |
MDA-MB-231 |
PhytoCAT-368 |
Halophila ovalis extract |
Halophila ovalis |
Bcl-2, PARP, Nrf-2, SOD-2, HO-1, Caspase 3 |
MCF-7 |
PhytoCAT-369 |
Cratoxylum cochinchinense extract |
Cratoxylum cochinchinense |
NA |
MDA-MB-468 |
PhytoCAT-370 |
Hyperelodiones A |
Hypericum elodeoides |
NA |
HeLa, MCF-7 |
PhytoCAT-371 |
Hyperelodiones B |
Hypericum elodeoides |
NA |
HeLa, MCF-7 |
PhytoCAT-372 |
Hyperelodiones C |
Hypericum elodeoides |
NA |
HeLa, MCF-7 |
PhytoCAT-373 |
Hypericum salsugineum extracts |
Hypericum salsugineum |
Tyrosinase |
MCF-7, MDA-MB-231 |
PhytoCAT-374 |
2-Methoxystypandrone |
Polygonum cuspidatum |
STAT-3 |
NA |
PhytoCAT-375 |
Crocin |
Crocus sativus |
ERα, HDAC2 |
MKN-28, MCF-7, MDA-MB-231, Caco-2, BALB/c mice |
PhytoCAT-376 |
Ursolic acid |
Prinsepia utilis |
Fas receptor, Caspase 8, Caspase 3, Caspase 9, PARP, Bax, Bcl-2, cyt-c, Nrf2, NQO1, Keap1, miR-499a-5p, mTOR, AKT, MMP2, u-PA, NF-κB, Cyclin D, Cyclin E, CDK4, CDK2, PI3K, AKT, ERK, FoxO1/FoxO3a, DR4, DR5, Cyclin D1, PCNA, p21Waf1/Cip1, PLK1, CCNB1, ABCC1, MiR-186-5p, MAPK1/3, ABCG2 |
A549, HCT116, MDA-MB-231, and CCRF-CEM, 4T1, ,MCF-7, BEL-7402, SPC-A-1, SGC-7901, HeLa, HT-29 , Caco-2, HepG2, HT-29, HDFn, SKBR-3, HeLa S3, KB, HL60, MDA-MB-468, Hep3B |
PhytoCAT-377 |
Vitisin B |
Iris lactea |
FAS |
MDA-MB-231 |
PhytoCAT-378 |
Juglanin |
Juglans mandshurica |
Caspase 3, Caspase 8, Caspase 9, LC3B-II, JNK |
SKBR-3, MCF-7, MDA-MB-231, BT-474, mouse xenograft model |
PhytoCAT-379 |
Martynoside |
Ajuga chamaecistus |
ICI182780, IGFBP3 |
MCF-7 |
PhytoCAT-380 |
Acteoside |
Anisomeles indica |
NA |
MCF-7 |
PhytoCAT-381 |
Ovatodiolide |
Anisomeles indica |
Oct4, Nanog, Hsp27, SMURF2 |
AS-B145, BT-474 |
PhytoCAT-382 |
2alpha-hydroxyursolic acid |
Cunila lythrifolia |
NF-κB |
HepG2, MCF-7, Caco-2 |
PhytoCAT-383 |
Hedeoma drummondii extract |
Mexican poleo |
NA |
MCF-7, HeLa |
PhytoCAT-384 |
Eriocalyxin B |
Isodon eriocalyx |
NF-κBp65, STAT-3 , Bax, Bcl-2, MMP, Caspase 3 |
MCF-7, MDA-MB-231 / MDA-MB-231 xenograft model |
PhytoCAT-385 |
Lavandula angustifolia extract and essential oil |
Lavandula angustifolia |
Bax, PARP |
HeLa, MCF-7 |
PhytoCAT-386 |
Lavandula Coronopifolia extract |
Lavandula coronopifolia |
NA |
MDA-MB-321 |
PhytoCAT-387 |
Motherwort extract |
Leonurus japonicus |
NA |
MCF-7, MDA-MB-231 |
PhytoCAT-388 |
Marrubium crassidens extract |
Marrubium crassidens |
NA |
MCF-7 |
PhytoCAT-389 |
Marrubium persicum extract |
Marrubium persicum |
NA |
MCF-7 |
PhytoCAT-390 |
Melissa officinalis extract |
Melissa officinalis |
NA |
SKOV3, MCF-7 and PC-3, A549 |
PhytoCAT-391 |
14-Deoxy-11,12-didehydroandrographolide |
Andrographis paniculata |
GADD45A/p38 MAPK/DDIT3 |
T-47D |
PhytoCAT-392 |
1,8-cineole |
Nepeta menthoides |
NA |
MCF-7, T47D, MDA-MB-231, A2780 |
PhytoCAT-393 |
Ocimum gratissimum extract |
Ocimum gratissimum |
MMP2, MMP9 |
MDA-MB-231 |
PhytoCAT-394 |
Isothymusin |
Ocimum tenuiflorum |
COX- 2, 5-LOX, CatD, DHFR, hyaluronidase, ODC1 |
NA |
PhytoCAT-395 |
Origanum acutidens extract |
Origanum acutidens |
Caspase 7 |
MCF-7, MDA-MB-468, MDA-MB-231 |
PhytoCAT-396 |
Origanum majorana extract |
Origanum majorana |
Caspase 7, HO-1 , TNF-α, Caspase 8, Caspase 3, PARP, p53, Survivin, γ-H2AX |
MCF-7 |
PhytoCAT-397 |
Salvibuchanic acid |
Salvia buchananii |
NA |
Jurkat, HeLa, MCF-7 |
PhytoCAT-398 |
Hyptadienic acid |
Salvia buchananii |
NA |
Jurkat, HeLa, MCF-7 |
PhytoCAT-399 |
7β-acetoxy-20-hydroxy-19,20-epoxyroyleanone (compound 1) |
Salvia corrugata |
ERK1/2 kinase |
MCF-10A, SKBR-3, BT-474 |
PhytoCAT-400 |
6,7-dehydroroyleanone (3) |
Salvia deserta |
NA |
A549, MDA-MB-231, KB, KB-VIN, and MCF-7 |
PhytoCAT-401 |
7-O-methylhorminone (5) |
Salvia deserta |
NA |
A549, MDA-MB-231, KB, KB-VIN, and MCF-7 |
PhytoCAT-402 |
14-deoxycoleon U (8) |
Salvia deserta |
NA |
A549, MDA-MB-231, KB, KB-VIN, and MCF-7 |
PhytoCAT-403 |
Neotanshinlactone |
Salvia digitaloides |
NA |
HL-60, SMMC-7721, A-549, SKBR-3, PANC-1 |
PhytoCAT-404 |
Salvia fruticosa extract |
Salvia fruticosa |
NA |
MCF-7, T47D, ZR-75-1, BT-474 |
PhytoCAT-405 |
Tanshinone IIA |
Salvia miltiorrhiza |
LC3-II |
MDA-MB-468, PC9, MCF-7, SKBR-3 |
PhytoCAT-406 |
15,16-Dihydrotanshinone I |
Salvia miltiorrhiza |
ERp57 |
MDA-MB-231 |
PhytoCAT-407 |
Salvia miltiorrhiza extract |
Salvia miltiorrhiza |
Nrf2, HO-1 |
MCF-7 |
PhytoCAT-408 |
Salvianolic acid A |
Salvia miltiorrhiza |
Transgelin 2, ABC transporter |
MCF-7/PTX |
PhytoCAT-409 |
Cryptotanshinone |
Salvia miltiorrhiza |
p38/JNK, Erk1/2 |
HepG2 , MCF-7, HA22T |
PhytoCAT-410 |
Rosemary extract |
Rosmarinus officinalis |
TNF-α, IL-1β, iNOS, COX-2 |
HL60, K562, MCF-7, MDA-MB-468, MDA-MB-231 |
PhytoCAT-411 |
Sclareol |
Salvia sclarea |
IL-4, IFN-γ |
MCF-7, breast-cancer-bearing Balb/c mice, HeLa |
PhytoCAT-412 |
Salvia syriaca extract |
Salvia syriaca |
NA |
MCF-7, T47D, ZR-75-1, BT-474 |
PhytoCAT-413 |
Maslinic acid |
Salvia tomentosa |
NA |
MDA-MB-231 |
PhytoCAT-414 |
6-Hydroxyflavone |
Scutellaria baicalensis |
NA |
ZR-75-1 |
PhytoCAT-415 |
Scutellaria baicalensis extract |
Scutellaria baicalensis |
PGE(2) |
HepG2, MCF-7, PC-3, LNCaP, KM-12, HCT-15, KB, SCC-25 |
PhytoCAT-416 |
Wogonoside |
Scutellaria baicalensis |
MST1 |
TNBC cell xenograft model, HEC1A, BALB/c-nu mice |
PhytoCAT-417 |
Xanthomicrol |
Sideritis leucantha |
TNF-α, VEGF, MMP9, Ki67, Bax, Caspase 3, Caspase 9, miR21, miR27, miR125, miR29, miR34 |
4T1, Mouse fibroblast cells |
PhytoCAT-418 |
Hydroxytyrosol |
Teucrium polium |
Beclin-1, p62 |
MDA-MB-231 |
PhytoCAT-419 |
Thymus vulgaris L. essential oil |
Thymus vulgaris |
NA |
MCF-7, NCI-H460, MOLT-4 |
PhytoCAT-420 |
(-)-kunstleramide |
Beilschmiedia kunstleri |
NA |
A-549, Hela, MCF-7, IMR-32 |
PhytoCAT-421 |
Cinnamomum cassia extract |
Cinnamomum cassia |
NA |
MCF-7, MDA-MB-231, HT29 |
PhytoCAT-422 |
Cinnamic Acid |
Goniothalamus laoticus |
TNF-α, TNFR1 , Caspase 8, Caspase 3 |
MDA-MB-231, MCF-7, HeLa, K562 |
PhytoCAT-423 |
Goniothalamin |
Cryptocarya latifolia |
p38, JNK1/2, AKT, Bax, Bcl-2 |
SKBR-3 |
PhytoCAT-424 |
Methyl linderone (ML) |
Lindera erythrocarpa |
STAT-3, AP-1, MMP9, IL-8 |
MCF-7 |
PhytoCAT-425 |
Fisetin |
Acacia carneorum
Acacia buxifolia |
PTEN |
MDA-MB-231, MCF-7, BT-549 |
PhytoCAT-426 |
Acacia etbaica extract |
Acacia etbaica |
NA |
MCF-7, HEPG-2, HCT-116 |
PhytoCAT-427 |
Fraction 35 (F035) |
Acacia victoriae |
AKT |
MDA-MB-453, MDA-MB-435 |
PhytoCAT-428 |
5,7,3',4'-tetrahydroxyisoflavone (THIF) |
Ammopiptanthus mongolicus |
cdc2, Chk1, p53 |
T47D |
PhytoCAT-429 |
Butea monosperma extract |
Butea monosperma |
NA |
MCF-7 |
PhytoCAT-430 |
Sistosterol-3-beta-D-glycoside |
Cassia petersiana |
NA |
NA |
PhytoCAT-431 |
Christia vespertilionis extract |
Christia vespertilionis |
PCNA, Bax, cyt-c, Caspase 8, Caspase 3, Bcl-2 |
MCF-7 |
PhytoCAT-432 |
Chickpea protease inhibitor concentrate |
Cicer arietinum |
NA |
MDA-MB-231, PC-3, LNCaP |
PhytoCAT-433 |
Cyclopia genistoides extract |
Cyclopia genistoides |
NA |
MCF-7-BUS, MDA-MB-231 |
PhytoCAT-434 |
Butein |
Cyclopia subternata |
Aromatase |
MDA-MB-231, MCF-7 |
PhytoCAT-435 |
2',4'-dihydroxy-6'-methoxychalcone |
Erythrina abyssinica |
NA |
MCF-7, A549 |
PhytoCAT-436 |
Isoneorautenol |
Erythrina excelsa |
NA |
MDA-MB-231, CCRF-CEM, HCT116, U87MG |
PhytoCAT-437 |
Derrone |
Erythrina orientalis |
Aurora kinases |
MCF-7, HeLa, KPL4, H1299 |
PhytoCAT-438 |
Gleditsia sinensis extract |
Gleditsia sinensis |
NA |
MCF-7, MDA-MB-231, HepG2 , SLMT-1 |
PhytoCAT-439 |
Isoliquiritigenin |
Glycyrrhiza glabra |
Arg-1, HO-1, iNOS, microRNA 155, SHIP1, STAT-3, STAT6, PLA2, COX-2, CYP4A, PGE2, COX-1, FLAP, 5-LOX, LTB4, HIF-1α, VEGF, MMP2, MM9, Aromatase |
MCF-7, A-549, BGC-823, MDA-MB-231, HepG2 |
PhytoCAT-440 |
Glycyrrhizin |
Glycyrrhiza glabra |
NA |
MDA-MB-231, HeLa, MCF-7 |
PhytoCAT-441 |
Glycyrrhetinic acid |
Glycyrrhiza glabra |
TOPO 2A |
MDA-MB-231 |
PhytoCAT-442 |
Pinocembrin |
Glycyrrhiza glabra |
Cyclin B1, Cdc2, PARP-1, Bcl-2, Survivin, PARP-1, Caspase 3, Caspase 9, Bax, ABCG2 |
MDA-MB-231, MCF-7, HeLa |
PhytoCAT-443 |
Glycybridin D (4) |
Glycyrrhiza glabra |
PTP1B |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-444 |
Glycybridin A (1) |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-445 |
Glycybridin B (2) |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-446 |
Glycybridin C (3) |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-447 |
Glycybridin E (5) |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-448 |
Glycybridin F (6) |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-449 |
Glycybridin G (7) |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-450 |
Glycybridin H (8) |
Glycyrrhiza glabra |
PTP1B |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-451 |
Glycybridin I (9) |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-452 |
Glycybridin J (10) |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-453 |
Glycybridin K (11) |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-454 |
Kanzonol W |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-455 |
3′-hydroxy-4′-O-methylglabridin |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-456 |
Glabrene |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-457 |
Hispaglabridin A (16) |
Glycyrrhiza glabra |
PTP1B |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-458 |
Hispaglabridin B |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-459 |
Kanzonol X |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-460 |
8-prenyl-phaseollinisoflavan |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-461 |
3,4-didehydroglabridin |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-462 |
Kanzonol U |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-463 |
2′-O-demethybidwillol |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-464 |
Glyinflanin H |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-465 |
Kanzonol Y |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-466 |
Glabrone (35) |
Glycyrrhiza glabra |
PTP1B |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-467 |
Lupiwighteone |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-468 |
2,3-dehydrokievitone |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-469 |
Parvisoflavones-A |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-470 |
Isoglabrone |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-471 |
1″,2″-dehydrocyclokievitone |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-472 |
7,2′-dihydroxy-4′-methoxy-8-(3-methyl-2-butenyl) isoflavanone |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-473 |
Glabrol |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-474 |
Xambioona |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-475 |
Shinflavanone |
Glycyrrhiza glabra |
PTP1B |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-476 |
(2S)-abyssinone I |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-477 |
Euchrenone a5 |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-478 |
Kanzonol Z |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-479 |
(2R,3R)-3,4′,7-trihydroxy-3′-prenylflavane |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-480 |
3-hydroxyglabrol |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-481 |
Liquiritigenin |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-482 |
Abyssinone II |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-483 |
[6″,6″-dimethylpyrano(2″,3″:4,5)]-3′-γ,γ-dimethylallyl-2′,3,4′-trihydroxychalcone |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-484 |
Kanzonol C |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-485 |
Kanzonol B |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-486 |
Licoagrochalcone A |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-487 |
Paratocarpins B |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-488 |
Isobavachalcone |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-489 |
Erybacin |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-490 |
Licoagrocarpin |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-491 |
Dehydroglyceollin I |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-492 |
Shinpterocarpin |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-493 |
Glycyrrhiza glabra extract |
Glycyrrhiza glabra |
P450 1B1, CYP1B1, CYP1A1 |
MDA-MB-468 |
PhytoCAT-494 |
Dibenzoylmethane |
Glycyrrhiza inflata |
MMP9 |
MCF‑7 |
PhytoCAT-495 |
Licochalcone A (LCA) |
Glycyrrhiza inflata |
p53, Sp1, PRMT6 |
MDA-MB-231, MCF-7, MCF-10A |
PhytoCAT-496 |
Licochalcone B (LCB) |
Glycyrrhiza glabra |
Cyclin A, CDK2, Cdc25 A, p21, Caspase 3, Caspase 9, Bax, Bcl-2, p53 |
MCF-7 |
PhytoCAT-497 |
Chinese licorice extract |
Glycyrrhiza uralensis |
p53, Bax, p21(waf1/cip1), CDK 2, Cyclin E |
MCF-7 |
PhytoCAT-498 |
2,4-di-tert-butylphenol (HU-2) |
Humboldtia unijuga |
p53 |
MCF-7 |
PhytoCAT-499 |
erythrodiol-3-acetate (HU-1) |
Humboldtia unijuga |
Caspase 7 |
MCF-7, A431 |
PhytoCAT-500 |
Benzo[b]tryptanthrin |
Indigofera tinctoria |
topo I, topo II, MDR1, Caspase 3, PARP |
HCT15, MCF-7 |
PhytoCAT-501 |
2,3,9-Trimethoxypterocarpan |
Pisum sativum |
NA |
MCF-7, T47D, HS578T |
PhytoCAT-502 |
Hyperoside |
Lotus ucrainicus |
Bcl-2, Bax, IL-6 |
MDA-MB-231 |
PhytoCAT-503 |
Barbigerone |
Millettia ferruginea |
P-gp ATPase |
MCF-7/ADR |
PhytoCAT-504 |
Cucurbitacin E |
Hemsleya delavayi |
Cyclin D1, Survivin, XIAP, Bcl-2, Mcl-1, JNK, AKT, ERK |
MDA-MB-231, MDA-MB-468, SW527, MCF-7 |
PhytoCAT-505 |
Deguelin |
Mundulea sericea |
NA |
MDA-MB-231 |
PhytoCAT-506 |
Artemisia santolina extract |
Artemisia santolina |
NA |
AGS, HeLa, HT-29, MCF-7 |
PhytoCAT-507 |
Ebenfuran I |
Onobrychis ebenoides |
IGFBP-3 |
MCF-7, MC3T3-E1, HeLa |
PhytoCAT-508 |
Ebenfuran II |
Onobrychis ebenoides |
NA |
MCF-7, MC3T3-E1, HeLa |
PhytoCAT-509 |
Ebenfuran III |
Onobrychis ebenoides |
NA |
MCF-7, MC3T3-E1, HeLa |
PhytoCAT-510 |
Onobrychis ebenoides extract |
Onobrychis ebenoides |
IGFBP3 |
MCF-7, KS483, HeLa |
PhytoCAT-511 |
Ebenosin |
Onobrychis ebenoides |
NA |
MCF-7, MDA-MB-231 |
PhytoCAT-512 |
Kievitone |
Phaseolus vulgaris |
EGFR kinase |
MCF-7, T47D, SKBR-3 |
PhytoCAT-513 |
7-O-beta-D-glucopyranosylchrysin |
Podocytisus caramanicus |
NA |
MCF-7 |
PhytoCAT-514 |
Psoralen |
Psoralea corylifolia |
Rh123, P-gp, Fra-1, Axin2, β-catenin |
MCF-7/ADR, MCF-7, MDA-MB-231, BALB/c nude mice |
PhytoCAT-515 |
Matrine |
Sophora flavescens |
PTEN, miR-21 , AKT, Bad, p21(/WAF1/CIP1), p27(/KIP1), Bcl-2, Bax, VEGF, VEGFR-2, Caspase 3, Caspase 9, P-gp, MRP1, IKKβ, GRP78, eIF2α, CHOP, p62, mTOR, Topo I, LIN28A/Let-7 |
MCF-7, 4T1 Balb/c mice, MCF-7/ADR, MDA-MB-231, BT-474, MDA-MB-468 |
PhytoCAT-516 |
Sophopterocarpan A |
Sophora flavescens |
NA |
MCF-7 |
PhytoCAT-517 |
Sophora interrupta extract (SEA) |
Sophora interrupta |
NA |
MCF-7, PC-3 |
PhytoCAT-518 |
Piceatannol (PCT)/(PIC) |
Sophora interrupta |
NA |
MCF-7, SKBR-3 |
PhytoCAT-519 |
Tonkinensine B |
Sophora tonkinensis |
Bax, Bcl-2, Caspase 3, Caspase 9 |
MDA-MB-231, 4T1 |
PhytoCAT-520 |
Caulis Spatholobi extract (SET) |
Spatholobus suberectus |
NA |
4T1 / mice model |
PhytoCAT-521 |
Tephrosin |
Tephrosia uniflora |
ABCG2, P-gp |
MCF-7/MX, EPG85.257RDB |
PhytoCAT-522 |
Trigonella berythea extract |
Trigonella berythea |
NA |
MCF-7, U937 |
PhytoCAT-523 |
Fenugreek extract |
Trigonella foenum-graecum |
PI3K, Bax, Bcl-2 |
MCF-7, MDA-MB-231, KAIMRC1, SK-BR3, HL60, K562, HCT8, HCT116 |
PhytoCAT-524 |
Hexadecanoic acid |
Vicia monantha |
NA |
MCF-7, HCT-116, HepG2 |
PhytoCAT-525 |
β-sitosterol |
Vicia monantha |
NA |
MCF-7, HCT-116, HepG2 |
PhytoCAT-526 |
β-amyrin |
Vicia monantha |
NA |
MCF-7, HCT-116, HepG2 |
PhytoCAT-527 |
β-sitosterol-glucoside |
Vicia monantha |
NA |
MCF-7, HCT-116, HepG2 |
PhytoCAT-528 |
Adzuki bean extract |
Phaseolus angularis |
PR mRNA and protein |
MCF-7 |
PhytoCAT-529 |
Allium atroviolaceum extract (FAA) |
Allium atroviolaceum |
p53, Bcl-2, CDK-1, Caspase 3 |
MCF-7, MDA-MB-231 |
PhytoCAT-530 |
Allium autumnale extract |
Allium autumnale |
NA |
MCF-7, MDA-MB-231 |
PhytoCAT-531 |
Allium bakhtiaricum extracts |
Allium bakhtiaricum |
NA |
MDA-MB-231, MCF-7, 4T1 BALB/c mice, HepG2, HT-29 |
PhytoCAT-532 |
2-Methylpyridine-1-ium-1-sulfonate |
Allium hirtifolium |
Bax, Bcl-2, Caspase 3, Caspase 9, VEGF, MMP2, MMP9, p21, p27, p53 |
MCF-7, MDA-MB-231 |
PhytoCAT-533 |
Allium hirtifolium extract |
Allium hirtifolium |
NA |
HeLa, MCF-7 , L929 |
PhytoCAT-534 |
Allicin |
Allium sativum |
Caspase 3, Caspase 8, Caspase 9, NOXA, p21, Bak, Bcl-xL |
HeLa , MCF-7, L929, A549, HT29, HUVEC, HCC-70 |
PhytoCAT-535 |
Alliin |
Allium sativum |
NA |
MCF-7, HCC-70 |
PhytoCAT-536 |
Thiosulfinates |
Allium tuberosum |
NA |
MCF-7, SW480, HepG2, LNCaP.FGC, mice |
PhytoCAT-537 |
Diallyl disulphide |
Allium vineale |
Bax, Bcl-2, Bcl-w, Bcl-xL |
MCF-7 |
PhytoCAT-538 |
Aloe perryi extract |
Aloe perryi |
NA |
HepG2, HCT-116, MCF-7, A-549, PC-3, HEp-2 and HeLa |
PhytoCAT-539 |
Aloe-emodin |
Aloe vera |
Bcl-2, Bax, NF-κB, p38, ERK, miR-15a, miR-16-1, IL-1β, IL-6, VEGF, MMP2, MMP9 |
MCF-10A, MCF-10AT, MCF-7, MDA-MB-231, 4T1 |
PhytoCAT-540 |
Aloe vera extract |
Aloe vera |
Cyclin D1, CYP 1A1, CYP 1A2, Bax, p21 |
MCF-7, Hela |
PhytoCAT-541 |
Aloin |
Aloe vera |
Topo II alpha, Cyclin B1 |
MCF-7, SKBR-3 |
PhytoCAT-542 |
Gracillin (NSC-698787) |
Dioscorea collettii |
NA |
CCRF-CEM, RPMT-8226, KM12, SF-539, U251, M14, 786-0, DU-145, MDA-MB-435 |
PhytoCAT-543 |
5,6-anhydrohupehenine |
Fritillaria hupehensis |
NA |
MCF-7, HepG2 |
PhytoCAT-544 |
Kwanzoquinones A |
Hemerocallis fulva |
NA |
NA |
PhytoCAT-545 |
Kwanzoquinones B |
Hemerocallis fulva |
NA |
NA |
PhytoCAT-546 |
Kwanzoquinones C |
Hemerocallis fulva |
NA |
NA |
PhytoCAT-547 |
Kwanzoquinones E |
Hemerocallis fulva |
NA |
NA |
PhytoCAT-548 |
Hyacinthus orientalis extract |
Hyacinthus orientalis |
NA |
Balb/C mice, MCF-7, T47D, EMT6/P |
PhytoCAT-549 |
Liriopem I (1) |
Liriope muscari |
NA |
MDA-MB-435 |
PhytoCAT-550 |
Liriopem II (2) |
Liriope muscari |
NA |
MDA-MB-435 |
PhytoCAT-551 |
Liriope platyphylla extract |
Liriope platyphylla |
AKT, Bcl-2, Bcl-xL, Survivin |
MCF-7, MDA-MB-231, Huh-7, Hep 3B, A549 |
PhytoCAT-552 |
Polyphyllin VI |
Paris polyphylla Sm |
Rell2, miR-18a |
Mouse mammary carcinoma 4T1, MDA-MB-231 |
PhytoCAT-553 |
Polyphyllin D |
Paris polyphylla |
Beclin-1, Caspase 3 |
NA |
PhytoCAT-554 |
Smilax china extract |
Smilax china |
TIMP1, TIMP2, uPA, uPAR |
MDA-MB-231 |
PhytoCAT-555 |
(+)-Dihydrokaempferol |
Manilkara zapota. |
NA |
BT-474, Chago-K1, HepG2, KATO-III, SW620 |
PhytoCAT-556 |
Smilax spinosa extract |
Smilax spinosa Miller |
CYP1A1, p21, STAT-3, Caspase 9, Caspase 8, Caspase 3 |
MCF-7, MDA-MB-231, HL60 |
PhytoCAT-557 |
Secoisolariciresinol diglucoside |
Linum usitatissium |
ps2, Bcl-2, IGF-1R, ERα, ERbeta, EGFR, Bcl-2 mRNA, PMAPK protein, p65, NF-κB |
C57BL/6 mice, E0771, MDA-MB-231, MCF-7 |
PhytoCAT-558 |
Colchicine |
Buddleja davidii |
NA |
Mgc-803, BCap-37, MDA-MB-435, MDA-MB-231, OVCAR3 |
PhytoCAT-559 |
Strychnos nux-vomica extract |
Strychnos nux-vomica |
NA |
MCF-7, Hep-2, HCT |
PhytoCAT-560 |
Kaempferol-7 glucoside |
Strychnos nux-vomica |
NA |
MCF-7, Hep-2, HCT |
PhytoCAT-561 |
7-Hydroxy coumarin |
Strychnos nux-vomica |
NA |
MCF-7, Hep-2, HCT |
PhytoCAT-562 |
Quercetin-3-rhamnoside |
Strychnos nux-vomica |
NA |
MCF-7, Hep-2, HCT |
PhytoCAT-563 |
Kaempferol 3-rutinoside |
Strychnos nux-vomica |
NA |
MCF-7, Hep-2, HCT |
PhytoCAT-564 |
Dendrophthoe pentandra extract |
Dendrophthoe pentandra |
TUBB3, MAP4 |
MCF-7 |
PhytoCAT-565 |
Corosolic acid |
Lagerstroemia speciosa |
NA |
ACHN , A498, MDA-MB-231, SK-Hep1, Huh7, T47D, HT-29, K-562, MCF-7 |
PhytoCAT-566 |
Delphinidin |
Punica granatum |
Cyclin B1, CDK-1, NF-κB, NF-κB/p65, PKCalpha, IKKalpha/beta, IkappaBalpha, STAT-3, MMP9, HER2, PARP, Caspase 3, Bcl-2, BAX, EGFR, AKT, MAPK, PI3K |
MDA-MB-453, AU-565, MCF-10A, MCF-7, BT-474 |
PhytoCAT-567 |
Punica granatum extract |
Punica granatum |
Sp1, Sp3, Sp4, miR-27a, ZBTB10, SHIP-1, miRNA-155, AKT |
BT-474, MDA-MB-231, MCF-7 |
PhytoCAT-568 |
Tricetin |
Punica granatum |
Bax, Bak, p21, cdc2, cdc25C, Cyclin B, Bcl-2, Bcl-xL, ABCG2 |
MCF-7 |
PhytoCAT-569 |
Punicalagin |
Punica granatum |
NA |
MCF-7, Hs578T |
PhytoCAT-570 |
Gomisin H |
Schisandra viridis |
NA |
MCF-7, CAL27, HEK293 |
PhytoCAT-571 |
Schisandrin |
Schisandra viridis |
NA |
MCF-7, CAL27, HEK293 |
PhytoCAT-572 |
Angeloylgomisin H |
Schisandra viridis |
NA |
MCF-7, CAL27, HEK293 |
PhytoCAT-573 |
(+)-gomisin M2 |
Schisandra viridis |
NA |
MCF-7, CAL27, HEK293 |
PhytoCAT-574 |
Schisanol |
Schisandra viridis |
NA |
MCF-7, CAL27, HEK293 |
PhytoCAT-575 |
Strobilanthes crispa extract |
Strobilanthes crispa |
Caspase 8 |
HepG-2, MDA-MB-231 |
PhytoCAT-576 |
Betulin |
Hibiscus Syriacus |
Bax, NOXA, PUMA, PERP, Bcl-x, TAp63, p21, Caspase 3, Bak, Caspase 7, Caspase 9, PARP |
HBL-100, MDA-MB-231, H184B5F5/M10, MCF-7, K562, HeLa, HepG2, A549, SK-HEP-1, PC-3, NCI-H460 |
PhytoCAT-577 |
Hibiscus syriacus extract |
Hibiscus syriacus |
AKT |
MDA-MB-231, HBL-100 |
PhytoCAT-578 |
Gossypol |
Cotton plant (Gossypium species), Thespesia populnea |
Bcl-2, Bcl-xL |
MCF-7, SiHa, Caco -2, HeLa, MCF-7/Adr, T-47D, HS 683, U373, U87 and U138 , C6 , SW-13 , SK-MEL-3, Colo 201 , KB, HT-29 |
PhytoCAT-579 |
Angustifolianin |
Aglaia angustifolia |
NA |
MCF-7 |
PhytoCAT-580 |
Amoora chittagonga extract |
Amoora chittagonga |
NA |
MCF-7, HTB-126, Panc-1, Mia-Paca2, Capan1 |
PhytoCAT-581 |
Aglaiabbreviatin E (AA-5) |
Aglaia abbreviata |
Caspase 9 |
MCF-7, MCF-7/ADM |
PhytoCAT-582 |
Aglaiabbreviatin F (AA-6) |
Aglaia abbreviata |
Caspase 9, P-gp |
MCF-7, MCF-7/ADM |
PhytoCAT-583 |
Amoora rohituka extract |
Amoora rohituka |
NA |
MCF-7, HTB-126, Panc-1, Mia-Paca2, and Capan1 |
PhytoCAT-584 |
Amooranin |
Amoora rohituka |
Caspase 8 |
MCF-7, MCF-7/TH, MCF-10A |
PhytoCAT-585 |
7α-hydroxy-β-sitosterol |
Chisocheton tomentosus |
Bax, Bcl-2, procaspase 9, procaspase 3, ERK1/2, FasL, Bim |
MCF-7, HMEC, HSC-4, HepG2 |
PhytoCAT-586 |
Rohitukine |
Dysoxylum binectariferum |
NA |
MCF-7, T47D, MDA-MB-273, SKOV3, NCI/ADR-RES |
PhytoCAT-587 |
Toosendanin (TSN) |
Melia azedarach |
ABCB1, PI3K P110α, P110β, Procaspase 3, Procaspase 9, Bcl-xL, LC3B, Beclin-1, PI3K |
MDA-MB-231, BT-549, 4T1 xenograft tumor |
PhytoCAT-588 |
Isotoosendanin (ITSN) |
Melia azedarach |
Procaspase 3, Procaspase 10, Bcl-xL, Beclin-1, LC3B |
MDA-MB-231, BT-549, 4T1 xenograft tumor |
PhytoCAT-589 |
17-ethylene-3,4-dihydroxy-14-methyl-18-norandrostene-16-one |
Melia azedarach. |
Bax, Bcl-2 |
T47D |
PhytoCAT-590 |
17-ethylene-3,4-dihydroxy-5-pregnene-16-one |
Melia azedarach. |
Bax, Bcl-2 |
T47D |
PhytoCAT-591 |
Turraea nilotica extract |
Turraea nilotica |
NA |
4T1, HEp2, Vero |
PhytoCAT-592 |
Turraea robusta extract |
Turraea robusta |
NA |
4T1, HEp2, Vero |
PhytoCAT-593 |
Azadirone |
Turraea nilotica
Turraea robusta |
NA |
4T1, HEp2, Vero |
PhytoCAT-594 |
12α-acetoxy-7-deacetylazadirone |
Turraea nilotica
Turraea robusta |
NA |
4T1, HEp2, Vero |
PhytoCAT-595 |
Mzikonone |
Turraea nilotica
Turraea robusta |
NA |
4T1, HEp2, Vero |
PhytoCAT-596 |
Azadironolide |
Turraea robusta |
NA |
4T1, HEp2, Vero |
PhytoCAT-597 |
11-epi-Toonacilin |
Turraea robusta |
NA |
4T1, HEp2, Vero |
PhytoCAT-598 |
Niloticin |
Turraea nilotica |
NA |
4T1, HEp2, Vero |
PhytoCAT-599 |
Hispidol B |
Turraea nilotica |
NA |
4T1, HEp2, Vero |
PhytoCAT-600 |
Piscidinol A |
Turraea nilotica |
NA |
4T1, HEp2, Vero |
PhytoCAT-601 |
Sinomenine |
Sinomenium acutum |
TRAP, OSCAR, c-Fos, NFATc1, hIL-8, IL-8/CXCR1, MMP2, MMP9 |
Tumor-bearing mice, MDA-MB-231 |
PhytoCAT-602 |
6,7-di-O-acetylsinococuline (FK-3000) |
Stephania delavayi |
NF-kB, COX-2, cyclin B, p-CDC2 |
MDA-MB-231 xenografted mice, MCF-7, MDA-MB-231, PC-3, HT-29 |
PhytoCAT-603 |
Sinococuline |
Stephania delavayi |
NA |
MDA-MB-231 xenografted mice, MCF-7, MDA-MB-231, PC-3, HT-29 |
PhytoCAT-604 |
Stephania delavayi extract |
Stephania delavayi |
NA |
MDA-MB-231 xenografted mice, MCF-7, MDA-MB-231, PC-3, HT-29 |
PhytoCAT-605 |
Cepharanthine |
Stephania epigaea |
Atg7, AMPK |
MDA-MB-231, HeLa, A549, MCF-7, PC3, HepG2, Hep3B, 50MT-1, HL-60, H1299, SMMC-7721, SW480 |
PhytoCAT-606 |
Isotrilobine |
Stephania japonica |
NA |
MCF-7/ADR |
PhytoCAT-607 |
Trilobine |
Stephania japonica |
NA |
MCF-7/ADR |
PhytoCAT-608 |
Cudraticusxanthone A |
Cudrania tricuspidata |
MMP9, IκBα |
MCF-7 cells, MDA-MB-231 |
PhytoCAT-609 |
Moringa oleifera (MOLSr) extracts (M1S9) |
Moringa oleifera |
SFRP1, Bax, p53, Caspase 8, CaN, SLC39A6, VEGF |
MDA-MB-231 xenograft breast tumor mice, MCF-7 |
PhytoCAT-610 |
Moringa stenopetala extract |
Moringa stenopetala |
MTAP, CDKN2A |
MCF-7, HepG2, HCT-116 |
PhytoCAT-611 |
Dichlorodiaportinol A |
Myoporum bontioides (endophytic fungus Trichoderma sp. 09) |
NA |
MCF-7, HepG2 |
PhytoCAT-612 |
(-)-5,6-dihydro-6-undecyl-2H-pyran-2-one |
Horsfieldia superba |
NA |
PC-3, HCT-116, MCF-7 |
PhytoCAT-613 |
(-)-5,6-dihydro-6-tridecyl-2H-pyran-2-one |
Horsfieldia superba |
NA |
PC-3, HCT-116, MCF-7 |
PhytoCAT-614 |
Anacardic acid |
Anacardium occidentale |
SCD, INSIG1,TGM2, PDK4, GPR176, ZBT20, GRP78, Hsp70, CDK-4, MMP9, Bcl-2, Mcl-1 , miR-378g, Cyclin D1, MYC, c-FOS, PPARγ, SIN3 |
MDA-MB-231, MCF-7 |
PhytoCAT-615 |
Erythro-austrobailignan-6 (EA6) |
Machilus thunbergii |
HER2/EGFR/integrinβ3, topo II |
MCF-7, 4T1 |
PhytoCAT-616 |
Meso-monomethyl dihydroguaiaretic acid |
Machilus thunbergii |
NA |
MCF-7, HT-29 |
PhytoCAT-617 |
Meso-dihydroguaiaretic acid (MDGA) |
Myristica argentea |
EGFR,Src, CDK-4, cyclin D1, integrin β3 |
MCF-7, 4T1, HT-29 |
PhytoCAT-618 |
Nectandrin-B |
Myristica argentea |
17beta-hydroxysteroid dehydrogenase, Aromatase |
MCF-7 |
PhytoCAT-619 |
(-)-Acuminatin |
Machilus thunbergii |
NA |
MCF-7, HT-29 |
PhytoCAT-620 |
Achyranthoside H methyl ester |
Achyranthes fauriei |
PARP |
MCF-7, MDA-MB-453 |
PhytoCAT-621 |
Ardisiphenol A |
Ardisia colorata |
NA |
FM3A |
PhytoCAT-622 |
Ardisiphenol B |
Ardisia colorata |
NA |
FM3A |
PhytoCAT-623 |
Ardisiphenol C |
Ardisia colorata |
NA |
FM3A |
PhytoCAT-624 |
Alkylresorcinol A |
Ardisia colorata |
NA |
FM3A |
PhytoCAT-625 |
Alkylresorcinol B |
Ardisia colorata |
NA |
FM3A |
PhytoCAT-626 |
Alkylresorcinol C |
Ardisia colorata |
NA |
FM3A |
PhytoCAT-627 |
AG36 |
Ardisia gigantifolia |
Cyclin B1, Cyclin D1, FAK, AKT, VEGF, VEGFR2, Caspase 3, Caspase 8, Bax, Bcl-2, Fas, FasL, TNFR1, DR5, cyt-c |
MCF-7, MDA-MB-231, SKBR-3, BALB/c nude mice |
PhytoCAT-628 |
2',4'-dihydroxy-6'-methoxy-3',5'-dimethylchalcone (ON-III) |
Eugenia aquea |
Bim, erbB-2, MAPK, AKT, PARP, Caspase 3, KDR |
MDA-MB-453, A549 |
PhytoCAT-629 |
Polymethoxyflavones |
Citrus sinensis |
NA |
MCF-7 |
PhytoCAT-630 |
Myrtus communis essential oil |
Myrtus communis |
NA |
MCF-7, P815 |
PhytoCAT-631 |
Psidium guajava essential oil |
Psidium guajava |
NA |
MCF-7, HeLa, M059J |
PhytoCAT-632 |
Glycitein |
Glycine max |
Bcl-2, Bax, MAPK, STAT-3 |
SKBR-3, MCF-7 |
PhytoCAT-633 |
Morin |
Psidium guajava
Cudranaia tricuspidata |
RAD51, H2AA.X, Caspase 3, Caspase 7, p38, JNK, PARP |
SKBR‑3 |
PhytoCAT-634 |
Clove |
Syzygium aromaticum |
NA |
MCF-7, MDA-MB-231, HeLa, DU-145 |
PhytoCAT-635 |
Syzygium aromaticum extract (SA-EXT) |
Syzygium aromaticum |
NA |
MCF-7, HeLa, NCI-H-460 |
PhytoCAT-636 |
Actinocephalus divaricatus extract |
Actinocephalus divaricatus |
NA |
LM3, LP07, MCF-7 |
PhytoCAT-637 |
Kelussia odoratissima Mozaff. extract |
Kelussia odoratissima |
Bax, Bcl-2, p21, p27 |
MCF-7, LA7, MCF-10A |
PhytoCAT-638 |
Amorphophallus paeoniifolius extract |
Amorphophallus paeoniifolius |
Bcl-2, Bax, Caspase 7, PARP |
MCF-7, MDA-MB-231 |
PhytoCAT-639 |
Yuehchukene |
Murraya paniculata |
NA |
MCF-7, MDA-MB-231 |
PhytoCAT-640 |
Genistein |
Genista tinctoria |
miR-155, BRCA1 , PI3K/AKT, CDK2, Cyclin D1, VEGF, MMP2, MMP9, uPA, Cyclin B1, mir-23b, NF-κB, p53, Chk2, GPR30-Akt, pRb105, FOXO3, PTEN, casein kinase, p27, UPR, GRP78, IRE1α, ATF4, Beclin-1, TGFβ, Foxp3, CD8a, PI, PIPK, Aromatase, ATRX, SUV39H1/H2, HP1BP3, KLf4, hTERT, CDK1, ER-beta, BRCA1, TNF, BARD1, p53, pS2, jun, BAX, BAP1, BARD1, BRCA2 |
MCF-7, MDA-MB-231, SK-N-SH, MDA-MB-468, T47D, MCF-12A, HepG2, PC12, BT-549, MDA-MB-435, G-292, SKBR-3, MMTV-Wnt-1 , BT-20, MDA468, GLC4/ADR, SW-1573/2R120, HT1080/DR4, MCF-7/Mitox, HL60/ADR, UACC-3199, MCF-10F, MDA-MB-435, Hs578t, |
PhytoCAT-641 |
Daidzein |
Glycine max |
BRCA1 ,BRCA2, VEGF-A, CXCL16, CDK1 , Cyclins A, Cyclin B, Cyclin D, CDK2, CDK4, p21(Cip1), p57(Kip2), caspase 9, ERα, c‑erbB‑2, AKR1BI, HRAS, GSTP1, p53, pS2, jun, GADD45, BAX, TNF, Rb1, p300 |
MCF-7, MDA MB-231, PC12, MCF10a, T47D, G-292, SKBR-3, HS578T, ZR‑75‑1 , MMTV-neu, MDA-MB-453 |
PhytoCAT-642 |
Glyceollin |
Glycine max |
NGFR |
HEK 293, MCF-7,nu/nu immune-compromised female ovariectomized mice, BG-1 |
PhytoCAT-643 |
Lunasin |
Glycine max |
MMP2, MMP9, NOS, IL-1, IL-6, TNF-α, Src, Akt, ERK, NF-κB, MCP-1 |
MDA-MB-231, 4T1 |
PhytoCAT-644 |
Coumestrol |
Glycine max |
BCRP, Aromatase, ER |
MCF-7, HCT116, T47D, MDA-MB-231 |
PhytoCAT-645 |
Bowman-Birk protease inhibitor |
Glycine max |
Atg5, Beclin-1, LC 3-II, Sequestosome1, Bax, Bcl-2 |
MDA-MB-231 |
PhytoCAT-646 |
(2S)-5,7,2',6'-tetrahydroxy-6,8-di (gamma,gamma-dimethylallyl) flavanone |
Patrinia villosa |
NA |
MCF-7, BEL-7402, HT-29, SGC-7901, K562, A498, A549 |
PhytoCAT-647 |
(2S)-5,7,2',6'-tetrahydroxy-6-lavandulylated flavanone |
Patrinia villosa |
NA |
MCF-7, BEL-7402, HT-29, SGC-7901, K562, A498, A549 |
PhytoCAT-648 |
(2S)-5,7,2',6'-tetrahydroxy-4'-lavandulylated flavanone |
Patrinia villosa |
NA |
MCF-7, BEL-7402, HT-29, SGC-7901, K562, A498, A549 |
PhytoCAT-649 |
(2S)-5,2',6'-trihydroxy-2'',2''-dimethylpyrano [5'', 6'': 6, 7] flavanone |
Patrinia villosa |
NA |
MCF-7, BEL-7402, HT-29, SGC-7901, K562, A498, A549 |
PhytoCAT-650 |
(2S, 3''S)-5,2',6'-trihydroxy-3''-gamma,gamma-dimethylallyl-2'',2''-dimethyl-3'',4''-dihydropyrano [5'', 6'': 6, 7] flavanone |
Patrinia villosa |
NA |
MCF-7, BEL-7402, HT-29, SGC-7901, K562, A498, A549 |
PhytoCAT-651 |
Licoagrochalcone B |
Patrinia villosa |
NA |
MCF-7, BEL-7402, HT-29, SGC-7901, K562, A498, A549 |
PhytoCAT-652 |
Gomisin J |
Schisandra chinensis |
p62, SQSTM1, LC3-I |
MCF-7, MDA-MB-231, BT-20, BT-549, T47D, SKBR-3, MDA-MB-453, HS578T, MDA-MB-468, HCT116, HT-29, HeLa, SiHa |
PhytoCAT-653 |
Erianin |
Dendrobium nobile |
Bcl-2 |
T47D, MDA-MB-231, MCF-7 |
PhytoCAT-654 |
Kaempferol-3-O-rhamnoside |
Schima wallichii |
Caspase 9, Caspase 3, PARP |
MCF-7, HC-04 |
PhytoCAT-655 |
Pseudolaric acid B |
Pseudolarix kaempferi |
HIF-1α, Caspase 8, Caspase 9, Cyclin B1 |
MDA-MB-468, MDA-MB-435, L929, MRC5, SW579, MCF-7 |
PhytoCAT-656 |
Croblongifolin |
Croton oblongifolius |
NA |
HEP-G2, SW620, CHAGO, KATO3, BT-474 |
PhytoCAT-657 |
Crovatin |
Croton oblongifolius |
NA |
HEP-G2, SW620, CHAGO, KATO3, BT-474 |
PhytoCAT-658 |
Nidorellol |
Croton oblongifolius |
NA |
HEP-G2, SW620, CHAGO, KATO3, BT-474 |
PhytoCAT-659 |
Jerantinine A |
Tabernaemontana corymbosa |
SF3B1, SF3B3 |
MCF-7, MDA-MB-468, T47D, MCF-10A |
PhytoCAT-660 |
Maesa macrophylla extract |
Maesa macrophylla |
NA |
MCF-7, HepG2, HeLa |
PhytoCAT-661 |
Artemisia indica extract |
Artemisia indica |
NA |
MCF-7, HepG2, HeLa |
PhytoCAT-662 |
Phlogacanthus thyrsiformis extract |
Phlogacanthus thyrsiformis |
NA |
MCF-7, HepG2, HeLa |
PhytoCAT-663 |
Pistacia integerrima extract |
Pistacia integerrima |
NA |
MCF-7 |
PhytoCAT-664 |
Nelumbo nucifera extract |
Nelumbo nucifera |
CTGF |
MDA-MB-231, SKBR-3, HCC1806 |
PhytoCAT-665 |
Camptothecine |
Miquelia dentata |
NA |
MDA-MB-273, NCI/ADR-RES, SKOV, HepG2, Hep3B, MDA-MB- 231, MCF-7, A549, Ca9-22, NCI/ADR-RES, Hela, HCT116, GI 101A, MDA-MB-157 |
PhytoCAT-666 |
Arctiin |
Forsythia koreana |
STAT3, TGF-β1, TLR4, NLRP3, VEGF, and cyclin D1 |
MCF-7, HeLa, SiHa |
PhytoCAT-667 |
Cabralealactone 3-acetate-24-methyl ether |
Forsythia koreana |
NA |
MCF-7 |
PhytoCAT-668 |
Fraxetin (FXT) |
Fraxinus bungeana |
Fas, FasL, Bax, Bcl-2 |
MCF-7, HCC827, H1650, A549, H460, PC-9, H1975 |
PhytoCAT-669 |
Olea europaea extract |
Olea europaea |
Aromatase, CYP19A1 |
MCF-7 |
PhytoCAT-670 |
Grammatophyllum speciosum extract |
Grammatophyllum speciosum |
AKT, β-catenin |
MCF-7 |
PhytoCAT-671 |
Crinum amabile extract |
Crinum amabile |
NA |
MCF-7, MDA-MB-231, HCT-116, HT-29 |
PhytoCAT-672 |
(2S)-5,2',6'-trihydroxy-6-lavandulyl-4''-(gamma,gamma-dimethylallyl)-2'',2''-dimethylpyrano-[5'',6'' : 7,8]-flavanone |
Spiranthes australis |
NA |
MCF-7, BEL-7402, HT-29, SGC-7901, K562, A498 |
PhytoCAT-673 |
Verbascoside |
Orobanche amethystea |
Caspase 3, Bax, Bcl-2, TLR4, MyD88, NF-κB |
4 T1, MCF-7, MDA-MB-231 |
PhytoCAT-674 |
Orobanche crenata extract |
Orobanche crenata |
NA |
HepG2, PC3, MCF-7, and HCT-116 |
PhytoCAT-675 |
Pancratium maritimum extract |
Pancratium maritimum |
Cyclin B1, Bcl-2, Ki67 |
C32, HeLa, MDA-MB-231, PC3, A549, MCF-7, and LNCaP |
PhytoCAT-676 |
Euterpe oleracea Mart. extract |
Euterpe oleracea |
NA |
MCF-7 |
PhytoCAT-677 |
Livistona chinensis extract |
Livistona chinensis |
PAK2, PKA, PKC, GSK-3alpha, CK2, MAPK, JNK1, EGF |
HeLa, A431, MCF-7, NPC-TW02 and -TW04 |
PhytoCAT-678 |
Lycorine |
Sternbergia clusiana |
Mcl-1, Bcl-xL, MMP2, MMP9, SHP-1, STAT-3 |
Nude mouse models, A549, HCT116, SK-OV-3, NCI-H460, K562, MCF-7 and HL-60 |
PhytoCAT-679 |
Formosanin C |
Trachycarpus fortunei |
NA |
MCF-7, MDA-MB-231 |
PhytoCAT-680 |
Pandanus amaryllifolius extract |
Pandanus amaryllifolius |
Caspase 8, Caspase 9, Caspase 3, Caspase 7 |
MDA-MB-231 |
PhytoCAT-681 |
Govaniadine |
Corydalis govaniana |
Bax, p53, Survivin, Caspase 7 |
MCF-7 |
PhytoCAT-682 |
Corydalis saxicola Bunting total alkaloids (CSBTA) |
Corydalis saxicola |
RANKL/OPG |
MDA-MB-231 |
PhytoCAT-683 |
Glaucine |
Corydalis turtschaninovii |
MMP9, NF-κB |
MDA-MB-231 |
PhytoCAT-684 |
Leptopidine |
Hypecoum leptocarpum |
FAS |
NA |
PhytoCAT-685 |
Noscapine |
Papaver somniferum |
Bcl-xL, Bcl-2 |
MCF-7 and MDA-MB-231 |
PhytoCAT-686 |
Sanguinarine |
Sanguinaria canadensis |
STAT-3 , XIAP, Caspase 3, Bcl-2, cIAP2, XIAP, c-FLIPs, p21, p27, Cyclin D1, Topoisomerase II |
NA |
PhytoCAT-687 |
Esculentoside A |
Phytolacca acinosa |
ALDH1A1, Sox2, Oct4, Bax, Caspase 3, Bcl-2, STAT3 |
BALB/c mice, MCF-7 |
PhytoCAT-688 |
Anemopsis californica extract |
Anemopsis californica |
ERK1/2 |
NA |
PhytoCAT-689 |
Piperlongumine |
Piper longum |
SETDB1, EGFR, STAT-3, ZBTB4, Sp1, Sp3, Sp4, Cyclin D1, Survivin, cMyc, EGFR |
A549, 786-O, SKBR-3, Female athymic nu/nu mice |
PhytoCAT-690 |
Crude extract of piperine free P. nigrum |
Piper nigrum |
p53, ER, E-cadherin, MMP9, MMP2, c-Myc, VEGF, E-cadherine, c-Myc |
mammary tumorigenesis rats and breast cancer cell lines MCF-7 and ZR-75-1. |
PhytoCAT-691 |
Asaricin |
Piper sarmentosum |
Bcl-2, Bax |
MDA-MB-231 |
PhytoCAT-692 |
Isoasarone |
Piper sarmentosum |
Bcl-2, Bax |
MDA-MB-231 |
PhytoCAT-693 |
Saururus chinensis extract |
Saururus chinensis |
VEGF, Cyclin D1, Bcl-2, Caspase-3 |
LNCaP, MCF-7 |
PhytoCAT-694 |
Sinapinic acid |
Limoniastrum guyonianum |
NA |
MCF-7, HeLa |
PhytoCAT-695 |
Plumbagin |
Plumbago zeylanica |
NQO1, NF-kB, MMP9, Akt, IKKalpha |
MCF-7, MDA-MB-231, HeLa, A549 |
PhytoCAT-696 |
Pterostilbene |
Vitis rupestris |
Beclin-1, LC3 II, hTERT, cMyc, Cyclin D1, Rac1, WAVE-2, Arp2/3 |
MCF-7,MDA-MB-231 , T-47D, NCI H-460 |
PhytoCAT-697 |
Maprang seed extract |
Bouea macrophylla |
Bax, Bcl-2 |
MCF-7 |
PhytoCAT-698 |
Kaempferol-3-O-β-D-(6″-n-butyl glucuronide) |
Calligonum polygonoides |
NA |
MCF-7, HepG2 |
PhytoCAT-699 |
Quercetin 3-O-β-D-(6″-n-butyl glucuronide) |
Calligonum polygonoides |
NA |
MCF-7, HepG2 |
PhytoCAT-700 |
Kaempferol-3-O-β-D-(6″-methyl glucuronide) |
Calligonum polygonoides |
NA |
MCF-7, HepG2 |
PhytoCAT-701 |
Dehydrodicatechin A |
Calligonum polygonoides |
NA |
MCF-7, HepG2 |
PhytoCAT-702 |
Catechin |
Calligonum polygonoides |
NA |
MCF-7, HepG2 |
PhytoCAT-703 |
Taxifolin |
Calligonum polygonoides |
SOS1, Grb2, CCL2 |
MCF-7, HepG2 |
PhytoCAT-704 |
Astragalin |
Calligonum polygonoides |
AKT, ZEB1, VEGF, and MMP9 |
MCF-7, HepG2 |
PhytoCAT-705 |
Quercetin-3-O-β-D-(6″-methyl glucuronide) |
Calligonum polygonoides |
NA |
MCF-7, HepG2 |
PhytoCAT-706 |
Quercetin-3-O-glucuronide |
Calligonum polygonoides |
NA |
MCF-7, HepG2 |
PhytoCAT-707 |
Kaempferol-3-O-glucuronide |
Calligonum polygonoides |
NA |
MCF-7, HepG2 |
PhytoCAT-708 |
Polygonum avicular extract |
Polygonum avicular |
p53 , Bcl-2 |
MCF-7 |
PhytoCAT-709 |
Polygonum cognatum extract |
Polygonum cognatum |
NA |
MDA-MB-231 |
PhytoCAT-710 |
Deoxyrhapontigenin |
Rheum undulatum |
GRP78, IRE1α, eIF2α, CHOP, JNK, p38 |
MCF-7, MCF-7/adr |
PhytoCAT-711 |
Rumex dentatus extract |
Rumex dentatus |
NA |
MCF-7, Hep-2, DU-145 |
PhytoCAT-712 |
Essential oil and methanol extract from Rumex nervosus |
Rumex nervosus |
NA |
MCF-7, MDA-MB-231 |
PhytoCAT-713 |
Rumex vesicarius extract |
Rumex vesicarius |
NA |
MCF-7, HepG2, Lovo, Caco-2 |
PhytoCAT-714 |
Mangifera indica peels extract |
Mangifera indica |
Aromatase |
MCF-7 |
PhytoCAT-715 |
Mangifera indica Extracts |
Mangifera indica |
PKM2 |
MDA-MB-231 |
PhytoCAT-716 |
Polyphenolics from mango |
Mangifera indica |
IR, IRS1, IGF-1R, mTOR |
Female athymic BALB/c nude mice |
PhytoCAT-717 |
Mangifera zeylanica extract |
Mangifera zeylanica |
Caspase 3, Caspase 7, Bcl-2-associated X , p53 |
MCF-7, MDA-MB-231 |
PhytoCAT-718 |
5-((8Z, 11Z, 14Z)-hexatriaconta-8, 11, 14-trienyl) benzene-1,3-diol |
Mangifera zeylanica |
Caspase 7 |
MCF-7 |
PhytoCAT-719 |
Saxifragifolin C |
Androsace umbellata |
p38 MAPK, ERK 1/2, JNK |
MCF-7, MDA-MB-231 |
PhytoCAT-720 |
Baneh extract |
Pistacia atlantica |
Caspase 3, PARP, Cyclin D1, CDK4 |
T47D |
PhytoCAT-721 |
Delcosine |
Aconitum barbatum
Aconitum napellus
Aconitum yesoense |
NA |
MCF-7, MDA-MB-231, A549, DU145,KB |
PhytoCAT-722 |
Sinchiangensine A |
Aconitum sinchiangense |
NA |
HL-60, A-549, SMCC-7721, MCF-7 and SW480 cell line. |
PhytoCAT-723 |
Actein |
Cimicifuga foetida |
VEGFR1, pJNK, pERK |
MCF-7, MDA-MB-361,SKBR-3, HT29, HepG2 and MKN28 / mouse xenograft model |
PhytoCAT-724 |
Cimicifoetiside A |
Cimicifuga foetida |
NA |
MDA-MB-A231 |
PhytoCAT-725 |
Cimicifoetiside B |
Cimicifuga foetida |
NA |
MDA-MB-A231 |
PhytoCAT-726 |
23-epi-26-deoxyactein |
Cimicifuga yunnanensis |
NA |
MCF-7, MDA-MB 231, SK-BR3 |
PhytoCAT-727 |
Cimigenol |
Cimicifuga yunnanensis |
NA |
MCF-7, MDA-MB 231, SK-BR3 |
PhytoCAT-728 |
Huanglian extract |
Coptis chinensis |
Cyclin B1 , cdc2 kinase |
MCF-7, MDA468, MKN-74 and HCT-116 |
PhytoCAT-729 |
Protoberberine |
Coptis chinensis |
NA |
MCF-7, MADB106, SGC7901 |
PhytoCAT-730 |
Jatrorrhizine |
Coptis chinensis |
TNIK |
MDA-MB-231, MCF-7 and 4T1 |
PhytoCAT-731 |
Schinus molle essential oil |
Schinus molle |
NA |
EMT-6, K562 |
PhytoCAT-732 |
Nigella sativa extract |
Nigella sativa |
Caspase 3, Caspase 8, Caspase 9, p53, Cyclin D1, p21 , PAK1, Bcl-2, VEGF |
MCF-7 |
PhytoCAT-733 |
Trans-epsilon-viniferin |
Paeonia lactiflora |
NA |
MCF-7, Hela, , HT-29, HePG2 |
PhytoCAT-734 |
Cis-epsilon-viniferin |
Paeonia lactiflora |
NA |
MCF-7, Hela, , HT-29, HePG2 |
PhytoCAT-735 |
Gnetin H |
Paeonia lactiflora |
NA |
MCF-7, Hela, , HT-29, HePG2 |
PhytoCAT-736 |
Paeoniflorin |
Paeonia lactiflora |
PI3K, AKT, HIF-1α, NOTCH‑1 and HES‑1 |
MDA-MB-231 |
PhytoCAT-737 |
Berberine |
Coptis chinensis |
EGFR, GPER1, ABCG2, CYP1A1, HMGB1, ABCG2, IL-1β, IL-6,TNF-α, NF-κB, Bax, Bcl-2, EGFR, AKT, P38, ERK1/2 |
Cytotoxic effect on MCF-7 cells, inhibitory effect on the growth of breast, liver and colon cancer cell lines (MCF-7, HepG2 and CACO-2, respectively). MDA-MB-231, the human ductal breast epithelial tumor cell line (T47D cell line) |
PhytoCAT-738 |
Extract of Spondias pinnata |
Spondias pinnata |
Caspase 3, Caspase 9, PARP, Bax |
MCF-7, A549 |
PhytoCAT-739 |
Trollius chinensis flavonoids |
Trollius chinensis |
Bcl-2, NF-κB, Caspase 9, Caspase 3 |
MCF-7 |
PhytoCAT-740 |
Frangula alnus extract |
Frangula alnus |
NA |
Jurkat, MCF-7, HeLa, and HT-29 |
PhytoCAT-741 |
Rutoside |
Frangula alnus |
NA |
Jurkat, MCF-7, HeLa, and HT-30 |
PhytoCAT-742 |
Trifolin |
Frangula alnus |
NA |
Jurkat, MCF-7, HeLa, HT-31 |
PhytoCAT-743 |
Protopheophorbide A |
Ziziphus lotus |
E-cadherin, Vimentin, β-catenin, FAK, Brk, Rac, Src |
MDA-MB-231, MCF-7 |
PhytoCAT-744 |
Agrimonia pilosa extract |
Agrimonia pilosa |
pS2, PR |
MCF-7 |
PhytoCAT-745 |
Annoglaxin |
Annona glabra |
NA |
MCF-7, A-498, PC-3, PACA-2 |
PhytoCAT-746 |
27-hydroxybullatacin |
Annona glabra |
NA |
MCF-7, A-498, PC-3, PACA-3 |
PhytoCAT-747 |
Ent-Kaur-16- en-19-oic acid |
Annona senegalensis |
NA |
MCF-7 |
PhytoCAT-748 |
Cleistochlamys kirkii extract |
Cleistochlamys kirkii |
NA |
MDA-MB-231 |
PhytoCAT-749 |
Chamanetin |
Cleistochlamys kirkii |
NA |
MDA-MB-231 |
PhytoCAT-750 |
Isochamanetin |
Cleistochlamys kirkii |
NA |
MDA-MB-231 |
PhytoCAT-751 |
E-acetylmelodorinol |
Cleistochlamys kirkii |
NA |
MDA-MB-231 |
PhytoCAT-752 |
Cleistenolide |
Cleistochlamys kirkii |
NA |
MDA-MB-231 |
PhytoCAT-753 |
Dichamanetin |
Cleistochlamys kirkii |
PARP1 |
MDA-MB-231, HT-29, DU145, |
PhytoCAT-754 |
Licania rigida extract |
Licania rigida |
NA |
MCF-7, Caco- 2 |
PhytoCAT-755 |
Apple extracts |
Malus domestica |
NA |
MCF-7 |
PhytoCAT-756 |
3β-trans-cinnamoyloxy-2α-hydroxy-urs-12-en-28-oic acid (CHUA) |
Malus pumila |
Bax, Bcl-2, cyt-c, Bcl-xL |
MDA-MB-231, MCF-7, HepG2, Caco-2, HeLa, A549/ old female nude mice (Balb/c-nu/nu) |
PhytoCAT-757 |
Pectic acid |
Malus domestica |
NA |
MDA-MB-231 |
PhytoCAT-758 |
13-methoxy-15-oxozoapatlin |
Parinari curatellifolia |
NA |
ZR-75-1, Athymic mice carrying KB cells |
PhytoCAT-759 |
2',4'-dihydroxy-3'-(2-hydroxybenzyl)-6'-methoxychalcone |
Ellipeiopsis cherrevensis |
NA |
BC, NCI-H187, KB |
PhytoCAT-760 |
Black Splendor plum extract |
Prunus salicina |
NA |
MCF-7, MDA-MB-435, MCF-10A |
PhytoCAT-761 |
3,10,11-trimethoxy-1,2-methylenedioxy-7-oxoaporphine |
Fissistigma oldhamii |
NA |
MCF-7 |
PhytoCAT-762 |
Selenium (Se)-containing polysaccharides |
Pyracantha fortuneana |
p53, Bax, PUMA, Noxa, Bcl-2, Bax, Caspase 3, Caspase 9, p53 |
MDA-MB-231 |
PhytoCAT-763 |
Cheliensisin A |
Goniothalamus cheliensis |
NA |
SKBR-3, HL-60, SMMC-7721, A-549, PANC-1 |
PhytoCAT-764 |
Styrylpyrone derivative |
Goniothalamus tamirensis |
Bax |
MCF-7 |
PhytoCAT-765 |
Sanguiin H-6 |
Rubus coreanus |
Caspase 8, Caspase 3, PARP, Bax, Bcl-2 |
MCF-7, MDA-MB-231 |
PhytoCAT-766 |
Rubus crategifolius extract |
Rubus crategifolius |
Topoisomerase I |
MCF-7 |
PhytoCAT-767 |
1-(2-hydroxyphenyl)-4-methylpentan-1-one |
Rubus fairholmianus |
PARP |
MCF-7 |
PhytoCAT-768 |
2-[(3-methylbutoxy) carbonyl] benzoic acid |
Rubus fairholmianus |
PARP |
MCF-7 |
PhytoCAT-769 |
Blackberry extract |
Rubus fruticosus |
NA |
MCF-7, KB, CAL-27, HT-29, HCT116, LNCaP |
PhytoCAT-770 |
Ziyuglycoside II |
Sanguisorba officinalis |
Bax, Fas/FasL, Bcl-2, EMT |
MCF-7 and MDA-MB-231 |
PhytoCAT-771 |
(6E,10E) isopolycerasoidol |
Pseuduvaria monticola |
Bcl-2 |
MCF-7, MDA-MB-231 |
PhytoCAT-772 |
(6E,10E) Isopolycerasoidol Methyl Ester |
Pseuduvaria monticola |
Caspase 3, Caspase 7, Caspase 9, Bcl-2, p38 MAPK |
MCF-7,MDA-MB-231 |
PhytoCAT-773 |
Calycopterin |
Dracocephalum kotschyi |
Bax, Bcl-2 |
MDA-MB-231, MCF-7 |
PhytoCAT-774 |
7, 3', 5'-trihydroxyflavanone |
Hydnophytum formicarum |
Bcl-2, Bax |
MCF-7 |
PhytoCAT-775 |
3β, 6β, 19α, 24-tetrahydroxy-urs-12-en-28-oic acid |
Mitragyna diversifolia |
NA |
MCF-7, HT-29 |
PhytoCAT-776 |
Rotundic acid |
Mitragyna diversifolia |
NA |
MCF-7, HT-29 |
PhytoCAT-777 |
23-nor-24-exomethylene- 3β, 6β, 19α-trihydroxy-urs-12-en-28-oic acid |
Mitragyna diversifolia |
NA |
MCF-7, HT-29 |
PhytoCAT-778 |
Nordamnacanthal |
Morinda citrifolia |
NA |
MDA-MB-231, MCF-7 and 4T1/ Balb/C mice |
PhytoCAT-779 |
Oldenlandia diffusa extract |
Oldenlandia diffusa |
p53, p21WAF1/Cip1 |
MCF-7 |
PhytoCAT-780 |
Chlorogenic acid |
Pavetta indica |
NA |
MDA-MB-435, MCF-7, MDA-MB-231, T-47D and BJ-hTERT |
PhytoCAT-781 |
Carvacrol |
Xylopia aromatica |
TRPM7 |
BT-483, BT-474, MCF-7, MDA-MB-231, and MDA-MB-453 |
PhytoCAT-782 |
Thymol |
Xylopia sericea |
NA |
MDA-MB-231, PC-3, DU145, KLN205 |
PhytoCAT-783 |
Mollugin |
Rubia cordifolia |
FAS |
SKBR-3 , SK-OV-3 |
PhytoCAT-784 |
Alizarin |
Rubia tinctorum |
NA |
MDA-MB-231 |
PhytoCAT-785 |
Isoquercitrin |
Tetrastigma hemsleyanum |
LSD1 |
MDA-MB-231 |
PhytoCAT-786 |
Uncaria tomentosa extract |
Uncaria tomentosa |
NA |
MCF-7 |
PhytoCAT-787 |
Mitraphylline |
Uncaria tomentosa |
NA |
HAE, BEAS-2B, SK-N-SH, HepG2, HEK293, MKN45, DLD1, A549, MCF7, LNCaP |
PhytoCAT-788 |
Angelica sinensis polysaccharide |
Angelica sinensis |
PARP, Bax, Bcl-2, Bcl-xL, Apaf1 |
T47D, nude mice xenograft model |
PhytoCAT-789 |
8-hydroxyartabonatine C |
Pseuduvaria trimera |
NA |
HepG2, MDA-MB-231 |
PhytoCAT-790 |
Aegle marmelos extract |
Aegle marmelos |
NA |
MCF-7, MDA-MB-231/ Female Charles Foster strain rats |
PhytoCAT-791 |
Marmin |
Aegle marmelos |
NA |
T47D |
PhytoCAT-792 |
Auraptene |
Aegle marmelos |
VEGF, VEGFR2, VCAM-1, TNFR-1, COX-2, IFNγ |
T47D, 4T, MDA-MB-231, HUVEC |
PhytoCAT-793 |
Acacia catechu extract (ACME) |
Acacia catechu |
Bax, Bcl-2 |
MCF-7 |
PhytoCAT-794 |
Alpinia nantoensis extract |
Alpinia nantoensis |
EGFR |
MDA-MB-231, MCF-7 |
PhytoCAT-795 |
Sauromatum giganteum extract |
Sauromatum giganteum |
NA |
MCF-7, SMMC-7721, SGC-7901 |
PhytoCAT-796 |
8,2'-Diprenylquercetin 3-methyl ether |
Sinopodophyllum hexandrum |
NA |
MDA-231 and T47D |
PhytoCAT-797 |
Ampelopsin |
Ampelopsis grossedentata |
p21, Cyclin A, CDK2, IκBα, NF-κB p65 , CD44, MRP1, β-catenin, KLF4 |
MDA-MB-231, MDA-MB-231/IR |
PhytoCAT-798 |
Murraya koenigii leaf extract |
Murraya koenigii |
NA |
MDA-MB-231 |
PhytoCAT-799 |
Mukonal |
Murraya koenigii |
PARP, Caspase 3, Bcl-2, Beclin-1, LC3B-I, LC3B-II |
MDA-MB-231, CAMA-1, MDA-MB-435, SKBR-3/ xenografted mice models |
PhytoCAT-800 |
Emodic-acid |
Asphodelus microcarpus |
JNK, p38, ERK, IL-1β, IL-6, VEGF, MMP2, MMP9 |
4T1 |
PhytoCAT-801 |
4-vinylphenol (4VP) |
Hedyotis diffusa |
PI3K/AKT, p38 MAPK, NF-κB |
C57BL/6 mice |
PhytoCAT-802 |
Eupatolide |
Inula britannica |
Vimentin , E-cadherin, EMT |
MCF-7, MDA-MB-231 and MDA-MB-453 |
PhytoCAT-803 |
Aucklandia Lappa Decne extract |
Aucklandia lappa |
NA |
T47D, HeLa, HEp-2 |
PhytoCAT-804 |
Saponin glycoside |
Fagonia indica |
PARP, Caspase 3 |
MDA-MB-468, Caco-2, MCF-7 |
PhytoCAT-805 |
Quinovic acid |
Fagonia indica |
Caspase 3, Caspase 8, PARP |
NA |
PhytoCAT-806 |
Robustaflavone A |
Selaginella trichoclada |
VDAC2 channel, Nedd4 E3 ubiquitin ligase |
MCF-7 |
PhytoCAT-807 |
Didymin |
Citrus latipes |
NA |
MDA-MB-231 |
PhytoCAT-808 |
Patrinia scabiosaefolia extract (EAE-PS) |
Patrinia scabiosaefolia |
Bcl-2, Bcl-xL |
MCF-7, HepG2, A375, A549, PC-3 |
PhytoCAT-809 |
Diosmetin |
Dictamnus dasycarpus |
Bcl-2, Cyclin D1, p53, Bax, Caspase 3, Caspase 9, Caspase 3 |
MDA-MB-468, MCF-7, MDA-MB-231 |
PhytoCAT-810 |
Lanostane |
Lyonia ovalifolia |
Bax, Bcl-2 |
SKBR-3, MB-157 |
PhytoCAT-811 |
Girinimbine |
Murraya euchrestifolia |
NA |
MDA-MB-453 |
PhytoCAT-812 |
Mahanine |
Bergera koenigii |
NA |
MDA‑MB‑157, MCF‑7, MDA-MB-231 |
PhytoCAT-813 |
Paramignya trimera extract (PTL) |
Paramignya trimera |
NA |
MCF-7, MiaPaCa-2, HT29, A2780, H460, A431, Du145, BE2-C, U87, SJ-G2, and SMA |
PhytoCAT-814 |
Paratrimerin I |
Paramignya trimera |
NA |
MCF-7, HepG2 |
PhytoCAT-815 |
Protocatechuic acid (PCA) |
Bauhinia variegata |
NA |
MCF-7, C-6, HCT-15 |
PhytoCAT-816 |
Harmine |
Peganum harmala |
Twist1, TAZ, p‑Erk, p‑Akt, Bcl‑2, Bax |
BT-549 |
PhytoCAT-817 |
Harmine hydrochloride |
Peganum harmala |
PI3K, AKT, mTOR, FOXO3a |
MCF-7, MDA-MB-231 |
PhytoCAT-818 |
Peganum harmala extract |
Peganum harmala |
NA |
MCF-7, Jurkat, HeLa, and HT-29 |
PhytoCAT-819 |
Cynaroside |
Peganum harmala |
NA |
MCF-7, Jurkat, HeLa, and HT-29 |
PhytoCAT-820 |
Nitidine chloride |
Zanthoxylum nitidum |
PARP, Bax, Caspase 9, Caspase 3, Bcl-2 |
MCF-7, MDA-MB-231 |
PhytoCAT-821 |
Sichuan pepper extracts |
Zanthoxylum piperitum |
Cyclin D1, PAK1 |
MDA-MB-231 xenograft in mice |
PhytoCAT-822 |
Alpha-Santalol |
Santalum album |
NA |
MDA-MB 231, MCF-7 |
PhytoCAT-823 |
Escin Ia |
Aesculus chinensis |
LOXL2 |
Female athymic nude mice, MCF-7, MDA-MB-231 |
PhytoCAT-824 |
Descurainia sophia volatile oil |
Descurainia sophia |
NA |
MCF-7, HeLa |
PhytoCAT-825 |
Pouteria torta leaf extract |
Pouteria torta |
NA |
OSCC-3 and MCF-7 |
PhytoCAT-826 |
Halofuginone |
Dichroa febrifuga |
MMP9 |
MDA-MB-231, PC3 |
PhytoCAT-827 |
Galangin |
Alpinia officinarum |
STAT-3, p-JAK2, Bcl-2, Caspase 3, PARP, Ki67, Nrf2 , NQO-1, HO-1, GSTP1-1 |
MDA-MB-231, MCF-7, HCT-116, HeLa, BT-474, MGC 803 |
PhytoCAT-828 |
1'S-1'-acetoxyeugenol acetate |
Alpinia conchigera |
NA |
MCF-7, HMEC |
PhytoCAT-829 |
Alpinia galanga rhizhome extract |
Alpinia galanga |
NA |
MCF-7 |
PhytoCAT-830 |
Galangal extract (GE) |
Alpinia galanga |
NA |
4T1 |
PhytoCAT-831 |
Pinostrobin chalcone |
Alpinia mutica |
NA |
KB, MCF-7, A549, Caski, HCT116, HT29 |
PhytoCAT-832 |
Eicosapentaenoic acid |
Alpinia oxyphylla |
NA |
MCF-7 |
PhytoCAT-833 |
Alpha-Turmerone |
Curcuma longa |
NA |
HepG2, MCF-7, MDA-MB-231 |
PhytoCAT-834 |
Terpecurcumin D |
Curcuma longa |
NA |
MDA-MB-231, A549, HepG2 |
PhytoCAT-835 |
Terpecurcumin F |
Curcuma longa |
NA |
MDA-MB-231, A549, HepG2 |
PhytoCAT-836 |
Terpecurcumin G |
Curcuma longa |
NA |
MDA-MB-231, A549, HepG2 |
PhytoCAT-837 |
Bisabolocurcumin ether |
Curcuma longa |
p38, p53 |
MDA-MB-231, A549, HepG2 |
PhytoCAT-838 |
Demethoxybisabolocurcumin ether |
Curcuma longa |
NA |
MDA-MB-231, A549, HepG2 |
PhytoCAT-839 |
Terpecurcumin Q |
Curcuma longa |
NA |
MCF-7 |
PhytoCAT-840 |
Curcumin |
Curcuma longa |
c-Myc, Cyclin D1, Bcl-2, ABCB1, ABCC1, ABCG2, CXCL1, CXCL2, CXCR4, PTEN, BMI1, EGFR, CRP, EZH2, FABP5, ABCB4, DYRK2, HR.SERPINE1, PGAP3, MAP3K1, MAPK1, TCF, MTOR, AKT1, BIRC5, CCND1 , NQO1, PRMT5, MEP50, AURKA, CDK2, CDK1, FOS, H2AX, KIF11, SOD2, STAT-3, TNF, APC, ARNT,AXIN1, HIAP1, CRAF1, TRAF6, CASP1, CASP2, CASP3, CASP4, HPRT, GADD45, MCL-1, NIP1, Bcl-2L2, TRAP3, GSTP1, DAXX, PIG11, UBC, PIG3, PCNA, CDC10, JNK1, RBP2, TRAIL, TNFR, AP13, IGFBP3, SARP3, PKB, IGFBP, CASP7, CASP9, TNFSF6, TRICK2A, CAS, TRAIL-R2, RATS1, hTRIP, TNFb, TNFRSF5, CASP9, COL4A1, DAXX, DVL2, ENPP2, ERP29, FASN, ISG15, MYBL1 , PDK1, VEGF-A, XIAP, PARP, HER-2, NF-kB, Caspase 3, Caspase 7, skp2, p27, Cadherin-11, Plasminogen |
MDA-MB-231, MCF-7, MD-MB-468, AU565, HCT116, A549, A375, T47D, DLD-1,MDA-MB-435, breast cancer xenograft model |
PhytoCAT-841 |
Xanthorrhizol |
Curcuma xanthorrhiza |
Bcl-2, p53, PARP-1, pS2 |
MDA-MB-231 and MCF-7 |
PhytoCAT-842 |
[10]-gingerol |
Zingiber officinale |
NA |
MDA-MB-231, MDA-MB-468, mouse (4T1, E0771), MCF-7, T47D |
PhytoCAT-843 |
Ginger polysaccharides |
Zingiber officinale |
NA |
MCF-7, H1975, HCT116, MCF-7 |
PhytoCAT-844 |
6-gingerol |
Zingiber officinale |
p53, Bax, Bcl-2, cyt-c |
MDA-MB-231 and MCF-7 |
PhytoCAT-845 |
6-methoxy-2E,9E-humuladien-8-one |
Zingiber zerumbet |
NA |
MDA-MB-231 |
PhytoCAT-846 |
Zerumbone |
Zingiber zerumbet |
Bax, Caspase 7, Caspase 9, Bcl-2 |
MCF-7 |
PhytoCAT-847 |
Melognine |
Melodinus fusiformis |
Caspase 3, p53, Bcl-2 |
BT-549 |
PhytoCAT-848 |
Scrophularia atropatana extract |
Scrophularia atropatana |
Tp53, Survivin |
MCF-7, L929 |
PhytoCAT-849 |
2,3-seco-taraxer-14-en-2,3-lactone (pycanocarpine) |
Pleiocarpa pycnantha |
NA |
MCF-7 |
PhytoCAT-850 |
Minecoside |
Veronica peregrina |
CXCR4 |
MDA‑MB‑231, PANC1, SW480, HCT116, A2780, U266, A549, MCF-7 |
PhytoCAT-851 |
Ailanthone |
Ailanthus altissima |
Bax, Bcl-2 |
MCF-7 |
PhytoCAT-852 |
Bruceantin |
Brucea javanica |
NA |
MCF-7, Lu1, LNCaP |
PhytoCAT-853 |
Brucea javanica Seed extract |
Brucea javanica |
ULK1, Beclin-1, p62 |
MDA-MB-231 |
PhytoCAT-854 |
Bruceae fructus oil (BO) |
Brucea javanica |
mTOR, 4E-BP1 |
MDA-MB-231 and BT-20 / Female Balb/c nude mice |
PhytoCAT-855 |
9-methoxycanthin-6-one |
Eurycoma longifolia |
PKM, ANXA2, LGAL3, HNRNP1A1, PRDX3, GAPDH, ACAA2, ALDH1A1, CAPG,MDH2, EEF1A1, TPI1 |
MCF-7, A2780, SKOV-3, HT29, A375, HeLa, DU-145, RD, CaOV-3, MDBK, A-549 |
PhytoCAT-856 |
Canthin-6-one |
Eurycoma longifolia |
NA |
HCC 1395, DU 145, Vero E6, A549, MCF-7, HL60 , AZ521, SKBR-3 |
PhytoCAT-857 |
Eurycoma longifolia extract |
Eurycoma longifolia |
Bax, Bcl-2, p53 |
MDA-MB-231, MCF-7 |
PhytoCAT-858 |
Picrasidine G |
Picrasma quassioides |
Caspase 3, PARP, STAT-3, EGFR, Survivin |
MDA-MB-468 |
PhytoCAT-859 |
Simalikalactone D |
Simarouba tulae |
NA |
MDA-MB-435, MDA-MB-231, A2780CP20, 4T1, MCF10A, PC3, HCT-116, SH-SY5Y |
PhytoCAT-860 |
Lycium barbarum extract |
Lycium barbarum |
NA |
MCF-7 |
PhytoCAT-861 |
Lycium barbarum polysaccharides(LBGP-I-3) |
Lycium barbarum |
NA |
MCF-7 |
PhytoCAT-862 |
Isopicrinine |
Rhazya stricta |
PUMA, Survivin |
MCF-7 |
PhytoCAT-863 |
Rhazyaminine |
Rhazya stricta |
Bcl-2 |
MCF-7 |
PhytoCAT-864 |
Strophanthidin |
Strophanthus kombe |
MEK1, PI3K, AKT, mTOR, Gsk3α, β-catenin |
MCF-7, A549, and HepG2 |
PhytoCAT-865 |
Affinisine |
Tabernaemontana catharinensis |
NA |
MCF-7, U251, NCI-ADR/RES, 786-0, NCI-H460, HT-29, K562 , PC-3 |
PhytoCAT-866 |
Viscosalactone B |
Withania somnifera |
EGFR, HER2, estrogen and NF-κB receptors |
MCF-7, NCI-H460, HCT-116, SF-268 |
PhytoCAT-867 |
Withaniasomnifera root extracts (WRE) |
Withania somnifera |
TGFβ, EMT, Vimentin, fibronectin, E-cadherin |
MDA-MB-231, MCF-7, T47D, Hs578-T |
PhytoCAT-868 |
Pomolic acid |
Euscaphis japonica |
NA |
Human breast cancer cells, MCF-7 and MDA-MB-231, and human umbilical vascular endothelial cells (HUVEC). |
PhytoCAT-869 |
Mansorin-A |
Mansonia gagei |
NA |
MCF-7, HepG2, HCT-116, HeLa |
PhytoCAT-870 |
Mansorin-B |
Mansonia gagei |
NA |
MCF-7, HepG2, HCT-116, HeLa |
PhytoCAT-871 |
Mansorin-C |
Mansonia gagei |
NA |
MCF-7, HepG2, HCT-116, HeLa |
PhytoCAT-872 |
Mansorin-I |
Mansonia gagei |
NA |
MCF-7, HepG2, HCT-116, HeLa |
PhytoCAT-873 |
Mansorin-II |
Mansonia gagei |
NA |
MCF-7, HepG2, HCT-116, HeLa |
PhytoCAT-874 |
Mansorin III |
Mansonia gagei |
NA |
MCF-7, HepG2, HCT-116, HeLa |
PhytoCAT-875 |
Mansonone-G |
Mansonia gagei |
NA |
MCF-7, HepG2, HCT-116, HeLa |
PhytoCAT-876 |
Mansonone-N |
Mansonia gagei |
NA |
MCF-7, HepG2, HCT-116, HeLa |
PhytoCAT-877 |
Tamarix articulata extract |
Tamarix articulata |
NA |
MCF-7, RKO |
PhytoCAT-878 |
α-conidendrin |
Taxus yunnanensis |
p21 , Bcl-2, p53 , Bax, Caspase 3, Caspase 9, Cyclin D1, CDK4 |
MCF-7 and MDA-MB-231 |
PhytoCAT-879 |
Actinidia chinensis extract |
Actinidia chinensis |
Bax, E-cadherin, Cyclin D1, Survivin, Bcl-2, N-cadherin, Snail |
MDA-MB-231 and MDA-MB-453 |
PhytoCAT-880 |
Oleiferoside B |
Camellia oleifera |
NA |
MCF-7, SMMC-7721 |
PhytoCAT-881 |
Theaflavins |
Black tea |
p53, Bax |
MCF-7, MDA-MB-231, ZR-75-1 |
PhytoCAT-882 |
Camellia sinensis extract |
Camellia sinensis |
Bax, Bcl-2, Caspase 8, Caspase 3 |
4T1/ BALB/c mice |
PhytoCAT-883 |
Gallic acid |
Ceriops tagal |
EGFR, Src, AKT/p65, MMP9 |
HeLa, MDA-MB23, MCF-7 |
PhytoCAT-884 |
Camellianin A |
Adinandra nitida |
NA |
MCF-7, HepG2 |
PhytoCAT-885 |
Daphne gnidium L. extract |
Daphne gnidium |
COX-2 |
MCF-7 |
PhytoCAT-886 |
P. macrocarpa fruit ethyl acetate fraction (PMEAF) |
Phaleria macrocarpa |
Bax, Bid, Caspase 3, Caspase 8, cyt-c, p21, p27, p53, SMAC, Bcl-2, Bcl-w, XIAP, Survivin |
MDA-MB-231 |
PhytoCAT-887 |
Chamaejasmenin B |
Stellera chamaejasme |
β3 integrin-TβRII, TGF-beta |
MDA-MB-231, ZR75-1 and 4T1 |
PhytoCAT-888 |
Thymelaea hirsuta L. extracts |
Thymelaea hirsuta |
NA |
MCF-7 and OVCAR |
PhytoCAT-889 |
Petiolaticin A |
Elaeocarpus petiolatus |
NA |
MDA-MB-468, MDA-MB-231, MCF-7, and SW48 |
PhytoCAT-890 |
Luehea candicans extract |
Luehea candicans |
NA |
MCF-7, NCI-ADR, NCI-460, UACC-62, 786-0, OVCAR, PCO-3, HT-29, K-562 |
PhytoCAT-891 |
Trapa acornis husks (TAH) extract |
Trapa acornis |
VEGF, p-Her2, p-ERK1/2, VEGF, MMP2, MMP9, uPA |
Female BALB/C-nu mice, SKBR-3 |
PhytoCAT-892 |
Saikosaponin A |
Bupleurum chinense |
VEGFR2, PLCγ1, FAK, Src, AKT |
4T1, MCF-7, HCT-15, AGS, HepG2 |
PhytoCAT-893 |
Bupleurum marginatum extract |
Bupleurum marginatum |
Caspase 3, Caspase 7 |
MCF-7, Caco-2, CCL-81, CCRF-CEM, COS-7, HL-60, MIA PaCa-2, PANC-1 |
PhytoCAT-894 |
Falcarinol |
Chaerophyllum aureum |
NA |
MCF-7 |
PhytoCAT-895 |
Beta-carotene |
Daucus carrota |
AF040958, AK001555, g41894, hshsp90r, U83857, AB014509, AF126028, AF053641, AF117386, AF050127,NM_012177, humtopi, AJ250915, U37547, U78798, NM_004849, NM_005346, AF004711, NM_006595, NM_001418, AB015051 |
MCF-7, MD-MB-231, HCT-116, AGS , NCI-H460 |
PhytoCAT-896 |
Daucus carota oil extract |
Daucus carota |
BAX, Bcl-2, Caspase 3, PARP, ERK |
MCF-7, MDA-MB-231, HT-29, Caco-2 |
PhytoCAT-897 |
Asafoetida |
Ferula assa-foetida |
NA |
4T1 |
PhytoCAT-898 |
Ferulin C |
Ferula ferulaeoides |
NA |
MCF-7 and MDA-MB-231 |
PhytoCAT-899 |
Conferone |
Ferula gummosa |
NA |
MCF-7/Dox |
PhytoCAT-900 |
Feselol |
Ferula gummosa |
NA |
MCF-7/Dox |
PhytoCAT-901 |
Ferula hermonis Boiss. extract |
Ferula hermonis |
NA |
MDA-MB-231/ Wistar albino rats |
PhytoCAT-902 |
Umbelliprenin |
Ferula szowitsiana |
NA |
MCF-7, M4Beu, A549, PC3, PA1 |
PhytoCAT-903 |
Galbanic acid |
Ferula szowitsiana |
NA |
MCF-7 |
PhytoCAT-904 |
Ferulago carduchorum essential oil |
Ferulago carduchorum |
NA |
T47D, HEP-G2, HT-29 |
PhytoCAT-905 |
Oliveria decumbens essential oil |
Oliveria decumbens |
NA |
MCF-7, T47D, MDA- MB-231 |
PhytoCAT-906 |
Prim-O-glucosylcimifugin |
Saposhnikovia divaricata |
Arg-1, iNOS |
B16-F10, (4 T1) mouse tumour models |
PhytoCAT-907 |
Perillyl alcohol |
Trachyspermum anethifolium |
Cyclin D1 mRNA |
T47D, MCF-7, MDA-MB-231 |
PhytoCAT-908 |
Artelastin |
Artocarpus elasticus |
NA |
MCF-7 |
PhytoCAT-909 |
Artonin E |
Artocarpus elasticus |
p21, Cyclin D, cyt-c, Bax, Caspase 7, Caspase 9, MAPK |
MCF-7, MDA-MB-231, 1A9, HCT-8 |
PhytoCAT-910 |
Artocarpin |
Artocarpus heterophyllus |
Caspase 8, Caspase 10 |
T47D |
PhytoCAT-911 |
Artocarpus heterophyllus extract |
Artocarpus heterophyllus |
NA |
T47D, TH29 and B16F10 |
PhytoCAT-912 |
Boehmeriasin A |
Boehmeria siamensis |
Cyclin E2, Cyclin D1 |
MDA-MB-231 |
PhytoCAT-913 |
Broussoflavonol B |
Broussonetia papyrifera |
c-Myc , p16(INK4a), p19(INK4D), p21(WAF1/CIP1), Cyclin B1, cdc2, cdc25C, ER-α36, Epidermal growth factor receptor |
MDA-MB-231 |
PhytoCAT-914 |
Ficus carica extracts |
Ficus carica |
NA |
MDA-MB-231 |
PhytoCAT-915 |
Ficus crocata extracts |
Ficus crocata |
p53, Procaspase 8, Procaspase 3 |
MDA-MB-231 |
PhytoCAT-916 |
Ficus hispida extract |
Ficus hispidaf |
NA |
SKBR-3, HL60, A549, KB, Hela, HT29, HepG2 |
PhytoCAT-917 |
Ficus salicifolia latex |
Ficus salicifolia |
ERK2, CREB, AKT2 |
MDA-MB-231 |
PhytoCAT-918 |
Ficus septica extract |
Ficus septica |
PARP |
T47D |
PhytoCAT-919 |
Vanillic acid |
Ficus septica |
NA |
MDA MB 468, HBL 100, PC3, MCF-7 |
PhytoCAT-920 |
Arisaema tortuosum extract |
Arisaema tortuosum |
NA |
MCF-7 |
PhytoCAT-921 |
Valerian extract |
Valeriana officinalis |
NA |
MCF-7 and MDA-MB-231 |
PhytoCAT-922 |
Valeric acid |
Valeriana officinalis |
NA |
MCF-7, MDA-MB-231, MCF-10A |
PhytoCAT-923 |
Avicennia marina extract |
Avicennia marina |
MMP2, MMP9, Cyclin B, Vimentin, snail |
MDA-MB-231, AU565, BT483 |
PhytoCAT-924 |
Rhoifolin (RFL) |
Callicarpa nudiflora |
NA |
MDA-MB-231 |
PhytoCAT-925 |
Apigenin |
Clerodendrum viscosum |
Cyclin D1, Cyclin D3, CDK4, HER2/neu , AKT, CTSS, C3, LAMC2, TLR2, GPRC5B, CNTNAP1, CLDN1, NFATC2, CXCL10, CXCL11, IRAK3, NR3C2, IL32, IL-24, SLIT2, TMEM132A, TMEM171, STAP2, MLKL, KDR, BMPER, KLHL36, STAT-3, YAP/TAZ, CTGF, CYR61, Caspase 3, VEGF, Progestrone receptor, PI3K, JAK3, PLD2, CYP1A1,CYP1B1 |
MDA-MB-453, T47D, ZR-75-1, PC-3, MCF-7, HT-29, HeLa, A549, MDA-MB-231, ChaGo-I , NIH/3T3, A431, MDA-MB-468, Hs578T, SKBR-3 |
PhytoCAT-926 |
Lippia origanoides extract |
Lippia origanoides |
NA |
MDA-MB-231 |
PhytoCAT-927 |
1-O-trans-p-coumaroyl-2-O-trans-caffeoyl-α-L-rhamnopyranose |
Premna odorata |
c-met |
MCF-7, BT-474 cells, and MDA-MB-468 |
PhytoCAT-928 |
Icetexane-1 |
Premna tomentosa |
NA |
MCF-7, HT-29, Hep-G2, A-431, and A-549 |
PhytoCAT-929 |
Icetexatriene-3 |
Premna tomentosa |
NA |
MCF-7, HT-29, Hep-G2, A-431, and A-549 |
PhytoCAT-930 |
Vitex rotundifolia extract |
Vitex rotundifolia |
Bax, Bcl-2 , Caspase 3, Caspase 7, Caspase 9 |
MCF-7 |
PhytoCAT-931 |
Ampelopsin A |
Vitis thunbergii |
AKT |
MDA-MB-231 |
PhytoCAT-932 |
Ampelopsin C |
Vitis thunbergii |
AXL, Dtk (TYRO3), EphA2, EphA6, Fyn, Hck, SRMS |
MDA-MB-231 |
PhytoCAT-933 |
Caffeic acid |
Thalassodendron ciliatum |
NA |
MCF-7/Adr, MCF-7/wt, MDA-MB-231, T47D |
PhytoCAT-934 |
Thalassosterol |
Thalassodendron ciliatum |
NA |
MCF-7 ,HeLa , HepG2 |
PhytoCAT-935 |
Alpinia pahangensis extract |
Alpinia pahangensis |
NA |
MCF-7, A549, KB, Ca Ski and HCT 116 |
PhytoCAT-936 |
Cardamonin |
Amomum subulatum |
FOXO3a, p21, p27, Bim |
MDA-MB 231 and MCF-7 |
PhytoCAT-937 |
Ramonanin A |
Guaiacum sanctum and Guaiacum officinale |
NA |
SKBR-3, MD-MBA-468, MD-MBA 231 |
PhytoCAT-938 |
Nordihydroguaiaretic acid (NDGA) |
Larrea divaricata |
p16INK4a |
HepG2, MDA-MB-468, T47D, RKO |
PhytoCAT-939 |
Larrea divaricata extract |
Larrea divaricata |
NA |
MCF-7 |
PhytoCAT-940 |
Larrea tridentata extract |
Larrea tridentata |
ERK1/2 |
MCF-7/AZ |
PhytoCAT-941 |
Pothobanol |
Pothos scandens |
NA |
T47D, MCF-7 |
PhytoCAT-942 |
Typhonium flagelliforme tuber extract |
Typhonium flagelliforme |
Survivin, Caspase 9, Caspase 3 |
Breast cancer stem cells (bCSCs) |
PhytoCAT-943 |
Allium sivasicum (AS) extract |
Allium sivasicum |
NA |
MDA-MB-231, MDA-MB-468, MCF-7 |
PhytoCAT-944 |
Taiwanin E |
Eleutherococcus trifoliatus |
pRb, CDK4, p21, p27, CDK6, Cyclin D3, Cyclin D4 |
MCF-7 |
PhytoCAT-945 |
Ochradenus arabicus extract |
Ochradenus arabicus |
NA |
MCF-7 |
PhytoCAT-946 |
Extract of Origanum munzurense (OME) |
Origanum munzurense |
NA |
MCF-7 |
PhytoCAT-947 |
Tinospora cordifolia extract |
Tinospora cordifolia |
NA |
MDA-MB-231 and MCF-7 |
PhytoCAT-948 |
Epoxy clerodane diterpene |
Tinospora cordifolia |
CYP1A, GPX, GSK3β, TNF-α, NF-κB, CDKn2A, Rb1, p53, Bax, Caspase 3, Caspase 8, Caspase 9, p21, Bcl-2, mdm2, PCNA |
MCF-7 |
PhytoCAT-949 |
Oplopandiol |
Oplopanax horridus |
NA |
MCF-7 (RPMI-1640), HCT-116 and SW-480 , IEC-6 |
PhytoCAT-950 |
Oplopandiol acetate |
Oplopanax horridus |
NA |
MCF-7, HCT-116, SW-480 |
PhytoCAT-951 |
Oplopantriol A |
Oplopanax horridus |
NA |
MCF-7, HCT-116, SW-480 |
PhytoCAT-952 |
Panaxydol |
Panax ginseng |
EGFR |
MCF-7 , PC3 and Renca mouse renal cancer cells |
PhytoCAT-953 |
Micranthin B |
Isodon lophanthoides |
NA |
MCF-7, A549, HeLa |
PhytoCAT-954 |
Rabdosia rubescens extract |
Rabdosia rubescens |
AKT |
MDA-MB-231 and HUVEC |
PhytoCAT-955 |
Oridonin |
Isodon rubescens |
Bcl-2, Caspase 3, PARP, AKT |
MDA-MB-231 , MCF-7, A375-S2 |
PhytoCAT-956 |
20(S)-25-methoxyl-dammarane-3beta, 12beta, 20-triol [20(S)-25-OCH3-PPD] |
Panax notoginseng |
NA |
MCF-7, MDA-MB-468, A172 , T98G, HPAC, Panc-1, A549, H1299, H358, H838, LNCaP, PC3 |
PhytoCAT-957 |
Azadirachta indica extract |
Azadirachta indica |
Bax, Cyclin D1, CYP 1A1, CYP 1A2 |
MCF-7, HeLa |
PhytoCAT-958 |
Annomocherin |
Annona cherimolia |
NA |
MCF-7, A-498 |
PhytoCAT-959 |
Annonacin |
Annona cherimolia |
Cyclin D1, Bcl-2, HIF-1 |
MCF-7 xenografts in nude mice, MDA-MB-231, MCF-7, T47D |
PhytoCAT-960 |
Annomontacin |
Annona cherimolia |
NA |
MDA-MB-231, MCF-7 |
PhytoCAT-961 |
Annona cherimola ethanolic leaf extract (AELE) |
Annona cherimola |
Bax, Bcl-2, p21, cyt-c |
MDA-MB-231 and MCF-7 |
PhytoCAT-962 |
Houttuyninum |
Houttuynia cordata |
ERK1/2, AKT |
MDA-MB-468, BT-474, A431, N87 xenografts |
PhytoCAT-963 |
Solajiangxin I |
Solanum lyratum |
NA |
MCF-7, HCT-8, A-549, SGC-7901 and BEL-7402 |
PhytoCAT-964 |
7-Hydroxylsolajiangxin I |
Solanum lyratum |
NA |
MCF-7, HCT-8, A-549, SGC-7901 and BEL-7402 |
PhytoCAT-965 |
Solajiangxin H |
Solanum lyratum |
Bcl-2, Survivin, Bcl-2-like 4, Caspase 3, c-Caspase 9 |
MCF-7, HCT-8, A-549, SGC-7901 and BEL-7402 |
PhytoCAT-966 |
Lyratol D |
Solanum lyratum |
B-cell lymphoma (Bcl)-2, Survivin, Bcl-2-like protein 4, (c)-Caspase 3, c-Caspase 9 |
MCF-7, HCT-8, A-549, SGC-7901 and BEL-7402 |
PhytoCAT-967 |
Dehydrovomifoliol |
Solanum lyratum |
NA |
MCF-7, HCT-8, A-549, SGC-7901 and BEL-7402 |
PhytoCAT-968 |
Blumenol A |
Solanum lyratum |
NA |
MCF-7, HCT-8, A-549, SGC-7901 and BEL-7402 |
PhytoCAT-969 |
Solajiangxin A |
Solanum lyratum |
NA |
MCF-7, HCT-8, A-549, SGC-7901 and BEL-7402 |
PhytoCAT-970 |
Solajiangxin B |
Solanum lyratum |
NA |
MCF-7, HCT-8, A-549, SGC-7901 and BEL-7402 |
PhytoCAT-971 |
Solajiangxin C |
Solanum lyratum |
NA |
MCF-7, HCT-8, A-549, SGC-7901 and BEL-7402 |
PhytoCAT-972 |
Solajiangxin D |
Solanum lyratum |
NA |
MCF-7, HCT-8, A-549, SGC-7901 and BEL-7402 |
PhytoCAT-973 |
Solajiangxin E |
Solanum lyratum |
NA |
MCF-7, HCT-8, A-549, SGC-7901 and BEL-7402 |
PhytoCAT-974 |
2-Hydroxysolajiangxin E |
Solanum lyratum |
NA |
MCF-7, HCT-8, A-549, SGC-7901 and BEL-7402 |
PhytoCAT-975 |
Lyratol A |
Solanum lyratum |
NA |
MCF-7, HCT-8, A-549, SGC-7901 and BEL-7402 |
PhytoCAT-976 |
Lyratol B |
Solanum lyratum |
NA |
MCF-7, HCT-8, A-549, SGC-7901 and BEL-7402 |
PhytoCAT-977 |
Lyratol C |
Solanum lyratum |
NA |
MCF-7, HCT-8, A-549, SGC-7901 and BEL-7402 |
PhytoCAT-978 |
Cyanidin-3-O-(6''-O-α-rhamnopyranosyl- β-glucopyranoside |
Acer palmatum |
NA |
T47D, LLC |
PhytoCAT-979 |
Cyanidin-3-O- β- glucopyranoside |
Acer palmatum |
NA |
T47D, LLC |
PhytoCAT-980 |
Cyanidin-3-O-[2''-O-(galloyl)-6''-O-(rhamnosyl)-β-glucoside] |
Acer palmatum |
NA |
T47D, LLC |
PhytoCAT-981 |
Cyanidin-3-O-[2''-O-(galloyl)- β-glucopyranoside] |
Acer palmatum |
NA |
T47D, LLC |
PhytoCAT-982 |
Dehydrocorydaline |
Corydali syanhusuo |
CDK1, CCND1, Bcl-2, MMP2, MMP9, Caspase 3, Caspase 8, Caspase 9, Bax, Bcl-2 |
MDA‑MB‑231 , MCF-7 |
PhytoCAT-983 |
Protopine |
Corydalis yanhusuo |
EGFR, ICAM-1, αv-integrin, β1-integrin, β5-integrin |
MCF-7, MDA-MB-231 |
PhytoCAT-984 |
Aristolochia foetida Kunth extract |
Aristolochia foetida |
NA |
MCF-7 |
PhytoCAT-985 |
8,8′-Oxo-biplumbagin |
Diospyros shimbaensis |
NA |
MDA-MB-231 |
PhytoCAT-986 |
Trans-isoshinanolone |
Diospyros shimbaensis |
NA |
MDA-MB-231 |
PhytoCAT-987 |
Cis-isoshinanolone |
Diospyros shimbaensis |
NA |
MDA-MB-231 |
PhytoCAT-988 |
3,3′-Biplumbagin |
Diospyros shimbaensis |
NA |
MDA-MB-231 |
PhytoCAT-989 |
Diospyros shimbaensis extract (Methanol extract) |
Diospyros shimbaensis |
NA |
MDA-MB-231 |
PhytoCAT-990 |
Diospyros shimbaensis extract (Isohexane extract) |
Diospyros shimbaensis |
NA |
MDA-MB-231 |
PhytoCAT-991 |
Diospyros shimbaensis extract (Dichloromethane extract) |
Diospyros shimbaensis |
NA |
MDA-MB-231 |
PhytoCAT-992 |
Diospyros shimbaensis extract (Methanol crude extract from the root barks) |
Diospyros shimbaensis |
NA |
MDA-MB-231 |
PhytoCAT-993 |
Diospyros shimbaensis extract (Dichloromethane crude extract from the leaves) |
Diospyros shimbaensis |
NA |
MDA-MB-231 |
PhytoCAT-994 |
Diospyros shimbaensis extract (Methanol crude extract from the leaves) |
Diospyros shimbaensis |
NA |
MDA-MB-231 |
PhytoCAT-995 |
Methyl angolensate |
Soymida febrifuga |
KU70, KU80 |
T47D |
PhytoCAT-996 |
Khat (Extract of Catha edulis) |
Catha edulis |
Bax, Bcl-2, p-JNK, p-ERK |
MDA-MB-231 |
PhytoCAT-997 |
Tanacetum Polycephalum extract (TPHE) |
Tanacetum polycephalum |
NA |
MCF-7 |
PhytoCAT-998 |
Methyl β-lilacinobioside |
Caralluma retrospiciens |
topo II |
MCF-7 |
PhytoCAT-999 |
Leptadenia pyrotechnica extract |
Leptadenia pyrotechnica |
NA |
MCF-7 |
PhytoCAT-1000 |
Wedelolactone |
Sphagneticola calendulacea |
ERα, ERβ, SoX2, ABCG2 |
NA |
PhytoCAT-1001 |
Eupafolin |
Eupatorium album |
Bax, Caspase 3, Bcl-2, PI3K, AKT, mTOR |
EO771 |
PhytoCAT-1002 |
Evodiamine |
Evodia rutaecarpa |
MMP9, uPA, uPAR, ERK, p38 MAPK, topo I, Bax, Bcl-2, Caspase 3, Survivin |
MDA-MB-231, MCF-7, A375-S2, HeLa, THP-1, L929 |
PhytoCAT-1003 |
Cephalinone D |
Cephalantheropsis gracilis |
NA |
MCF-7, NCI-H460, and SF-269 |
PhytoCAT-1004 |
Flavanthrin |
Cephalantheropsis gracilis |
NA |
MCF-7, NCI-H460, and SF-270 |
PhytoCAT-1005 |
Tryptanthrin |
Cephalantheropsis gracilis |
NA |
MCF-7, NCI-H460, and SF-268, HCT-15 |
PhytoCAT-1006 |
Julibroside (J29) |
Albizia julibrissin |
NA |
MDA-MB-435, PC-3M-1E8, HeLa |
PhytoCAT-1007 |
Julibroside (J30) |
Albizia julibrissin |
NA |
MDA-MB-435, PC-3M-1E8, HeLa |
PhytoCAT-1008 |
Julibroside (J31) |
Albizia julibrissin |
NA |
MDA-MB-435, PC-3M-1E8, HeLa |
PhytoCAT-1009 |
Voacamine |
Voacanga africana |
NA |
MDA-MB-231, HEPG-2, A375, SH-SY5Y, CT26 |
PhytoCAT-1010 |
19-epi-voacristine |
Voacanga africana |
NA |
MDA-MB-231, HEPG-2, A375, SH-SY5Y, CT26 |
PhytoCAT-1011 |
Vobasine |
Voacanga africana |
NA |
MDA-MB-231, HEPG-2, A375, SH-SY5Y, CT26 |
PhytoCAT-1012 |
Voacristine |
Voacanga africana |
NA |
MDA-MB-231, HEPG-2, A375, SH-SY5Y, CT26 |
PhytoCAT-1013 |
Galanal A |
Boesenbergia rotunda |
NA |
MCF-7, LK-2, A549, ECC4, HeLa, DU145 |
PhytoCAT-1014 |
Galanal B |
Boesenbergia rotunda |
NA |
MCF-7, LK-2, A549, ECC4,HeLa, DU145 |
PhytoCAT-1015 |
Voacangine |
Voacanga africana |
NA |
MDA-MB-231, HEPG-2, A375, SH-SY5Y, CT27 |
PhytoCAT-1016 |
Pyranocycloartobiloxanthone A (PA) |
Artocarpus obtusus |
Bax, Bcl-2 |
MCF-7, K562, HL-60 |
PhytoCAT-1017 |
Curcumin and berberine combination |
Curcumin - Curcuma longa Berberine - Thalictrum delavayi |
Bcl-2, JNK, Beclin-1 |
MCF-7, MDA-MB-231 |
PhytoCAT-1018 |
Ent-1β,3β,16β,17-tetrahydroxyatisane |
Euphorbia fischeriana |
NA |
MCF-7, HepG-2 , SGC-7901 |
PhytoCAT-1019 |
Ent-1β,3α,16β,17-tetrahydroxyatisane |
Euphorbia fischeriana |
NA |
MCF-7, HepG-2 , SGC-7901 |
PhytoCAT-1020 |
Euphorbia hirta extract |
Euphorbia hirta |
Caspase 2, Caspase 6, Caspase 8, Caspase 9 |
MCF-7 |
PhytoCAT-1021 |
Ginsenoside Rg3 |
Panax ginseng |
CXCR4, STXBP5-AS1, RFX3-AS1 , EEF2, MYCBP2, STXBP5, GRM1, RFX3, SLC1A1, WT1 |
MDA-MB-231, MCF-7, MCF-10A |
PhytoCAT-1022 |
Formononetin |
Astragalus membranaceus |
hTERT,c-MYC,Bcl-2, Ha-ras, QR, C3, COX7RP, SULT1A3, ERα, miR-375, AKT, Bcl-2, MMP2, MMP9, TIMP-1, TIMP-2, TNF-α, IL-6 and IL-1β, nitrite, PGE2, iNOS, COX-2 |
MCF-7, MDA-MB-231, 4T1, ER-positive MCF-7, T47D, Caco-2, SKBR-3, HUVEC, LNCaP, PC-3 |
PhytoCAT-1023 |
Quercetin |
Melia azedarach |
PTEN, CYP1B1, EGFR, AKR1C3, PIP, SULT1E1, CDK6, STAT-3,UCA1, CAT, Bcl-2, EGFR, RRM2B, CYP3A4, POTEE, Bax, FAS, MMP2, MMP9, MYC, CASP3, CCND1, CD34, CDK2, CXCL10, CXCL11, DVL2, HSF2, RRM2B, PIG8, CD95, PIDD, Tp53INP, Noxa, p21, PUMA, AMPK, COX-2, PI, HER-2, VEGFR-2, PI3K, AKT, PKB, CYP1A1, CYP1B1 |
HeLa, MDA-MB-231, HEP-2, RD, MCF-7, HepG-2, HCT-116, HeLa, CYP1B1, T47D, 143B, HT - 29, MDA-MB-231 - estrogen-negative breast cancer, MDA-MB-435, MDA-MB-468, HCC-38, BT-474, SK-Br3, TAMR-MCF-7, C6 and COLO-205,KBCHR8-5, DLD-1, DLD-1 human colorectal cancer xenograft model in nude mice, NUDE MICE created from green fluorescent protein-tagged MDA-MB-435 bone metastatic variant |
PhytoCAT-1024 |
Epigallocatechin gallate (EGCG) |
Limoniastrum guyonianum |
EGFR, GOLM1,, FAS, ERα, PTEN, p21, Bax, p-PDK1, AKT, Cyclin D1, Bcl-2 |
MDA-MB-231, 4T1, , MCF-7, MCF-7tam,Hs578T, T47D, WI38VA, Caco-2, Hs578T, SUM-149, SUM-190, BT-20, BT-549, MDA-MB-435, HFF |
PhytoCAT-1025 |
Artahongkongol A |
Artabotrys hongkongensis |
NA |
MCF-7, HL-60, SMMC-7721, A-549, SW480 |
PhytoCAT-1026 |
1a-hydroxy-5,11-
eudesmadiene |
Artabotrys hongkongensis |
NA |
MCF-7, HL-60, SMMC-7721, A-549, SW480 |
PhytoCAT-1027 |
5-eudesmene-1b,4a-diol |
Artabotrys hongkongensis |
NA |
MCF-7, HL-60, SMMC-7721, A-549, SW480 |
PhytoCAT-1028 |
1b,11-dihydroxy-5- eudesmene |
Artabotrys hongkongensis |
NA |
MCF-7, HL-60, SMMC-7721, A-549, SW480 |
PhytoCAT-1029 |
1b-hydroxy-11-methoxy-5- eudesmene |
Artabotrys hongkongensis |
NA |
MCF-7, HL-60, SMMC-7721, A-549, SW480 |
PhytoCAT-1030 |
2a-hydroxy pterodontic acid |
Artabotrys hongkongensis |
NA |
MCF-7, HL-60, SMMC-7721, A-549, SW480 |
PhytoCAT-1031 |
1b,9b-dihydroxy-4aH-eudesma-5,11(13)- dien-12-oic acid |
Artabotrys hongkongensis |
NA |
MCF-7, HL-60, SMMC-7721, A-549, SW480 |
PhytoCAT-1032 |
1b,3a-dihydroxyeudesma-5,11(13)-dien-12-oic acid |
Artabotrys hongkongensis |
NA |
MCF-7, HL-60, SMMC-7721, A-549, SW480 |
PhytoCAT-1033 |
Lentinula edodes mycelia extract |
Lentinula edodes(mushroom) |
SOD1 |
MCF-7 and MDA-MB-231 cells. |
PhytoCAT-1034 |
Caesalpinia spinosa extract (P2Et) |
Caesalpinia spinosa |
Caspase 3, Caspase 9, CD4, CD8, Calreticulin , IFN-γ |
B16F10, A375, 4T1 |
PhytoCAT-1035 |
Grifolin |
Albatrellus confluens |
Bax, Bcl-2, Caspase 8, Caspase 9, Caspase 3, DAPK1 |
MCF-7, HL-60, SMMC-7721, A-549 |
PhytoCAT-1036 |
(4α,5α,8β,10β)-4,10-dihydroxy-1,11(13)-guaidien-12,8-olide |
Chrysophthalmum montanum |
NA |
MCF-7, MDA-MB 231, HT-29, PC3 |
PhytoCAT-1037 |
Achyrobichalcone |
Achyrocline satureioides |
Caspase 9, Caspase 3, Caspase 7 |
MDA-MB-231 and MCF-12A |
PhytoCAT-1038 |
Luteolin |
Avicennia marina |
Cyclin E2, Bcl-2, Caspase 3, Bax, VEGF, YAP/TAZ, ABCG2, CD44, EMT, VEGF, MPA, Aromatase, CYP1A1, CYP1B1 |
MDA-MB-468, MCF-7, MDA-MB-453, MDA-MB-231, Hs578T, Progestin-dependent xenograft, LNM35, HT29, HepG2 |
PhytoCAT-1039 |
6-prenylnaringenin (6-PN) |
Humulus lupulus |
NA |
MDA-MB-231, T-47D, PC-3, HT-29, A-2780 |
PhytoCAT-1040 |
8-prenylnaringenin (8-PN) |
Humulus lupulus |
NA |
MDA-MB-231, T-47D, PC-3, HT-29, A-2780 |
PhytoCAT-1041 |
Ziyuglycoside I |
Sanguisorba officinalis |
p53, p21WAF1, Bax, Bcl-2 |
MDA-MB-231 |
PhytoCAT-1042 |
Quercitrin |
Mangifera pajang |
ABCG2 |
MCF-7, HeLa, HT-29 |
PhytoCAT-1043 |
Artemisia herba alba extracts |
Artemisia herba |
NA |
MCF-7, HeLa |
PhytoCAT-1044 |
Kigelia Africana, Ximenia Caffra and Mimusops Zeyheri Seed Oils |
Kigelia Africana, Ximenia Caffra and Mimusops Zeyheri |
CD62P, CD63 |
MCF-7, MDA-MB-231 |
PhytoCAT-1045 |
Camphoratin F |
Taiwanofungus camphoratus |
NA |
MCF-7, Hep2, Hela |
PhytoCAT-1046 |
Camphoratin E |
Taiwanofungus camphoratus |
NA |
MCF-7, Hep2, Hela |
PhytoCAT-1047 |
Antrocamphin A |
Taiwanofungus camphoratus |
NA |
MCF-7, Hep2, Hela |
PhytoCAT-1048 |
Antcin A |
Taiwanofungus camphoratus |
NA |
MCF-7, Hep2, Hela |
PhytoCAT-1049 |
Costunolide |
Costus speciosus |
p21WAF1, Cdc2, Cyclin B1, Fas, Caspase 8, Caspase 3, Cyclin D1, Cyclin D3, CDK-4, CDK-6, p18 INK4c, p27 KIP1 |
MDA-MB-231, MCF-7 |
PhytoCAT-1050 |
(6S,9S)-roseoside |
Abutilon theophrasti |
NA |
MCF-7 |
PhytoCAT-1051 |
Abutilon theophrasti extract |
Abutilon theophrasti |
NA |
MCF-7, CCRF-CEM and CEM/ADR5000 |
PhytoCAT-1052 |
3-hydroxyflavone |
Acacia retinodes |
NA |
MCF-7/BUS |
PhytoCAT-1053 |
Ginnalin A |
Acer rubrum |
Cyclin A, Cyclin D1 |
MCF-7, HCT-116 |
PhytoCAT-1054 |
Ageratum conyzoides extract |
Ageratum conyzoides |
MMP9 |
T47D, 4T1 |
PhytoCAT-1055 |
Ajuga bracteosa extract |
Ajuga bracteosa |
NA |
MCF-7, Hep-2 |
PhytoCAT-1056 |
Diallyl disulfide |
Allium sativum |
Bax, Bcl-2, Bcl-xL, Bcl-w |
MCF-7 |
PhytoCAT-1057 |
Diallyl trisulfide |
Allium sativum |
Bcl-2, PARP, JNK |
MCF-7 |
PhytoCAT-1058 |
Kaempferol |
Justicia gendarussa |
IQGAP3, CYP1A1, CYP1B1, Survivin, PR, AHR, ERα, GREB1, Aromatase |
MCF-7, HCT-15, T47D, C-6, BT-549, A549, HEK293,MDA-MB-231, MDA-MB-468 |
PhytoCAT-1059 |
γ-Tocotrienol |
Amaranthus cruentus |
Cyclin D1, CDK2, CDK4, CDK6, Rb, E2F1, p27, p16 |
MCF-7, MDA-MB-231 |
PhytoCAT-1060 |
Gamma-linolenic acid (GLA) |
Anemone cylindrica |
Her-2/neu |
BT-474, SK-Br3, MDA-MB-453, SK-OV3, NCI-N87 |
PhytoCAT-1061 |
Ferulic acid |
Angelica sinensis |
HER2, ESR1 |
MCF-7, BT-474, MDA- MB-231, SKBR-3 |
PhytoCAT-1062 |
Alpha-lipoic acid |
Arabidopsis thaliana |
p27(kip1), Bax, Bcl-2 |
MCF-7, SK-N-SH, Hela |
PhytoCAT-1063 |
3,3'-diindolylmethane (DIM) |
Arundo donax |
FoxM1, CXCR4, CXCL12, p21, Cadherin-11, Plasminogen |
MDA-MB-231, MCF-7, MDA-MB-468, SKBR-3, BALB/c mice, T47D, Saos2 |
PhytoCAT-1064 |
Desacetyl nimbinene (DAN) |
Azadirachta indica |
JNK, p38, SOD1, SOD2 |
MCF-7, MDA-MB-231 |
PhytoCAT-1065 |
Bacopa monnieri extract |
Bacopa monnieri |
NA |
MCF-7, MDA-MB 231 |
PhytoCAT-1066 |
Boerhaavia diffusa extract |
Boerhaavia diffusa |
NA |
NA |
PhytoCAT-1067 |
Allyl Isothiocyanate |
Brassica nigra |
TRPA1 |
MCF-7, MDA-MB-231 |
PhytoCAT-1068 |
Broccoli sprouts (BSp) |
Brassica oleracea |
DNMT1, HDAC1 |
PC3, BPH-1, LnCaP, MCF-7 |
PhytoCAT-1069 |
Brazilin |
Caesalpinia sappan |
p38, p53, DNMT1, p21 |
SiHa, MDA-MB-231, A549, NCI- H1299 |
PhytoCAT-1070 |
Cajanin stilbene acid |
Cajanus cajan |
MYC |
MCF-7 |
PhytoCAT-1071 |
Calcitrinone A |
Callistemon citrinus |
NA |
MDA-MB-231 |
PhytoCAT-1072 |
Sasanquasaponin (SQS) |
Camellia oleifera |
p21, Cyclin D1 |
MCF-7, HepG2 |
PhytoCAT-1073 |
Epicatechin |
Garcinia mangostana |
DR4/DR5, Bad, Bax |
MCF-7, T47D, MDA-MB-231, HCT116 |
PhytoCAT-1074 |
Epicatechin gallate |
Garcinia mangostana |
HIF-1, GLUT-1, VEGF, CDKN1A |
T47D, MCF-7 |
PhytoCAT-1075 |
Δ9-tetrahydrocannabinolic acid |
Cannabis sativa |
NA |
MDA-MB-231, HCT-116 |
PhytoCAT-1076 |
Capsicum annuum extract (CAP) |
Capsicum annuum |
VEGF |
MCF-7, MDA-MB-231, MDA-MB-435 |
PhytoCAT-1077 |
Chestnoside B |
Castanea sativa |
NA |
MCF-7, PC3 |
PhytoCAT-1078 |
Luteolin-7-O-glucoside |
Celosia argentea |
NA |
MCF-7, SiHa, HCT |
PhytoCAT-1079 |
1-(4-hydroxy-2-methoxybenzofuran-5-yl)-3-phenylpropane-1,3-dione |
Celosia argentea |
NA |
MCF-7, SiHa, HCT |
PhytoCAT-1080 |
Ukrain |
Chelidonium majus |
NA |
SKBR-3, 4T07, TUBO, MDA-MB-231, PA-TU-8902, CCL-221 , U-138MG |
PhytoCAT-1081 |
25-O-acetyl-7,8-didehydrocimigenol-3-O-β-d-(2-acetyl)xylopyranoside (ADHC-AXpn) |
Cimicifuga foetida |
ERK1, ERK2, Raf,AKT |
MCF-7, HepG2, HepG2/ADM, HeLa,PC3 |
PhytoCAT-1082 |
Citrus lemon extract |
Citrus limon |
JAK1, JAK2, TYK2, IRF7, IRF3 |
MDA-MB-231, Vero |
PhytoCAT-1083 |
Osthole |
Cnidium monnieri |
GPX1, SOD2, GCL-c, G6pdh, NOX2, ACOX, FASN, c-met, c-FLIP, Bax, Akt, mTOR, p53, p21, Cdk2, cyclin D1 Caspase 3, Caspase 9 |
MDA-MB-231, MDA-MB-435, Caki, U251MG, |
PhytoCAT-1084 |
Falcarindiol |
Cnidium officinale |
Bax , p53, Bcl-2 |
MCF-7, HCT-116 |
PhytoCAT-1085 |
Kahweol |
Coffea arabica |
PEA3, AP-2, FASN, SREBP-1c, mTOR |
SKBR-3 |
PhytoCAT-1086 |
Hawthorn fruit (HF) extract |
Crataegus pinnatifida |
Caspase 3, Caspase 9 |
MCF-7, SKOV-3 |
PhytoCAT-1087 |
Saffron extract |
Crocus sativus |
NA |
MCF-7 |
PhytoCAT-1088 |
Cucumol B |
Cucumis melo |
NA |
SKOV-3, MCF-7, and HCT-116 |
PhytoCAT-1089 |
Cuscutamine |
Cuscuta chinensis |
NA |
MCF-7, T47D |
PhytoCAT-1090 |
Cuscutic resinoside A |
Cuscuta chinensis |
NA |
MCF-7, T47D |
PhytoCAT-1091 |
Cynanchum paniculatum extract |
Cynanchum paniculatum |
MMP2 |
MDA-MB-231, MCF-7, ZR-75-1 |
PhytoCAT-1092 |
Cyperus rotundus extract (EECR) |
Cyperus rotundus |
Bcl-2, Bax |
MDA-MB-231, MDA-MB-468 |
PhytoCAT-1093 |
Dioscorea bulbifera extract |
Dioscorea bulbifera |
NA |
MDA-MB-231, MCF-7, HCT116 |
PhytoCAT-1094 |
Dioscin |
Dioscorea villosa |
GATA3, DNMT3A, TET2, TET3, ZFPM2 , E-cad, TET1, VIM, MMP9, Bcl-2, cIAP-1, Mcl-1 |
MCF-7, MDA-MB-231, T47D |
PhytoCAT-1095 |
Diospyros lotus extract |
Diospyros lotus |
NA |
MCF-7, COR-L23, CaCo-2, C32, ACHN, A375, A549, Huh-7D12 and LNCaP |
PhytoCAT-1096 |
Dittrichia viscosa extract |
Dittrichia viscosa |
NA |
MDA-MB-231, PC3 |
PhytoCAT-1097 |
Syringin |
Eleutherococcus senticosus |
PARP, XIAP, MAP2K1, PIK3CA, HRAS, EGFR, Caspase3, and PTGS2 |
MCF-7, MDA-MB-231 |
PhytoCAT-1098 |
Embelin |
Embelia ribes |
SOD1, ERK1, ERK2, Bax, Bcl-2, XIAP |
MCF-7, 4T1 |
PhytoCAT-1099 |
Erucin |
Eruca sativa |
SOD1, ERK1, ERK2, Bax, Bcl-2, XIAP |
MDA-MB-231, SKBR-3, T47D, MCF-7 |
PhytoCAT-1100 |
F1012-2 |
Eupatorium lindleyanum |
Cyclin B1, cdc2, p21, p-cdc2. |
MDA-MB-231, MDA-MB-468, MDA-MB-231 xenografts |
PhytoCAT-1101 |
Dihydroconiferyl alcohol |
Euterpe oleracea |
NA |
MCF-7 |
PhytoCAT-1102 |
(+)-lariciresinol |
Euterpe oleracea |
NA |
MCF-7 |
PhytoCAT-1103 |
(+)-pinoresinol |
Euterpe oleracea |
p53 |
MCF-7, MDA-MB-231, HCT116, LNCaP |
PhytoCAT-1104 |
(+)-syringaresinol |
Euterpe oleracea |
NA |
HeLa, Hep3B, MCF-7 |
PhytoCAT-1105 |
Protocatechuic acid methyl ester |
Euterpe oleracea |
NA |
MCF-7 |
PhytoCAT-1106 |
Açai extract |
Euterpe oleracea |
NA |
MCF-7 |
PhytoCAT-1107 |
Ferula assa-foetida essential oil |
Ferula assa-foetida |
NA |
4T1 |
PhytoCAT-1108 |
Farnesiferol A |
Ferula persica |
NA |
MCF-7 |
PhytoCAT-1109 |
Tannic acid |
Forsythia suspensa |
CXCL12, CXCR4 |
MCF-7, MDA-MB-231 |
PhytoCAT-1110 |
Arctigenin |
Arctium lappa |
4EBP1, STAT-3, RAD51, Survivin, β-catenin, Cyclin D1 |
MDA-MB-231, MCF-7 |
PhytoCAT-1111 |
Gambogenic acid |
Garcinia hanburyi |
Fas, Caspase 3,-8,-9, Bax, Bcl-2 |
MDA-MB-231 |
PhytoCAT-1112 |
Ginkgolic acid C15:1 |
Ginkgo biloba |
FAS |
MCF-7, A549, HL-60 |
PhytoCAT-1113 |
Ginkgolic acid C17:2 |
Ginkgo biloba |
FAS |
MCF-7, A549, HL-60 |
PhytoCAT-1114 |
Ginkgolic acid C17:1 |
Ginkgo biloba |
FAS |
MCF-7, A549, HL-60 |
PhytoCAT-1115 |
Ginkgolic acid C13:0 |
Ginkgo biloba |
uPA, PAI-1, CXCR4, MMP9 |
MCF-7 and MDA-MB 231 |
PhytoCAT-1116 |
Ginkgo biloba extract |
Ginkgo biloba |
Caspase 3, Bcl-2, Bax, CYP1B1, Aryl hydrocarbon receptor |
MDA-MB-231, MCF-7 |
PhytoCAT-1117 |
Glaucium flavum extract |
Glaucium flavum |
NA |
MDA-MB-435, MDA-MB-231, Hs578T |
PhytoCAT-1118 |
Glehnia littoralis extract |
Glehnia littoralis |
CDK4, Cyclin D1 , p21, p27 |
MCF-7 |
PhytoCAT-1119 |
Tectochrysin |
Hedychium spicatum |
ABCG2 |
MDA-MB-231 |
PhytoCAT-1120 |
Phytoene |
Hibiscus syriacus |
NA |
T47D, MCF-7, ECC-1 |
PhytoCAT-1121 |
St. John's Wort extract (SJWE) |
Hypericum perforatum |
Bcl-2 and Bcl-xL |
MDA-MB-231, MCF-7 |
PhytoCAT-1122 |
2-Methoxyestrone |
Imperata cylindrica |
NA |
BT-549, HT-29 |
PhytoCAT-1123 |
11, 16-Dihydroxypregn-4-ene-3, 20-dione |
Imperata cylindrica |
NA |
BT-549, HT-29 |
PhytoCAT-1124 |
Daucosterol linolenate (DLA) |
Ipomoea batatas |
Caspase 3, Caspase 9, PARP-1 , Ki67, VEGF, Bcl-2,Bax, Bcl-xL |
MCF-7 xenograft in nude mice, MDA-MB-231, 4T1 |
PhytoCAT-1125 |
5,7- dihydroxy-3,4'-dimethoxyflavone |
Juglans regia |
NA |
MCF-7, BHY |
PhytoCAT-1126 |
Regiolone |
Juglans regia |
NA |
MCF-7, BHY |
PhytoCAT-1127 |
Juglans regia extract |
Juglans regia |
NA |
MCF-7, NCI-H460, HeLa, HepG2 |
PhytoCAT-1128 |
Effususin B |
Juncus effusus |
NA |
SHSY-5Y, SMMC-7721, HepG2, Hela, and MCF-7 |
PhytoCAT-1129 |
Essential oil of Juniperus communis |
Juniperus communis |
NA |
MCF-7 |
PhytoCAT-1130 |
Lawsonia inermis extract |
Lawsonia inermis |
NA |
MCF-7, A549, C6 and COLO-205 |
PhytoCAT-1131 |
Aviculin |
Lespedeza cuneata |
PARP, Caspase 9, Caspase 7, Bax, Bcl-2 |
MCF-7 |
PhytoCAT-1132 |
Methyl jasmonate |
Lonicera japonica |
Caspase 3, PAL |
MDA-MB-435, MCF-7, A549 |
PhytoCAT-1133 |
Cudraxanthone I |
Maclura cochinchinensis |
Caspase 3, Caspase 7, Caspase 8, Caspase 9 |
MDA-MB-231 BCRP |
PhytoCAT-1134 |
Tetramethoxystilbene |
Maclura pomifera |
CYP1A1 , CYP1B1, Nqo1 , IL-8 |
MCF-7 |
PhytoCAT-1135 |
Pomiferin |
Maclura pomifera |
NA |
MCF-7, MDA-MB-231 |
PhytoCAT-1136 |
Honokiol |
Magnolia obovata |
c-Src, EGFR, AKT, mTOR , 4E-BP and p70 S6 kinase, Caspase 3, Caspase 8, Caspase 9, Bid, Bcl-2, Neu1, NO, COX-2, NF-kB, IL-6, miR-188-5p, FBXW7 |
Female Sprague Dawlely (SD) rats, MCF-7/ADR, MCF-7, 4T1, MDA-MB-231 |
PhytoCAT-1137 |
Hirsutine |
Uncaria tomentosa |
γH2AX, Caspase 3, Caspase 7 |
MCF-7, MDA-MB-231, MDA-MB-468, MDA-MB-453, ZR-75-1, BT-474 |
PhytoCAT-1138 |
Magnolol |
Magnolia officinalis |
miR-200c |
T47D, MCF-7, Hela, A549 |
PhytoCAT-1139 |
Mango polyphenolics |
Mangifera indica |
PI3K, AKT, HIF-1α, VEGF mRNA, pAKT, AKT, pPI3K (p85), VEGF, NF-κB , NF-κB (p65), PARP |
BT-474, xenografts in mice |
PhytoCAT-1140 |
Dihydro-β-agarofuran |
Maytenus cuzcoina, Maytenus canariensis, Maytenus magellanica, Maytenus chubutensis |
P-gp |
MDA-MB-231, NIH-3T3, NIH-3T3 MDR-G185, MDCKII, MDCKII-MRP2,MDA-MB-231-BCRP |
PhytoCAT-1141 |
Endophytes of noni |
Morinda citrifoliainn |
NA |
LU-1, PC-3, MCF-7 |
PhytoCAT-1142 |
Phenethyl Isothiocyanate |
Nasturtium officinale |
MTDH , CDH1, TSC2, sfRON |
MCF-7, MDA-MB-231, PC-3, DU145, U87, HCT116, HepG2, SKBR-3 |
PhytoCAT-1143 |
Isoliensinine |
Nelumbo nucifera |
p38 MAPK, JNK, CDK2, p21, AKT, GSK3α |
MCF-7, MDA-MB-231, HeLa, A549, PC3, HepG2, Hep3B, H1299 |
PhytoCAT-1144 |
Neferine (NEF) |
Nelumbo nucifera |
miR-374a/FGFR-2 |
MDA-MB-231, MCF-7 |
PhytoCAT-1145 |
Thymoquinone (TQ) |
Nigella sativa |
HSPA6, CXCR4, p53, DNMT1,3A,3B, G9A, HDAC1,4,9, KDM1B, KMT2A,B,C,D,E, DLC1, PPARG, ST7, FOXO6, TET2, CYP1B1, SALL4, DDIT3, RASL11B, RASD1, GNG3, BAD, BIK |
MCF-7, MBD-MB 231 |
PhytoCAT-1146 |
Ocimum basilicum (OB) extract |
Ocimum basilicum |
AMPK |
HeLa, MCF-7, Jurkat, HT-29, T24, MIAPaCa-2 |
PhytoCAT-1147 |
Oleuropein |
Olea europaea |
CASP1, CASP14, FADD, TNFRSF21, GADD45A, CYCS, BNIP2, BNIP3, BID, BCL10, CFLAR, BFAR, BRAF, IAP, BIRC3, RIPK2, TNFRSF10A, CASP4, CASP6, PYD, PAYCARD, BIRC5, TNFRSF11B, HDAC2, HDAC3 |
MDA-MB-468, MDA-MB-231, SKBR-3 |
PhytoCAT-1148 |
Ophiopogonin D |
Ophiopogon japonicus |
TGF-β1, ITGB1, MMP9, FAK, Src, AKT |
MDA-MB-231, Hs 578Bst |
PhytoCAT-1149 |
Oplopanax horridus extract |
Oplopanax horridus |
NA |
SW-480, HCT-116, HT-29, MCF-7, NSCLC |
PhytoCAT-1150 |
Rh2 |
Panax ginseng |
Cyclin D3, CIP1, RNF217, RNA STXBP5-AS1 |
MCF-7 |
PhytoCAT-1151 |
Pennogenin 3-O-α-L-rhamnopyranosyl-(1→4)-[α-L-rhamnopyranosyl-(1→2)]-β-D-glucopyranoside |
Paris quadrifolia |
NA |
HL-60, HeLa and MCF-7 |
PhytoCAT-1152 |
Pennogenin 3-O-α-L-rhamnopyranosyl-(1→4)-α-L-rhamnopyranosyl-(1→4)-[α-L-rhamnopyranosyl-(1→2)]-β-D-glucopyranoside |
Paris quadrifolia |
NA |
HL-60, HeLa and MCF-7 |
PhytoCAT-1153 |
Parkinsonia aculeata extract |
Parkinsonia aculeata |
NA |
MCF-7, HepG-2 |
PhytoCAT-1154 |
Peucedanum japonicum Thunb (PJT) extract |
Peucedanum japonicum |
MMP9 |
MCF-7 |
PhytoCAT-1155 |
Pinolenic acid |
Pinus koraiensis |
COX-2 |
MDA-MB-231 |
PhytoCAT-1156 |
Pinus nigra Arn. bark extracts from Mokra gora (MG) and Tara mountains |
Pinus nigra |
NA |
MCF-7, HeLa,HT-29, MRC-5 |
PhytoCAT-1157 |
Baneh gum |
Pistacia atlantica |
p53, Caspase 3 |
MCF-7 |
PhytoCAT-1158 |
Pithecellobium dulce extract |
Pithecellobium dulce |
Bax, p21, p53 , TNF, fasBcl-2, NF-κB, CDK |
MCF-7 |
PhytoCAT-1159 |
Aucubin |
Plantago media |
NA |
MCF-7, MDA-MB-231, HeLaS3, A549, and KB |
PhytoCAT-1160 |
Plantago major extract |
Plantago major |
TNF-α, IL-1β, IL-6, IFN-γ |
MCF-7, MDA-MB-231, HeLaS3, A549, and KB |
PhytoCAT-1161 |
Jaboticaba peel extract (JPE) |
Plinia cauliflora |
NA |
MDA-MB-231, L929 |
PhytoCAT-1162 |
Podophyllum hexandrum extract |
Podophyllum hexandrum |
Catalase, Superoxide dismutase, Glutathione peroxidase |
MCF-7, A-549, PC-3, Colo-25, IMR-32, SF-295, MDA-MB-231 |
PhytoCAT-1163 |
Polygonatum odoratum extract |
Polygonatum odoratum |
Bcl-2, Bax |
MDA-MB-231 |
PhytoCAT-1164 |
Neohesperidin |
Poncirus trifoliata |
p53, Bax, Bcl-2 |
MDA-MB-231, MCF-7 |
PhytoCAT-1165 |
Chinese propolis extract (CPWE) |
Populus tremula (poplar) |
Caspase 3 |
MCF-7, MDA-MB-231, HeLa, and A549 |
PhytoCAT-1166 |
Prosopis juliflora extract |
Prosopis juliflora |
NA |
MCF-7, HepG2 , LS-174T |
PhytoCAT-1167 |
Betulinic acid |
Prunus dulcis |
GRP78, NOP2, p120, WDR12, S6 ribisomal protein, p21 |
MCF-7, HepG2, A549, HL-60,HCT-116, PC-3, HeLa |
PhytoCAT-1168 |
Amygdalin |
Prunus spinosa |
Bcl-2, PARP, Bax, Caspase 3, Survivin, XIAP, GAS5, MALAT1 |
MDA-MB-231, Hs578T, MCF-7, HepG2 |
PhytoCAT-1169 |
3beta-trans-p-coumaroyloxy-2alpha-hydroxyolean-12-en-28-oic acid |
Psidium guajava |
NA |
MCF-7, HepG2, Caco-2 |
PhytoCAT-1170 |
Eleostearic acid (alpha-ESA) |
Momordica charantia |
HER2/HER3, PTEN |
MDA-MB-231, SKBR-3, T47D |
PhytoCAT-1171 |
Pomegranate extract |
Punica granatum |
MRE11, RAD50, NBS1, RAD51, BRCA1, BRCA2, BRCC3, miR-183, miR-24 |
MCF-7, MDA-MB-231, HEC-1A, SiHa, HeLa, SKOV3, MCF-10A |
PhytoCAT-1172 |
Emodin |
Rheum palmatum |
IRF4, STAT6, Runx2, Bcl-2, Bax, Cytochrome c, MMP9, activator -1, NF-κB, miR-34a, IRF4, EMT |
MCF-7, 4T1, ZR-75-1, MDA-MB-453, MDA-MB-231, mice bearing EO771 or 4T1
|
PhytoCAT-1173 |
Rhus verniciflua Stokes extract (PPEF) |
Rhus verniciflua |
NA |
MCF-7, MDA-MB-231, SKBR-3, AGS, SNU-668, SNU-638, A549, NCI-H157, HCT116, HepG2 |
PhytoCAT-1174 |
Carnosic acid |
Rosmarinus officinalis |
AKR1C2, TNXRD1, HMOX1, GDF15, PHLDA1, DDIT3, ID3, CDKN2C, Cyclin B1 |
MDA-MB-453, NCI-H82 , DU-145 , Hep-3B , K-562 , MCF-7, PC-3, MDA-MB-231 |
PhytoCAT-1175 |
Carnosol |
Rosmarinus officinalis |
STAT-3, MMP9, Cyclin B1 |
MDA-MB-231, Hs578T, MCF-7,T47D |
PhytoCAT-1176 |
Bigelovii A |
Salicornia bigelovii |
Bcl-2, Cyclin D1, NF‑κB‑regulated gene products, Cyclin D1, COX‑2 |
MDA‑MB‑231, MDA‑MB‑468HL-60, MCF-7, HepG2, A549 |
PhytoCAT-1177 |
3β-[(α-L-arabinopyranosyl)oxy]-19α,23-dihydroxyolean-12-en-28-oic acid 28-[6-O-acetyl-β-D-glucopyranosyl] ester |
Sanguisorba officinalis |
NA |
MCF-7, HeLa, HepG2, SGC-7901, NCI-H460, and BGC-823 |
PhytoCAT-1178 |
2α,3β,19α,23-tetrahydroxyurs-12-en-28-oic acid 28-[6-O-acetyl-β-D-glucopyranosyl] ester |
Sanguisorba officinalis |
NA |
MCF-7, HeLa, HepG2, SGC-7901, NCI-H460, and BGC-823 |
PhytoCAT-1179 |
3β-[(α-L-arabinopyranosyl)oxy]-19α-hydroxyurs-12,20(30)-dien-28-oic acid 28-[6-O-acetyl-β-D-glucopyranosyl] ester |
Sanguisorba officinalis |
NA |
MCF-7, HeLa, HepG2, SGC-7901, NCI-H460, and BGC-823 |
PhytoCAT-1180 |
Schisandrin B |
Schisandrae Chinensis |
NOX4, TGF-β |
4T1, siha, MCF-7, A2780 |
PhytoCAT-1181 |
Schisandrin A |
Schisandrae Chinensis |
p65, STAT-3 |
MDA-MB-231, BT-549, MDA-MB-231 xenograft mouse model |
PhytoCAT-1182 |
Scutellarein |
Erigeron breviscapus |
CYP1A1, CYP1B1 |
MDA-MB-468, MCF-7, MCF10A |
PhytoCAT-1183 |
Baicalin |
Scutellaria baicalensis |
miR-338-3p, MORC4, ALPP, DUSP1, CYR61, ALPPL2, SPP1, TLR4, EMT |
T-47D, MCF-7, MDA-MB-231 |
PhytoCAT-1184 |
Baicalein-8-sodium sulfonate (BcS) |
Scutellaria baicalensis |
NA |
MCF-7 |
PhytoCAT-1185 |
Scutebata A |
Scutellaria barbata |
NA |
MCF-7, LoVo, SMMC-7721, HCT-116 |
PhytoCAT-1186 |
Bezielle (BZL101) |
Scutellaria barbata |
Cyclin A2, Cyclin D1, CDK2, CDK4, ERα |
MCF-7, MDA-MB-231, LNCaP, PC3 |
PhytoCAT-1187 |
Semecarpus anacardium nut extract (SA) |
Semecarpus anacardium |
HIF-1, Bcl-2, Bax, cyt-c, Caspase 3, Caspase 9, PARP |
T47D, Cancer rats |
PhytoCAT-1188 |
Solanum nigrum extract |
Solanum nigrum |
ABCG2, ADAM23, BRCA1, CCNA1, CSF1, EGF, EGFR, ESR2, GSTP1, IL-6, Notch1, SERPINE1, VEGFA, ABCB1, Bcl-2, CCND1, CDH13, ESR1, KRT19, PGR, PTG |
MCF-7, AU565 |
PhytoCAT-1189 |
Oxymatrine |
Sophora flavescens |
αⅤβ3 integrin, E-cadherin, FAK, PI3K, and Akt |
MCF-7, MDA-MB-231 and 4T1 |
PhytoCAT-1190 |
Eugenol |
Syzygium aromaticum |
LC3, NUp62, E2F1/survivin |
MCF-7, HeLa, MDA-MB-231 |
PhytoCAT-1191 |
Tagetone A |
Tagetes minuta |
NA |
MCF-7 and A549 |
PhytoCAT-1192 |
Tamarix aphylla essential oil |
Tamarix aphylla |
NA |
MCF-7, Caco-2, Panc-1 |
PhytoCAT-1193 |
Arjunolic acid (AA) |
Terminalia arjuna |
NA |
MCF-7, HeLa |
PhytoCAT-1194 |
Chebulinic acid (CA) |
Terminalia chebula |
SOD1 |
MDA-MB-231, MCF-7, S115, HOS-1, PC-3 |
PhytoCAT-1195 |
Epoxy clerodane diterpene (ECD) |
Tinospora cordifolia |
Bax, Caspase 3, Caspase 8, Caspase 9, p21, Bcl-2, mdm2, PCNA |
MCF-7 |
PhytoCAT-1196 |
Torilis japonica extract (TJE) |
Torilis japonica |
EGFR, EMT |
MCF-7 |
PhytoCAT-1197 |
Tragopogon porrifolius extract |
Tragopogon porrifolius (Salsify) |
CAT |
MDA-MB-231 |
PhytoCAT-1198 |
23,24-Dihydrocucurbitacin B |
Trichosanthes kirilowli |
NA |
Bcap37, HeLa, SW620, SMMC-7721, K562, MCF-7 |
PhytoCAT-1199 |
Cucurbitacin D |
Trichosanthes kirilowli |
STAT-3 |
MDA-MB-231 |
PhytoCAT-1200 |
Trichosanthes kirilowii extract |
Trichosanthes kirilowli |
STAT-3 |
MDA-MB-231 |
PhytoCAT-1201 |
Celastrol |
Tripterygium wilfordii Hook F |
CXCR4, NF- kB, MMP9, DCLK1, ALDH1, CD133 |
MDA-MB-231, MCF-7 |
PhytoCAT-1202 |
Uncaria rhynchophylla (UPAs) |
Uncaria rhynchophylla |
Bax, Bcl-2 , Caspase 3 |
MDA-MB-231 |
PhytoCAT-1203 |
Proanthocyanidin |
Uncaria rhynchophylla |
NA |
MCF-7, A549, HS578T and HEK293 |
PhytoCAT-1204 |
Prodelphinidin B-2 3,3'-di-O-gallate |
Myrica rubra |
p53, p21/WAF1 |
MCF-7 |
PhytoCAT-1205 |
Jatamanvaltrate P |
Valeriana jatamansi Jones |
PARP, Cyclin B1, Cyclin D1, Cdc-2 |
MCF-7, MDA-MB-231, MDA-MB-453, MDA-MB-468, MCF-10A |
PhytoCAT-1206 |
Valeriana officinalis extract |
Valeriana officinalis |
NA |
MDA-MB-231, MCF-7, MCF-10A |
PhytoCAT-1207 |
Linoleic acid |
Vitex agnus-castus |
BRCA1, ER |
MDA-MB-231, MCF-7, mouse mammary tumor, T47D, Ishikawa cells |
PhytoCAT-1208 |
Anthocyanin |
Vitis coignetiae Pulliat |
TNF-α, NF-kappaB, COX-2, C-myc, MMP2, MMP9, ICAM-1, VEGF |
MDA-MB-435, HCT-116, MCF-7, NCI-H460, SF-268, AGS |
PhytoCAT-1209 |
Bis(4-hydroxy-2H-chromen-2-one) coumarin (4HC) |
NA |
CYP19A1, Bcl-2, Bax, Caspase 3, |
MCF-7 |
PhytoCAT-1210 |
Withaferin A |
Withania somnifera |
STAT-3, Notch2, Notch 4, ATR, CHK1 |
MCF-7, SUM159, MDA-MB-231 |
PhytoCAT-1211 |
(-)-Xanthatin |
Xanthium strumarium |
GADD45γ, c-fos |
MDA-MB-231 |
PhytoCAT-1212 |
6-shogaol |
Zingiber officinale (Ginger) |
MT1-MMP, c-Src kinase, cortactin, JNK, NF-κB, STAT-3, CCL2, Aromatase |
MDA-MB-231, A549 |
PhytoCAT-1213 |
Zingiber officinale extract (ZOME) |
Zingiber officinale (Ginger) |
NA |
HeLa, MDA-MB-231 |
PhytoCAT-1214 |
Jujuboside B |
Zizyphus jujuba |
PARP, Caspase 3, LC3-II |
MDA-MB-231 and MCF-7 xenografts |
PhytoCAT-1215 |
Indole-3-carbinol |
Brassica oleracea |
BRCA1, EGFR , MUC1, BRCA1, BRCA2, p53, MDM2, GATA3, ERalpha |
MDA-MB-231, T47D, MCF-7, MDA-MB-468, PC3, LNCaP, DU-145, 10AT-Her2, tumor xenograft |
PhytoCAT-1216 |
Daucosterol Linoleate |
Ipomoea batatas |
Ki67, VEGF, Bcl-2, PI3K/AKT/NF-kB, XIAP, Bax, Bad |
MDA-MB-231, MCF-7, 4T1, MCF-7 xenograft nude mice |
PhytoCAT-1217 |
Clausehainanines A |
Clausena hainanensis |
NA |
HL-60, SMMC-7721, A-549, MCF-7, SW480 |
PhytoCAT-1218 |
Clausehainanines B |
Clausena hainanensis |
NA |
HL-60, SMMC-7721, A-549, MCF-7, SW480 |
PhytoCAT-1219 |
Clausehainanines C |
Clausena hainanensis |
NA |
HL-60, SMMC-7721, A-549, MCF-7, SW480 |
PhytoCAT-1220 |
Clausehainanines D |
Clausena hainanensis |
NA |
HL-60, SMMC-7721, A-549, MCF-7, SW480 |
PhytoCAT-1221 |
Clausehainanines E |
Clausena hainanensis |
NA |
HL-60, SMMC-7721, A-549, MCF-7, SW480 |
PhytoCAT-1222 |
Adenium obesum extract |
Adenium obesum |
NA |
MCF-7 |
PhytoCAT-1223 |
Dentatin (DTN) |
Clausena excavata Burm |
Bcl-2, Bax, Caspase 9, Caspase 3, Caspase 7, cyt-c |
MCF-7 |
PhytoCAT-1224 |
Clausena excavata root extract |
Clausena excavata Burm |
NA |
HL-60, HT-29, HepG2, MCF-7, HeLa |
PhytoCAT-1225 |
Clausena excavata stem bark extract |
Clausena excavata Burm |
NA |
NA |
PhytoCAT-1226 |
Genipin |
Rothmannia wittii |
UCP2 |
MCF-7, MDA-MB-231, NCI-H187, T47D |
PhytoCAT-1227 |
10-O-acetylmacrophyllide |
Rothmannia wittii |
NA |
MCF-7, NCI-H187 |
PhytoCAT-1228 |
Garjasmine |
Rothmannia wittii |
NA |
MCF-7, NCI-H187 |
PhytoCAT-1229 |
1,2,3,4,6-Penta-O-galloyl-β-d-glucose |
Macaranga tanarins |
Skp2, FoxO1, p27 |
MDA-MB-231, BT-474 |
PhytoCAT-1230 |
Mimusops zeyheri seed oil |
Mimusops zeyheri |
CD62P, CD63 |
MCF-7, MDA-MB-231 |
PhytoCAT-1231 |
Oroxylum indicum (PHO) extract |
Oroxylum indicum |
MMP9, ICAMP1, Caspase 3 |
MDA-MB-231, MCF-7, WRL-68 |
PhytoCAT-1232 |
Rhinacanthin A |
Rhinacanthus nasutus |
NA |
MCF-7 |
PhytoCAT-1233 |
Siegesbeckia orientalis extract |
Siegesbeckia orientalis |
Caspase 3, Caspase 8, Caspase 9, Bad, Bak, Bax, Bcl-2 |
MDA-MB-231, A549, Hep G2, FaDu , LNCaP |
PhytoCAT-1234 |
Pinostilbene |
Commiphora africana |
NA |
MCF-7, A549, PC3, HepG2 |
PhytoCAT-1235 |
5-methoxy-(E)-resveratrol 3-O-rutinoside |
Commiphora africana |
NA |
MCF-7, A549, PC3, HepG2 |
PhytoCAT-1236 |
Commiphora africana extract |
Commiphora africana |
NA |
MCF-7, A549, PC3, HepG2 |
PhytoCAT-1237 |
Salvisertin A |
Salvia deserta |
NA |
A549, MDA-MB-231, KB, KB-VIN, and MCF-7 |
PhytoCAT-1238 |
Horminone |
Salvia deserta |
NA |
A549, MDA-MB-231, KB, KB-VIN, and MCF-7 |
PhytoCAT-1239 |
Sugiol |
Salvia deserta |
NA |
A549, MDA-MB-231, KB, KB-VIN, and MCF-7 |
PhytoCAT-1240 |
Demethylcryptojaponol |
Salvia deserta |
NA |
A549, MDA-MB-231, KB, KB-VIN, and MCF-7 |
PhytoCAT-1241 |
Ximenia caffra seed oil |
Ximenia caffra |
CD62P, CD63 |
MCF-7, MDA-MB-231 |
PhytoCAT-1242 |
Zantholic acid |
Zanthoxylum zanthoxyloides |
NA |
WRL-68, CaCO2, MCF-7, PC-3 |
PhytoCAT-1243 |
Bergapten (Bg) |
Ficus carica |
p53, PTEN |
MDA-MB-231, MCF-7, ZR75 |
PhytoCAT-1244 |
Antroquinonol (AQ) |
Antrodia camphorata |
IL-10, PTGS2, IL-6 |
MCF-7, MDA-MB-231, Hep3B, HepG2, DU-145, LNCaP |
PhytoCAT-1245 |
Icaritin |
Epimedium diphyllum |
EGFR, GPER1 |
MDA-MB-231, MCF-7, MDA-MB-453 , 4T1,SKBR-3 |
PhytoCAT-1246 |
Xanthohumol |
Humulus lupulus (Common hop) |
EGFR, STAT-3, PHB2, NIS |
MDA-MB-231, SKBR-3, MCF-7, HT-29, A-2780 |
PhytoCAT-1247 |
quercetin 3-O-β-d-xylopyranosyl-(1‴→2″)-O-β-d-glucopyranoside |
Callistemon viminalis |
NA |
MCF-7, HepG2 |
PhytoCAT-1248 |
Kaempferol 3-O-β-d-mannuronopyranoside |
Callistemon viminalis |
NA |
MCF-7, HepG2 |
PhytoCAT-1249 |
Kaempferol 3-O-β-d-mannopyranoside |
Callistemon viminalis |
NA |
MCF-7, HepG2 |
PhytoCAT-1250 |
Quercetin 3-O-β-d-mannuronopyranoside |
Callistemon viminalis |
NA |
NA |
PhytoCAT-1251 |
Scutestrigillosins A |
Scutellaria strigillosa |
NA |
HONE-1, P-388, MCF-7 and HT29 |
PhytoCAT-1252 |
Scutestrigillosins B |
Scutellaria strigillosa |
NA |
HONE-1, P-388, MCF-7 and HT29 |
PhytoCAT-1253 |
Scutestrigillosins C |
Scutellaria strigillosa |
NA |
HONE-1, P-388, MCF-7 and HT29 |
PhytoCAT-1254 |
Scutestrigillosins D |
Scutellaria strigillosa |
NA |
HONE-1, P-388, MCF-7 and HT29 |
PhytoCAT-1255 |
Scutestrigillosins E |
Scutellaria strigillosa |
NA |
HONE-1, P-388, MCF-7 and HT29 |
PhytoCAT-1256 |
Artahongkongene A |
Artabotrys hongkongensis |
NA |
HL-60, SMMC-7721, A-549, MCF-7 and SW480 |
PhytoCAT-1257 |
Artahongkongene B |
Artabotrys hongkongensis |
NA |
HL-60, SMMC-7721, A-549, MCF-7 and SW480 |
PhytoCAT-1258 |
Artahongkongene C |
Artabotrys hongkongensis |
NA |
HL-60, SMMC-7721, A-549, MCF-7 and SW480 |
PhytoCAT-1259 |
Artahongkongene D |
Artabotrys hongkongensis |
NA |
HL-60, SMMC-7721, A-549, MCF-7 and SW480 |
PhytoCAT-1260 |
Artahongkongene E |
Artabotrys hongkongensis |
NA |
HL-60, SMMC-7721, A-549, MCF-7 and SW480 |
PhytoCAT-1261 |
Artahongkongene F |
Artabotrys hongkongensis |
NA |
HL-60, SMMC-7721, A-549, MCF-7 and SW480 |
PhytoCAT-1262 |
Lucidimine B |
Ganoderma lucidum |
NA |
MCF-7 |
PhytoCAT-1263 |
Urs-12-ene-3beta,6beta,16beta-triol-3-O-beta-galactopyranosyl-(1-->2)-beta-glucopyranoside |
Silphium radula Nutt |
NA |
MDA-MB-231 |
PhytoCAT-1264 |
Wedebicoside A |
Wedelia biflora |
NA |
HeLa, MCF-7 and NCI-H460 |
PhytoCAT-1265 |
Wedebicoside B |
Wedelia biflora |
NA |
HeLa, MCF-7 and NCI-H460 |
PhytoCAT-1266 |
Wedebicoside C |
Wedelia biflora |
NA |
HeLa, MCF-7 and NCI-H460 |
PhytoCAT-1267 |
Wedebicoside E |
Wedelia biflora |
NA |
HeLa, MCF-7 and NCI-H460 |
PhytoCAT-1268 |
Ganoderma lucidum extract |
Ganoderma lucidum |
EGFR, Bax, Cyclin D1, p21/Waf1 |
MCF-7 human breast cancer cell, MDA-MB-231 cells, prostate cancer PC-3 cell, human umbilical vein endothelial cells. |
PhytoCAT-1269 |
Coriolus versicolor extract |
Coriolus versicolor |
p53, Bcl-2, IL-6, IL-8, MMP-9, TLR4, p-IκB |
HUVEC , MDA-MB-231, MCF-7 and T-47D, HL-60 cells. |
PhytoCAT-1270 |
2'-Hydroxyflavanone |
Citrus sinensis |
Ki67, CD31, Vimentin, Survivin, Bcl-2, Bax, E-cadherin, PARP, RLIP76 |
MCF-7 or SKBR-3 BC cells, MDA-MB-231, TMD231, MCF10a and T47D cells. |
PhytoCAT-1271 |
Flaxseed |
Linum usitatissimum |
Insulin-like growth factor I, Epidermal growth factor receptor |
MCF-7, MDA-MB-435 and MDA-MB-231, SKBR-3, athymic mice with MCF-7 xenografts |
PhytoCAT-1272 |
Amorphophalli rhizoma extract |
Amorphophallus konjac
Amorphophallus rivieri
Amorphophallus sinensis |
KNL-1, OLFML2A, RTKN2 |
MDA-MB-231, MDA-MB-231BO |
PhytoCAT-1273 |
Ferulago angulata extract |
Ferulago angulata |
PCNA, Ki67, Bax, p53, Caspase 3 |
MCF-7 |
PhytoCAT-1274 |
Anastatica hierochuntica extracts |
Anastatica hierochuntica (L) |
Tp53, CDKN1A, Caspase 3, Caspase 9, Bax |
MCF-7 |
PhytoCAT-1275 |
Pink Lady apples' peel-flavonoids (Peel-F) |
Malus domestica 'Cripps Pink' |
NA |
LoVo, MCF-7 |
PhytoCAT-1276 |
Pink Lady apples' flesh-flavonoids (Flesh-F) |
Malus domestica 'Cripps Pink' |
NA |
LoVo, MCF-7 |
PhytoCAT-1277 |
Adonioside A |
Adonis multiflora Nishikawa & Koki Ito |
NA |
HCT-116, HepG2, HeLa, SK-OV-3, and SK-MEL-5, and SKBR-3 |
PhytoCAT-1278 |
Adonioside B |
Adonis multiflora Nishikawa & Koki Ito |
NA |
HCT-116, HepG2, HeLa, SK-OV-3, and SK-MEL-5, and SKBR-3 |
PhytoCAT-1279 |
Cymarin |
Adonis multiflora Nishikawa & Koki Ito |
NA |
HCT-116, HepG2, HeLa, SK-OV-3, and SK-MEL-5, and SKBR-3 |
PhytoCAT-1280 |
Phaitanthrin A |
Cephalantheropsis gracilis |
NA |
MCF-7, NCI-H460, and SF-268 |
PhytoCAT-1281 |
Lampranthus glaucus extract |
Lampranthus glaucus |
NA |
MCF-7, HepG2, HCT-116 |
PhytoCAT-1282 |
Condensed tannins |
Phaseolus vulgaris |
MMP2, MMP9, VEGF |
HEL 299, Caco-2, MCF-7, Hs578T, DU 145 |
PhytoCAT-1283 |
Guggulsterone |
Commiphora mukul |
NA |
MCF-7, MDA-MB-231, HMEC |
PhytoCAT-1284 |
Biochanin A |
Trifolium pratense |
hTERT, c-MYC, Bcl-2, Ha-ras, QR, C3, COX7RP, p18, MSH2, NF2, WT1, ER?, miR-375, Aromatase |
MCF-7, MDA435/LCC6 , MCF-7/ADR, T47-D, MDA-MB-468, MCF-7 MX100,SK-BR3,MCF12A
HeLa, NCI-H460, HMEC |
PhytoCAT-1285 |
5-hydroxymethyl-2-furalclehyde |
Ardisia Crenata |
NA |
MDA-MB-231 |
PhytoCAT-1286 |
n-butyl-alpha-D-fructofuranoside |
Ardisia Crenata |
NA |
MDA-MB-231 |
PhytoCAT-1287 |
Ardisiacrispins B |
Ardisia Crenata |
NA |
MDA-MB-231 |
PhytoCAT-1288 |
Toonayunnanin B |
Toona ciliata var yunnanensis |
NA |
HL-60, SMMC-7721, A-549, MCF-7 and SW480 |
PhytoCAT-1289 |
Ziziphus jujube extract |
Ziziphus jujube |
Bax, Bad, Bid |
MCF-7, SKBR-3, OV2008 |
PhytoCAT-1290 |
Glaucocalyxin H |
Isodon japonica Hara var glaucocalyx |
NA |
CE-1, U87, A-549, MCF-7, Hela, K-562, HepG-2 |
PhytoCAT-1291 |
5,4'-dihydroxy-3'-methoxyflavanone-7-(6''-O-α-L-rhamnopyranosyl)-β-D-glucopyranoside |
Satureja spicigera |
NA |
T47D |
PhytoCAT-1292 |
2α-O-trans-p-coumaroyl-3β,19α-dihydroxy-urs-12-en-28-oic acid |
Prinsepia utilis Royle |
NA |
A549, HCT116, MDA-MB-231, CCRF-CEM |
PhytoCAT-1293 |
3-O-trans-p-coumaroyltormentic acid |
Prinsepia utilis Royle |
NA |
A549, HCT116, MDA-MB-231, CCRF-CEM |
PhytoCAT-1294 |
3-O-cis-p-coumaroyltormentic acid |
Prinsepia utilis Royle |
NA |
A549, HCT116, MDA-MB-231, CCRF-CEM |
PhytoCAT-1295 |
3-O-trans-p-coumaroyl-2α-hydroxyursolic acid |
Prinsepia utilis Royle |
NA |
A549, HCT116, MDA-MB-231, CCRF-CEM |
PhytoCAT-1296 |
3-O‑cis-p-coumaroyl-2α-hydroxyursolic acid |
Prinsepia utilis Royle |
NA |
A549, HCT116, MDA-MB-231, CCRF-CEM |
PhytoCAT-1297 |
3-O-trans-p-coumaroylmaslinic acid |
Prinsepia utilis Royle |
NA |
A549, HCT116, MDA-MB-231, CCRF-CEM |
PhytoCAT-1298 |
3-O-cis-p-coumaroylmaslinic acid |
Prinsepia utilis Royle |
NA |
A549, HCT116, MDA-MB-231, CCRF-CEM |
PhytoCAT-1299 |
Nexrutine |
Phellodendron amurense |
CDK2, p21, p27, Cyclin D1, PGE2 synthase (mPGES), PPAR? |
SKBR-3, MDA-MB 231 |
PhytoCAT-1300 |
Garcimangostanol |
Garcinia mangostana |
NA |
MCF-7, A549, Hep-G2, CNE |
PhytoCAT-1301 |
8-deoxygartanin |
Garcinia mangostana |
NA |
MCF-7, A549, Hep-G2, CNE and HT-29 |
PhytoCAT-1302 |
1-isomangostin |
Garcinia mangostana |
NA |
MCF-7, A549, Hep-G2 and CNE |
PhytoCAT-1303 |
Garcinone C |
Garcinia mangostana |
CDK2 |
MCF-7, A549, Hep-G2, CNE, 22Rν1and MDA-MB-231 |
PhytoCAT-1304 |
Wheatgrass extract |
Triticum aestivum |
Bax, Cyclin D1 |
MCF-7, HeLa |
PhytoCAT-1305 |
DLBS1425 |
Phaleria macrocarpa |
BAD, Bax |
MDA-MB-231, MCF-7 |
PhytoCAT-1306 |
Foeniculum vulgare extract |
Foeniculum vulgare |
NA |
MCF-7, MDA-Mb, Hela |
PhytoCAT-1307 |
Cordatine |
Macleaya cordata |
NA |
MCF-7 and SF-268 |
PhytoCAT-1308 |
8-methoxydihydrochelerythrine |
Macleaya cordata |
NA |
MCF-7, SF-269 |
PhytoCAT-1309 |
Baicalein |
Scutelleria baicalensis |
PTEN, STAT-3, CYP1A1 , CDKN1A, CXCL9, CXCL10, FKBP5, ZBTB4, GILZ, EMT |
HT-29, Caco-2, HepG2, SW480, MCF-7, MDA-MB-231, MCF10A., SKBR-3, MDA-MB-468 , MMTV-PyMT |
PhytoCAT-1310 |
Wogonin |
Scutelleria baicalensis |
H2AX, Cyclin D1, p21, Cdc25A |
MCF-7, MDA?MB?231, MCF-7/DOX,SKBR-3, HepG2, SW480 and MCF-7 |
PhytoCAT-1311 |
Khz (fusion of Ganoderma lucidum and Polyporus umbellatus) |
Ganoderma lucidum and Polyporus umbellatus |
Caspase 7, Caspase 8, Caspase 9 |
MCF?7 |
PhytoCAT-1312 |
Red ginseng extract |
Korean red ginseng |
P-gp , Bax, Bak, BAD, Bcl-2, Bcl-xL, Fas, FasL |
MCF-7, MCF-10A |
PhytoCAT-1313 |
1-hydroxy-5-pentyl-Quinone |
Juglans mandshurica |
NA |
MDA-MB-231, HepG2, SNU638 |
PhytoCAT-1314 |
4-(5-hydroxy-1,4-dioxo-1,4-dihydro-naphthalen-2-ylamino)-butyric acid methyl ester |
Juglans mandshurica |
NA |
MDA-MB-231, HepG2, SNU638 |
PhytoCAT-1315 |
5-hydroxy-2-(2-hydroxy-ethylamino)-(1,4) naphthoquinone |
Juglans mandshurica |
NA |
MDA-MB-231, HepG2, SNU638 |
PhytoCAT-1316 |
Juglone |
Juglans mandshurica |
NA |
MDA-MB-231, HepG2, SNU638 |
PhytoCAT-1317 |
Phaleria macrocarpa extract (PMEAF) |
Phaleria macrocarpa (Scheff) Boerl |
Bax, Bid, Caspase 3, Caspase 8, cyt-c, p21, p27, p53, SMAC, Bcl-2, Bcl-w, XIAP, Survivin |
MDA-MB-231 |
PhytoCAT-1318 |
Oroxylin A |
Scutellaria baicalensis |
NA |
HepG2, SW480, MCF-7 |
PhytoCAT-1319 |
Alisma canaliculatum extract |
Alisma canaliculatum |
CXCR3, CXCL10, IKK-NF-kappaB |
MDA-MB-231 |
PhytoCAT-1320 |
Hibiscus extract |
Hibiscus syriacus |
p21 |
MCF-7, MDA-MB-231, HBL-100 and normal human skin fibroblast cell line. |
PhytoCAT-1321 |
Apigenin 4'-geranyl-8-glucopyranosyl-7-O-α-glucopyranoside |
Cupressus sempervirens |
NA |
HepG2, MCF-7, HCT116 and A549 |
PhytoCAT-1322 |
Apigenin 7-O-β-d-glucopyranoside |
Cupressus sempervirens |
NA |
HepG2, MCF-7, HCT116 and A549 |
PhytoCAT-1323 |
Querctine-3-O-glucoside |
Cupressus sempervirens |
NA |
HepG2, MCF-7, HCT116 and A549 |
PhytoCAT-1324 |
Apigenin 4'-pernyl-8-glucopyranosyl -7-O-α-glucopyranoside |
Cupressus sempervirens |
NA |
HepG2, MCF-7, HCT116 and A549 |
PhytoCAT-1325 |
Artemisinin |
Artemisia annua |
CDK4, Cyclin-B1, Cyclin D1, Cyclin E, ER , miR-34a ,TSP50 |
MCF-7, MDA-MB-231, P-388, A-549, HT-29, KB |
PhytoCAT-1326 |
Ardicrenin |
Ardisia crenata |
NA |
A549, MCF-7, HepG2 and MDA-MB-231 |
PhytoCAT-1327 |
3-O-methylchangnanic acid |
Schisandra chinensis |
NA |
MCF-7, A549, HeLa and RPMI8226 |
PhytoCAT-1328 |
PH-1 (4-methyl-5-oxo-tetrahydrofuran-3-yl acetate) |
Polygonum hydropiper |
NA |
MCF-7, HeLA, NIH/3T3 |
PhytoCAT-1329 |
ChalcEA (2',4'-dihydroxy-6-methoxy-3,5-dimethylchalcone) |
Eugenia aquea |
ERα , Caspase 3 |
T47D, A549, MCF-7. |
PhytoCAT-1330 |
Bavachin |
Psoralea corylifolia |
ABCG2 |
MCF-7/MX, EPG85.257RDB, HT-29, Caco-2, LLC-PK1, MCF-7 |
PhytoCAT-1331 |
Artemisia princeps extract |
Artemisia princeps |
Bcl-2, Caspase 3, Caspase 8, Caspase 9 |
MCF-7 |
PhytoCAT-1332 |
Entelon |
Vitis vinifera |
IL1A |
4T1, MDA-MB-231, Hs578T, MDA-MB-468 |
PhytoCAT-1333 |
Chelidonium majus extract |
Chelidonium majus |
NA |
A549, H460, HCT 116, SW480, MDA-MB 231, MCF-7 |
PhytoCAT-1334 |
Benzyl isothiocyanate |
Cruciferous vegetables |
STAT-3, XIAP, Caspase 9, Caspase 3, Caspase 8, Bax, Bcl-2, Bcl-xL, Bak, sfRON, MFN2, MAPK, JNK, p38, E-cadherin, Vimentin, Fibronectin, Notch2, FocO1, PUMA, Ron, AKT |
MDA-MB-231, MCF-7, MCF-10A, MDA-MB-453, MDA-MB-361, Female athymic mice, SUM159, HCT-1, MCF-12A |
PhytoCAT-1335 |
Oleanolic acid |
Gleditsia sinensis |
ABCB1, CDK2, CDK4, CD34, Cyclin E, Cyclin D1, p-JNK, p-ERK, p21, p27, p53, cyt-c, Bax, PARP-1, VEGF-B, AMPK, VEGFR-2, Caspase 3, mTOR/FRAP1, RAPTOR, RICTOR, VEGF |
A549, MDA-MB-231, PC-3, MCF-7, DU145, U87, HT-29, HDFn, HepG-2, Bel-7402, HeLa, MDA-MB-468, HCT-116, T-47D, HL-60/HAR, K562, A354-S2 |
PhytoCAT-1336 |
Cedrelone |
Toona ciliata, Trichilia catigua |
EGFR, MMP9, MMP |
HL-60, SMMC-7721, A-549, MCF-7, SW480, MDA-MB-231 |
PhytoCAT-1337 |
Dysobinin |
Toona ciliata
Chisocheton siamensis |
NA |
HL-60, SMMC-7721, A-549, MCF-7, SW480, NCI-H187, KB |
PhytoCAT-1338 |
Epoxyazadiradione |
Toona ciliata, Neem |
MMP9 |
HL-60, SMMC-7721, A-549, MCF-7, SW480, MDA-MB-231 |
PhytoCAT-1339 |
Daidzin |
Glycine max |
ER |
ZR-75-1, MDA-MB-231, MCF-7 |
PhytoCAT-1340 |
Anoectochilus formosanus extract |
Anoectochilus formosanus Hayata |
FasL, FAST, phospholipase C, kinase C, the type 1 inositol 1,4,5-triphosphate receptor (IP3R-1), c-Jun N-terminal kinase (JNK), c-Jun |
MCF-7 |
PhytoCAT-1341 |
Extract of Serenoae repentis fructus |
Serenoa repens |
NA |
MCF-7, MDA-MB-231, LNCaP, Caki-1, A549, HCT 116, J82 |
PhytoCAT-1342 |
Artemisia princeps smoke and water extracts |
Artemisia princeps |
Caspase 3, Caspase 8, Caspase 9, Bcl-2 |
MCF-7 |
PhytoCAT-1343 |
Bilberry extract |
Vaccinium myrtillus (Bilberry ) |
NA |
MCF-7 |
PhytoCAT-1344 |
Extract of Centella asiatica |
Centella asiatica |
NA |
MCF-7 |
PhytoCAT-1345 |
Picrorhiza kurroa extracts |
Picrorhiza kurroa |
NA |
MCF-7, MDA-MB 231, HeLa, SiHa, Hep3B, PC-3, MDA-MB-435S |
PhytoCAT-1346 |
Extracts of Rheum emodi Wall. ex Meissn. rhizome. |
Rheum emodi |
NA |
MDA-MB-435S, Hep3B, PC-3, HepG2, MDA-MB-231 and NIH/3T3 |
PhytoCAT-1347 |
Lemon extract |
Citrus limon |
JAK1, JAK2, TYK2, IRF7, IRF3 gene, p53, Caspase 3, Bax, Bcl-2, cyt-c, PARP |
Vero, MDA-MB-231, MCF-12F, MCF-7 |
PhytoCAT-1348 |
Pistacia atlantica sub kurdica extract |
Pistacia atlantica |
Cyclin D1, Caspase 3, p53 , CDK4, Cyclin-D1 |
T47D |
PhytoCAT-1349 |
Gugulipid |
Commiphora mukul |
TCF-4, Cyclin D1, C-myc, Survivin |
MCF-7, MDA-MB-231 |
PhytoCAT-1350 |
Extract of garden cress |
Lepidium sativum |
Caspase 6, Caspase 7 |
MCF-7 |
PhytoCAT-1351 |
Isoflavones extracted from chickpea sprouts (ICS) |
Cicer arietinum |
Bax, Bcl-2, Caspase 7, Caspase 9, p53, P21 |
SKBR-3, MCF-7 |
PhytoCAT-1352 |
Mango kernel extract |
Mangifera indica |
Bax, cyt-c, MDA, p53, Bcl-2 |
MDA-MB-231, MCF-7 |
PhytoCAT-1353 |
Erythronium japonicum extracts |
Erythronium japonicum |
MMP2, MMP9 |
MDA-MB-231 |
PhytoCAT-1354 |
Scrophularia oxysepala extract |
Scrophularia oxysepala |
Caspase 3, Caspase 9 mRNA, Bcl-2 gene, NF-?B gene |
MCF-7 |
PhytoCAT-1355 |
Polyphenols of Artichoke |
Cynara scolymus |
p16(INK4a), p21 (Cip1/Waf1) |
MDA-MB-231 |
PhytoCAT-1356 |
Diospyros lycioides extract |
Diospyros lycioides |
p53, Bcl-2, enolase, pyruvate kinase, glyceraldehyde-3-phosphate |
MCF-7 |
PhytoCAT-1357 |
Purple-fleshed sweet potato (PFSP) Tainung 73 |
Ipomoea batatas |
NF-κβ, TNF-α, Caspase 3, IL-6 |
MCF-7, SNU-1, WiDr |
PhytoCAT-1358 |
Urtica dioica extract |
Urtica dioica |
miR-21, Caspase 3, Caspase 9, Bcl-2, MMP1, MMP9, MMP13, Vimentin, CXCR4, E-Cadherin, ODC1, ADA |
MDA-MB-468, MCF - 7 |
PhytoCAT-1359 |
Extracts of Paeonia suffruticosa |
Paeonia suffruticosa |
IL-6, IL-2, IL-24, Fas, Bcl-2, TNF-α |
MDA-MB-231 |
PhytoCAT-1360 |
Phyllanthus niruri extract |
Phyllanthus niruri |
MMP2, MMP9, HIF1-α , AP-1, c-Jun-, c-myc, elongation factor 2 , Hsp90, stress-70 s, Hsp60 |
MCF-7 |
PhytoCAT-1361 |
Papaya leaf extract |
Carica papaya |
NA |
MCF-7 |
PhytoCAT-1362 |
Echinophora platyloba extract |
Echinophora Platyloba |
Bcl-2, p27, Bax |
MDA-MB-231, MCF-10a |
PhytoCAT-1363 |
Satureja khuzestanica total extract |
Satureja khuzestanica |
Bax, Bcl-2, Cyclin D1 |
MCF-7 |
PhytoCAT-1364 |
Euphorbia szovitsii Fisch & C.A. Mey extract |
Euphorbia szovitsii Fisch & CAMey |
NA |
MDA-MB-231 |
PhytoCAT-1365 |
Graviola extract |
Annona muricata (Graviola) |
NA |
MCF-7 |
PhytoCAT-1366 |
Artemisia annua herbal preparation |
Artemisia annua |
Caspase 3 |
MDA-MB-231, MCF-7,MIA PaCa-2, PC-3, A459, MDA-MB-231 xenografts grown on CAM as well as in nude mice. |
PhytoCAT-1367 |
Red guava extracts |
Psidium guajava (Guava) |
Caspase 3, PARP |
MCF-10A, MCF-7, NIH-3T3, MDA-MB-231 and MDA-MB-468 |
PhytoCAT-1368 |
Ajwa Dates Pulp Extract |
Phoenix dactylifera |
p53, Bax, Bcl-2, Fas, FasL, Caspase 3 |
MDA-MB-231, MCF-7 |
PhytoCAT-1369 |
Cuscuta chinensis extract |
Cuscuta chinensis |
Bax, Bcl-2 , Caspase 3, PTEN |
MDA-MB-468, MCF-7, HT29, Hela, PC3, T47D |
PhytoCAT-1370 |
Melaleuca Alternifolia Concentrate |
Melaleuca Alternifolia |
Caspase 3, Caspase 7 |
MCF-7, LNCaP |
PhytoCAT-1371 |
Isocryptotanshinone |
Salvia miltiorrhiza |
JNK, ERK, p38 MAPK |
MCF-7, MDA-MB-231, HepG2, A459 |
PhytoCAT-1372 |
Antcin-A |
Antrodia cinnamomea |
p53, E-cadherin, occludin, N-cadherin, Vimentin, ZEB1 |
MCF-7 and MDA-MB-231 |
PhytoCAT-1373 |
Epipremnum pinnatum extract |
Epipremnum pinnatum (L) |
Caspase 3, p53, c-myc |
T-47D |
PhytoCAT-1374 |
Bauhinia variegata extract |
Bauhinia variegata |
NA |
DU-145, HOP-62, IGR-OV-1, MCF-7, and THP-1 |
PhytoCAT-1375 |
Eurycoma longifolia Jack extract |
Eurycoma longifolia Jack |
cyt-c, Caspase 3, Bax, Bcl-2, Bax, p53, Caspase -8, Caspase -7 |
MCF-7, MCF-10A, KB, DU-145, RD, CaOV-3, MDA-MB-231 |
PhytoCAT-1376 |
Sutherlandia frutescens extract |
Sutherlandia frutescens |
MEK5, PIAS1 , SMPD3, MMP16, MMP21, MYC2L |
MCF-7 |
PhytoCAT-1377 |
9-methoxy-18,19-dehydrocamptothecin |
Nothapodytes foetida |
NA |
HepG2, Hep3B, MDA-MB- 231, MCF-7, A549, and Ca9-22 |
PhytoCAT-1378 |
9-methoxy-camptothecin |
Nothapodytes foetida |
NA |
HepG2, Hep3B, MDA-MB- 231, MCF-7, A549, and Ca9-22 |
PhytoCAT-1379 |
5-hydroxycamptothecin |
Nothapodytes foetida |
NA |
HepG2, Hep3B, MDA-MB- 231, MCF-7, A549, and Ca9-22 |
PhytoCAT-1380 |
5-hydroxy-9-methoxycamptothecin |
Nothapodytes foetida |
NA |
HepG2, Hep3B, MDA-MB- 231, MCF-7, A549, and Ca9-22 |
PhytoCAT-1381 |
Isoadenolin I |
Isodon adenolomus |
NA |
HL-60, SMMC-7721, A-549, MCF-7, and SW-480 |
PhytoCAT-1382 |
lasiokaurin |
Isodon adenolomus |
NA |
HL-60, SMMC-7721, A-549, MCF-7, and SW-480 |
PhytoCAT-1383 |
Xerophilusin N |
Isodon adenolomus |
NA |
HL-60, SMMC-7721, A-549, MCF-7, and SW-480 |
PhytoCAT-1384 |
Effusanin B |
Isodon adenolomus |
NA |
HL-60, SMMC-7721, A-549, MCF-7, and SW-480 |
PhytoCAT-1385 |
Longikaurin E |
Isodon adenolomus |
NA |
HL-60, SMMC-7721, A-549, MCF-7, and SW-480 |
PhytoCAT-1386 |
Xerophilusin B |
Isodon adenolomus |
NA |
HL-60, SMMC-7721, A-549, MCF-7, and SW-480 |
PhytoCAT-1387 |
Elaeis guineensis extract |
Elaeis guineensis |
NA |
MCF-7 |
PhytoCAT-1388 |
Conophylline |
Tabernaemontana divaricata, Tabernaemontana corymbosa |
NA |
HL-60, SMMC-7721, A-549, MCF-7, SW480, KB, PC-3, LNCaP, MDA-MB-231, HT-29, and HCT 116 |
PhytoCAT-1389 |
Lineariifolianoid E |
Inula lineariifolia Turcz |
NA |
MCF-7, MDA-MB-231 |
PhytoCAT-1390 |
Dehydrooopodin |
Ferula oopoda |
NA |
MCF-7 and K562 |
PhytoCAT-1391 |
Antiaroside A |
Antiaris toxicaria |
NA |
KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9 and S-KMEL-2 |
PhytoCAT-1392 |
Convallatoxal |
Antiaris toxicaria |
NA |
KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9 and S-KMEL-2 |
PhytoCAT-1393 |
Convallatoxin |
Antiaris toxicaria |
NA |
KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2, HCT-116, SF-268, HL-60, BT-474, MDA-MB-231 |
PhytoCAT-1394 |
Desglucocheirotoxin |
Antiaris toxicaria |
NA |
KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9 and S-KMEL-2 |
PhytoCAT-1395 |
α-antiarin |
Antiaris toxicaria |
NA |
KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
PhytoCAT-1396 |
Periplorhamnoside |
Antiaris toxicaria |
NA |
KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
PhytoCAT-1397 |
Cheiranthoside |
Antiaris toxicaria |
NA |
KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
PhytoCAT-1398 |
Strophanthidol |
Antiaris toxicaria |
NA |
KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
PhytoCAT-1399 |
Cannogenol |
Antiaris toxicaria |
NA |
KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
PhytoCAT-1400 |
Strophathojavoside |
Antiaris toxicaria |
NA |
KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
PhytoCAT-1401 |
Strophalloside |
Antiaris toxicaria |
NA |
KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
PhytoCAT-1402 |
Convalloside |
Antiaris toxicaria |
NA |
KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
PhytoCAT-1403 |
Glucostrophalloside |
Antiaris toxicaria |
NA |
KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
PhytoCAT-1404 |
Antiaroside C |
Antiaris toxicaria |
NA |
KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
PhytoCAT-1405 |
Antiaroside D |
Antiaris toxicaria |
NA |
KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
PhytoCAT-1406 |
Malayoside |
Antiaris toxicaria |
NA |
KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
PhytoCAT-1407 |
Antialloside |
Antiaris toxicaria |
NA |
KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
PhytoCAT-1408 |
Toxicarioside B |
Antiaris toxicaria |
NA |
KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
PhytoCAT-1409 |
β-antiarin |
Antiaris toxicaria |
NA |
KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
PhytoCAT-1410 |
Antiaroside E |
Antiaris toxicaria |
NA |
KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
PhytoCAT-1411 |
Antiaroside F |
Antiaris toxicaria |
NA |
KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
PhytoCAT-1412 |
Antiaroside G |
Antiaris toxicaria |
NA |
KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
PhytoCAT-1413 |
Antiaroside H |
Antiaris toxicaria |
NA |
KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
PhytoCAT-1414 |
Antiaroside I |
Antiaris toxicaria |
NA |
KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
PhytoCAT-1415 |
Antiarotoxinin A |
Antiaris toxicaria |
NA |
KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
PhytoCAT-1416 |
Curcuma zedoaria extract |
Curcuma zedoaria |
E-cadherin, SDF-1, CXCR4, CCR7, CYP3A4, PXR, MDR1, BCRP |
MDA-MB-231, Ca Ski, TNBC xenograft mice model,HCT-116 |
PhytoCAT-1417 |
Lobatoside N |
Actinostemma lobatum |
NA |
HCT-116, HT-29, MCF-7, A549 |
PhytoCAT-1418 |
Tupichinolide |
Adonis multiflora, Tupistra chinensis |
NA |
HCT-116, HepG2, HeLa, SK-OV-3, SK-MEL-5, SKBR-3, HL-60, SMMC-7721,A-549,MCF-7,SW480 |
PhytoCAT-1419 |
Cryptojaponol |
Clerodendrum kiangsiense |
NA |
HL-60, SMMC-7721, A-549 and MCF-7 |
PhytoCAT-1420 |
Fortunin E |
Clerodendrum kiangsiense |
NA |
HL-60, SMMC-7721, A-549 and MCF-7 |
PhytoCAT-1421 |
12-methoxy-6,11,14,16-tetrahydroxy-17(15→16)-abeo-5,8,11,13-abietatetraen-3,7-dione |
Clerodendrum kiangsiense |
NA |
HL-60, SMMC-7721, A-549 and MCF-7 |
PhytoCAT-1422 |
Peganum harmala's extract |
Peganum harmala |
Bax, Puma, TRAIL, Caspase 8, Bid, Bcl-2, Caspase 6, Caspase 9 |
MDA-MB-231, A2780, PC3, A549, HepG2, HT-29, HeLa, Jurkat,HL-60, HCT-116 , SGC-7901 |
PhytoCAT-1423 |
Lansiumarin C |
Clausena hainanensis |
NA |
HL-60, SMMC-7721, A-549, MCF-7, SW480 |
PhytoCAT-1424 |
Lansiumarin A |
Clausena hainanensis |
NA |
HL-60, SMMC-7721, A-549, MCF-7, SW480 |
PhytoCAT-1425 |
8-[(2E)-6-oxo-3,7-dimethyloct-2-enyloxylpsoralen |
Clausena hainanensis |
NA |
HL-60, SMMC-7721, A-549, MCF-7, SW480 |
PhytoCAT-1426 |
Claucoumarin D |
Clausena hainanensis |
NA |
HL-60, SMMC-7721, A-549, MCF-7, SW480 |
PhytoCAT-1427 |
Melicotriphyllin A |
Clausena hainanensis |
NA |
HL-60, SMMC-7721, A-549, MCF-7, SW480 |
PhytoCAT-1428 |
Melicotriphyllin C |
Clausena hainanensis |
NA |
HL-60, SMMC-7721, A-549, MCF-7, SW480 |
PhytoCAT-1429 |
Nauclorienine |
Nauclea orientalis |
NA |
HL-60, SMMC-7721, A-549, MCF-7, SW480 |
PhytoCAT-1430 |
Antirhine |
Nauclea orientalis |
NA |
HL-60, SMMC-7721, A-549, MCF-7, SW480 |
PhytoCAT-1431 |
Iso-antirhine |
Nauclea orientalis |
NA |
HL-60, SMMC-7721, A-549, MCF-7, SW480 |
PhytoCAT-1432 |
Alangine |
Nauclea orientalis |
NA |
HL-60, SMMC-7721, A-549, MCF-7, SW480 |
PhytoCAT-1433 |
Artahainanol A |
Artabotrys hainanensis |
NA |
HL-60, SMMC-7721, A-549, MCF-7, SW480 |
PhytoCAT-1434 |
Flexuvarol B |
Artabotrys hainanensis |
NA |
HL-60, SMMC-7721, A-549, MCF-7, SW480 |
PhytoCAT-1435 |
Uvamalol C |
Artabotrys hainanensis |
NA |
HL-60, SMMC-7721, A-549, MCF-7, SW480 |
PhytoCAT-1436 |
Flexuvarol A |
Artabotrys hainanensis |
NA |
HL-60, SMMC-7721, A-549, MCF-7, SW480 |
PhytoCAT-1437 |
Tripterregeline A |
Tripterygium regelii |
NA |
HL-60, SMMC-7721, A-549, MCF-7, SW480 |
PhytoCAT-1438 |
Triptobenzene H |
Tripterygium regelii |
NA |
HL-60, SMMC-7721, A-549, MCF-7, SW480 |
PhytoCAT-1439 |
Triptinin A |
Tripterygium regelii |
NA |
HL-60, SMMC-7721, A-549, MCF-7, SW480 |
PhytoCAT-1440 |
Triptinin B |
Tripterygium regelii |
NA |
HL-60, SMMC-7721, A-549, MCF-7, SW480 |
PhytoCAT-1441 |
Triptobenzene D |
Tripterygium regelii |
NA |
HL-60, SMMC-7721, A-549, MCF-7, SW480 |
PhytoCAT-1442 |
Triptoquinone A |
Tripterygium regelii |
NA |
HL-60, SMMC-7721, A-549, MCF-7, SW480 |
PhytoCAT-1443 |
Triptobenzene S |
Tripterygium regelii |
NA |
HL-60, SMMC-7721, A-549, MCF-7, SW480 |
PhytoCAT-1444 |
Phlomis viscosa Poiret extract |
Phlomis viscosa Poiret |
NA |
U-87, MCF-7, HEK293 |
PhytoCAT-1445 |
Isocowanin |
Garcinia tetrandra |
NA |
Hep G2, HeLa S3, MCF-7, HT-29, KB |
PhytoCAT-1446 |
Parvifolixanthone C |
Garcinia tetrandra |
NA |
Hep G2, HeLa S3, MCF-7, HT-29, KB |
PhytoCAT-1447 |
Rosmarinus officinalis extract |
Rosmarinus officinalis |
ER-α, HER2 |
MCF-7, LoVo, HeLa, RAW 264.7, FMM-1, NIH3T3, MDA-MB-231, 5637,Jurkat, K562, HL60, NCI-H82, DU-145, Hep-3B, PC-3, LNCaP |
PhytoCAT-1448 |
Polyphyllin V |
Paris polyohylla var chinensis |
NA |
MDA-MB-231, HeLa |
PhytoCAT-1449 |
Capsanthin |
Capsicum annuum |
p53, Bax, Bcl-2, p-gp |
MCF-7, MDA-MB-231, MDR-1 gene-transfected L1210 mouse lymphoma cells |
PhytoCAT-1450 |
Cryptoyunnane D |
Cryptocarya yunnanensis |
NA |
A549, HCT-116, MDA-MB-231, PC-3, HeLa |
PhytoCAT-1451 |
Obolactone |
Cryptocarya yunnanensis |
NA |
A549, HCT-116, MDA-MB-231, PC-3, HeLa |
PhytoCAT-1452 |
Cryptoyunnane A |
Cryptocarya yunnanensis |
NA |
HCT-116, MDA-MB-231 and PC-3 |
PhytoCAT-1453 |
Cryptoyunnane B |
Cryptocarya yunnanensis |
NA |
HCT-116, MDA-MB-231, PC-3 |
PhytoCAT-1454 |
7',8'-Dihydroobolactone |
Cryptocarya yunnanensis |
NA |
HCT-116, MDA-MB-231, PC-3 |
PhytoCAT-1455 |
Phlomis russeliana extract |
Phlomis russeliana |
Bcl-2 |
MCF-7 |
PhytoCAT-1456 |
Ziziphus spina-christi extract |
Ziziphus spina-christi |
Bax, Bcl-2 |
MCF-7 |
PhytoCAT-1457 |
Lupinalbin D |
Ficus altissima |
NA |
HepG2, MCF-7, MDA-MB-231 |
PhytoCAT-1458 |
Curcumol |
Curcuma wenyujin |
Bcl-2, Bak, IDH1, PUMA, p73 |
MDA-MB-231, MDA-MB-468, MGC-803 |
PhytoCAT-1459 |
Physalis minima extract |
Physalis minima |
c-myc , p53, Caspase 3 |
T-47D, Caov-3 |
PhytoCAT-1460 |
9 - hydroxycalabaxanthone |
Garcinia tetrandra |
NA |
MCF-7, HT-29, KB, Hep G2, and HeLa S3 |
PhytoCAT-1461 |
20-O-salicyl-kidjoranin |
Cynanchum wilfordii |
NA |
HL-60, MCF-7 |
PhytoCAT-1462 |
Rostratamin |
Cynanchum wilfordii |
NA |
MCF-7 |
PhytoCAT-1463 |
Abifadine E |
Abies fargesii |
NA |
B16, MCF-7, HepG2 |
PhytoCAT-1464 |
15-hydroxydehydroabietic acid |
Abies fargesii |
NA |
B16, MCF-7, and HepG2 |
PhytoCAT-1465 |
Isojiangrubesin B |
Isodon rubescens |
NA |
HL-60, SMMC-7721, A-549, MCF-7, RAW264.7 SW480 |
PhytoCAT-1466 |
Isojiangrubesin E |
Isodon rubescens |
NA |
HL-60, SMMC-7721, A-549, MCF-7, RAW264.7 SW481 |
PhytoCAT-1467 |
Effusanin A |
Isodon rubescens |
NA |
HL-60, SMMC-7721, A-549, MCF-7, RAW264.7 SW482 |
PhytoCAT-1468 |
Longikaurin A |
Isodon rubescens |
NA |
HL-60, SMMC-7721, A-549, MCF-7, RAW264.7 SW483 |
PhytoCAT-1469 |
7,14- O-(1-methylethylidene)oridonin |
Isodon rubescens |
NA |
HL-60, SMMC-7721, A-549, MCF-7, RAW264.7 SW484 |
PhytoCAT-1470 |
Hederagenin 3-O-β-D-glucopyranosyl-(1→4)-β-D-glucopyranosyl-(1→3)-α-L-rhamnopyranosyl-(1→2)-α-L-arabinopyranoside |
Lonicera similis Hemsl |
NA |
HepG2, MCF-7, A-549 |
PhytoCAT-1471 |
Caroguaianolide A |
Carpesium abrotanoides |
NA |
HGC-27, MDA-MB-231 |
PhytoCAT-1472 |
Caroguaianolide B |
Carpesium abrotanoides |
NA |
HGC-27, MDA-MB-231 |
PhytoCAT-1473 |
Caroguaianolide C |
Carpesium abrotanoides |
NA |
HGC-27, MDA-MB-231 |
PhytoCAT-1474 |
Akihalin |
Carpesium abrotanoides |
NA |
HGC-27, MDA-MB-231 |
PhytoCAT-1475 |
4β-hydroxy,10β-hydroperoxyl,5αH,7αH,8βH-guaia-1,11(13)-dien-8α,12-olide |
Carpesium abrotanoides |
NA |
HGC-27, MDA-MB-231 |
PhytoCAT-1476 |
(3aR,4aS,5S,7aS,8S,9aR)-5-hydroxy-4a,8-dimethyl-3-methylen-decahydroazuleno[6,5-b]furan-2(3H)-on |
Carpesium abrotanoides |
NA |
HGC-27, MDA-MB-231 |
PhytoCAT-1477 |
2-desoxy-4-epi-pulchellin |
Carpesium abrotanoides |
NA |
HGC-27, MDA-MB-231 |
PhytoCAT-1478 |
Kopsifoline I |
Kopsia fruticosa |
NA |
HS-1, HS-4, SCL-1, A431, BGC-823, MCF-7, and W480 |
PhytoCAT-1479 |
Kopsifoline J |
Kopsia fruticosa |
NA |
HS-1, HS-4, SCL-1, A431, BGC-823, MCF-7, and W480 |
PhytoCAT-1480 |
Kopsifoline K |
Kopsia fruticosa |
NA |
HS-1, HS-4, SCL-1, A431, BGC-823, MCF-7, and W480 |
PhytoCAT-1481 |
Chrysin |
Scutellaria baicalensis |
BRCA1, FTO, H2AX, MMP2, MMP9, RAD51, STAT-3, Aromatase |
MCF-7, BT-474, HeLa, HepG-2, MDA-MB-468, BCRP-MDCKII, Caco-2, 518A2, HCT-116 colon, KB-V1/Vbl cervix, MCF-7/Topo, MDA-MB-231, A549 , T47D, MV4-11, LoVo |
PhytoCAT-1482 |
Sulforaphane |
Cruciferous vegetables (Brassica oleracea) |
MMP7, MMP14, p38, Caspase 7, Bax, EMT, CR1, CRIPTO-3/TDGF1P3 (CR3, a homologue of CR1), Nanog, ALDH1A1, Wnt3, Notch4, KLF4, hTERT, CDKN2A, PTEN, RARbeta2, DNMT1, p53, p21, PBR, vimentin, Twist1, POU5F1, IL-1beta, IL-6, TNF-alpha, IFN-gamma,IL-4, PDGF, VEGF. |
MCF-7, MDA-MB-231, SKBR-3, MCF-12A, HeLa |
PhytoCAT-1483 |
Antrodin C |
Antrodia cinnamomea |
E-cadherin, occludin, N-cadherin, Vimentin, MMP2, MMP9 |
MCF-7 |
PhytoCAT-1484 |
5,7,8,4'-tetramethoxyflavone |
Citrus hystrix |
NA |
U87, A549, MCF-7 |
PhytoCAT-1485 |
Citracridone I |
Citrus hystrix |
NA |
U87, A549, MCF-7 |
PhytoCAT-1486 |
Citronellol |
Citrus hystrix |
Bcl-2 |
MDA-MB-231 |
PhytoCAT-1487 |
Citronellal |
Citrus hystrix |
Bcl-2 |
MDA-MB-231 |
PhytoCAT-1488 |
Fresh Yellow Onion |
Allium cepa |
CEA, CA125 |
NA |
PhytoCAT-1489 |
Ellagic acid |
Rubus idaeus |
CDK6, ACTN4, AKT/mTOR |
MCF-7, HeLa, HUVEC, HEL 299, Caco-2, Hs 578T, DU 145, C32, A375 |
PhytoCAT-1490 |
Fucoidan |
Brown algae |
TGFRI and TGFRII proteins, Smad2/3, Smad4 , TGF?, Bid, Caspase 7, Caspase 8, Caspase 9, PARP |
MDA-MB-231, MCF-7, T47D, 4T1 xenograft female Balb/c mice |
PhytoCAT-1491 |
Nobiletin |
Arisaema franchetianum Engl , citrus fruits (lemons, oranges, tangerines, and grapefruits) |
CXCR4, MMP9, CYP1A1, CYP1B1 |
MCF-7, MDA-MB-231, H-29, Hs578T, BT-549 |
PhytoCAT-1492 |
α-linolenic acid |
Linum usitatissimum (Flaxseed) |
FAS, liver X receptor (LXR), and farnesoid X receptor (FXR) |
TM2H, MCF-7, BT-474, MDA-MB-231, MDA-MB-468 |
PhytoCAT-1493 |
Glycyrrhizic acid |
Glycyrrhiza glabra |
p62, Beclin-1-associated protein |
MDA-MB-231 |
PhytoCAT-1494 |
Ellipticine |
Berrywood tree, Asparagus cochinchinensis |
ALDH1A1, Bax, Bcl-2, XIAP, cyt-c, Caspase 3, Caspase 9, p53, KIP1/p27 |
MCF-7, MDA-MB-231/ HCT116 xenograft mouse tumor |
PhytoCAT-1495 |
Nemorosone |
Clusia rosea |
ESR2, GRB7, MAPK3, MLH1, MYC, Notch1, PRDM2, THBS1, Tp53, VEGFA, APC, CCND1, CCNE1, ESR1, IGFBP3, KRT19, MKI6, MUC1, PG |
MCF-7 BUS, MCF-7, MDA-MB-231 |
PhytoCAT-1496 |
Mistletoe extract (PS76A2) |
Viscum album |
TNF, H2A histone family member X, Plasminogen |
MCF-7, HT-144, SK-MEL-28, SK-MLS-1, S-UT-1B, Kpl-1, Mfm-223 |
PhytoCAT-1497 |
Hesperetin |
Citrus plant |
CDK4, P21, Caspase 9, caspace-3, Bax, Bcl-2, eNOS, aromatase, p53, PPARG, NOTCH1, CDK2, Cyclin D, Mir-486-5p And H19 Lncrna, ICAM-1, HER2 |
MCF-7, MDA-MB-435 |
PhytoCAT-1498 |
Punicic acid |
Punica granatum |
NA |
MDA-MB-231, MDA-ERalpha7, HepG2, Huh7, HT29 , HCT116, DU145 |
PhytoCAT-1499 |
Pomegranate whole seed ethanolic extract |
Punica granatum |
NA |
ACHN, A375, C32, MCF-7, LNCaP, HeLa, COR-L23, 142BR |
PhytoCAT-1500 |
β-Caryophyllene oxide |
Psidium guajava, Origanum vulgare, Cinnamomum spp, Eugenia caryophyllata, Piper nigrum |
Bcl-2, Bcl-xL, IAP-1, IAP-2, COX-2, VEGF, p53, p21, Cyclin D1 |
PC-3, MCF-7, MCF-7, MDA-MB-231, Ehrlich solid tumor bearing mice |
PhytoCAT-1501 |
Isolate f6l |
Cassia alata |
NA |
MCF-7,a breast carcinoma, SKBR-3, another breast carcinoma, T24 a bladder carcinoma, Col 2, a colorectal carcinoma, and A549, a non- small cell lung adenocarcinoma. |
PhytoCAT-1502 |
Piperine |
Piper nigrum
Piper longum |
MMP2 and -9 mRNA, GLO1, SREBP-1, FAS, CXCL7, sICAM-1, L-selectin |
A549, MDA-MB-231, HepG2, MCF-7 |
PhytoCAT-1503 |
Rosmarinic acid |
Melissa officinalis, Rosemary plant
Salvia officinalis |
MDM2, ZEB1, ABCB1, PTEN, TWIST1, COX-2, Tyrosinase |
MDA-MB-231, MCF-7, HCT116, NCI-H460, NCI-H460/R , MCR-5, NCI-H82, DU-145, Hep-3B, K-562, PC-3 |
PhytoCAT-1504 |
Panaxadiol |
Panax ginseng |
MMP9, CDK2, CDK4, p21, p27, Cyclin D1, CDK6, EGFR,HER2 |
MCF-7, A549 |
PhytoCAT-1505 |
Sesamol |
Sesamum indicum |
pS2, GREB1, DNMT3A, DNMT3B, miR-370-3p |
MDA-MB-231, HUVEC and Hs-578T cells. |
PhytoCAT-1506 |
Ergost-25-ene-3,6-dione,5,12-dihydroxy-,(5.alpha.,12.beta.) |
Solanum torvum |
BRCA1 |
MCF-7 |
PhytoCAT-1507 |
Daucosterol |
Pterospermum yunnanense |
NA |
MCF-7 and BHY |
PhytoCAT-1508 |
Oxyresveratrol |
Artocarpus lakoocha Wall ex |
Rad51 |
MCF-7, HepG2, PC–3, RAW 264.7 and A–549 |
PhytoCAT-1509 |
Papain |
Carica papaya |
NA |
MDA-MB-231, A2058, MCF-7 |
PhytoCAT-1510 |
Glabridin |
Glycyrrhiza glabra(licorine) |
GLUT1, miR-148a, FAK/Src complex, AKT, ERK1/2 |
MDA-MB-231, HEK-293, K562, MCF-7, HeLa, HepG2 and WRL-68 |
PhytoCAT-1511 |
Stachydrine hydrochloride |
Leonurus cardiaca |
Caspase 3, Bcl-2, AKT, ERK |
MCF-7 , T47D |
PhytoCAT-1512 |
Tanshinone IIA (Tan IIA) and andrographolide (Andro) combination |
Tanshinone IIA - Salvia miltiorrhiza Andrographolide - Andrographis paniculata |
p53 |
MCF-7, BGC823, SMMC7721 |
PhytoCAT-1513 |
Julibroside J19 |
Albizzia julibrissin Durazz |
NA |
HeLa, Bel-7402 and MDA-MB-435 |
PhytoCAT-1514 |
Julibroside J18 |
Albizzia julibrissin Durazz |
NA |
HeLa, Bel-7402 and MDA-MB-435 |
PhytoCAT-1515 |
Merulin C |
Endophytic fungus of Xylocarpus granatum |
NA |
BT-474, SW621 |
PhytoCAT-1516 |
Rocaglamide |
Aglaia odorata |
NA |
HL-60, SMMC-7721, A-549, MCF-7 and SW480 |
PhytoCAT-1517 |
Eichlerianic acid |
Aglaia odorata |
NA |
HL-60, SMMC-7721, A-549, MCF-7 and SW480 |
PhytoCAT-1518 |
Vibsanol C |
Viburnum odoratissimum |
NA |
HL-60, SMMC-7721, A-549, MCF-7, and SW-480 |
PhytoCAT-1519 |
Eucalrobusone C |
Eucalyptus robusta |
NA |
HepG2, MCF-7, and U2OS |
PhytoCAT-1520 |
Nitidulin |
Dalbergia velutina |
NA |
KB, HeLa-S3, MCF-7, HepG-2, and HT-29 |
PhytoCAT-1521 |
Dalvelutinane B |
Dalbergia velutina |
NA |
KB, HeLa-S3, MCF-7, HepG-2, and HT-29 |
PhytoCAT-1522 |
Clauhainanin A |
Clausena hainanensis |
NA |
HL-60, SMMC-7721, A-549, MCF-7 and SW480 |
PhytoCAT-1523 |
Clausenalansimin A |
Clausena hainanensis |
NA |
HL-60, SMMC-7721, A-549, MCF-7 and SW480 |
PhytoCAT-1524 |
Mappiodoinin A |
Mappianthus iodoies |
NA |
HL-60, SMMC-7721, A-549, MCF-7 and SW-480 |
PhytoCAT-1525 |
Mappiodoinin B |
Mappianthus iodoies |
NA |
HL-60, SMMC-7721, A-549, MCF-7 and SW-480 |
PhytoCAT-1526 |
Mappiodoinin C |
Mappianthus iodoies |
NA |
HL-60, SMMC-7721, A-549, MCF-7 and SW-480 |
PhytoCAT-1527 |
Conocarpan |
Mappianthus iodoies |
NA |
HL-60, SMMC-7721, A-549, MCF-7 and SW-480 |
PhytoCAT-1528 |
Odoratisol A |
Mappianthus iodoies |
NA |
HL-60, SMMC-7721, A-549, MCF-7 and SW-480 |
PhytoCAT-1529 |
Trichobenzolignan |
Mappianthus iodoies |
NA |
HL-60, SMMC-7721, A-549, MCF-7 and SW-480 |
PhytoCAT-1530 |
Prunustosanan AI |
Mappianthus iodoies |
NA |
HL-60, SMMC-7721, A-549, MCF-7 and SW-480 |
PhytoCAT-1531 |
Simulanol |
Mappianthus iodoies |
NA |
HL-60, SMMC-7721, A-549, MCF-7 and SW-480 |
PhytoCAT-1532 |
Woorenogenin |
Mappianthus iodoies |
NA |
HL-60, SMMC-7721, A-549, MCF-7 and SW-480 |
PhytoCAT-1533 |
4-O-methylbalanophonin |
Mappianthus iodoies |
NA |
HL-60, SMMC-7721, A-549, MCF-7 and SW-480 |
PhytoCAT-1534 |
Cassyformin |
Mappianthus iodoies |
NA |
HL-60, SMMC-7721, A-549, MCF-7 and SW-480 |
PhytoCAT-1535 |
(3S)-7-hydroxy-8,2′-dimethoxy-4′,5′-methylenedioxyisoflavane |
Spatholobus suberectus |
NA |
MCF-7, MDA-MB-231 |
PhytoCAT-1536 |
(S)-sativan |
Spatholobus suberectus |
NA |
MCF-7, MDA-MB-231 |
PhytoCAT-1537 |
Cratochinone B |
Cratoxylum cochinchinense |
NA |
KB, HeLa S-3, HT-29, MCF-7 and Hep G2 |
PhytoCAT-1538 |
Macluraxanthone |
Cratoxylum cochinchinense |
NA |
KB, HeLa S-3, HT-29, MCF-7 and Hep G2 |
PhytoCAT-1539 |
Pruniflorone G |
Cratoxylum cochinchinense |
NA |
KB, HeLa S-3, HT-29, MCF-7 and Hep G2 |
PhytoCAT-1540 |
Merulin A |
Endophytic fungus of Xylocarpus granat |
NA |
BT-474, SW620 |
PhytoCAT-1541 |
Balanophonin |
Mappianthus iodoies, Cornus kousa, Eria bambusifolia |
NA |
HL-60, SMMC-7721, A-549, MCF-7 and SW-480 |
PhytoCAT-1542 |
(-)-maackiain |
Spatholobus suberectus |
NA |
MDA-MB-231, MCF-7, Hep3B, H1299, HeLa, MCF-7, BHY, Miapaca‑2, Colo‑205, A-549 |
PhytoCAT-1543 |
(3S)-7,2'-Dihydroxy-8,4'-dimethoxyisoflavane |
Spatholobus suberectus |
NA |
MDA-MB-231, MCF-7 |
PhytoCAT-1544 |
Achyranthes bidentata Blume extract |
Achyranthes bidentata Blume |
TNF-α |
MCF-7 |
PhytoCAT-1545 |
Ouabain |
Acokanthera oppositifolia, Acokanthera schimperi |
NA |
CasKi, SiHa and Hela, MDA-MB-321 and MCF-7, A549, SW480, HPAF-II |
PhytoCAT-1546 |
Oleamide |
Moringa oleifera |
Bcl-2 |
MDA-MB-231 |
PhytoCAT-1547 |
Sarchookloide A |
Sarcococca hookeriana |
NA |
Hela, A549, MCF-7, SW480, and CEM |
PhytoCAT-1548 |
Sarchookloide B |
Sarcococca hookeriana |
NA |
Hela, A549, MCF-7, SW480, and CEM |
PhytoCAT-1549 |
Sarchookloide C |
Sarcococca hookeriana |
NA |
Hela, A549, MCF-7, SW480, and CEM |
PhytoCAT-1550 |
Rhizoxin |
Rhizopus chinensis |
NA |
B16 melanoma, M5076 sarcoma, LOX melanoma, MX-1 breast cancer, A549 |
PhytoCAT-1551 |
Dehydrothyrsiferol |
Laurencia viridis sp nov |
NA |
T47D, ZR-75-1, and Hs578T |
PhytoCAT-1552 |
Acetoxyscirpendiol |
Paecilomyces tenuipes |
Cyclin C, Mad-1 |
MCF-7 |
PhytoCAT-1553 |
Beta-sitosteryl-3beta-glucopyranoside-6'-O-palmitate |
Plumbago zeylanica |
NA |
MCF-7, Bowes |
PhytoCAT-1554 |
Farnesylthiosalicylic acid (FTS) |
NA |
s6k1, mTOR |
MCF-7 |
PhytoCAT-1555 |
Laurenditerpenol |
Laurenciaintricata |
HIF-1, VEGF |
T47D |
PhytoCAT-1556 |
Vincristine |
Catharanthus roseus |
Tp53, Bax, Bcl-2 mRNA , miR-222-3p |
BT-20, SKBR- 3, MCF-7 |
PhytoCAT-1557 |
Vinblastine |
Catharanthus roseus |
Tp53, Bax, Bcl-2 mRNA , miR-222-3p |
BT-20, SKBR- 3 |
PhytoCAT-1558 |
11,11'-dideoxyverticillin |
Shiraia bambusicola |
EGFR, VEGFR-1/Flt-1, HER2/ErbB-2, Erk1/2, Flt-1, KDR/Flk-1 |
MDA-MB-468, HUVEC, Mice |
PhytoCAT-1559 |
6-Prenylchrysin |
NA |
ABCG2 |
HEK-293, MDA-MB-231 |
PhytoCAT-1560 |
Salvicine |
Chinese herb |
topo II, mdr-1, Bcl-2, p38 MAPK, ERK, DNA-dependent kinase (DNA-PK(CS)) |
MCF-7, MDA-MB-435, MDR K562/A02, K562/A02, KB/VCR and MCF-7/ADR, K562, KB |
PhytoCAT-1561 |
Glossogyne tenuifolia extract |
Glossogyne tenuifolia |
NA |
MCF-7, MDA-MB-231, Hep G2, Hep 3B |
PhytoCAT-1562 |
Putranjivain A |
Euphorbia jolkini |
p21, WAF1 |
MCF-7 |
PhytoCAT-1563 |
Cladonia rangiformis extract |
Cladonia rangiformis |
NA |
MCF-7 |
PhytoCAT-1564 |
Cladonia convolute extract |
Cladonia convolute |
NA |
MCF-7 |
PhytoCAT-1565 |
Coprinellus sp. (CME) |
NA |
NA |
MCF-7, MDA-MB-231, BT-20 |
PhytoCAT-1566 |
Flammulina velutipes extract (FVE) |
NA |
NA |
MCF-7, MDA-MB-231, BT-20 |
PhytoCAT-1567 |
3,5,7,3',4'-pentahydroxyflavonol-3-O-beta-D-glucopyranoside |
Cranberry |
NA |
HepG2, MCF-7 |
PhytoCAT-1568 |
Red grape wine extract (RWPF) |
Vitis palmata |
NA |
MCF-7 |
PhytoCAT-1569 |
Danshen |
Salvia miltiorrhizae Binge |
AKT, p27, Rb, Cyclin D1, p53, p65, p50, NF-kB, HER2 |
MCF-7, MCF-7 vec cells and MCF-7 HER2 cells |
PhytoCAT-1570 |
Salvianolic Acid B |
Salvia miltiorrhizae Binge |
Glutathione, TNF-?, MMP8, Cyclin D1, Ki67, Caspase 3, p53, COX-2 |
MCF-7, ESC treated mice |
PhytoCAT-1571 |
Phytofluene |
Hibiscus syriacus |
NA |
T47D, MCF-7, ECC-1 |
PhytoCAT-1572 |
Cephalinone-F |
Cephalanceropsis gracilis |
NA |
MCF-7, NCI-H460, and SF-268 |
PhytoCAT-1573 |
White button mushroom |
Agaricus bisporous |
Bak-1 |
MCF-7, MCF-10A, MDA-MB-231, BT-20 |
PhytoCAT-1574 |
Tricin |
Sasa borealis |
NA |
MDA MB 468, MCF-7, SW480 |
PhytoCAT-1575 |
Kaempferol-3-O-methyl ether |
Zingiber zerumbet |
NA |
MCF-7 |
PhytoCAT-1576 |
Kaempferol-3,4' -O-dimethyl ether |
Zingiber zerumbet |
NA |
MCF-7 |
PhytoCAT-1577 |
2a,3ß-dihydroxylup-20(29)-ene-27,28-dioic acid |
Ampelozizyphus amazonicus Ducke |
NA |
SKBR-3, C-8161 |
PhytoCAT-1578 |
Epimedium brevicornum extract |
Epimedium brevicornum |
ERalpha, Progesteron receptor |
MCF-7 |
PhytoCAT-1579 |
Epimedonin L |
Epimedium brevicornum |
NA |
HL-60, SMMC-7721, A-549, MCF-7, and SW-480 |
PhytoCAT-1580 |
Ginsenoside Rg1 |
Panax ginseng |
NA |
MCF-7, HEK293 |
PhytoCAT-1581 |
Arachidonic acid |
Staphisagria macrosperma |
p38, ER, TP53, Ki67 |
HeLa, MCF-7, MDA-MB-231, HT-29 |
PhytoCAT-1582 |
Triphala |
NA |
p53 |
HeLa, MCF-7, T47D, MD-MB-231 |
PhytoCAT-1583 |
Diosgenin |
Trigonella foenum-graecum
Paris polyphylla |
XIAP, Survivin, Bcl-2, AKT, JNK, mTOR, Cyclin D1, CDK-2, CDK-4, FAS |
MCF-7, T47D, MDA-MB-231, C6, T98G, MCF-7 and MDA-231 xenografts in nude mice |
PhytoCAT-1584 |
Oleic acid |
Olea europaea |
Her-2/neu (erbB-2), BCRP, FAS |
MCF-7, MDA-MB-231, SKBR-3, caco-2, A549 |
PhytoCAT-1585 |
Beta-Sitosterol |
Styrax perkinsiae
Gastrodia elata Blume
Zanthoxylum nitidum
Goniothalamus laoticus |
Caspase 8, Caspase 9 |
HT29, MCF-7, PC3, MDA-MB-231 and U-87 MG |
PhytoCAT-1586 |
3,3',4,4',5,5'-hexahydroxystilbene (M8) |
NA |
p53, MnSOD |
ZR-75-1, MDA-MB-231, T47D |
PhytoCAT-1587 |
Cotylenin A |
NA |
Cyclin G2, AKT, mTOR |
MCF-7 and A549 |
PhytoCAT-1588 |
Rhodiola crenulata extract |
Rhodiola crenulata |
HIF1, MYCN |
MDA-MB-231, mice bearing tumor graft, NB-1691 |
PhytoCAT-1589 |
Yanhusuo extract |
Corydalis yanhusuo |
p38, MMP9 |
MDA-MB-231 |
PhytoCAT-1590 |
Quercetin-3-O-beta-D-arabinofuranoside |
Malus domestica |
NA |
HepG2, MCF-7 |
PhytoCAT-1591 |
Monosporasols A |
Monosporascus eutypoides |
NA |
HeLa, HCT-8, A549, MCF-7 |
PhytoCAT-1592 |
Monosporasols B |
Monosporascus eutypoides |
NA |
HeLa, HCT-8, A549, MCF-7 |
PhytoCAT-1593 |
3-(4-methoxyphenyl) quinolin-4(1H)-one |
NA |
SerRS mRNA, VEGFA |
MDA-MB-231, 4T1 / BALB/c mice |
PhytoCAT-1594 |
Kaempferol 3-O-β-D-rutinoside |
Cassia glauca |
NA |
MCF-7, HepG-2 |
PhytoCAT-1595 |
Mycoleptodiscin B |
Endophytic fungus Mycoleptodiscus sp |
NA |
In silico |
PhytoCAT-1596 |
Naringin |
Rhizoma drynariae |
p21, Survivin |
MCF-7, MDA-MB-231 xenograft mice |
PhytoCAT-1597 |
Phenylacetaldehyde |
NA |
STAT-3, IL-6 |
MCF-7, MDA-MB-231 |
PhytoCAT-1598 |
Rukamtenol |
Flacourtia rukam Zoll & Moritzi |
NA |
MDA-MB-231, HepG2, and RD |
PhytoCAT-1599 |
7-octenoic acid |
Moringa oleifera |
Bcl-2 |
MDA-MB-231 |
PhytoCAT-1600 |
1-phenyl-2-pentanol |
Moringa oleifera |
Bcl-2 |
MDA-MB-231 |
PhytoCAT-1601 |
Hesperidin |
Yucca aloifolia variegata |
p21, Cyclin D1, p53 |
MCF-7, HepG2, MDA-MB-231 |
PhytoCAT-1602 |
4-Acetylantroquinonol B (4-AAQB) |
Antrodia camphorata |
NA |
MCF-7 |
PhytoCAT-1603 |
Tricholopardin C |
Mushroom Tricholoma pardinum |
NA |
MCF-7. HeLa |
PhytoCAT-1604 |
Novel cold-water-soluble polysaccharide (BEP) |
Boletus edulis |
Bax, Bcl-2, cyt-c, Caspase 3, Caspase 9 |
MDA-MB-231 and Ca761 |
PhytoCAT-1605 |
Strobilanthes crispus extract |
Strobilanthes crispus |
Bcl-2, Cyclin A2, Bax, Caspase 9 |
MDA-MB-231 |
PhytoCAT-1606 |
Scutellaria barbata extract (BZL101) |
Scutellaria barbata |
NA |
Clinical trial |
PhytoCAT-1607 |
Porphyridium cruentum sulfated polysaccharides |
Porphyridium cruentum |
IL-6, TNF-α |
HTC-116, U-937, HL-60, MCF-7, NCI-H460, HGF-1/ male Balb/C mice |
PhytoCAT-1608 |
Hydroxyl safflower yellow B (HSYB) |
NA |
Caspase 9, Bax, Caspase 3 |
MCF-7 |
PhytoCAT-1609 |
Quercetin 3-O-β-d-mannuronpyranoside |
Callistemon viminalis |
5-LOX |
MCF-7, HepG2 |
PhytoCAT-1610 |
Senecio rhizomatus Rusby (SrR) extract |
Senecio rhizomatus Rusby |
NA |
MCF-7 |
PhytoCAT-1611 |
Lampranthus aurantiacus extract |
Lampranthus aurantiacus |
NA |
MCF-7, HepG2, HCT-116 |
PhytoCAT-1612 |
Clinacanthus nutans extract (CN) |
Clinacanthus nutans |
IL-6, IL-1β, TNF-α. |
MDA-MB-231 |
PhytoCAT-1613 |
Jacein |
Centaurea schmidii |
XBP1, sXBP1, ATF-4, ChoP |
MCF-7 and MDA-MB 231 |
PhytoCAT-1614 |
3-demethyljacein |
Centaurea schmidii |
XBP1, sXBP1, ATF-4, ChoP |
MCF-7, MDA-MB 231 |
PhytoCAT-1615 |
Diosmin |
NA |
AURKA, CDK1, KIF11. |
MCF-7, MDA-MB-231, SKBR-3 |
PhytoCAT-1616 |
Eriocitrin |
NA |
STAT-3, Bcl-2 |
MCF-7 |
PhytoCAT-1617 |
Extracts of Agaricus albus |
Agaricus albus |
NA |
MCF-7 |
PhytoCAT-1618 |
Clerodendrum viscosum extract |
Clerodendrum viscosum |
NA |
MCF-7 |
PhytoCAT-1619 |
Prunus amygdalus Batsch (bitter almond extract) |
Prunus amygdalus Batsch |
NA |
MCF-7 |
PhytoCAT-1620 |
2-methoxy mucic acid |
Rhizophora apiculata |
NA |
HeLa, MDA-MB-231 |
PhytoCAT-1621 |
Atraric acid (PF-2) |
Pseudevernia furfuracea |
NA |
PA-1, MCF-7 |
PhytoCAT-1622 |
(+)-Torreyol |
Lignosus rhinocerotis |
NA |
MCF-7 |
PhytoCAT-1623 |
α-cadinol |
Lignosus rhinocerotis |
NA |
MCF-7 |
PhytoCAT-1624 |
Sargassum angustifolium extract |
Sargassum angustifolium |
NA |
HT-29, HeLa and MCF-7 |
PhytoCAT-1625 |
Sargassum oligocystum extract |
Sargassum oligocystum |
NA |
HT-29, HeLa and MCF-7 |
PhytoCAT-1626 |
Sargassum boveanum extract |
Sargassum boveanum |
NA |
HT-29, HeLa and MCF-7 |
PhytoCAT-1627 |
Cordyceps sinensis extract |
Cordyceps sinensis |
NA |
orthotopic mouse tumor model 4T1 |
PhytoCAT-1628 |
Indole[3,2-b] carbazole |
Cruciferous vegetables |
Vimentin, E-cadherin, MMP2, MMP9, FAK |
MCF-7 and MDA-MB-231 |
PhytoCAT-1629 |
Russula delica extract |
Russula delica |
NA |
HepG2, MCF-7 |
PhytoCAT-1630 |
Violaxanthin |
Dunaliella tertiolecta |
NA |
MCF-7, MDA-MB-231, A549 , LNCaP |
PhytoCAT-1631 |
Dunaliella tertiolecta extract |
Dunaliella tertiolecta |
NA |
MCF-7, MDA-MB-231, A549 , LNCaP |
PhytoCAT-1632 |
1-naphthyl isothiocyanate |
Cruciferous vegetables |
NA |
MCF-7/Adr, MCF-7/wt |
PhytoCAT-1633 |
beta-phenethyl isothiocyanate |
Cruciferous vegetables |
NA |
MCF-7/Adr, MCF-7/wt |
PhytoCAT-1634 |
Tocotrienol-alpha + Genistein |
Palm oil and Soybean respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1635 |
Tocotrienol-alpha + Narigenin |
Palm oil and Grapefruit respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1636 |
Tocotrienol-alpha + Hesperetin |
Palm oil and Oranges respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1637 |
Tocotrienol-alpha + Tangeretin |
Palm oil and Tangerine respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1638 |
Tocotrienol-alpha + Nobiletin |
Palm oil and Tangerine respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1639 |
Tocotrienol-alpha + Quercetin |
Palm oil and various plants respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1640 |
Tocotrienol-alpha + Apigenin |
Palm oil and various plants respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1641 |
Tocotrienol-gamma + Genistein |
Palm oil and Soybean respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1642 |
Tocotrienol-gamma + Narigenin |
Palm oil and Grapefruit respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1643 |
Tocotrienol-gamma + Hesperetin |
Palm oil and Oranges respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1644 |
Tocotrienol-gamma + Tangeretin |
Palm oil and Tangerine respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1645 |
Tocotrienol-gamma + Nobiletin |
Palm oil and Tangerine respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1646 |
Tocotrienol-gamma + Quercetin |
Palm oil and various plants respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1647 |
Tocotrienol-gamma + Apigenin |
Palm oil and various plants respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1648 |
Tocotrienol-delta + Genistein |
Palm oil and Soybean respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1649 |
Tocotrienol-delta + Narigenin |
Palm oil and Grapefruit respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1650 |
Tocotrienol-delta + Hesperetin |
Palm oil and Oranges respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1651 |
Tocotrienol-delta + Tangeretin |
Palm oil and Tangerine respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1652 |
Tocotrienol-delta + Nobiletin |
Palm oil and Tangerine respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1653 |
Tocotrienol-delta + Quercetin |
Palm oil and various plants respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1654 |
Tocotrienol-delta + Apigenin |
Palm oil and various plants respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1655 |
Guizhi Fuling Decoction (GFD) |
NA |
HRAS, EGFR, PTK2, SOS1, ITGB1 |
MDA-MB-231 |
PhytoCAT-1656 |
Matcha green tea (MGT) |
NA |
NA |
MCF-7 |
PhytoCAT-1657 |
Pseurotin A |
Aspergillus fumigatus |
PCSK9 |
BT-474, T47D |
PhytoCAT-1658 |
Fucoxanthin |
Undaria pinnatifida |
TIMP‐1, MMP2, MMP9 |
MDA-MB-231 |
PhytoCAT-1659 |
Qingdu granule (QDG) |
QDG is composed of eleven herbs, such as Bupleuri Radix (Bupleurum chinense DC, root), Citri Reticulatae Pericarpium (Citrus reticulata Blanco, peel), Curcumae Radix (Curcuma wenyujin Y H Chen et Cing, root tuber), Sophorae Flos (Sophora japonica, flower), Moutan Cortex (Paeonia suffruticosa Andr, root bark), Arnebiae Radix (Arnebia euchroma (Royle) Johnst, root), Prunellae Spica (Prunella vulgaris, ear), Salviae Miltiorrhizae Radix et Rhizoma (Salvia miltiorrhiza Bge, root and rhizome), Curcumae Rhizoma (Curcuma phaeocaulis Val, root tuber), Astragali Radix (Astragalus membranaceus (Fisch) Bge var mongholicus (Bge) Hsiao, root), and Glycyrrhizae Radix et Rhizoma (Glycyrrhiza uralensis Fisch, root and rhizome) |
VEGF, VEGFR2, NFATc3 |
Breast cancer xenograft model |
PhytoCAT-1660 |
Leucobryum bowringii extract |
Leucobryum bowringii Mitt |
MMP2, MMP9 |
MCF-7 |
PhytoCAT-1661 |
Antcamphin A |
Antrodia camphorata |
NA |
MDA-MB-231, A549, HS68 |
PhytoCAT-1662 |
Antcamphin B |
Antrodia camphorata |
NA |
MDA-MB-231, A549, HS68 |
PhytoCAT-1663 |
Antcamphin E |
Antrodia camphorata |
NA |
MDA-MB-231, A549, HS68 |
PhytoCAT-1664 |
Antcamphin F |
Antrodia camphorata |
NA |
MDA-MB-231, A549, HS68 |
PhytoCAT-1665 |
Antcamphin G |
Antrodia camphorata |
NA |
MDA-MB-231, A549, HS68 |
PhytoCAT-1666 |
Antcamphin H |
Antrodia camphorata |
NA |
MDA-MB-231, A549, HS68 |
PhytoCAT-1667 |
Antcamphin I |
Antrodia camphorata |
NA |
MDA-MB-231, A549, HS68 |
PhytoCAT-1668 |
Antcamphin J |
Antrodia camphorata |
NA |
MDA-MB-231, A549, HS68 |
PhytoCAT-1669 |
Antcamphin K |
Antrodia camphorata |
NA |
MDA-MB-231, A549, HS68 |
PhytoCAT-1670 |
Antcamphin L |
Antrodia camphorata |
NA |
MDA-MB-231, A549, HS68 |
PhytoCAT-1671 |
Pulveraven A |
Pulveroboletus ravenelii |
Caspase 8, Caspase 7, Bax, Bcl-2 |
MCF-7 |
PhytoCAT-1672 |
Phoenix Dan Cong tea |
Phoenix Dan Cong tea |
NA |
L02, WI38, MDA-MB-231, SW480, HepG2, HeLa |
PhytoCAT-1673 |
Luteolin and its oxidovanadium(IV) complex [VO(lut)(H2O)2]Na·3H2O (VOlut) |
NA |
NA |
MDA-MB-231, CT26, A549, Balb/C mice |
PhytoCAT-1674 |
Parmotrema reticulatum extract |
Parmotrema reticulatum |
Bax, Bcl-2 , Caspase |
MCF-7, A549, WI-38 |
PhytoCAT-1675 |
Maizediterpene B |
Zea mays |
NA |
HCT-116, MDA-MB-23, SK-HEP-1 and SNU-638 |
PhytoCAT-1676 |
4-desoxynivalenol |
Zea mays |
NA |
HCT-116, MDA-MB-23, SK-HEP-1 and SNU-639 |
PhytoCAT-1677 |
Icariol |
Zea mays |
NA |
HCT-116, MDA-MB-23, SK-HEP-1 and SNU-640 |
PhytoCAT-1678 |
(-)-Oleocanthal (OC) |
Olea europaea |
EGFR |
BT-474 and SKBR-3 |
PhytoCAT-1679 |
Kuwanon C |
Morus nigra |
NA |
MCF-7, HepG2 |
PhytoCAT-1680 |
2',3,4'-trimethoxy-5-hydroxy-trans-stilbene |
Morus nigra |
NA |
MCF-7, HepG2 |
PhytoCAT-1681 |
Isoforrethin-D |
Isodon forrestii var forrestii |
NA |
SMMC-7721, A-549, MCF-7, SW-480 |
PhytoCAT-1682 |
Zhumeria majdae essential oil |
Zhumeria majdae |
NA |
A375, MCF-7 |
PhytoCAT-1683 |
Triphenylethylene-Coumarin Hybrid 5c |
NA |
NA |
SKBR-3 |
PhytoCAT-1684 |
Walnuts |
NA |
NA |
NA |
PhytoCAT-1685 |
Hibiscus rosa-sinesis extract |
Hibiscus rosa-sinesis |
NA |
MDA-MB-231 and MCF-7 cells |
PhytoCAT-1686 |
Santonin |
NA |
NA |
SKBR-3 |
PhytoCAT-1687 |
3-(5-oxohexyl)plumbagin |
Diospyros undulata |
NA |
NCI-H187, MCF-7, KB |
PhytoCAT-1688 |
Saikosaponin b2 (SSb2) |
Radix Bupleuri |
STAT-3, VASP, MMP2, MMP9, c-myc, Cyclin D1 |
MCF-7 |
PhytoCAT-1689 |
Scrophularia umbrosa Dumort extract |
Scrophularia umbrosa Dumort |
NA |
MCF-7 |
PhytoCAT-1690 |
Meriandra dianthera essential oil (MDEO) |
Meriandra dianthera |
NA |
MCF-7, LOVO |
PhytoCAT-1691 |
Evolvulin I |
Evolvulus alsinoides |
NA |
MCF-7 |
PhytoCAT-1692 |
Cordycepin |
Cordyceps militaris |
NA |
MCF-7 |
PhytoCAT-1693 |
(3S)-7-hydroxy-8,2′,4′-trimethoxyisoflavane |
Spatholobus suberectus |
NA |
MCF-7, MD-MB-231 |
PhytoCAT-1694 |
Erythrina corallodendron essential oil |
Erythrina corallodendron |
NA |
MDA-MB-231, MCF-7, HMLE |
PhytoCAT-1695 |
Sinoflavonoidgs A |
Sinopodophyllum hexandrum |
NA |
MCF-7, HepG2, HeLa, KB |
PhytoCAT-1696 |
Sinoflavonoidgs B |
Sinopodophyllum hexandrum |
NA |
MCF-7, HepG2, HeLa, KB |
PhytoCAT-1697 |
3-methoxyquercetin |
Sinopodophyllum hexandrum |
NA |
HeLa |
PhytoCAT-1698 |
Cystoseira barbata extract (CBAE) |
Cystoseira barbata |
NA |
A549, HT-29, MCF-7, MCF10A |
PhytoCAT-1699 |
Alysicarpus vaginalis extract |
Alysicarpus vaginalis |
Bax, Bcl-2, Bcl-xL, PARP-1 |
Sprague-Dawley rats, MCF-7 and MDA-MB-453 |
PhytoCAT-1700 |
Acridocarpus orientalis extract |
Acridocarpus orientalis |
NA |
MCF-7, MDA-MB-231, MCF-10A, HeLa |
PhytoCAT-1701 |
4',6'-dihydroxy-2',4-dimethoxy-5'-(2″-hydroxybenzyl)dihydrochalcone |
Cyathostemma argenteum |
Caspase 3, Caspase 8, Caspase 9, ATM, ATR |
MDA-MB-231 and MCF-7 |
PhytoCAT-1702 |
Salvia africana extract |
Salvia africana |
NA |
HepG2, HeLa, MCF-7 |
PhytoCAT-1703 |
Unguinol |
Aspergillus |
Aromatase |
MDA-MB-231 |
PhytoCAT-1704 |
Aspergillusidone D |
Aspergillus |
NA |
MDA-MB-231 |
PhytoCAT-1705 |
Candidone |
Tephrosia candida, Pongamia pinnata,onchocarpus costaricensis |
ABCG2 |
MCF-7/MX, EPG85.257RDB |
PhytoCAT-1706 |
Antcamphorol H |
Antrodia camphorata |
NA |
MCF-7, U251, SW480 |
PhytoCAT-1707 |
Grape leaves extract |
Vitis vinifera |
Bax, Bcl-2 |
HepG2, MCF-7 |
PhytoCAT-1708 |
Machilin D |
Saururus chinensis |
IL-6, IL-8, NF-κB |
MCF-7, MDA-MB-231 |
PhytoCAT-1709 |
Tangeretin |
Citrus tankan |
Caspase 3,Caspase 8, Caspase 9, Bax, Bid, tBid, p53, p21/cip1, Fas, FasL, PIK3CA, MMP9, PTGS2, IKK, PCNA |
MDA-MB-435, MCF-7, HT-29, MDA-MB-231 |
PhytoCAT-1710 |
Coleus hybridus extract |
Coleus hybridus |
NA |
MCF-7 |
PhytoCAT-1711 |
Celastrus hindsii extract |
Celastrus hindsii |
NA |
MCF-7, A549, HeLa, HK2. |
PhytoCAT-1712 |
Solanum chacoense extract |
Solanum chacoense |
Bax, Bcl-2, STAT-3, CCND1, NF-κB |
MCF-7 |
PhytoCAT-1713 |
Hygrophorus eburneus extract (HEAE) |
Hygrophorus eburneus |
NA |
HCT-116, MDA-MB-231 |
PhytoCAT-1714 |
Sargassum linearifolium extract |
Sargassum linearifolium |
Bcl-2, Bax, Beclin-1 |
MCF-7 |
PhytoCAT-1715 |
Cystoseira crinita extract |
Cystoseira crinita |
Bcl-2, Bax, Beclin-2 |
MCF-7 |
PhytoCAT-1716 |
2'-hydroxy-3',4',6'-trimethoxychalcone |
Persicaria maculosa |
NA |
4T1 |
PhytoCAT-1717 |
Pashanone |
Persicaria maculosa |
NA |
4T1 |
PhytoCAT-1718 |
Pentadecanoic acid |
Staphisagria macrosperma |
Caspase 3, Caspase 7, caspase 8, caspase 9, β-catenin, MDR1, MRP1-and epithelial-mesenchymal transition (EMT) markers-snail, slug, MMP9, MMP2. |
MCF-7, MDA-MB-231 |
PhytoCAT-1719 |
Aurovertin B |
Calcarisporium arbuscular |
DUSP1 |
MDA-MB-231, MCF-7 |
PhytoCAT-1720 |
Datura stramonium (DS) and Datura inoxia (DI) ethyl acetate leaf extract |
Datura stramonium (DS) and Datura inoxia (DI) |
NA |
PC-3, MDA-MB 231 and MCF-7 |
PhytoCAT-1721 |
4-hydroxyisophthalic acid (4-HIPA) |
Decalepis hamiltonii |
NA |
MCF-7, MDA-MB-468, MCF-10 |
PhytoCAT-1722 |
Arnicolide D |
Centipeda minima |
NA |
MDA-MB-231 xenograft mouse model, MDA-MB-231, MDA-MB-468 |
PhytoCAT-1723 |
Elephantopus mollis Kunth extract |
Elephantopus mollis Kunth |
PCNA, Bid, Bak, Bcl-2, p53 |
MCF-7, A549, T47D, HepG2, DLD-1, NCI-H23 |
PhytoCAT-1724 |
Quercetin-3-O-beta-D-arabinofuranoside |
Malus domestica |
NA |
HepG2, MCF-7 |
PhytoCAT-1725 |
Pleurotus ostreatus extracts |
Pleurotus ostreatus (oyster mushroom) |
NA |
MCF-7, MDA-MB-231, HT-29, HCT-116 |
PhytoCAT-1726 |
Grape seed extract |
Vitis vinifera |
AKT, S6 kinase, S6 , VEGF, HIF-1alpha |
MDA-MB-231, MCF-7, U251, MDA-MB-468 |
PhytoCAT-1727 |
Cordyceps militaris extract(AECM) |
Cordyceps militaris |
Caspase 3, AKT |
MDA-MB-231 |
PhytoCAT-1728 |
Eugenia jambolana extract (JFE) |
Eugenia jambolana |
NA |
MDA-MB-231 |
PhytoCAT-1729 |
Sumadain C |
Alpinia katsumadai |
NA |
HepG2, MCF-7 and BT-549 |
PhytoCAT-1730 |
Caffeic acid phenethyl ester (CAPE) |
Propolis, Euonymus alatus (Winged Spindle Tree) |
TLR4, MyD88, IRAK4, TRIF, NF-κB p65 |
MDA-MB-231, MCF-7, Hs578T, HaCaT |
PhytoCAT-1731 |
Saikosaponin-d (SSd) |
Bupleurum falcatum |
NA |
MCF-7, HeLa, MDA-MB-231 |
PhytoCAT-1732 |
Phyllanthus amarus extract |
Phyllanthus amarus Schum & Thon |
NA |
MDA-MB-435S, MCF-7 |
PhytoCAT-1733 |
Scutellaria litwinowii extract |
Scutellaria litwinowii |
NA |
AGS, HeLa, MCF-7, PC12 and NIH 3T3 |
PhytoCAT-1734 |
Loquat extract |
Eriobotrya japonica |
NA |
MDA-MB-231 |
PhytoCAT-1735 |
Deoxyelephantopin |
Elephantopus scaber |
p21(Waf1/Cip1), MMP9, NF-kB |
MDA-MB-231, MCF-7 |
PhytoCAT-1736 |
Delphinidin-3-glucoside (Dp-3-gluc) |
NA |
NA |
MCF-7 |
PhytoCAT-1737 |
Mangifera pajang kernel extract |
Mangifera pajang |
NA |
MCF-7, MDA-MB-231 |
PhytoCAT-1738 |
Pterogynine (PGN) |
Pterogyne nitens |
NA |
ZR-7530 |
PhytoCAT-1739 |
Pterogynidine (PGD) |
Pterogyne nitens |
NA |
ZR-7530 |
PhytoCAT-1740 |
Malabaricone C (mal C) |
NA |
NA |
MCF-7 |
PhytoCAT-1741 |
Camphoratin J |
Taiwanofungus camphoratus |
NA |
Hep2, MCF-7, Hela |
PhytoCAT-1742 |
Phaseollin |
Phaseolus vulgaris |
NA |
MCF-7 |
PhytoCAT-1743 |
Euphorbia factor L1 |
Euphorbia lathyris |
ABCB1 |
C6, MCF-7, KBv200 |
PhytoCAT-1744 |
Origanum compactum essential oil |
Origanum compactum |
NA |
MCF-7 |
PhytoCAT-1745 |
Bromelain |
Ananas comosus |
NA |
MCF-7 , KB, SK-MEL-28, GI-101A |
PhytoCAT-1746 |
Taspine |
Radix et Rhizomaeonticis |
ER, PR |
ZR-75-30 human breast cancer xenografts in athymic mice |
PhytoCAT-1747 |
Alterporriol K |
NA |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1748 |
Alterporriol L |
NA |
NA |
MDA-MB-435 and MCF-7 |
PhytoCAT-1749 |
Ethyl-beta-D-fructopyranoside |
Ardisia Crenata |
NA |
NA |
PhytoCAT-1750 |
Syringic acid |
Ardisia Crenata |
NA |
NA |
PhytoCAT-1751 |
n-butyl-beta-D-fructofuranoside |
Ardisia Crenata |
NA |
NA |
PhytoCAT-1752 |
Methyl-alpha-D-fructofuranoside |
Ardisia Crenata |
NA |
NA |
PhytoCAT-1753 |
(+)-Bergenin |
Ardisia Crenata |
NA |
NA |
PhytoCAT-1754 |
Asperuloside acid |
Ardisia Crenata |
NA |
NA |
PhytoCAT-1755 |
Sartoryglabin B |
Neosartorya glabra |
NA |
MCF-7, NCI-H460, A375-C5 |
PhytoCAT-1756 |
Androstan glycoside |
Caralluma tuberculata |
NA |
MDA-MB-469 |
PhytoCAT-1757 |
Rheum emodi extract |
Rheum emodi |
NA |
MDA-MB-435S, Hep3B, PC-3 |
PhytoCAT-1758 |
Brusatol |
Brucea javanica |
NA |
HL-60, SMMC-7721, A-549, MCF -7, SW480 |
PhytoCAT-1759 |
Bruceine B |
Brucea javanica |
NA |
HL-60, SMMC-7721, A-549, MCF -7, SW480 |
PhytoCAT-1760 |
(20R)-O-(3)-β-D-glucopyranosyl-(1→2)-α-L-arabinopyranosyl-pregn-5-en-3β,20-diol |
Brucea javanica |
NA |
HL-60, SMMC-7721, A-549, MCF -7, SW480 |
PhytoCAT-1761 |
Coffee extract |
Coffea arabica |
NA |
MDA-MB-231, MCF-7 |
PhytoCAT-1762 |
Longirostrerones A |
Chaetomium longirostre |
NA |
MCF-7 |
PhytoCAT-1763 |
1-benzyl-I3C |
NA |
CD40, CDK6 |
MCF-7, MDA-MB-231 |
PhytoCAT-1764 |
Vinorelbine |
NA |
Caspase 3, Caspase 9, Caspase 8, cyt-c, Bid, HER2, Tp53, Bax, Bcl-2 mRNA , miR-222-3p |
MX-1, MCF-7 |
PhytoCAT-1765 |
Ophiobolin O |
Aspergillus ustus 094102 |
JNK, p38 MAPK, ERK, Bcl-2 phosphorylation (Ser70) |
MCF-7 |
PhytoCAT-1766 |
Coprinus comatus extract |
Coprinus comatus |
Ikappaalpha |
MCF-7 |
PhytoCAT-1767 |
Ganoderiol E |
Ganoderma sinense |
NA |
MCF-7 |
PhytoCAT-1768 |
Geranyl (3-GAP) |
NA |
p53, cyt-c, Bax, Caspase 3, Caspase 7, Caspase 9 |
MCF-7, HT1080 |
PhytoCAT-1769 |
Toxicarioside M |
Antiaris toxicaria |
NA |
KB, HCT-116, SF-268, MCF-7, HL-60, PC-3, MRC-5 |
PhytoCAT-1770 |
Brevione A |
Penicillium sp |
NA |
MCF-7 |
PhytoCAT-1771 |
Brevione I |
Penicillium sp |
NA |
MCF-7 |
PhytoCAT-1772 |
Horse chestnut extract (HCE) |
Aesculus hippocastanum |
MMP, VEGF |
Jurkat, CEM, HeLa, and MCF-7 |
PhytoCAT-1773 |
Strigolactones |
NA |
ATM, ATR, DNA-PKcs, PARP-1, RAD51 |
NA |
PhytoCAT-1774 |
Schizophyllan |
Schizophyllum commune |
NA |
Female adult swiss albino mice |
PhytoCAT-1775 |
1-O-methyl-6-acetoxy-5-(pentadec-10Z-enyl)resorcinol |
Labisia pumila |
NA |
PC3, HCT116 and MCF-7 |
PhytoCAT-1776 |
1-O-methyl-6-acetoxy-5-pentadecylresorcinol |
Labisia pumila |
NA |
PC3, HCT116 and MCF-7 |
PhytoCAT-1777 |
Neocaesalpin AA |
Caesalpinia minax |
NA |
Hela, HCT-8, HepG-2, MCF-7 and A549 |
PhytoCAT-1778 |
Neocaesalpin AB |
Caesalpinia minax |
NA |
Hela, HCT-8, HepG-2, MCF-7 and A549 |
PhytoCAT-1779 |
Neocaesalpin AC |
Caesalpinia minax |
NA |
Hela, HCT-8, HepG-2, MCF-7 and A549 |
PhytoCAT-1780 |
Neocaesalpin AD |
Caesalpinia minax |
NA |
Hela, HCT-8, HepG-2, MCF-7 and A549 |
PhytoCAT-1781 |
Neocaesalpin AE |
Caesalpinia minax |
NA |
Hela, HCT-8, HepG-2, MCF-7 and A549 |
PhytoCAT-1782 |
12α-methoxyl,5α,14β-dihydroxy-1α,6α,7β-triacetoxycass-13(15)-en-16,12-olide |
Caesalpinia minax |
NA |
Hela, HCT-8, HepG-2, MCF-7 and A549 |
PhytoCAT-1783 |
Tubeimu |
Bolbostemma paniculatum |
NA |
MDA-MB-231, SKBR-3 |
PhytoCAT-1784 |
Methyl antcinate A |
Antrodia camphorata, Antrodia cinnamomea |
Bax, Bak, PUMA. |
KB, TSCCa, GNM, OC-2, and OEC-M1 , Panc-1 , BT-474, PC-3, OVCAR-3, HeLa, and U2OS, ER+ T47D |
PhytoCAT-1785 |
Methyl antcinate B |
Antrodia camphorata, Antrodia cinnamomea |
NA |
KB, TSCCa, GNM, OC-2, and OEC-M1 , Panc-1 , BT-474, PC-3, OVCAR-3, HeLa, U2OS, ER+ T47D |
PhytoCAT-1786 |
Dehydroeburicoic acid |
Antrodia camphorata |
NA |
KB, TSCCa, GNM, OC-2, and OEC-M1 , Panc-1 , BT-474, PC-3, OVCAR-3, HeLa, and U2OS, ER+ T47D |
PhytoCAT-1787 |
Protoapigenone |
Macrothelypteris torresiana |
(MAPK) ERK, JNK, p38, Bcl-2, Bcl-xL |
HepG2, Hep3B, A549, MDA-MB-231,MCF-7 |
PhytoCAT-1788 |
Puerarin |
Pueraria lobata |
NA |
MCF-7 |
PhytoCAT-1789 |
Potentilla fulgens (PRE) extract |
Potentilla fulgens |
PARP1, Survivin |
MCF-7 |
PhytoCAT-1790 |
Songaricalarin D |
Ligularia songarica |
NA |
A-549, MCF-7, KB, and KBVIN |
PhytoCAT-1791 |
Garlic extract |
Allium sativum |
hsp27, sam68 |
MCF-7, MDA-MB-231, U937, U-87 |
PhytoCAT-1792 |
Sulfuretin |
Calanticaria bicolor |
MMP9 |
MCF-7 |
PhytoCAT-1793 |
Iris Nertschinskia extract |
Iris Nertschinskia |
AKT1, AKT2 |
Hs578Tand MDA-MB-231 |
PhytoCAT-1794 |
(-)-Gossypol-enriched cottonseed oil [(-)-GPCSO] |
Gossypium herbaceum |
Bcl-2 |
MDA-MB-231, MCF-7 |
PhytoCAT-1795 |
Artemisia Stolonifera extract (AST) |
Artemisia Stolonifera |
NA |
HS578T, T47D |
PhytoCAT-1796 |
Artemisia Selengensis extract(ASE) |
Artemisia Selengensis |
NA |
HS578T, T47D |
PhytoCAT-1797 |
Artemisia Keiskeana extract (AKE) |
Artemisia Keiskeana |
NA |
HS578T, T47D |
PhytoCAT-1798 |
Calycosin |
Radix astragali |
RASD1, Bax, Bcl-2 |
MCF-7 |
PhytoCAT-1799 |
Timosaponin AIII |
Anemarrhena asphodeloidea Bunge |
COX2, c-met, MMP9, ERK |
MDA-MB-231 |
PhytoCAT-1800 |
Yuanhuacine |
Daphne genkwa |
NA |
MCF-7, MDA-MB-231, Huh7, AGS, HT-29, B 16, Colo 205, A549, A2058 |
PhytoCAT-1801 |
Daphnoretin |
Daphne genkwa |
NA |
MCF-7, MDA-MB-231, Huh7, AGS, HT-29, B 16, Colo 205, A549, A2058 |
PhytoCAT-1802 |
Genkwanin |
Daphne genkwa |
NA |
MCF-7, MDA-MB-231, Huh7, AGS, HT-29, B 16, Colo 205, A549, A2058 |
PhytoCAT-1803 |
Tiliroside |
Daphne genkwa |
NA |
MCF-7, MDA-MB-231, Huh7, AGS, HT-29, B 16, Colo 205, A549, A2058 |
PhytoCAT-1804 |
Yuanhuadine |
Daphne genkwa |
NA |
MCF-7, MDA-MB-231, Huh7, AGS, HT-29, B 16, Colo 205, A549, A2058 |
PhytoCAT-1805 |
Genkwanin III |
Daphne genkwa |
NA |
MCF-7, MDA-MB-231, Huh7, AGS, HT-29, B 16, Colo 205, A549, A2058 |
PhytoCAT-1806 |
Genkwanin VIII |
Daphne genkwa, Daphne mezereum |
NA |
MCF-7, MDA-MB-231, Huh7, AGS, HT-29, B 16, Colo 205, A549, A2058 |
PhytoCAT-1807 |
Salvia hormium extract |
Salvia hormium |
NA |
MCF-7, T47D, ZR-75-1, BT-474 |
PhytoCAT-1808 |
Salvia dominica extract |
Salvia dominica |
NA |
MCF-7, T47D, ZR-75-1, BT-474 |
PhytoCAT-1809 |
18β-glycyrrhetinic acid |
NA |
NA |
MCF-7 |
PhytoCAT-1810 |
Falcarindiol 3-acetate |
Daucus carota |
NA |
HEK293 |
PhytoCAT-1811 |
Falcarindiol 3,8-diacetate |
NA |
NA |
NA |
PhytoCAT-1812 |
Radix ranunculus ternati polysaccharides |
Ranunculus ternatus Thunb |
NA |
MCF-7 |
PhytoCAT-1813 |
3alpha-O-acetyl-8,24-dien-tirucallic acid |
Boswellia carteri |
NA |
Hep-G2, MCF-7, RAW 264.7 |
PhytoCAT-1814 |
Verticilla-4(20),7,11-triene |
Boswellia carteri |
COX-1, COX-2 |
Hep-G2, MCF-7, RAW 264.7 |
PhytoCAT-1815 |
Desoxyrhaponticin |
Rheum tanguticum Maxim ex Balf (rhubarb) |
Fatty acid synthase (FAS) |
MCF-7 |
PhytoCAT-1816 |
Rhaponticin |
Rheum tanguticum Maxim ex Balf (rhubarb) |
Fatty acid synthase (FAS) |
MCF-7 |
PhytoCAT-1817 |
Terminalia belerica extract |
Terminalia belerica |
Bax, Bcl-2 |
A549, MCF-7 |
PhytoCAT-1818 |
α-eleostearic acid (α-ESA) |
Momordica charantia |
Bcl-2, BAD, HER2, PTEN, HER3 |
SKBR-3, T47D, MCF-7 |
PhytoCAT-1819 |
9β,13β-epoxy-7-abietene |
Tetradenia riparia |
NA |
MDA-MB-435, HCT-8, SF-295, HL-60 |
PhytoCAT-1820 |
Coriandrum sativum extract |
Coriandrum sativum |
Catalase, Superoxide dismutase, Glutathione peroxidase, Caspase 3, Caspase 8, Caspase 9 |
MCF-7 |
PhytoCAT-1821 |
Dillenia suffruticosa extract(EADs) |
Dillenia suffruticosa |
SOD1, SOD2, p53, p21. |
MCF-7 |
PhytoCAT-1822 |
Quercetin-4'-O-sulphate |
NA |
NA |
MCF-7, Caco-2, BxPC-3 |
PhytoCAT-1823 |
p-hydroxybenzoic acid |
Tetrastigma hemsleyanum
Honey |
NA |
MCF-7, HeLa |
PhytoCAT-1824 |
Fevicordin-A (FevA) |
Phaleria macrocarpa (Scheff) Boerl |
NA |
MCF-7, T47D |
PhytoCAT-1825 |
Thymus caramanicus extract (TCE) |
Thymus caramanicus Jalas |
NA |
MCF-7 |
PhytoCAT-1826 |
Furanodiene |
Curcuma wenyujin |
integrin αV , β-catenin, FAK, AKT, PI3 kinase p85 |
MDA-MB-231 |
PhytoCAT-1827 |
Tocopherols |
Palm oil/Palm fruits |
p21, p27, Caspase 3, peroxisome proliferator activated receptor-gamma, AKT, OCT4, CD44, SOX-2, trefoil factor (TFF)/pS2, cathepsin D, PR, SERPINA1 |
MCF-7 and MDA-MB 231 |
PhytoCAT-1828 |
Hawaiinolide A |
Paraconiothyrium hawaiiense |
NA |
A549, T24, HeLa, HCT116, and MCF-7 |
PhytoCAT-1829 |
Saussurea lappa extract(ESL) |
Saussurea lappa |
NA |
MCF-7 |
PhytoCAT-1830 |
Boswellia ovalifoliolata extract (BL EthOH) |
Boswellia ovalifoliolata |
NA |
MDA-MB-231 and MDA-MB-453 |
PhytoCAT-1831 |
Ouregidione |
Pseuduvaria trimera |
NA |
HepG2, MDA-MB-231 |
PhytoCAT-1832 |
11α-hydroxy-lup-20(29)-ene-3β-palmitate |
Saussurea phyllocephala |
NA |
MCF-7, HeLa, HepG2, SGC-7901, NCI-H460 and BGC-823 |
PhytoCAT-1833 |
28-hydroxy-20-oxo-30-norlupane-3β-palmitate |
Saussurea phyllocephala |
NA |
(MCF-7, HeLa, HepG2, SGC-7901, NCI-H460 and BGC-824 |
PhytoCAT-1834 |
1β,11α,28-tyrihydroxy oleana-9(11),12-dien-3β-palmitate |
Saussurea phyllocephala |
NA |
MCF-7, HeLa, HepG2, SGC-7901, NCI-H460 and BGC-825 |
PhytoCAT-1835 |
Derivatives of caffeic acid (fraction F-I ) |
Peach and Plum |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1836 |
Elaeodendroside B |
Elaeodendron orientale |
NA |
HeLa, A-549, MCF-7 and HL-60, normal Vero cells |
PhytoCAT-1837 |
Elaeodendroside C |
Elaeodendron orientale |
NA |
HeLa, A-549, MCF-7 and HL-60, normal Vero cells |
PhytoCAT-1838 |
Affinoside T |
Elaeodendron orientale |
NA |
HeLa, A-549, MCF-7 and HL-60, normal Vero cells |
PhytoCAT-1839 |
Isoxanthohumol |
Humulus lupulus |
NA |
MDA-MB-231, T-47D, PC-3, HT-29, A-2780 |
PhytoCAT-1840 |
6,8-diprenylnarigenin (6,8-diPN) |
Humulus lupulus |
NA |
MDA-MB-231 |
PhytoCAT-1841 |
Coptisine |
Coptidis rhizoma |
NA |
MDA-MB-231 |
PhytoCAT-1842 |
Cyclopside 1 |
Acacia cyclops |
NA |
MCF-7, OVAR |
PhytoCAT-1843 |
2α,3β-dihydroxy-urs-20(30)-en-28-oic acid |
Sour jujube |
NA |
HepG2, MCF-7 |
PhytoCAT-1844 |
2α,3β,28-trihydroxy-urs-20(30)-ene |
Sour jujube |
NA |
HepG2, MCF-7 |
PhytoCAT-1845 |
Bisdemethylcurcumin |
NA |
NA |
SKBR-3, MCF-7 |
PhytoCAT-1846 |
3,5-bis((E)-3,4-dimethoxystyryl)isoxazole |
NA |
NA |
SKBR-3, MCF-7 |
PhytoCAT-1847 |
Cladosporium oxysporum extract |
Cladosporium oxysporum |
NF-κB, Bcl-2, Bcl-xL, Bax, cyt-C, Caspase 3 |
T47D |
PhytoCAT-1848 |
Boswellia thurifera extract |
Boswellia thurifera |
p53 |
MDA-MB-231 |
PhytoCAT-1849 |
Citrus aurantifolia extract |
Citrus aurantifolia |
p53, Bcl-2 |
MCF-7 |
PhytoCAT-1850 |
Kochia scoparia extract (MEKS) |
Kochia scoparia Scharder |
Caspase 3, Caspase 8, Caspase 9,PARP |
MDA-MB-231 |
PhytoCAT-1851 |
Panepoxydone |
Penicillium griseum |
LDH-B, LDH-A, NF-κB |
MDA-MB-231, MDA-MB-468, MDA-MB-453 |
PhytoCAT-1852 |
Trichothecinol A |
Engleromyces goetzii |
NA |
HL-60, SMMC-7721, A549, MCF-7, SW-480 |
PhytoCAT-1853 |
Deacetyl-mycoepoxydiene |
Plant endophytic fungi Phomosis sp |
Caspase 3, Bax, Caspase 9, PARP, p21, Bcl-2 |
MCF-7, nude mice with human breast carcinoma xenografts. |
PhytoCAT-1854 |
Icacinlactone F |
Icacina trichantha |
NA |
MDA-MB-435, MDA-MB-231, OVCAR3 |
PhytoCAT-1855 |
Indole diketopiperazines |
Endophytic Chaetomium sp 88194 |
NA |
MCF-7 |
PhytoCAT-1856 |
(+)- altholactone |
Goniothalamus elegants Ast |
NA |
KB, MCF-7 and NCI-H187 |
PhytoCAT-1857 |
Sesamin |
Sesamum indicum,
Zanthoxylum capense,
Zanthoxylum paracanthum Kokwaro,
Peperomia pellucida,
Zanthoxylum nitidum,
Homalomena wendlandii,
Stemona pierrei,
Knema glauca,
Triclisia sacleuxii,
Zanthoxylum setulosum |
CDK2, CDK4, CDK6, E2F1, PDK1, Bax, Caspase 3, p53 |
MCF-7,+SA, MDA-MB-231, Caco-2, HEK295, mouse |
PhytoCAT-1858 |
Bruceine D |
Brucea javanica |
NA |
MCF-7, MDA-MB-231, HS 578T |
PhytoCAT-1859 |
KTH-13-amine-monophenyl |
Cordyceps bassiana |
Caspase 3, Caspase 9, Caspase-3, Caspase 8, Caspase 9, Bcl-2 |
MDA-MB-231,HeLa ,C6 glioma |
PhytoCAT-1860 |
Flavokawain A |
Piper methsyticum |
IFN-γ, IL-2, NO, iNOS, NF-κB, ICAM, COX-2 |
Breast cancer murine model |
PhytoCAT-1861 |
Apodytes dimidiata extract |
Apodytes dimidiata |
NA |
Jurkat, Ehrlich's ascites carcinoma, SKBR-3 |
PhytoCAT-1862 |
Dahliane B |
Verticillium dahliae |
NA |
MCF-7 |
PhytoCAT-1863 |
Dahliane C |
Verticillium dahliae |
NA |
MCF-7 |
PhytoCAT-1864 |
Pelingo apple juice |
Pelingo apple |
p21, ERK1/2, LC3B |
MCF-7 , MDA-MB-231 |
PhytoCAT-1865 |
Methyl caffeate |
Solanum torvum |
Bcl-2, Bid, Bax, cyt-c |
MCF-7, A549, COLO320, HepG-2, Vero |
PhytoCAT-1866 |
Solanum torvum extract |
Solanum torvum |
NA |
MCF-7, A549, COLO320, HepG-2, Vero |
PhytoCAT-1867 |
Conjugated linoleic acid |
Agaricus bisporous,Momordica charantia |
LXR, PTPgamma, c-myc |
MDA-MB-231, MCF-7, SG652, 639V, ADF, PC3, LNCaP, SK-HEP-1, HepG2, MCF-7aro, MDA-wt, MDA-ERalpha7, M21-HPB, HT-29 |
PhytoCAT-1868 |
Shikonin |
Lithospermum erythrorhizon |
DUSP1, DUSP2, ERα, GPER, EGFR, p-ERK, RIP1K, RIP3K, E-cadherin, N-cadherin, vimentin, Snail |
MDA-MB-468, MDA-MB-231, MCF-7, SKBR-3 |
PhytoCAT-1869 |
Salacia oblonga extract |
Salacia oblonga |
NA |
MDA-MB-231 |
PhytoCAT-1870 |
Norstictic acid |
Usnea strigosa |
NA |
MDA-MB-231 |
PhytoCAT-1871 |
Corilagin |
Euphorbia fischeriana |
Hes1, Notch1, mTOR |
MCF-7, HepG2, CCA |
PhytoCAT-1872 |
Galium aparine extract (GA MeOH) |
Galium aparine |
NA |
MCF-7, MDA-MB-231, MCF-10A |
PhytoCAT-1873 |
Geraniin |
Phyllanthus urinariainn
Nephelium lappaceum |
Bcl-2, PARP, Caspase 3 |
MCF-7 |
PhytoCAT-1874 |
Cladosporium cladosporioides 2 |
Vernonia amygdalina |
NA |
MCF-7 |
PhytoCAT-1875 |
Cinnamaldehyde |
Cinnamomum cassia |
BRCA1, TOPO1, ERCC1 |
HT-29, LoVo, T47D, NCI-H322 |
PhytoCAT-1876 |
Myricetin |
Withania coagulans |
p53, BRCA1, GADD45, Bax, Bcl-2 |
MCF-7, T47D, MDA-MB-231 |
PhytoCAT-1877 |
Vernonilide A |
Vernonia anthelmintica |
NA |
A549, HeLa, MDA-MB-231 |
PhytoCAT-1878 |
Vernodalin |
Vernonia anthelmintica,
Vernonia extensa,
Centratherum anthelminticum (L) |
NA |
HepG2, MCF-7, MDA-MB-231, HeLa, A549 |
PhytoCAT-1879 |
Vernomelitensin |
Vernonia anthelmintica,
Vernonia guineensis Benth (Asteraceae) |
NA |
MDA-MB-231, MCF-7, HCT-116, HL-60, A549, A375, OVCAR3, PC-3, DU-145 |
PhytoCAT-1880 |
Vernolepin |
Vernonia anthelmintica |
NA |
HeLa, MDA-MB-231, HepG2 |
PhytoCAT-1881 |
Perovskia abrotanoides extract |
Perovskia abrotanoides |
NA |
MCF-7 and Hela |
PhytoCAT-1882 |
Germacrone |
Curcuma wenyujin |
TFF1, GREB1, CCND1, ERG3, PKIB, CTSD, CXCL12, PGR, MYC |
MCF-7 |
PhytoCAT-1883 |
Boldine |
Lindera umbellata |
p38, ERK, JNK |
MCF-7, MDA-MB-231, Tumor-bearing mice |
PhytoCAT-1884 |
Soyabean aglycone rich extracts (SARE) |
NA |
NA |
MCF-7 and MDA-MB-231 |
PhytoCAT-1885 |
Flaxseed aglycone rich extracts (FSARE) |
NA |
NA |
MCF-7 and MDA-MB-231 |
PhytoCAT-1886 |
Clinacanthus nutans extract (CN) |
Clinacanthus nutansindau |
Bcl-2 |
MCF-7, HTB-22, HeLa, CCL-2, NIH 3T3, CRL-1658 |
PhytoCAT-1887 |
3,4-bis-3,4,5-trimethoxybenzylidene-dihydrofuran (BTMB) |
Taiwania cryptomerioides |
CDC2, Cyclin D1, Cyclin E |
MDA-MB-468 |
PhytoCAT-1888 |
Withania somnifera extract |
Withania somnifera |
CCL2, Caspase 3 |
MDA-MB-231, MCF-7, HCT116, HepH2, Transgenic (MMTV/Neu) mice |
PhytoCAT-1889 |
Polysaccharide SpaTA |
Sparganii Rhizoma |
ERα |
ZR-75-1, MDA-MB-231 |
PhytoCAT-1890 |
Boletus edulis extract |
Boletus edulis |
NA |
MCF-7 |
PhytoCAT-1891 |
Cratoxy formosum extract |
Cratoxy formosum |
Rac1, CDK6, p21, Cyclin D1, MMP2, MMP9 |
MCF - 7 |
PhytoCAT-1892 |
5, 7, 4′-trihydroxy-3′-(3-methylbut-2-enyl)-3-methoxy flavone |
Sinopodophyllum hexandrum |
NA |
T47D, MCF-7, MDA-MB-231 |
PhytoCAT-1893 |
Sinopodophylline B |
Sinopodophyllum hexandrum |
NA |
T47D, MCF-7, MDA-MB-231 |
PhytoCAT-1894 |
Citrusinol |
Sinopodophyllum hexandrum |
NA |
T47D, MCF-7, MDA-MB-231 |
PhytoCAT-1895 |
6-prenylquercetin 3-methyl ether |
Sinopodophyllum hexandrum |
NA |
T47D, MCF-7, MDA-MB-231 |
PhytoCAT-1896 |
1, 3, 7, 8-tetrahydroxyxanthone |
Sinopodophyllum hexandrum |
NA |
T47D, MCF-7, MDA-MB-231 |
PhytoCAT-1897 |
Tanshinones |
Radix Salviae Miltiorrhizae |
Caspase3, Caspase 9, ATF-4 , PARP, p-eIF2 α, P-JNK, Caspase 12 |
MCF-7, A549, MKN-45, HGC-27, PC9, QGY-7703, HCT116, U266/ RPMI8226 |
PhytoCAT-1898 |
Apomorphine |
NA |
NA |
MCF-7 |
PhytoCAT-1899 |
Comophoroside A |
Commiphora opobalsamum |
NA |
HepG-2, MCF-7 |
PhytoCAT-1900 |
3β-hydroxy-30-(4-phenyl-1-piperazinyl)olean-12-ene-11,30-dione |
NA |
NA |
MCF-7, HeLa, HepG2,A549 |
PhytoCAT-1901 |
Antrodia cinnamomea extract |
Antrodia cinnamomea |
skp2 |
GBM 8401, A549, THP-1, HepG2, SW620, MDA-MB-231, HS68, 3T3, BALB/c , tamoxifen-resistant MCF-7, T47D BC cell. |
PhytoCAT-1902 |
Tetrandrine (Tet) |
Radix stephaniae tetrandrae |
NA |
MDA-MB-231 |
PhytoCAT-1903 |
ω-Hydroxyundec-9-enoic acid (ω-HUA) |
NA |
p38 |
MDA-MB-231, MDA-MB-435 |
PhytoCAT-1904 |
Pine honey |
NA |
NA |
MCF-7, SKBR-3, MDA -MB - 231 |
PhytoCAT-1905 |
Cladosporol A |
Cladosporium cladosporioides |
p21 |
MCF-7 |
PhytoCAT-1906 |
Grifola frondosa extract (GFPs) |
Grifola frondosa |
NA |
MCF-7, MDA-MB-231 |
PhytoCAT-1907 |
Annurca apple polyphenol extract (APE) |
Malus pumila Miller cv Annurca |
p53, p21, Cyclin D1, ERK1/2 phosphorylation, Bax, Bcl-2 , Caspase 9,Caspase 6, Caspase 7, PARP |
MCF-7 |
PhytoCAT-1908 |
Artemisinic acid |
Artemisia herba alba |
NA |
MCF-7, HeLa |
PhytoCAT-1909 |
Scopolin |
Artemisia herba alba |
NA |
MCF-7, HeLa |
PhytoCAT-1910 |
Isoschaftoside |
Artemisia herba alba |
NA |
MCF-7, HeLa |
PhytoCAT-1911 |
Trametes versicolor extract |
Trametes versicolor |
NA |
MCF-7, HepG2 |
PhytoCAT-1912 |
10-hydroxy camptothecin |
Nothapodytes nimmoniana |
p21 |
MCF-7, BGC823 and HepG2 |
PhytoCAT-1913 |
Ziyang green tea (ZTP) |
Ziyang green tea |
p53, CDK2, Bax, Bcl-2 , Caspase 3, Caspase 9 |
MCF-7 |
PhytoCAT-1914 |
(+)-Tengerensine |
Ficus fistulosa |
NA |
MDA-MB-468, MDA-MB-231, and MCF-7 |
PhytoCAT-1915 |
Tengechlorenine |
Ficus fistulosa |
NA |
MDA-MB-468, MDA-MB-231, and MCF-7 |
PhytoCAT-1916 |
Phyllanthus amarus (PAM) extract |
Phyllanthus amarus |
NA |
MiaPaCa-2 , HT29, A2780, H460, A431, Du145, BE2-C , MCF-7, MCF-10A, U87, SJ-G2, SMA |
PhytoCAT-1917 |
Phloridzin |
Malus pumila |
NA |
MDA-MB-231, MCF-7 |
PhytoCAT-1918 |
Mangostanaxanthone VII |
Garcinia mangostana |
NA |
A549, MCF-7 |
PhytoCAT-1919 |
Huaier extract |
Trametes robiniophila murr |
H19, ATM, miR-203, miR-675-5p, MMP2, MMP9, VEGF, ERK, p65, JNK, STAT-3, CBL, ATM |
T47D, ZR-75-1, MCF-7, MDA-MB-231, M7-TR, M7-FR, RAW264.7 murine macrophage, 4T1 tumor bearing mice |
PhytoCAT-1920 |
Lentinan (LNT) |
Lentinus edodes |
p53, p-ERK1/2, cleaved-Caspase 3, PARP 1, MDM2, TERT, NF-κB (NF-κB) p65, Bcl-2, ERα, PI3K, p-AKT, mTOR |
MCF-7 |
PhytoCAT-1921 |
Baker's yeast |
Saccharomyces cerevisiae |
NA |
The metastatic murine 4T1 line, the murine Ehrlich ascites carcinoma (EAC) line, and the human breast cancer MCF-7 cell line. |
PhytoCAT-1922 |
Clematis hederagenin saponin (CHS) |
Clematis ganpiniana |
NA |
MCF-7 and MDA-MB-231 |
PhytoCAT-1923 |
Gomisin G |
Schisandra chinesis |
AKT phosphorylation, retinoblastoma tumor suppressor (Rb), phosphorylated Rb, Cyclin D1 |
MDA-MB-231 and MDA-MB-468 |
PhytoCAT-1924 |
Chlorella minutissimma extract |
Chlorella minutissima |
MMP1, MMP2, MMP9, TIMP-3, c-Jun |
MDA-MB-231 |
PhytoCAT-1925 |
Trigohowimine A |
Trigonostemon howii |
NA |
HL-60, SMMC-7721, A-549, MCF-7 and SW480. |
PhytoCAT-1926 |
Hebecarposide C |
Lyonia ovalifolia var hebecarpa |
NA |
SMMC-7721, HL-60, SW480, MCF-7, and A-549 |
PhytoCAT-1927 |
Hebecarposide H |
Lyonia ovalifolia var hebecarpa |
NA |
SMMC-7721, HL-60, SW480, MCF-7, and A-549 |
PhytoCAT-1928 |
Clauselenisin A |
Clausena lenis |
NA |
HL-60, SMMC-7721, A-549, MCF-7 and SW480 |
PhytoCAT-1929 |
Cis-khellactone |
Angelica amurensis |
VDAC1, Bax, Bak |
MCF-7, MDA-MB-231, BT-20, BT-549, T47D, SKBR-3, MDA-MB-453, HS578T, MDA-MB-468, HCT116, HT-29, HeLa, SiHa, HEK293T, HEK293 |
PhytoCAT-1930 |
Satureja khuzestanica extract |
Satureja khuzestanica Jamzad |
Bax, Bcl-2 |
MCF-7 |
PhytoCAT-1931 |
Tebesinone B |
Salvia tebesana Bunge |
NA |
MCF-7, B16F10, PC-3, C26 |
PhytoCAT-1932 |
Aegyptinone A |
Salvia tebesana Bunge |
NA |
MCF-7, B16F10, PC-3, C27 |
PhytoCAT-1933 |
Graviola extract |
Annona muricata |
EGFR |
MDA-MB-231, MCF-7, MDA-MB-468 |
PhytoCAT-1934 |
Vulpinic Acid |
Candelaria concolor lichen |
p53 |
MCF-7, SKBR-3 |
PhytoCAT-1935 |
Pteris Quadriureta (PQ) extract |
Pteris Quadriureta |
Bcl-2, Cyclin D2 |
MCF-7 and BT47 |
PhytoCAT-1936 |
Ginsenoside Rg5 |
Black ginseng |
p53, p21(WAF1/CIP1), p15(INK4B), Cyclin D1, Cyclin E2, CDK4 |
BALB/c nude mouse model of human breast cancer, MCF-7 |
PhytoCAT-1937 |
Pseuderanthemum palatiferum (Nees) extract |
Pseuderanthemum palatiferum |
NA |
MDA-MB-231 |
PhytoCAT-1938 |
Astragaloside IV |
Astragali radix |
P-gp, BCRP, Nrf2 |
Wild-type C57BL/6 mice |
PhytoCAT-1939 |
Santolina corsica extracts |
Santolina corsica Jord |
COX-2 |
A549, HeLa, PC3, MCF-7, MDA-MB-231 |
PhytoCAT-1940 |
Dicranopteris linearis extract (MEDL) |
Dicranopteris linearis |
NA |
A549, HeLa, HepG2, HT-29, MCF-7, MDA-MB-231 |
PhytoCAT-1941 |
Boswellia frereana extract (BFE) |
Boswellia frereana |
NA |
BT-549 and MDA-MB-231 |
PhytoCAT-1942 |
(E)-resveratrol 3-O-rutinoside |
Commiphora africana |
NA |
MCF-7, A549, PC3, and HepG2 |
PhytoCAT-1943 |
Oolong Tea Extract |
NA |
NA |
MCF-7, T47D, SKBR-3, MDA-MB-231, MDA-MB-435, MDA-MB-468 |
PhytoCAT-1944 |
Ganoderic acid A (GA-A) |
Ganoderma lucidum |
STAT-3 |
MDA-MB-231 |
PhytoCAT-1945 |
Stigmasterol |
Citrus hystrix
Garcinia penangiana
Decaschistia parviflora |
NA |
HT29, MCF-7, PC3, U-87 MG |
PhytoCAT-1946 |
Pachypodium lamerei extract |
Pachypodium lamerei Drake |
NA |
MDA-MB-231 |
PhytoCAT-1947 |
(+)-pinoresinol di-O-β-d-allopyranoside |
Cimicifuga dahurica (Turcz.) Maxim. |
c-Myc, Cyclin D1, Bcl-2 |
MCF-7 |
PhytoCAT-1948 |
2'-Hydroxycinnamaldehyde |
Cinnamomum cassia Blume |
E-cadherin, KLF17, Id-1, EMT |
MCF-7, T47D, MDA-MB-231, MDA-MB-435, mice model |
PhytoCAT-1949 |
Red-fleshedapple peel extract |
Malus niedzwetzkyana |
pAKT, pBad, Bcl-2, cyt-c, Cle-Caspase 9, Cle-Caspase 3, Cle-PARP, p-p53, p21, PCNA, Cyclin D1 |
MDA-MB-231 |
PhytoCAT-1950 |
Red-fleshedapple flesh extract |
Malus niedzwetzkyana |
pAKT, pBad, Bcl-2, cyt-c, Cle-Caspase 9, Cle-Caspase 3, Cle-PARP, p-p53, p21, PCNA, Cyclin D1 |
MDA-MB-231 |
PhytoCAT-1951 |
Raspberry oil emulsion: cold pressed (ROCOP) |
Rubus idaeus |
NA |
MCF-7, MCF-7/DX, A549, LoVo, LoVo/DX |
PhytoCAT-1952 |
Raspberry oil emulsion: supercritical CO2 (ROSCO2) |
Rubus idaeus |
NA |
MCF-7, MCF-7/DX, A549, LoVo, LoVo/DX |
PhytoCAT-1953 |
Theaflavin-3-gallate |
Camellia sinensis |
HSP90, MMP9, VEGFA, SPP1 |
MCF-7, Caco-2 |
PhytoCAT-1954 |
Ent-17-acetoxy-16β-hydroxykauran-3-one |
Chloranthus anhuiensis |
NA |
MDA-MB-231, 4T1, HepG2, PC12 |
PhytoCAT-1955 |
(5R, 10S)-5,6,7,8-tetrahydro-8-mehtyl-5-(1-methylethyl)-2-naphthalenol |
Chloranthus anhuiensis |
NA |
MDA-MB-231, 4T1, HepG2, and PC12 |
PhytoCAT-1956 |
Tetrahydropalmatine (THP) and Berberine (Ber) |
Corydalis yanhusuo W. T. Wang |
NA |
MDA-MB-231 |
PhytoCAT-1957 |
Triregelin K |
Tripterygium regelii |
NA |
MCF-7, A2780, HepG2 |
PhytoCAT-1958 |
Neotriptonoterpene |
Tripterygium regelii |
NA |
MCF-7, A2780, HepG2 |
PhytoCAT-1959 |
Triregelin I |
Tripterygium regelii |
NA |
MCF-7, A2780, HepG2 |
PhytoCAT-1960 |
7-acetylaltholactone |
Goniothalamus macrocalyx Ban |
NA |
KB, HepG2, Lu, MCF-7 |
PhytoCAT-1961 |
Pentagalloyl glucose |
Quercus aliena |
GRO-α/CXCL1, IƙBKE, MAPK, DR4, DR5, TNF |
MDA-MB-468, MDA-MB-231 |
PhytoCAT-1962 |
Dihydrocapsaicin |
Capsicum annuum.
Zingiber officinale Roscoe |
Caspase family CASP9, CASP3, Bax |
MDA-MB-231 |
PhytoCAT-1963 |
Wikstrol B |
Wikstroemia scytophylla |
NA |
HL-60, SMMC-7721, A549, MCF-7, and SW480 |
PhytoCAT-1964 |
3-(1, 3-benzodioxol-5-ylmethyl)-4-[(3, 4-dimethoxyphenyl)methyl]dihydro-, (3S-cis)-2(3H)-furanone |
Wikstroemia scytophylla |
NA |
HL-60, SMMC-7721, A549, MCF-7, and SW480 |
PhytoCAT-1965 |
4-[(R)-1, 3-benzodioxol-5-ylhydroxymethyl]-3-(1, 3-benzodioxol-5-ylmethyl)dihydro-, (3S, 4R)-2(3H)-furanone |
Wikstroemia scytophylla |
NA |
HL-60, SMMC-7721, A549, MCF-7, and SW480 |
PhytoCAT-1966 |
(-)-dihydrosesamin |
Wikstroemia scytophylla |
NA |
HL-60, SMMC-7721, A549, MCF-7, and SW480 |
PhytoCAT-1967 |
4, 4’-dihydroxy-3, 3’, 9-trimethoxy-9, 9’-epoxylignan |
Wikstroemia scytophylla |
NA |
HL-60, SMMC-7721, A549, MCF-7, and SW480 |
PhytoCAT-1968 |
(+)-1-hydroxypinoresinol |
Wikstroemia scytophylla |
NA |
HL-60, SMMC-7721, A549, MCF-7, and SW480 |
PhytoCAT-1969 |
Usnic Acid |
Niebla homalea |
hsa-miR-5006-5p, hsa-miR-892c-3p, hsa-miR-4430, hsa-miR-5194, hsa-miR-3198, hsa-miR-3171, hsa-miR-933, hsa-miR-185-3p |
A2780, HeLa, MCF-7, SKBR-3, HT-29, HCT-116 p53(+/+), HCT-116 p53(-/-), HL-60 and Jurkat |
PhytoCAT-1970 |
Atranorin |
Stereocaulon alpinum |
NA |
A2780, HeLa, MCF-7, SKBR-3, HT-29, HCT-116 p53(+/+), HCT-116 p53(-/-), HL-60 and Jurkat |
PhytoCAT-1971 |
Fumarprotocetraric acid |
Cetraria islandica |
NA |
T-47D and Panc-1 |
PhytoCAT-1972 |
Gyrophoric acid |
NA |
NA |
A2780, HeLa, MCF-7, SKBR-3, HT-29, HCT-116 p53(+/+), HCT-116 p53(-/-), HL-60 and Jurkat |
PhytoCAT-1973 |
Parietin |
NA |
NA |
A2780, HeLa, MCF-7, SKBR-3, HT-29, HCT-116 p53(+/+), HCT-116 p53(-/-), HL-60 and Jurkat |
PhytoCAT-1974 |
Acalypha fruticosa Forssk extract |
Acalypha fruticosa Forssk |
NA |
MDA-MB-435S, Hep3B |
PhytoCAT-1975 |
Pheophorbide-a |
Scutellaria barbata |
JNK, ERK |
MDA-MB-231 |
PhytoCAT-1976 |
Parthenolide |
Tanacetum parthenium |
AMPK, JNK, NF-κB, STAT-3, MAP kinase, FAK1 |
Hs605T, MCF-7, SiHa, MCF-7/HER2, MDA-MB-231, BT-474 |
PhytoCAT-1977 |
1,7-Bis(4-hydroxyphenyl)-1,4-heptadien-3-one |
Viscum coloratum |
NA |
HeLa, SGC-7901, MCF-7, and U251 |
PhytoCAT-1978 |
5-hydroxy-3,7,3'-trimethoxyflavone-4'-O-beta-D-glucoside |
Viscum coloratum |
NA |
HeLa, SGC-7901, MCF-7, and U251 |
PhytoCAT-1979 |
Demethylzeylasteral (T-96) |
Tripterygium wilfordii Hook F |
Vimentin, fibronectin, α-SMA |
MDA-MB-231, 4T1 mouse model |
PhytoCAT-1980 |
Maytansinoids |
Putterlickia pyracantha |
NA |
NA |
PhytoCAT-1981 |
1,3,6-Trihydroxy-7-methyl-9,10-anthracenedione |
Lindera |
Fatty acid synthase |
MDA-MB-231 |
PhytoCAT-1982 |
Stachys pilifera Benth. extract |
Stachys pilifera Benth. |
NA |
HL-60, K562, MCF-7 |
PhytoCAT-1983 |
Stachys persica S.G.Gmel. ex C.A.Mey extract |
Stachys persica S.G.Gmel. ex C.A.Mey |
NA |
HL-60, K562, MCF-7 |
PhytoCAT-1984 |
Stachys byzantina C. Koch extract |
Stachys byzantina C. Koch |
NA |
HL-60, K562, MCF-7 |
PhytoCAT-1985 |
2,3,5,4'-Tetrahydroxystilbene-2-O-β-d-glucoside (THSG) |
Polygonum multiflorum Thunb. |
Bax, Bcl-2, Caspase 3 |
MCF-7, H1299 and LNC |
PhytoCAT-1986 |
Andrographolide |
Andrographis paniculata |
Heme oxygenase-1, MMP9, COX-2 |
MCF-7 |
PhytoCAT-1987 |
Fennel essential oil |
Foeniculum vulgare |
Bax, Bcl-2 |
MCF-7 |
PhytoCAT-1988 |
Trans-anethole (TA) |
Foeniculum vulgare |
NA |
NA |
PhytoCAT-1989 |
Macrooxazole C |
Ethyl acetate (EtOAc) extracts of Phoma sp. JS0228 cultures, an endophytic fungus of Morus alba (M. alba) |
NA |
MCF-7, LNCaP |
PhytoCAT-1990 |
SANT, a novel Chinese herbal monomer combination |
Astragaloside IV - Astragalus membranaceus,
α-solanine - Solanum nigruminn,
neferine - otus plumule, and
2,3,5,6-tetramethylpyrazine -igusticum |
ATG16L1, ATG9B, ATG4D, HB-EGF, thrombospondin-2, amphiregulin, leptin, IGFBP-9, EGF, coagulation factor III, and MMP9, serpin E1, platelet factor 4 |
MDA-MB-231 hpa (231-Hpa) and MDA-MB-231 mock (231-Mock), BALB/c nude mice |
PhytoCAT-1991 |
Xanthone V |
Vismia laurentii |
Caspase 3, Caspase 7 |
CCRF-CEM, CEM/ADR5000, PF-382, HL-60, MiaPaCa-2, Capan-1, MCF-7, SW-680, 786-0, U87MG, A549, Colo-38, HeLa, Caski |
PhytoCAT-1992 |
2-acetylfuro-1,4-naphthoquinone |
Newbouldia laevis |
NA |
CCRF-CEM, CEM/ADR5000, PF-382, HL-60, MiaPaCa-2, Capan-1, MCF-7, SW-680, 786-0, U87MG, A549, Colo-38, HeLa, Caski |
PhytoCAT-1993 |
2β-hydroxy-8β-[5′-hydroxytigloyloxy]-costunolide |
Eupatorium fortunei |
NA |
PC3, SKOV3, A549, MCF-7, HEp-2 |
PhytoCAT-1994 |
Pygenic acid A (PA) |
Prunella vulgaris |
cIAP1, cIAP2, Survivin, p21, Cyclin D1, p-STAT-3, HO-1, IRE1α, p-elF2α, LC3B I, LC3B II |
MDA-MB-231 cells (human) and 4T1 cells (mouse) |
PhytoCAT-1995 |
(+)-baphicacanthcusines A |
Baphicacanthus cusia |
NA |
MCF-7 |
PhytoCAT-1996 |
(-)-baphicacanthcusines A |
Baphicacanthus cusia |
NA |
MCF-7 |
PhytoCAT-1997 |
(-)-baphicacanthcusines B |
Baphicacanthus cusia |
NA |
MCF-7 |
PhytoCAT-1998 |
Alternate C |
Alternaria alternata, an endophyte isolated from Paeonia lactiflora. |
NA |
A-549, MDA-MB-231, MCF-7, KB, KB-VIN |
PhytoCAT-1999 |
3-Deoxy-2β,16-dihydroxynagilactone E (B6) |
Podocarpus nagi |
JAK-2, IL-6, STAT-3 |
MDA-MB-231, MDA-MB-468 |
PhytoCAT-2000 |
1,5,8-trihydroxy-3-methoxyxanthone (XD) |
Swertia chirata |
Bax, Bcl-2 |
MCF-7, MDA-MB-231, Ehrlich ascites carcinoma (EAC), a mouse transplantable breast carcinoma cell line |
PhytoCAT-2001 |
Crassin (C4) |
Croton crassifolius |
pAKT, pERK |
MDA-MB-231 |
PhytoCAT-2002 |
Phenyl glucuronide |
Euclea crispa |
Her2 |
In-silico |
PhytoCAT-2003 |
Hydrocortisone acetate |
Euclea crispa |
Her2 |
In-silico |
PhytoCAT-2004 |
6-(4,6-dioxo-1,4,5,6-tetrahydropyrimidin-2-yl-amino)hexanoic acid trifluoroacetate |
Euclea crispa |
Her2 |
In-silico |
PhytoCAT-2005 |
Flavensomycinoic acid |
Culture filtrate of endophytic Streptomyces sp. YIM66017 from Alpinia oxyphylla |
NA |
MCF-7 |
PhytoCAT-2006 |
Artichoke Polyphenols |
Cynara cardunculus |
FEN1 |
MCF-7, MDA-MB-231 |
PhytoCAT-2007 |
Amplexicaule A |
Polygonum amplexicaule D. Don var. sinense Forb |
Caspase 3,-8,-9, PARP, MCL-1, Bcl-2 |
MCF-7, MDA-MB-435, Female Kunming nude mice |
PhytoCAT-2008 |
Bikaverin |
Fusarium oxysporum EPH2RAA endophytic in Ephedra fasciculata |
CK2 |
MCF-7, A427, A431 |
PhytoCAT-2009 |
(2'R)-6-(2'-acetoxytridecyl)-2-methoxy-1,4-dihydroxybenzene |
Ardisia virens |
NA |
MCF-7, NCI-H460, SF-268 |
PhytoCAT-2010 |
1-acetoxy-2-methoxy-6-pentadecyl-4-hydroxybenzene |
Ardisia virens |
NA |
MCF-7, NCI-H460, SF-268 |
PhytoCAT-2011 |
1-acetoxy-2-methoxy-6-tridecyl-4-hydroxybenzene |
Ardisia virens |
NA |
MCF-7, NCI-H460, SF-268 |
PhytoCAT-2012 |
(2'R)-1-acetoxy-6-(2'-acetoxy-tridecyl)-2-methoxy-4-hydroxybenzene |
Ardisia virens |
NA |
MCF-7, NCI-H460, SF-268 |
PhytoCAT-2013 |
Ardisianone |
Ardisia virens |
NA |
MCF-7, NCI-H460, SF-268 |
PhytoCAT-2014 |
Cornudentanone |
Ardisia virens |
NA |
MCF-7, NCI-H460, SF-268 |
PhytoCAT-2015 |
Ardisianol |
Ardisia virens |
NA |
MCF-7, NCI-H460, SF-268 |
PhytoCAT-2016 |
Berbamine |
Berberis amurensis |
SNAP29, VAMP8, BNIP3, VAMP8, Bcl-2, Bax, pro-MMP9/pro-MMP2, c-met , AKT, nuclear factor kappaB p-65, Bcl-2/Bax, osteopontin, VEGF, MMP9, MMP2 |
MDA-MB-231, MDA-MB-435S |
PhytoCAT-2017 |
Tylophorine |
Tylophora indica |
Caspase 3, Caspase 9 |
T47D |
PhytoCAT-2018 |
Trans-nerolidol (NER) |
Myrica rubra |
NA |
MCF-7, MDA-MB-231, Ehrlich solid tumor bearing mice |
PhytoCAT-2019 |
β-elemene |
Zanthoxylum setulosum |
SNAI1, SNAI2, TWIST, SIP1, TGF-β1, Smad3, EGFR, GLUT1, LDHA, PKM-2, importin α5, PTEN, Pgp, PKM2, EMT |
MCF-7/Adr, MCF-7/Doc, MCF-7 |
PhytoCAT-2020 |
Physagulide P |
Physalis angulate. |
JNK |
MDA-MB-231, MDA-MB-468 |
PhytoCAT-2021 |
5-hydroxy-8,8-dimethyl-4-phenyl-9,10-dihydro-8H-pyrano-[2,3-f]chromen-2-one |
Marila pluricostata |
NA |
MCF-7, H-460, SF-268 |
PhytoCAT-2022 |
5-hydroxy-8,8-dimethyl-4-phenyl-6-propionyl-9,10-dihydro-8H-pyrano-[2,3-f]chromen-2-one |
Marila pluricostata |
NA |
MCF-7, H-460, SF-268 |
PhytoCAT-2023 |
5,7-dihydroxy-8-(3-methylbut-2-enyl)-4-phenylchromen-2-one |
Marila pluricostata |
NA |
MCF-7, H-460, SF-268 |
PhytoCAT-2024 |
Mammea A/AA |
Marila pluricostata |
NA |
MCF-7, H-460, SF-268 |
PhytoCAT-2025 |
Mammea A/BA |
Marila pluricostata |
NA |
MCF-7, H-460, SF-268 |
PhytoCAT-2026 |
Mammea A/AA cyclo D |
Marila pluricostata |
NA |
MCF-7, H-460, SF-268 |
PhytoCAT-2027 |
Mammea A/AB cyclo D |
Marila pluricostata |
NA |
MCF-7, H-460, SF-268 |
PhytoCAT-2028 |
Mammea A/AD cyclo D |
Marila pluricostata |
NA |
MCF-7, H-460, SF-268 |
PhytoCAT-2029 |
Isomesuol |
Marila pluricostata |
NA |
MCF-7, H-460, SF-268 |
PhytoCAT-2030 |
Mammea A/AB |
Marila pluricostata |
NA |
MCF-7, H-460, SF-268 |
PhytoCAT-2031 |
Mammea A/AD |
Marila pluricostata |
NA |
MCF-7, H-460, SF-268 |
PhytoCAT-2032 |
Mammea A/BB |
Marila pluricostata |
NA |
MCF-7, H-460, SF-268 |
PhytoCAT-2033 |
Isodispar B |
Marila pluricostata |
NA |
MCF-7, H-460, SF-268 |
PhytoCAT-2034 |
Mammea A/AA cyclo F |
Marila pluricostata |
NA |
MCF-7, H-460, SF-268 |
PhytoCAT-2035 |
Disparinol A |
Marila pluricostata |
NA |
MCF-7, H-460, SF-268 |
PhytoCAT-2036 |
Mammea A/AB cyclo F |
Marila pluricostata |
NA |
MCF-7, H-460, SF-268 |
PhytoCAT-2037 |
Mammea A/AD cyclo F |
Marila pluricostata |
NA |
MCF-7, H-460, SF-268 |
PhytoCAT-2038 |
3b,16b,23,28-tetrahydroxy-11a-methoxy-olean-12-ene 3-O-b-Dfucopyranoside |
Bupleurum chinense |
NA |
A549, HepG2, Hep3B, BCap-37, MCF-7 |
PhytoCAT-2039 |
3b,16b, 28-trihydroxyl-11a-methoxy-olean-12-ene-O-b-D-fucopyranoside |
Bupleurum chinense |
NA |
A549, HepG2, Hep3B, BCap-37, MCF-7 |
PhytoCAT-2040 |
3b,16b-dihydroxy-23-O-acetyl-13b,28b-epoxyolean-11-ene 3-O-b-D-fucopyranoside. |
Bupleurum chinense |
NA |
A549, HepG2, Hep3B, BCap-37, MCF-7 |
PhytoCAT-2041 |
3b, 23, 28-trihydroxy-11, 13(18)-diene-16-one 3-O-b-D-glucopyranosyl-(1→3)-b-Dfucopyranoside. |
Bupleurum chinense |
NA |
A549, HepG2, Hep3B, BCap-37, MCF-7 |
PhytoCAT-2042 |
Saikosaponin-b4 |
Bupleurum chinense |
NA |
A549, HepG2, Hep3B, BCap-37, MCF-7 |
PhytoCAT-2043 |
Saikogenin G |
Bupleurum chinense |
NA |
A549, HepG2, Hep3B, BCap-37, MCF-7 |
PhytoCAT-2044 |
Prosaikogenin F |
Bupleurum chinense |
NA |
A549, HepG2, Hep3B, BCap-37, MCF-7 |
PhytoCAT-2045 |
Saikosaponin-A |
Bupleurum chinense |
NA |
A549, HepG2, Hep3B, BCap-37, MCF-7 |
PhytoCAT-2046 |
Saikosaponin-D |
Bupleurum chinense |
NA |
A549, HepG2, Hep3B, BCap-37, MCF-7 |
PhytoCAT-2047 |
Saikosaponin-E |
Bupleurum chinense |
NA |
A549, HepG2, Hep3B, BCap-37, MCF-7 |
PhytoCAT-2048 |
2''-O-Acetylsaikosaponin A |
Bupleurum chinense |
NA |
A549, HepG2, Hep3B, BCap-37, MCF-7 |
PhytoCAT-2049 |
3''-O-Acetylsaikosaponin A |
Bupleurum chinense |
NA |
A549, HepG2, Hep3B, BCap-37, MCF-7 |
PhytoCAT-2050 |
6''-O-Acetylsaikosaponin A |
Bupleurum chinense |
NA |
A549, HepG2, Hep3B, BCap-37, MCF-7 |
PhytoCAT-2051 |
23-O-Acetylsaikosaponin-a |
Bupleurum chinense |
NA |
A549, HepG2, Hep3B, BCap-37, MCF-7 |
PhytoCAT-2052 |
Saikosaponin C |
Bupleurum chinense |
NA |
A549, HepG2, Hep3B, BCap-37, MCF-7 |
PhytoCAT-2053 |
6''-O-Acetylsaikosaponin D |
Bupleurum chinense |
NA |
A549, HepG2, Hep3B, BCap-37, MCF-7 |
PhytoCAT-2054 |
Prosaikogenin D |
Bupleurum chinense |
NA |
A549, HepG2, Hep3B, BCap-37, MCF-7 |
PhytoCAT-2055 |
Prosaikogenin A |
Bupleurum chinense |
NA |
A549, HepG2, Hep3B, BCap-37, MCF-7 |
PhytoCAT-2056 |
Saikosaponin-b1 |
Bupleurum chinense |
NA |
A549, HepG2, Hep3B, BCap-37, MCF-7 |
PhytoCAT-2057 |
23- hydroxy-13b,28b-epoxy-olean-11-ene-16-one 3-O-b-D-glu-copyranosyl-(1 → 3)-b-D-fucopyranoside |
Bupleurum chinense |
NA |
A549, HepG2, Hep3B, BCap-37, MCF-7 |
PhytoCAT-2058 |
2-acetyl-7-methoxynaphtho[2,3-b]furan-4,9-quinone (AMNQ) |
Millettia versicolor |
NA |
MDA-MB-231/BCRP, HepG2, CCRF-CEM |
PhytoCAT-2059 |
Juniperus communis extract (#46) |
Juniperus communis. |
p53, CDK2, p21, Bcl-2, Caspase 9 |
A549, MCF-7, TK6, U937 |
PhytoCAT-2060 |
Cotinus coggygria extract |
Cotinus coggygria Scop. |
p27, p21 |
A549, MCF-7, TK6, U937 |
PhytoCAT-2061 |
4-coumaric acid methyl ester |
Punica granatum |
ERα, ERβ, ERγ |
In-silico |
PhytoCAT-2062 |
Ferutinin |
Ferula ovina |
NA |
MCF-7, TCC, HFF3 |
PhytoCAT-2063 |
7-hydroxy, 5-methoxy, methyl cinnamate (1) |
Phyllostachys heterocycla var. pubescens |
EGFR tyrosine kinase |
MCF-7, HepG2 |
PhytoCAT-2064 |
Cercosporamide |
Endophytic fungus Phoma species ZJWCF006 in Arisaema erubescens |
NA |
HT-29, SMMC-772, MCF-7, HL-60, MGC80-3, P388 |
PhytoCAT-2065 |
Tubeimoside-1 |
Bolbostemma paniculatum (Maxim) Franquet |
Mcl-1, Bcl-xL, Bcl-2 |
MDA-MB-231, T47D |
PhytoCAT-2066 |
(Z)-ethylidene-4,6-dimethoxycoumaran-3-one (Compound 1) |
Pogostemon quadrifolius (Benth.) |
NA |
Caco-2, HeLa, THP-1, MCF-7, Jurkat E6-1 |
PhytoCAT-2067 |
Senecio glaucus extract |
Senecio glaucus. |
NA |
MCF-7, HepG2, A549 |
PhytoCAT-2068 |
Brazilin A |
Caesalpinia sappan. |
NA |
MCF-7, A549 |
PhytoCAT-2069 |
Eugenia pyriformis (EP-EO) essential oil |
Eugenia pyriformis |
NA |
MCF-7, HeLa, M059J |
PhytoCAT-2070 |
Pergularia tomentosa extract |
Pergularia tomentosa |
NA |
HCT-116, HepG2, MCF-7 |
PhytoCAT-2071 |
Picraviane A |
Picramnia glazioviana Engl. |
NA |
MDA-MB-231 |
PhytoCAT-2072 |
Muscadine grape skin extract (MSKE) |
Vitis rotundifolia |
Snail, pSTAT-3 |
NA |
PhytoCAT-2073 |
Aspergillus nidulans extract |
Endophytic fungus Aspergillus nidulans, associated with Nyctanthes arbor-tristisinn. |
NA |
MCF-7, NCI-H460, HeLa |
PhytoCAT-2074 |
Sterigmatocystin |
Endophytic fungus Aspergillus nidulans, associated with Nyctanthes arbor-tristisinn. |
NA |
MCF-7, NCI-H460, HeLa |
PhytoCAT-2075 |
Onosma hookeri Clarke. var. longiforum Duthie (OHC-LD) extract |
Onosma hookeri |
NA |
MCF-7 |
PhytoCAT-2076 |
Jatrophone (JA) |
Jatropha gossypiifolia |
AXIN2, HMGA2, MYC, PCNA, CCND1, EMT |
MDA-MB-231, MDA-MB-157, HCC-38, MDA-MB-468 |
PhytoCAT-2077 |
Baeckea frutescens extracts |
Baeckea frutescens |
NA |
MCF-7, MDA-MB-231, MCF-10A |
PhytoCAT-2078 |
7,15-isopimaradien-3β,19-diol |
Aeollanthus rydingianus |
NA |
MDA-MB-231 |
PhytoCAT-2079 |
Polysaccharides from Taxus cuspidata |
Taxus cuspidata |
NA |
MCF-7, HepG2 |
PhytoCAT-2080 |
Quercus robur extract |
Quercus robur |
NA |
MCF-7, HeLa, Jurkat, HT-29 |
PhytoCAT-2081 |
Quercus macrocarpa extract |
Quercus macrocarpa |
NA |
MCF-7, HeLa, Jurkat, HT-29 |
PhytoCAT-2082 |
Scrophularia frigida Boiss extract |
Scrophularia frigida Boiss |
Human epidermal growth factor receptor 2, myeloid cell Leukemia-1, Caspase 3, Caspase 9 |
NA |
PhytoCAT-2083 |
Silvestrol |
Aglaia foveolata |
Cyclin B, Cyclin D |
MDA-MB-435 |
PhytoCAT-2084 |
Selaginella repanda extract |
Selaginella repanda |
NA |
A549, HCT-116, MCF-7 |
PhytoCAT-2085 |
Polydatin (PD) |
Polygonum cuspidatum |
Creb, Cyclin D1 |
MDA-MB-231, MCF-7 |
PhytoCAT-2086 |
Agave americana extract |
Agave americana |
NA |
MCF-7, Vero |
PhytoCAT-2087 |
Strychnos nuxvomica extract |
Strychnos nux-vomica. |
NA |
MCF-7, Vero |
PhytoCAT-2088 |
Areca catechu extract |
Areca catechu |
NA |
MCF-7, Vero |
PhytoCAT-2089 |
Morusin |
Morus alba |
E-cadherin, Vimentin, α2-, α6-, β1- integrin, MMP2, MMP9, iNOX, COX |
MCF-7, A549, HepG2, MDA-MB-231 |
PhytoCAT-2090 |
2',3,4',5,5'-pentahydroxy-cis-stilbene |
Morus nigra. |
NA |
MCF-7, HepG2 |
PhytoCAT-2091 |
Norartocarpetin |
Morus nigra. |
NA |
MCF-7, HepG2 |
PhytoCAT-2092 |
Cudraflavone A |
Morus nigra. |
NA |
MCF-7, HepG2 |
PhytoCAT-2093 |
Kuwanon G |
Morus nigra. |
NA |
MCF-7, HepG2 |
PhytoCAT-2094 |
Albafuran C |
Morus nigra. |
NA |
MCF-7, HepG2 |
PhytoCAT-2095 |
Mulberrofuran G |
Morus nigra. |
NA |
MCF-7, HepG2 |
PhytoCAT-2096 |
Ursolic acid-3-O-acetate |
Morus nigra. |
NA |
MCF-7, HepG2 |
PhytoCAT-2097 |
Uvaol |
Morus nigra. |
NA |
MCF-7, HepG2 |
PhytoCAT-2098 |
Heteroclitalactone A |
Kadsura heteroclita () Craib (Schizandraceae) |
NA |
Bel-7402, BGC-823, MCF-7, HL-60 |
PhytoCAT-2099 |
Heteroclitalactone C |
Kadsura heteroclita () Craib (Schizandraceae) |
NA |
Bel-7402, BGC-823, MCF-7, HL-60 |
PhytoCAT-2100 |
Heteroclitalactone D |
Kadsura heteroclita () Craib (Schizandraceae) |
NA |
Bel-7402, BGC-823, MCF-7, HL-60 |
PhytoCAT-2101 |
Heteroclitalactone E |
Kadsura heteroclita () Craib (Schizandraceae) |
NA |
Bel-7402, BGC-823, MCF-7, HL-60 |
PhytoCAT-2102 |
Schisandronic acid |
Kadsura heteroclita () Craib (Schizandraceae) |
NA |
Bel-7402, BGC-823, MCF-7, HL-60 |
PhytoCAT-2103 |
Nigranoic acid |
Kadsura heteroclita () Craib (Schizandraceae) |
NA |
Bel-7402, BGC-823, MCF-7, HL-60 |
PhytoCAT-2104 |
Changnanic acid |
Kadsura heteroclita () Craib (Schizandraceae) |
NA |
Bel-7402, BGC-823, MCF-7, HL-60 |
PhytoCAT-2105 |
Salvia atropatana extract |
Salvia atropatana |
NA |
PC3, MCF-7, MDA-MB-231 |
PhytoCAT-2106 |
Saprorthoquinone + Aethiopinone |
Salvia atropatana |
NA |
PC3, MCF-7, MDA-MB-231 |
PhytoCAT-2107 |
Atropatanene |
Salvia atropatana |
NA |
PC3, MCF-7, MDA-MB-231 |
PhytoCAT-2108 |
Rumex crispus L. extract |
Rumex crispus. |
NA |
MCF-7, HCT-116 |
PhytoCAT-2109 |
Ginsenoside Rp1 |
Panax ginseng |
IGF-1R |
MDA-MB-231, MCF-7, T-47D |
PhytoCAT-2110 |
6, 7-dimethoxy-1-(α-hydroxy-4-methoxybenzyl)-2-methyl-1, 2, 3, 4-tetrahydroisoquinoline |
Annona squamosa |
NA |
HepG-2, MCF-7, HCT-116 |
PhytoCAT-2111 |
Coclaurine |
Annona squamosa |
NA |
HepG-2, MCF-7, HCT-116 |
PhytoCAT-2112 |
Budlein A methylacrylate (BAM) |
Helianthus genus |
IκBα kinase, exportin-1 |
MDA-MB-231, MDA-MB-453, MDA-MB-435, MDA-MB-468, HCC1937, HCC2218, HCC1954, HCC202, HCC1500, MCF-7 |
PhytoCAT-2113 |
Quercus infectoria extract |
Quercus infectoria |
NA |
MDA-MB-231, HeLa, Hep G2, L929 |
PhytoCAT-2114 |
Pachymic acid |
Poria cocos |
Cyclin D1, Cyclin E, CDK2, CDK4, p53, p21, Bcl-2, Bax, Cyt-c, Caspase 3, Caspase 8, Caspase 9, MMP9, PKM2 |
SKBR-3, BALB/c nude mice/MDA-MB-231 |
PhytoCAT-2115 |
Luotonin A |
Peganum nigellastrum |
NA |
MCF-7, HeLa |
PhytoCAT-2116 |
Kola acuminate extract |
Kola acuminate |
NA |
MCF-7, MDA-MB-468, LNCaP |
PhytoCAT-2117 |
Xanthinosin |
Xanthium strumarium |
DR4, DR5, p53, CHOP, Bax, Caspase 3, Caspase 8, Caspase 9, Bcl-2 |
DLD1, DU145, HeLa, MCF-7, MDA-MB-231 |
PhytoCAT-2118 |
Glandora rosmarinifolia essential oil |
Glandora rosmarinifolia |
NA |
HA22T/VGH, HepG2, Hep3B, SUM 149, MDA-MB-231 |
PhytoCAT-2119 |
Schinensin C |
Schisandra chinensis |
NA |
MCF-7, A549, HeLa, RPMI8226 |
PhytoCAT-2120 |
Schinensin D |
Schisandra chinensis |
NA |
MCF-7, A549, HeLa, RPMI8226 |
PhytoCAT-2121 |
Shisanbilactone A |
Schisandra chinensis |
NA |
MCF-7, A549, HeLa, RPMI8226 |
PhytoCAT-2122 |
Kadsuphilactone B |
Schisandra chinensis |
NA |
MCF-7, A549, HeLa, RPMI8226 |
PhytoCAT-2123 |
Propinic lactone A |
Schisandra chinensis |
NA |
MCF-7, A549, HeLa, RPMI8226 |
PhytoCAT-2124 |
Polyphylloside A |
Paris polyohylla |
NA |
MCF-7, MDA-MB-231, A549, HeLa, HCT-116 |
PhytoCAT-2125 |
Polyphylloside B |
Paris polyohylla |
NA |
MCF-7, MDA-MB-231, A549, HeLa, HCT-116 |
PhytoCAT-2126 |
Polyphylloside C |
Paris polyohylla |
NA |
MCF-7, MDA-MB-231, A549, HeLa, HCT-116 |
PhytoCAT-2127 |
Polyphylloside D |
Paris polyohylla |
NA |
MCF-7, MDA-MB-231, A549, HeLa, HCT-116 |
PhytoCAT-2128 |
Polyphylloside E |
Paris polyohylla |
NA |
MCF-7, MDA-MB-231, A549, HeLa, HCT-116 |
PhytoCAT-2129 |
Polyphylloside F |
Paris polyohylla |
NA |
MCF-7, MDA-MB-231, A549, HeLa, HCT-116 |
PhytoCAT-2130 |
7-oxodioscin |
Paris polyohylla |
NA |
MCF-7, MDA-MB-231, A549, HeLa, HCT-116 |
PhytoCAT-2131 |
Isonarthogenin 3-O-α-L-rhamnopyranosyl-(1 → 2)-[α-L-rhamnopyranosyl-(1 → 4)]-β-D-glucopyranoside |
Paris polyohylla |
NA |
MCF-7, MDA-MB-231, A549, HeLa, HCT-116 |
PhytoCAT-2132 |
Trinervuloside C |
Paris polyohylla |
NA |
MCF-7, MDA-MB-231, A549, HeLa, HCT-116 |
PhytoCAT-2133 |
Caroguaianolide D |
Carpesium abrotanoides |
NA |
MDA-MB-231, HGC-27 |
PhytoCAT-2134 |
Caroguaianolide E |
Carpesium abrotanoides |
NA |
MDA-MB-231, HGC-27 |
PhytoCAT-2135 |
4α-hydroxy-9β,10β-epoxy-1βH,5αH-guaia11(13)-en-8α,12-olide |
Carpesium abrotanoides |
NA |
MDA-MB-231, HGC-27 |
PhytoCAT-2136 |
Carabrolactone B |
Carpesium abrotanoides |
NA |
MDA-MB-231, HGC-27 |
PhytoCAT-2137 |
4α-hydroxy1βH-guaia-9,11(13)-dien-12,8α-olide |
Carpesium abrotanoides |
NA |
MDA-MB-231, HGC-27 |
PhytoCAT-2138 |
8-epi-inuviscolide |
Carpesium abrotanoides |
NA |
MDA-MB-231, HGC-27 |
PhytoCAT-2139 |
Inuviscolide |
Carpesium abrotanoides |
NA |
MDA-MB-231, HGC-27 |
PhytoCAT-2140 |
6β, 14α-dihydroxy-15-acetoxysclareol |
Salvia reuterana |
NA |
MCF-7, HeLa |
PhytoCAT-2141 |
14α, 15- dihydroxy sclareol |
Salvia reuterana |
NA |
MCF-7, HeLa |
PhytoCAT-2142 |
14α-hydroxy-15-chlorosclareol |
Salvia reuterana |
NA |
MCF-7, HeLa |
PhytoCAT-2143 |
14α-hydroxy-15-acetoxysclareol |
Salvia reuterana |
NA |
MCF-7, HeLa |
PhytoCAT-2144 |
6β-hydroxy-14α-epoxysclareol |
Salvia reuterana |
NA |
MCF-7, HeLa |
PhytoCAT-2145 |
6β-hydroxysclareol |
Salvia reuterana |
NA |
MCF-7, HeLa |
PhytoCAT-2146 |
14α-epoxysclareol |
Salvia reuterana |
NA |
MCF-7, HeLa |
PhytoCAT-2147 |
Sinopodophylline C |
Sinopodophyllum hexandrum |
NA |
MCF-7, MDA-MB-231, T47D |
PhytoCAT-2148 |
Sinopodophylline A |
Sinopodophyllum hexandrum |
NA |
MCF-7, MDA-MB-231, T47D |
PhytoCAT-2149 |
Sinopodophylline D |
Sinopodophyllum hexandrum |
NA |
MCF-7, MDA-MB-231, T47D |
PhytoCAT-2150 |
Topazolin |
Sinopodophyllum hexandrum |
NA |
MCF-7, MDA-MB-231, T47D |
PhytoCAT-2151 |
Sinopodophylliside A |
Sinopodophyllum hexandrum |
NA |
MCF-7, MDA-MB-231, T47D |
PhytoCAT-2152 |
Quercetin-3-O-β-Dglucopyranoside |
Sinopodophyllum hexandrum |
NA |
MCF-7, MDA-MB-231, T47D |
PhytoCAT-2153 |
Quercetin-3-O-β-D-glucopyranoside5-methly ether |
Sinopodophyllum hexandrum |
NA |
MCF-7, MDA-MB-231, T47D |
PhytoCAT-2154 |
Quercetin-3-O-β-D-glucopyranoside7-methly ether |
Sinopodophyllum hexandrum |
NA |
MCF-7, MDA-MB-231, T47D |
PhytoCAT-2155 |
Kaempferol-3-O-β-D-glucopyranoside4′-methly ether |
Sinopodophyllum hexandrum |
NA |
MCF-7, MDA-MB-231, T47D |
PhytoCAT-2156 |
Stevioside |
Stevia rebaudiana |
Bax, Bcl-2, Caspase 9 |
MDA-MB-231, SKBR-3, MCF-7 |
PhytoCAT-2157 |
Lobeline |
Lobelia inflata |
P-gp |
Caco-2, CCRF-CEM, MDA-MB-231pcDNA3-BCRP-clone23 |
PhytoCAT-2158 |
(+/-)-trans-3-(3,4-dimethoxyphenyl)-4-[(E)-3,4-dimethoxystyryl]cyclohex-1-ene |
Zingiber cassumunar |
P-gp |
MCF-7/ADR |
PhytoCAT-2159 |
Thaliblastine (TBL) |
Thalictrum foliolosum |
P-gp |
MCF/AdR |
PhytoCAT-2160 |
Paris saponin VII |
Trillium tschonoskii |
NFR1, TRAIL R1/DR4, TRAIL R2/DR5, FADD, PARP, Caspase 8, Caspase 3, P-gp |
MCF-7/ADR |
PhytoCAT-2161 |
Sophoflavescenol |
Sophora flavescens |
NA |
MCF-7, HL-60, LLC, A549 |
PhytoCAT-2162 |
Thymbra Spicata extract |
Thymbra Spicata |
STAT-3, NF-kB |
MCF-7 |
PhytoCAT-2163 |
3'-hydroxygenkwanin |
Daphne genkwa |
NA |
MCF-7, MDA-MB-231, Huh7, AGS, HT-29, B 16, Colo 205, A549, A2058 |
PhytoCAT-2164 |
Rigidusol |
Haplopappus rigidus phil. |
NA |
ED50 = 3.8 μg/mL against MCF-7 |
PhytoCAT-2165 |
Scutellariae radix |
Scutellaria baicalensis |
BCRP, MRP2 |
Rats |
PhytoCAT-2166 |
Pomegranate seed oil (PSO) |
Punica granatum |
VEGF, IL-2, IL-6, IL-12, IL-17, IP-10, MIP-1α, MIP-1β, MCP-1, TNF-α |
MCF-7, MDA-MB-231, HT29, HepG2, HuH7, HCT116, DU145 |
PhytoCAT-2167 |
Xanthotoxol |
Angelica japonica |
ERα, PR, EGFR, mTOR |
In-silico |
PhytoCAT-2168 |
Extra-Virgin Olive Oil (EVOO) |
Olea Europea |
HER2, FASN |
MCF-7, SKBR3 |
PhytoCAT-2169 |
Valtrate |
Valeriana jatamansi Jones |
p-Akt, Cyclin B1, Caspase 8, p21, p-cdc2, Caspase 3, Caspase 9, MMP-9, MMP-2, PARP |
MCF-7, MDA-MB-231, MDA-MB-468, MDA-MB-453, MCF10A, SK-OV-3 |
PhytoCAT-2170 |
Spinasterol |
Pueraria mirifica
Pueraria lobata |
ERα, ERβ |
NA |
PhytoCAT-2171 |
Dendrosicyos socotrana extract |
Dendrosicyos socotrana |
NA |
MCF-7, A-427, LCLC-103H, 5637, RT-112 |
PhytoCAT-2172 |
Withanina aduensis extract |
Withanina aduensis |
NA |
MCF-7, A-427, LCLC-103H, 5637, RT-112 |
PhytoCAT-2173 |
Withania riebeckii extract |
Withania riebeckii |
NA |
MCF-7, A-427, LCLC-103H, 5637, RT-112 |
PhytoCAT-2174 |
Dracena cinnabari extract |
Dracaena cinnabari |
NA |
MCF-7, A-427, LCLC-103H, 5637, RT-112 |
PhytoCAT-2175 |
Buxus hildebrandtii extract |
Buxus hildebrandtii |
NA |
MCF-7, A-427, LCLC-103H, 5637, RT-112 |
PhytoCAT-2176 |
Porphyra dentata |
Porphyra dentata |
NA |
4T1 cell-implanted tumor BALB/c mice |
PhytoCAT-2177 |
Cedrelopsis grevei essential oil |
Cedrelopsis grevei |
NA |
MCF-7 |
PhytoCAT-2178 |
(Z)-β-farnesene |
Cedrelopsis grevei |
NA |
MCF-7 |
PhytoCAT-2179 |
3β,6β,16β-trihydroxy-lup-20(29)-ene |
Combretum leprosum |
NA |
MRC5, MCF-7, HepG2, T24, HCT116, HT29, CACO-2 |
PhytoCAT-2180 |
Hypericum adenotrichum extract |
Hypericum adenotrichum |
Caspase 3, PARP |
MCF-7, MDA-MB-231 |
PhytoCAT-2181 |
Nepeta deflersiana |
Nepeta deflersiana |
NA |
MCF-7, A549 |
PhytoCAT-2182 |
Carpesium cernuum extract |
Carpesium cernuum |
MMP9, CD44, COL4A2, TIMP1 |
MDA-MB-231, MCF-7, A549 |
PhytoCAT-2183 |
Solanum indicum extract |
Solanum indicum var. recurvatum |
NA |
NA |
PhytoCAT-2184 |
Triplaris gardneriana extracts |
Triplaris gardneriana |
NA |
MCF-7 |
PhytoCAT-2185 |
Helianthella quinquenervis extract |
Helianthella quinquenervis |
NA |
MCF-7, A549, HT-29 |
PhytoCAT-2186 |
Lithocarpus polystachyus extract |
Lithocarpus polystachyus |
PPARγ, Bax, Capase 3, Cyclin D1, Bcl-2 |
MCF-7 |
PhytoCAT-2187 |
Sageretia thea extract |
Sageretia thea |
NA |
MDA-MB-231 |
PhytoCAT-2188 |
Pumpkin |
Cucurbita maxima |
NA |
NA |
PhytoCAT-2189 |
Parvifloron D |
Plectranthus ecklonii |
NA |
MDA-MB-231 |
PhytoCAT-2190 |
Forskolin |
Coleus barbatus |
ERK1/2 |
MDA-MB-231, MDA-MB-468, MCF7, HeLa |
PhytoCAT-2191 |
Gelomulide K |
Suregada aequorea |
PARP-1 |
Xenograft model |