Phytochemical Name : (4α,5α,8β,10β)-4,10-dihydroxy-1,11(13)-guaidien-12,8-olide

Properties Information
PhytoCAT-ID PhytoCAT-1036
Phytochemical name or plant extracts (4α,5α,8β,10β)-4,10-dihydroxy-1,11(13)-guaidien-12,8-olide
PMID 30580030
Literature evidence Compound 4 exhibited strong and selective cell growth inhibition against HT-29 with viability 20.99% and was identified as a promising compound with high selectivity between cancer cells and normal human lung cells (BEAS-2B), especially against HT-29 (IC50 = 12.2 μg/mL) compared to that of cisplatin.
IUPAC name NA
Phytochemicals’ class or type of plant extracts Sesquiterpene lactone
Source of phytochemicals or plant Extracts Chrysophthalmum montanum
Geographical availability Southeastern, and Eastern parts of Turkey
Plant parts Aerial parts
Other cancers Breast cancer, Colon cancer, Lung cancer
Target gene or protein NA
Gene or Protein evidence NA
Target pathways NA
IC50 26.5±0.6 µg/mL against MCF-7
Potency In our study, we found that compound 4 has a low cytotoxicity against MCF-7 with IC50 value of >100 µg/mL by SRB assay
Cell line/ mice model MCF-7, MDA-MB 231, HT-29, PC3
Additional information  Compound 4 exhibited strong and selective cell growth inhibition against HT-29 with viability 20.99% and was identified as a promising compound with high selectivity between cancer cells and normal human lung cells (BEAS-2B), especially against HT-29 (IC50 = 12.2 μg/mL) compared to that of cisplatin.
PubChem ID NA
Additional PMIDs NA
Additional sources of information https://doi.org/10.1016/j.phytol.2020.01.003
Safety NA