| PhytoCAT-ID | Phytochemical name or plant extracts | Source of phytochemicals or plant Extracts | Target gene or protein | Cell line/ mice model |
|---|---|---|---|---|
| PhytoCAT-0 | Rocaglaol | Aglaia crassinervia | Bax, Bcl-xL, Caspase 9, Caspase 7, Cdc25c | Lu1, LNCaP, HL-60, SMMC-7721, A-549, MCF-7, W480 |
| PhytoCAT-2 | 1'-acetoxychavicol acetate | Alpinia galanga | STAT-3, MMP2, MMP9 | MCF-7, COR L23 |
| PhytoCAT-9 | Methyl ferulate | Calotropis procera | NA | MCF-7, HCT-116, HepG-2, A-549, SK-LU-1, KB |
| PhytoCAT-10 | Methyl 4-β-d-glucopyranosyl-ferulate | Calotropis procera | NA | MCF-7, HCT-116, HepG-2, A-549, SK-LU-1, KB |
| PhytoCAT-11 | Calotropagenin | Calotropis procera | NA | MCF-7, HCT-116, HepG-2, A-549, SK-LU-1, KB |
| PhytoCAT-16 | Kudolignan A | Sophora alopecuroides | NA | HeLa, Hep3B, MCF-7, H1299 |
| PhytoCAT-17 | Kudolignan B | Sophora alopecuroides | NA | HeLa, Hep3B, MCF-7, H1299 |
| PhytoCAT-18 | Stemophenanthrene A | Stemona tuberosa | NA | KB, MCF7, SK-LU-1, HepG2 |
| PhytoCAT-19 | Stemophenanthrene B | Stemona tuberosa | NA | KB, MCF7, SK-LU-1, HepG2 |
| PhytoCAT-20 | Stemophenanthrene C | Stemona tuberosa | NA | KB, MCF7, SK-LU-1, HepG2 |
| PhytoCAT-21 | Isopinosylvin A | Stemona tuberosa | NA | KB, MCF7, SK-LU-1, HepG2 |
| PhytoCAT-22 | Stemofuran X | Stemona pierrei | NA | KB, MCF7, SK-LU-1, HepG2 |
| PhytoCAT-23 | Stemofuran Y | Stemona tuberosa | NA | KB, MCF7, SK-LU-1, HepG2 |
| PhytoCAT-28 | Polyphenol mixtures of Euphorbia supina | Euphorbia supina | Snail1 , N-cadherin, MMP9, LOX, TNF-α-mediated VCAM-1 | MDA-MB-231 |
| PhytoCAT-29 | Caudatin | Cynanchum auriculatum | DR5, CHOP, p38 MAPK, JNK | MDA-MB-231, MCF-7/ nude mouse |
| PhytoCAT-33 | Berberiside A | Berberis tsarica | NA | A549, HepG2, MDA-MB-231 |
| PhytoCAT-34 | Berberiside D | Berberis tsarica | NA | A549, HepG2, MDA-MB-231 |
| PhytoCAT-41 | E/Z-acetoside | Tecoma stans | NA | Hep-G2, MCF-7 |
| PhytoCAT-55 | Isoazadironolide | Azadirachta indica | NA | HL60, A549, AZ521, SKBR-3 |
| PhytoCAT-61 | Bromelain proteinase (F9) | Ananas comosus | IL- 2, TNF-a | MCF-7, SK-MEL-28 |
| PhytoCAT-65 | Styrylpyrone dehydrogoniothalamin | Aniba heringeri | NA | PC-3, 786-0, HT-29, MCF-7, MDA-MB-231 |
| PhytoCAT-72 | Licania tomentosa extract | Licania tomentosa | NA | MCF-7, Caco-2 |
| PhytoCAT-87 | Lutein | Spinacia oleracea | HIF‑1α, Notch signaling, HES1, Bcl-2, Caspase 3, PARP, HO-1, SOD-1, Hsp-60 | MDA‑MB‑157, MCF‑7, BALB/c mice |
| PhytoCAT-89 | (-)-Cycloxanthochymol | Garcinia celebica | NA | HeLa, MCF-7, A549, B16 |
| PhytoCAT-90 | Isoxanthochymol | Garcinia celebica | NA | HeLa, MCF-7, A549, B16 |
| PhytoCAT-91 | Xanthochymol | Garcinia celebica | NA | HeLa, MCF-7, A549, B16 |
| PhytoCAT-94 | Trans-3-(3,4-dimethoxyphenyl)-4-[(E)-3,4-dimethoxystyryl]cyclohex-1-ene | Dryopteris fragrans | NA | A549, MCF-7, HepG2 |
| PhytoCAT-95 | Cis-3-(3,4-dimethoxyphenyl)-4-[(E)-3,4-dimethoxystyryl] cyclohex-1-ene | Dryopteris fragrans | NA | A549, MCF-7, HepG2 |
| PhytoCAT-97 | Aspidinol | Dryopteris fragrans | NA | A549, MCF-7, HepG2 |
| PhytoCAT-99 | (E)-caffeic acid-9-O-β-d-xylpyranosyl-(1→2)-β-d-glucopyranosyl ester | Dryopteris fragrans | NA | A549, MCF-7, SGC7901 , HUVEC |
| PhytoCAT-100 | Octyl gallate | Terminalia bellirica | Cyclin D1, Cyclin D3, CDK-4, CDK-6, p18 INK4, p21Waf-1, p27 KIP, MRP2 | MCF-7, MDA-MB-231 |
| PhytoCAT-108 | Thidiazuron | Nymphaea alba | uPAR, uPA, VEGF, MMP2, MMP9, TIMP-1/2 | NA |
| PhytoCAT-115 | 3R,8R-Dehydrofalcarindiol | Artemisia monosperma | NA | MDA231, MCF-7, LS174T, SKCO1, COLO320DM, WIDR |
| PhytoCAT-130 | Cichorin D | Cichorium intybus | NA | MDA-MB-468, MDA-MB-231, SK-N-MC, PC-3 |
| PhytoCAT-131 | Cichorin E | Cichorium intybus | NA | MDA-MB-468, MDA-MB-231, SK-N-MC, PC-3 |
| PhytoCAT-139 | 12-O-benzoyl-20-O-acetyl-3β,12β,14β,20β-tetrahydroxy-pregnan-3-ylO-β-D-glucopyranosyl-(1→4)-β-D-glucopyranosyl-(1 → 4)-3-methoxy-β-D-ribopyranoside | Caralluma tuberculata | PARP | MCF-7, MDA-MB-468 |
| PhytoCAT-140 | 7-O-acetyl-12-O-benzoyl-3β,7β,12β,14β-tetrahydroxy-17β-(3-methylbutyl-O-acetyl-1-yl)-androstan-3-ylO-β-D-glucopyranosyl-(1 → 4)-6-deoxy-β-D-allopyranosyl-(1 → 4)-β-D-cymaropyranosyl-(1 → 4)-β-D-cymapyranosyl-(1→ 4)-β-D-cymaropyranoside | Caralluma tuberculata | PARP | MCF-7, MDA-MB-469 |
| PhytoCAT-152 | Black raspberry | Rubus occidentalis | NA | KB, CAL-27, MCF-7, HT-29, HCT116, LNCaP |
| PhytoCAT-167 | 3,4-dihydroxy-phenylacetic acid (PAA) | Tragopogon orientalis | NA | T47D |
| PhytoCAT-175 | Cranberry extract | Vaccinium macrocarpon | NA | MDA-MB-435, MCF-7 |
| PhytoCAT-176 | 2-hydroxy-6-tridecylbenzoic acid | Ginkgo biloba | E-cadherin, N-cadherin, Vimentin, Snail, MMP2, MMP9 | MDA-MB-231, 4 T1 |
| PhytoCAT-184 | Camalexin | Arabidopsis thaliana | NA | SKBR-3, PREC |
| PhytoCAT-185 | Sinigrin | Armoracia rusticana | COX-1 | HCT-116, MCF-7, NCIH460, CNS, SF-268 |
| PhytoCAT-186 | Docosadienoic Acid (DDA) | Brassica carinata | IL-1β, IL-6, IFN-γ, MCP-1, TNF-α | SKBR-3 and MDA-MB-231 |
| PhytoCAT-187 | Docosatrienoic acid (DTA) | Brassica carinata | IL-1β, IL-6, IFN-γ, MCP-1, TNF-α | SKBR-3 and MDA-MB-231 |
| PhytoCAT-189 | P-coumaric acid | Carrichtera annua | p53, p21, CDK4 | SW 620, Hep G2, A549, T47D, HeLa, MCF-7 |
| PhytoCAT-201 | Snakegourd root polysaccharide | Trichosanthes cucumerina | Caspase 3, Caspase 8 | MCF-7 |
| PhytoCAT-209 | Benzoiisovanillin | Solanum nigrum | NA | MDA-MB-231, MCF-7 |
| PhytoCAT-210 | Mulberry leaf lectin | Morus alba | Caspase 3 | MCF-7, HCT-15 |
| PhytoCAT-212 | Moracin O | Morus alba | BCL‑XL, Bcl‑2, p65 subunit of NF‑κB | 4T1 |
| PhytoCAT-213 | Moracin P | Morus alba | BCL‑XL, Bcl‑2, p65 subunit of NF‑κB | 4T1 |
| PhytoCAT-218 | Strawberry extract | Fragaria ananassa | NA | KB, CAL-27, MCF-7, HT-29, HCT116, LNCaP |
| PhytoCAT-219 | Citrus sphaerocarpa extract | Citrus sphaerocarpa | MMP9 | MDA-MB-231 |
| PhytoCAT-221 | p-hydroxybenzoic acid-4-O-α-d-manopyranosyl-(1 → 3)-α-l-rhamnopyranoside | Melilotus officinalis | NA | MCF-7 |
| PhytoCAT-222 | 4-O-α-l-rhamnopyran-osyl-(1 → 6)-α-d-manopyranosyl-(1 → 3)-α-l-rhamnopyranoside | Melilotus officinalis | NA | MCF-7 |
| PhytoCAT-225 | Resveratrol | Juniperus polycarpos | PTEN, STAT-3, VDR, BRCA1, EDA, miR-125b-5p, miR-200c-3p, miR-409-3p, miR-122-5p, miR-542-3p, PCNA, Rb, p53, Bcl-2, aromatase, IL-6, p53, HNRNPA1, Caspase 3, MMP9, AURKA, PLK1, PAK1, Bax, CYP19, p21, RAD51, Twist1, EMT , EGF, AHR, ERα, CYP1A1, CYP1B1, GREB1, cAMP | MCF-7, HeLa, Seg-1, T47D, MDA-MB-231 , HCT116, PC12 , 4T1, ZR-75-1, MDA-MB-435, SKBR-3 |
| PhytoCAT-231 | Cannabidiolic acid | Cannabis sativa | COX-2 | MDA-MB-231 |
| PhytoCAT-232 | Pomaces from Muscadinia rotundifolia | Muscadinia rotundifolia | Cyclin A, p21 | MCF-7, MDA-MB-231 |
| PhytoCAT-235 | Salidroside | Rhodiola rosea | NA | MCF-7, Female BALB/c nude mice |
| PhytoCAT-236 | Fukinolic acid | Actaea racemosa | NA | MCF-7 |
| PhytoCAT-249 | Dioscorealide B | Dioscorea membranacea | Bax, Bak, Bcl-2, Caspase 8, Caspase 9, Caspase 7 | NA |
| PhytoCAT-250 | Arachidin-1 | Arachis hypogaea | Caspase 9, PARP, Survivin | MDA-MB-231, MDA-MB-435, MCF-10A |
| PhytoCAT-251 | Arachidin-3 | Arachis hypogaea | NA | MDA-MB-231, MDA-MB-435, MCF-10A |
| PhytoCAT-252 | Ampelopsin E | Dryobalanops rappa | PDGF, MMP2, MMP9, MMP14 | MDA-MB-231, MCF-7, HT-29, A-549, HeLa, 3T3, MCF10A |
| PhytoCAT-255 | Safflower yellow (SY) | Carthamus tinctorius | MMP9, p-Src | MBA-MD-231 |
| PhytoCAT-258 | Persin | Persea americana | NA | MCF-7, T-47D, MDA-MB-231 |
| PhytoCAT-301 | Rottlerin | Mallotus philippinensis | Atg12, Beclin-1, Bcl-2, Bcl-xL, XIAP, cIAP-1, LRP6 | MDA-MB-231, T47D, PC-3, DU145, MCF-7 |
| PhytoCAT-334 | Putranjiva roxburghii Seed Extract | Putranjiva roxburghii | NA | PANC-1, MDA-MB 231, HCT-116 |
| PhytoCAT-335 | 9-O-demethyltrigonostemone | Strophioblachia fimbricalyx | NA | NCI-H187, KB, MCF-7 |
| PhytoCAT-343 | Glyceryl 1-monopalmitate | Phyllostachys heterocycla | NA | MCF-7 |
| PhytoCAT-373 | Hypericum salsugineum extracts | Hypericum salsugineum | Tyrosinase | MCF-7, MDA-MB-231 |
| PhytoCAT-377 | Vitisin B | Iris lactea | FAS | MDA-MB-231 |
| PhytoCAT-379 | Martynoside | Ajuga chamaecistus | ICI182780, IGFBP3 | MCF-7 |
| PhytoCAT-380 | Acteoside | Anisomeles indica | NA | MCF-7 |
| PhytoCAT-408 | Salvianolic acid A | Salvia miltiorrhiza | Transgelin 2, ABC transporter | MCF-7/PTX |
| PhytoCAT-418 | Hydroxytyrosol | Teucrium polium | Beclin-1, p62 | MDA-MB-231 |
| PhytoCAT-420 | (-)-kunstleramide | Beilschmiedia kunstleri | NA | A-549, Hela, MCF-7, IMR-32 |
| PhytoCAT-422 | Cinnamic Acid | Goniothalamus laoticus | TNF-α, TNFR1 , Caspase 8, Caspase 3 | MDA-MB-231, MCF-7, HeLa, K562 |
| PhytoCAT-423 | Goniothalamin | Cryptocarya latifolia | p38, JNK1/2, AKT, Bax, Bcl-2 | SKBR-3 |
| PhytoCAT-424 | Methyl linderone (ML) | Lindera erythrocarpa | STAT-3, AP-1, MMP9, IL-8 | MCF-7 |
| PhytoCAT-430 | Sistosterol-3-beta-D-glycoside | Cassia petersiana | NA | NA |
| PhytoCAT-432 | Chickpea protease inhibitor concentrate | Cicer arietinum | NA | MDA-MB-231, PC-3, LNCaP |
| PhytoCAT-434 | Butein | Cyclopia subternata | Aromatase | MDA-MB-231, MCF-7 |
| PhytoCAT-435 | 2',4'-dihydroxy-6'-methoxychalcone | Erythrina abyssinica | NA | MCF-7, A549 |
| PhytoCAT-439 | Isoliquiritigenin | Glycyrrhiza glabra | Arg-1, HO-1, iNOS, microRNA 155, SHIP1, STAT-3, STAT6, PLA2, COX-2, CYP4A, PGE2, COX-1, FLAP, 5-LOX, LTB4, HIF-1α, VEGF, MMP2, MM9, Aromatase | MCF-7, A-549, BGC-823, MDA-MB-231, HepG2 |
| PhytoCAT-443 | Glycybridin D (4) | Glycyrrhiza glabra | PTP1B | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-444 | Glycybridin A (1) | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-445 | Glycybridin B (2) | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-446 | Glycybridin C (3) | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-447 | Glycybridin E (5) | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-448 | Glycybridin F (6) | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-449 | Glycybridin G (7) | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-450 | Glycybridin H (8) | Glycyrrhiza glabra | PTP1B | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-451 | Glycybridin I (9) | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-452 | Glycybridin J (10) | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-453 | Glycybridin K (11) | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-459 | Kanzonol X | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-462 | Kanzonol U | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-464 | Glyinflanin H | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-465 | Kanzonol Y | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-474 | Xambioona | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-477 | Euchrenone a5 | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-483 | [6″,6″-dimethylpyrano(2″,3″:4,5)]-3′-γ,γ-dimethylallyl-2′,3,4′-trihydroxychalcone | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-484 | Kanzonol C | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-485 | Kanzonol B | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-486 | Licoagrochalcone A | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-488 | Isobavachalcone | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-489 | Erybacin | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-490 | Licoagrocarpin | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-491 | Dehydroglyceollin I | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-494 | Dibenzoylmethane | Glycyrrhiza inflata | MMP9 | MCF‑7 |
| PhytoCAT-495 | Licochalcone A (LCA) | Glycyrrhiza inflata | p53, Sp1, PRMT6 | MDA-MB-231, MCF-7, MCF-10A |
| PhytoCAT-496 | Licochalcone B (LCB) | Glycyrrhiza glabra | Cyclin A, CDK2, Cdc25 A, p21, Caspase 3, Caspase 9, Bax, Bcl-2, p53 | MCF-7 |
| PhytoCAT-498 | 2,4-di-tert-butylphenol (HU-2) | Humboldtia unijuga | p53 | MCF-7 |
| PhytoCAT-505 | Deguelin | Mundulea sericea | NA | MDA-MB-231 |
| PhytoCAT-507 | Ebenfuran I | Onobrychis ebenoides | IGFBP-3 | MCF-7, MC3T3-E1, HeLa |
| PhytoCAT-508 | Ebenfuran II | Onobrychis ebenoides | NA | MCF-7, MC3T3-E1, HeLa |
| PhytoCAT-509 | Ebenfuran III | Onobrychis ebenoides | NA | MCF-7, MC3T3-E1, HeLa |
| PhytoCAT-518 | Piceatannol (PCT)/(PIC) | Sophora interrupta | NA | MCF-7, SKBR-3 |
| PhytoCAT-524 | Hexadecanoic acid | Vicia monantha | NA | MCF-7, HCT-116, HepG2 |
| PhytoCAT-525 | β-sitosterol | Vicia monantha | NA | MCF-7, HCT-116, HepG2 |
| PhytoCAT-531 | Allium bakhtiaricum extracts | Allium bakhtiaricum | NA | MDA-MB-231, MCF-7, 4T1 BALB/c mice, HepG2, HT-29 |
| PhytoCAT-532 | 2-Methylpyridine-1-ium-1-sulfonate | Allium hirtifolium | Bax, Bcl-2, Caspase 3, Caspase 9, VEGF, MMP2, MMP9, p21, p27, p53 | MCF-7, MDA-MB-231 |
| PhytoCAT-534 | Allicin | Allium sativum | Caspase 3, Caspase 8, Caspase 9, NOXA, p21, Bak, Bcl-xL | HeLa , MCF-7, L929, A549, HT29, HUVEC, HCC-70 |
| PhytoCAT-535 | Alliin | Allium sativum | NA | MCF-7, HCC-70 |
| PhytoCAT-536 | Thiosulfinates | Allium tuberosum | NA | MCF-7, SW480, HepG2, LNCaP.FGC, mice |
| PhytoCAT-537 | Diallyl disulphide | Allium vineale | Bax, Bcl-2, Bcl-w, Bcl-xL | MCF-7 |
| PhytoCAT-540 | Aloe vera extract | Aloe vera | Cyclin D1, CYP 1A1, CYP 1A2, Bax, p21 | MCF-7, Hela |
| PhytoCAT-549 | Liriopem I (1) | Liriope muscari | NA | MDA-MB-435 |
| PhytoCAT-550 | Liriopem II (2) | Liriope muscari | NA | MDA-MB-435 |
| PhytoCAT-553 | Polyphyllin D | Paris polyphylla | Beclin-1, Caspase 3 | NA |
| PhytoCAT-569 | Punicalagin | Punica granatum | NA | MCF-7, Hs578T |
| PhytoCAT-578 | Gossypol | Cotton plant (Gossypium species), Thespesia populnea | Bcl-2, Bcl-xL | MCF-7, SiHa, Caco -2, HeLa, MCF-7/Adr, T-47D, HS 683, U373, U87 and U138 , C6 , SW-13 , SK-MEL-3, Colo 201 , KB, HT-29 |
| PhytoCAT-585 | 7α-hydroxy-β-sitosterol | Chisocheton tomentosus | Bax, Bcl-2, procaspase 9, procaspase 3, ERK1/2, FasL, Bim | MCF-7, HMEC, HSC-4, HepG2 |
| PhytoCAT-589 | 17-ethylene-3,4-dihydroxy-14-methyl-18-norandrostene-16-one | Melia azedarach. | Bax, Bcl-2 | T47D |
| PhytoCAT-590 | 17-ethylene-3,4-dihydroxy-5-pregnene-16-one | Melia azedarach. | Bax, Bcl-2 | T47D |
| PhytoCAT-598 | Niloticin | Turraea nilotica | NA | 4T1, HEp2, Vero |
| PhytoCAT-599 | Hispidol B | Turraea nilotica | NA | 4T1, HEp2, Vero |
| PhytoCAT-600 | Piscidinol A | Turraea nilotica | NA | 4T1, HEp2, Vero |
| PhytoCAT-609 | Moringa oleifera (MOLSr) extracts (M1S9) | Moringa oleifera | SFRP1, Bax, p53, Caspase 8, CaN, SLC39A6, VEGF | MDA-MB-231 xenograft breast tumor mice, MCF-7 |
| PhytoCAT-612 | (-)-5,6-dihydro-6-undecyl-2H-pyran-2-one | Horsfieldia superba | NA | PC-3, HCT-116, MCF-7 |
| PhytoCAT-613 | (-)-5,6-dihydro-6-tridecyl-2H-pyran-2-one | Horsfieldia superba | NA | PC-3, HCT-116, MCF-7 |
| PhytoCAT-614 | Anacardic acid | Anacardium occidentale | SCD, INSIG1,TGM2, PDK4, GPR176, ZBT20, GRP78, Hsp70, CDK-4, MMP9, Bcl-2, Mcl-1 , miR-378g, Cyclin D1, MYC, c-FOS, PPARγ, SIN3 | MDA-MB-231, MCF-7 |
| PhytoCAT-621 | Ardisiphenol A | Ardisia colorata | NA | FM3A |
| PhytoCAT-622 | Ardisiphenol B | Ardisia colorata | NA | FM3A |
| PhytoCAT-623 | Ardisiphenol C | Ardisia colorata | NA | FM3A |
| PhytoCAT-624 | Alkylresorcinol A | Ardisia colorata | NA | FM3A |
| PhytoCAT-625 | Alkylresorcinol B | Ardisia colorata | NA | FM3A |
| PhytoCAT-626 | Alkylresorcinol C | Ardisia colorata | NA | FM3A |
| PhytoCAT-628 | 2',4'-dihydroxy-6'-methoxy-3',5'-dimethylchalcone (ON-III) | Eugenia aquea | Bim, erbB-2, MAPK, AKT, PARP, Caspase 3, KDR | MDA-MB-453, A549 |
| PhytoCAT-643 | Lunasin | Glycine max | MMP2, MMP9, NOS, IL-1, IL-6, TNF-α, Src, Akt, ERK, NF-κB, MCP-1 | MDA-MB-231, 4T1 |
| PhytoCAT-644 | Coumestrol | Glycine max | BCRP, Aromatase, ER | MCF-7, HCT116, T47D, MDA-MB-231 |
| PhytoCAT-645 | Bowman-Birk protease inhibitor | Glycine max | Atg5, Beclin-1, LC 3-II, Sequestosome1, Bax, Bcl-2 | MDA-MB-231 |
| PhytoCAT-651 | Licoagrochalcone B | Patrinia villosa | NA | MCF-7, BEL-7402, HT-29, SGC-7901, K562, A498, A549 |
| PhytoCAT-653 | Erianin | Dendrobium nobile | Bcl-2 | T47D, MDA-MB-231, MCF-7 |
| PhytoCAT-656 | Croblongifolin | Croton oblongifolius | NA | HEP-G2, SW620, CHAGO, KATO3, BT-474 |
| PhytoCAT-667 | Cabralealactone 3-acetate-24-methyl ether | Forsythia koreana | NA | MCF-7 |
| PhytoCAT-673 | Verbascoside | Orobanche amethystea | Caspase 3, Bax, Bcl-2, TLR4, MyD88, NF-κB | 4 T1, MCF-7, MDA-MB-231 |
| PhytoCAT-691 | Asaricin | Piper sarmentosum | Bcl-2, Bax | MDA-MB-231 |
| PhytoCAT-692 | Isoasarone | Piper sarmentosum | Bcl-2, Bax | MDA-MB-231 |
| PhytoCAT-693 | Saururus chinensis extract | Saururus chinensis | VEGF, Cyclin D1, Bcl-2, Caspase-3 | LNCaP, MCF-7 |
| PhytoCAT-694 | Sinapinic acid | Limoniastrum guyonianum | NA | MCF-7, HeLa |
| PhytoCAT-696 | Pterostilbene | Vitis rupestris | Beclin-1, LC3 II, hTERT, cMyc, Cyclin D1, Rac1, WAVE-2, Arp2/3 | MCF-7,MDA-MB-231 , T-47D, NCI H-460 |
| PhytoCAT-710 | Deoxyrhapontigenin | Rheum undulatum | GRP78, IRE1α, eIF2α, CHOP, JNK, p38 | MCF-7, MCF-7/adr |
| PhytoCAT-716 | Polyphenolics from mango | Mangifera indica | IR, IRS1, IGF-1R, mTOR | Female athymic BALB/c nude mice |
| PhytoCAT-718 | 5-((8Z, 11Z, 14Z)-hexatriaconta-8, 11, 14-trienyl) benzene-1,3-diol | Mangifera zeylanica | Caspase 7 | MCF-7 |
| PhytoCAT-733 | Trans-epsilon-viniferin | Paeonia lactiflora | NA | MCF-7, Hela, , HT-29, HePG2 |
| PhytoCAT-734 | Cis-epsilon-viniferin | Paeonia lactiflora | NA | MCF-7, Hela, , HT-29, HePG2 |
| PhytoCAT-735 | Gnetin H | Paeonia lactiflora | NA | MCF-7, Hela, , HT-29, HePG2 |
| PhytoCAT-743 | Protopheophorbide A | Ziziphus lotus | E-cadherin, Vimentin, β-catenin, FAK, Brk, Rac, Src | MDA-MB-231, MCF-7 |
| PhytoCAT-745 | Annoglaxin | Annona glabra | NA | MCF-7, A-498, PC-3, PACA-2 |
| PhytoCAT-746 | 27-hydroxybullatacin | Annona glabra | NA | MCF-7, A-498, PC-3, PACA-3 |
| PhytoCAT-751 | E-acetylmelodorinol | Cleistochlamys kirkii | NA | MDA-MB-231 |
| PhytoCAT-752 | Cleistenolide | Cleistochlamys kirkii | NA | MDA-MB-231 |
| PhytoCAT-754 | Licania rigida extract | Licania rigida | NA | MCF-7, Caco- 2 |
| PhytoCAT-757 | Pectic acid | Malus domestica | NA | MDA-MB-231 |
| PhytoCAT-759 | 2',4'-dihydroxy-3'-(2-hydroxybenzyl)-6'-methoxychalcone | Ellipeiopsis cherrevensis | NA | BC, NCI-H187, KB |
| PhytoCAT-762 | Selenium (Se)-containing polysaccharides | Pyracantha fortuneana | p53, Bax, PUMA, Noxa, Bcl-2, Bax, Caspase 3, Caspase 9, p53 | MDA-MB-231 |
| PhytoCAT-763 | Cheliensisin A | Goniothalamus cheliensis | NA | SKBR-3, HL-60, SMMC-7721, A-549, PANC-1 |
| PhytoCAT-765 | Sanguiin H-6 | Rubus coreanus | Caspase 8, Caspase 3, PARP, Bax, Bcl-2 | MCF-7, MDA-MB-231 |
| PhytoCAT-767 | 1-(2-hydroxyphenyl)-4-methylpentan-1-one | Rubus fairholmianus | PARP | MCF-7 |
| PhytoCAT-768 | 2-[(3-methylbutoxy) carbonyl] benzoic acid | Rubus fairholmianus | PARP | MCF-7 |
| PhytoCAT-769 | Blackberry extract | Rubus fruticosus | NA | MCF-7, KB, CAL-27, HT-29, HCT116, LNCaP |
| PhytoCAT-771 | (6E,10E) isopolycerasoidol | Pseuduvaria monticola | Bcl-2 | MCF-7, MDA-MB-231 |
| PhytoCAT-772 | (6E,10E) Isopolycerasoidol Methyl Ester | Pseuduvaria monticola | Caspase 3, Caspase 7, Caspase 9, Bcl-2, p38 MAPK | MCF-7,MDA-MB-231 |
| PhytoCAT-780 | Chlorogenic acid | Pavetta indica | NA | MDA-MB-435, MCF-7, MDA-MB-231, T-47D and BJ-hTERT |
| PhytoCAT-782 | Thymol | Xylopia sericea | NA | MDA-MB-231, PC-3, DU145, KLN205 |
| PhytoCAT-783 | Mollugin | Rubia cordifolia | FAS | SKBR-3 , SK-OV-3 |
| PhytoCAT-788 | Angelica sinensis polysaccharide | Angelica sinensis | PARP, Bax, Bcl-2, Bcl-xL, Apaf1 | T47D, nude mice xenograft model |
| PhytoCAT-796 | 8,2'-Diprenylquercetin 3-methyl ether | Sinopodophyllum hexandrum | NA | MDA-231 and T47D |
| PhytoCAT-801 | 4-vinylphenol (4VP) | Hedyotis diffusa | PI3K/AKT, p38 MAPK, NF-κB | C57BL/6 mice |
| PhytoCAT-804 | Saponin glycoside | Fagonia indica | PARP, Caspase 3 | MDA-MB-468, Caco-2, MCF-7 |
| PhytoCAT-815 | Protocatechuic acid (PCA) | Bauhinia variegata | NA | MCF-7, C-6, HCT-15 |
| PhytoCAT-824 | Descurainia sophia volatile oil | Descurainia sophia | NA | MCF-7, HeLa |
| PhytoCAT-827 | Galangin | Alpinia officinarum | STAT-3, p-JAK2, Bcl-2, Caspase 3, PARP, Ki67, Nrf2 , NQO-1, HO-1, GSTP1-1 | MDA-MB-231, MCF-7, HCT-116, HeLa, BT-474, MGC 803 |
| PhytoCAT-828 | 1'S-1'-acetoxyeugenol acetate | Alpinia conchigera | NA | MCF-7, HMEC |
| PhytoCAT-831 | Pinostrobin chalcone | Alpinia mutica | NA | KB, MCF-7, A549, Caski, HCT116, HT29 |
| PhytoCAT-832 | Eicosapentaenoic acid | Alpinia oxyphylla | NA | MCF-7 |
| PhytoCAT-833 | Alpha-Turmerone | Curcuma longa | NA | HepG2, MCF-7, MDA-MB-231 |
| PhytoCAT-834 | Terpecurcumin D | Curcuma longa | NA | MDA-MB-231, A549, HepG2 |
| PhytoCAT-835 | Terpecurcumin F | Curcuma longa | NA | MDA-MB-231, A549, HepG2 |
| PhytoCAT-836 | Terpecurcumin G | Curcuma longa | NA | MDA-MB-231, A549, HepG2 |
| PhytoCAT-837 | Bisabolocurcumin ether | Curcuma longa | p38, p53 | MDA-MB-231, A549, HepG2 |
| PhytoCAT-838 | Demethoxybisabolocurcumin ether | Curcuma longa | NA | MDA-MB-231, A549, HepG2 |
| PhytoCAT-840 | Curcumin | Curcuma longa | c-Myc, Cyclin D1, Bcl-2, ABCB1, ABCC1, ABCG2, CXCL1, CXCL2, CXCR4, PTEN, BMI1, EGFR, CRP, EZH2, FABP5, ABCB4, DYRK2, HR.SERPINE1, PGAP3, MAP3K1, MAPK1, TCF, MTOR, AKT1, BIRC5, CCND1 , NQO1, PRMT5, MEP50, AURKA, CDK2, CDK1, FOS, H2AX, KIF11, SOD2, STAT-3, TNF, APC, ARNT,AXIN1, HIAP1, CRAF1, TRAF6, CASP1, CASP2, CASP3, CASP4, HPRT, GADD45, MCL-1, NIP1, Bcl-2L2, TRAP3, GSTP1, DAXX, PIG11, UBC, PIG3, PCNA, CDC10, JNK1, RBP2, TRAIL, TNFR, AP13, IGFBP3, SARP3, PKB, IGFBP, CASP7, CASP9, TNFSF6, TRICK2A, CAS, TRAIL-R2, RATS1, hTRIP, TNFb, TNFRSF5, CASP9, COL4A1, DAXX, DVL2, ENPP2, ERP29, FASN, ISG15, MYBL1 , PDK1, VEGF-A, XIAP, PARP, HER-2, NF-kB, Caspase 3, Caspase 7, skp2, p27, Cadherin-11, Plasminogen | MDA-MB-231, MCF-7, MD-MB-468, AU565, HCT116, A549, A375, T47D, DLD-1,MDA-MB-435, breast cancer xenograft model |
| PhytoCAT-842 | [10]-gingerol | Zingiber officinale | NA | MDA-MB-231, MDA-MB-468, mouse (4T1, E0771), MCF-7, T47D |
| PhytoCAT-843 | Ginger polysaccharides | Zingiber officinale | NA | MCF-7, H1975, HCT116, MCF-7 |
| PhytoCAT-844 | 6-gingerol | Zingiber officinale | p53, Bax, Bcl-2, cyt-c | MDA-MB-231 and MCF-7 |
| PhytoCAT-850 | Minecoside | Veronica peregrina | CXCR4 | MDA‑MB‑231, PANC1, SW480, HCT116, A2780, U266, A549, MCF-7 |
| PhytoCAT-854 | Bruceae fructus oil (BO) | Brucea javanica | mTOR, 4E-BP1 | MDA-MB-231 and BT-20 / Female Balb/c nude mice |
| PhytoCAT-859 | Simalikalactone D | Simarouba tulae | NA | MDA-MB-435, MDA-MB-231, A2780CP20, 4T1, MCF10A, PC3, HCT-116, SH-SY5Y |
| PhytoCAT-861 | Lycium barbarum polysaccharides(LBGP-I-3) | Lycium barbarum | NA | MCF-7 |
| PhytoCAT-864 | Strophanthidin | Strophanthus kombe | MEK1, PI3K, AKT, mTOR, Gsk3α, β-catenin | MCF-7, A549, and HepG2 |
| PhytoCAT-866 | Viscosalactone B | Withania somnifera | EGFR, HER2, estrogen and NF-κB receptors | MCF-7, NCI-H460, HCT-116, SF-268 |
| PhytoCAT-878 | α-conidendrin | Taxus yunnanensis | p21 , Bcl-2, p53 , Bax, Caspase 3, Caspase 9, Cyclin D1, CDK4 | MCF-7 and MDA-MB-231 |
| PhytoCAT-883 | Gallic acid | Ceriops tagal | EGFR, Src, AKT/p65, MMP9 | HeLa, MDA-MB23, MCF-7 |
| PhytoCAT-886 | P. macrocarpa fruit ethyl acetate fraction (PMEAF) | Phaleria macrocarpa | Bax, Bid, Caspase 3, Caspase 8, cyt-c, p21, p27, p53, SMAC, Bcl-2, Bcl-w, XIAP, Survivin | MDA-MB-231 |
| PhytoCAT-889 | Petiolaticin A | Elaeocarpus petiolatus | NA | MDA-MB-468, MDA-MB-231, MCF-7, and SW48 |
| PhytoCAT-894 | Falcarinol | Chaerophyllum aureum | NA | MCF-7 |
| PhytoCAT-895 | Beta-carotene | Daucus carrota | AF040958, AK001555, g41894, hshsp90r, U83857, AB014509, AF126028, AF053641, AF117386, AF050127,NM_012177, humtopi, AJ250915, U37547, U78798, NM_004849, NM_005346, AF004711, NM_006595, NM_001418, AB015051 | MCF-7, MD-MB-231, HCT-116, AGS , NCI-H460 |
| PhytoCAT-897 | Asafoetida | Ferula assa-foetida | NA | 4T1 |
| PhytoCAT-918 | Ficus septica extract | Ficus septica | PARP | T47D |
| PhytoCAT-919 | Vanillic acid | Ficus septica | NA | MDA MB 468, HBL 100, PC3, MCF-7 |
| PhytoCAT-922 | Valeric acid | Valeriana officinalis | NA | MCF-7, MDA-MB-231, MCF-10A |
| PhytoCAT-927 | 1-O-trans-p-coumaroyl-2-O-trans-caffeoyl-α-L-rhamnopyranose | Premna odorata | c-met | MCF-7, BT-474 cells, and MDA-MB-468 |
| PhytoCAT-933 | Caffeic acid | Thalassodendron ciliatum | NA | MCF-7/Adr, MCF-7/wt, MDA-MB-231, T47D |
| PhytoCAT-934 | Thalassosterol | Thalassodendron ciliatum | NA | MCF-7 ,HeLa , HepG2 |
| PhytoCAT-936 | Cardamonin | Amomum subulatum | FOXO3a, p21, p27, Bim | MDA-MB 231 and MCF-7 |
| PhytoCAT-941 | Pothobanol | Pothos scandens | NA | T47D, MCF-7 |
| PhytoCAT-947 | Tinospora cordifolia extract | Tinospora cordifolia | NA | MDA-MB-231 and MCF-7 |
| PhytoCAT-949 | Oplopandiol | Oplopanax horridus | NA | MCF-7 (RPMI-1640), HCT-116 and SW-480 , IEC-6 |
| PhytoCAT-950 | Oplopandiol acetate | Oplopanax horridus | NA | MCF-7, HCT-116, SW-480 |
| PhytoCAT-951 | Oplopantriol A | Oplopanax horridus | NA | MCF-7, HCT-116, SW-480 |
| PhytoCAT-956 | 20(S)-25-methoxyl-dammarane-3beta, 12beta, 20-triol [20(S)-25-OCH3-PPD] | Panax notoginseng | NA | MCF-7, MDA-MB-468, A172 , T98G, HPAC, Panc-1, A549, H1299, H358, H838, LNCaP, PC3 |
| PhytoCAT-958 | Annomocherin | Annona cherimolia | NA | MCF-7, A-498 |
| PhytoCAT-959 | Annonacin | Annona cherimolia | Cyclin D1, Bcl-2, HIF-1 | MCF-7 xenografts in nude mice, MDA-MB-231, MCF-7, T47D |
| PhytoCAT-960 | Annomontacin | Annona cherimolia | NA | MDA-MB-231, MCF-7 |
| PhytoCAT-962 | Houttuyninum | Houttuynia cordata | ERK1/2, AKT | MDA-MB-468, BT-474, A431, N87 xenografts |
| PhytoCAT-986 | Trans-isoshinanolone | Diospyros shimbaensis | NA | MDA-MB-231 |
| PhytoCAT-987 | Cis-isoshinanolone | Diospyros shimbaensis | NA | MDA-MB-231 |
| PhytoCAT-998 | Methyl β-lilacinobioside | Caralluma retrospiciens | topo II | MCF-7 |
| PhytoCAT-1000 | Wedelolactone | Sphagneticola calendulacea | ERα, ERβ, SoX2, ABCG2 | NA |
| PhytoCAT-1003 | Cephalinone D | Cephalantheropsis gracilis | NA | MCF-7, NCI-H460, and SF-269 |
| PhytoCAT-1004 | Flavanthrin | Cephalantheropsis gracilis | NA | MCF-7, NCI-H460, and SF-270 |
| PhytoCAT-1018 | Ent-1β,3β,16β,17-tetrahydroxyatisane | Euphorbia fischeriana | NA | MCF-7, HepG-2 , SGC-7901 |
| PhytoCAT-1019 | Ent-1β,3α,16β,17-tetrahydroxyatisane | Euphorbia fischeriana | NA | MCF-7, HepG-2 , SGC-7901 |
| PhytoCAT-1024 | Epigallocatechin gallate (EGCG) | Limoniastrum guyonianum | EGFR, GOLM1,, FAS, ERα, PTEN, p21, Bax, p-PDK1, AKT, Cyclin D1, Bcl-2 | MDA-MB-231, 4T1, , MCF-7, MCF-7tam,Hs578T, T47D, WI38VA, Caco-2, Hs578T, SUM-149, SUM-190, BT-20, BT-549, MDA-MB-435, HFF |
| PhytoCAT-1037 | Achyrobichalcone | Achyrocline satureioides | Caspase 9, Caspase 3, Caspase 7 | MDA-MB-231 and MCF-12A |
| PhytoCAT-1043 | Artemisia herba alba extracts | Artemisia herba | NA | MCF-7, HeLa |
| PhytoCAT-1044 | Kigelia Africana, Ximenia Caffra and Mimusops Zeyheri Seed Oils | Kigelia Africana, Ximenia Caffra and Mimusops Zeyheri | CD62P, CD63 | MCF-7, MDA-MB-231 |
| PhytoCAT-1047 | Antrocamphin A | Taiwanofungus camphoratus | NA | MCF-7, Hep2, Hela |
| PhytoCAT-1053 | Ginnalin A | Acer rubrum | Cyclin A, Cyclin D1 | MCF-7, HCT-116 |
| PhytoCAT-1056 | Diallyl disulfide | Allium sativum | Bax, Bcl-2, Bcl-xL, Bcl-w | MCF-7 |
| PhytoCAT-1057 | Diallyl trisulfide | Allium sativum | Bcl-2, PARP, JNK | MCF-7 |
| PhytoCAT-1059 | γ-Tocotrienol | Amaranthus cruentus | Cyclin D1, CDK2, CDK4, CDK6, Rb, E2F1, p27, p16 | MCF-7, MDA-MB-231 |
| PhytoCAT-1060 | Gamma-linolenic acid (GLA) | Anemone cylindrica | Her-2/neu | BT-474, SK-Br3, MDA-MB-453, SK-OV3, NCI-N87 |
| PhytoCAT-1061 | Ferulic acid | Angelica sinensis | HER2, ESR1 | MCF-7, BT-474, MDA- MB-231, SKBR-3 |
| PhytoCAT-1062 | Alpha-lipoic acid | Arabidopsis thaliana | p27(kip1), Bax, Bcl-2 | MCF-7, SK-N-SH, Hela |
| PhytoCAT-1063 | 3,3'-diindolylmethane (DIM) | Arundo donax | FoxM1, CXCR4, CXCL12, p21, Cadherin-11, Plasminogen | MDA-MB-231, MCF-7, MDA-MB-468, SKBR-3, BALB/c mice, T47D, Saos2 |
| PhytoCAT-1064 | Desacetyl nimbinene (DAN) | Azadirachta indica | JNK, p38, SOD1, SOD2 | MCF-7, MDA-MB-231 |
| PhytoCAT-1067 | Allyl Isothiocyanate | Brassica nigra | TRPA1 | MCF-7, MDA-MB-231 |
| PhytoCAT-1068 | Broccoli sprouts (BSp) | Brassica oleracea | DNMT1, HDAC1 | PC3, BPH-1, LnCaP, MCF-7 |
| PhytoCAT-1070 | Cajanin stilbene acid | Cajanus cajan | MYC | MCF-7 |
| PhytoCAT-1071 | Calcitrinone A | Callistemon citrinus | NA | MDA-MB-231 |
| PhytoCAT-1076 | Capsicum annuum extract (CAP) | Capsicum annuum | VEGF | MCF-7, MDA-MB-231, MDA-MB-435 |
| PhytoCAT-1079 | 1-(4-hydroxy-2-methoxybenzofuran-5-yl)-3-phenylpropane-1,3-dione | Celosia argentea | NA | MCF-7, SiHa, HCT |
| PhytoCAT-1084 | Falcarindiol | Cnidium officinale | Bax , p53, Bcl-2 | MCF-7, HCT-116 |
| PhytoCAT-1090 | Cuscutic resinoside A | Cuscuta chinensis | NA | MCF-7, T47D |
| PhytoCAT-1097 | Syringin | Eleutherococcus senticosus | PARP, XIAP, MAP2K1, PIK3CA, HRAS, EGFR, Caspase3, and PTGS2 | MCF-7, MDA-MB-231 |
| PhytoCAT-1099 | Erucin | Eruca sativa | SOD1, ERK1, ERK2, Bax, Bcl-2, XIAP | MDA-MB-231, SKBR-3, T47D, MCF-7 |
| PhytoCAT-1101 | Dihydroconiferyl alcohol | Euterpe oleracea | NA | MCF-7 |
| PhytoCAT-1105 | Protocatechuic acid methyl ester | Euterpe oleracea | NA | MCF-7 |
| PhytoCAT-1109 | Tannic acid | Forsythia suspensa | CXCL12, CXCR4 | MCF-7, MDA-MB-231 |
| PhytoCAT-1112 | Ginkgolic acid C15:1 | Ginkgo biloba | FAS | MCF-7, A549, HL-60 |
| PhytoCAT-1113 | Ginkgolic acid C17:2 | Ginkgo biloba | FAS | MCF-7, A549, HL-60 |
| PhytoCAT-1114 | Ginkgolic acid C17:1 | Ginkgo biloba | FAS | MCF-7, A549, HL-60 |
| PhytoCAT-1115 | Ginkgolic acid C13:0 | Ginkgo biloba | uPA, PAI-1, CXCR4, MMP9 | MCF-7 and MDA-MB 231 |
| PhytoCAT-1122 | 2-Methoxyestrone | Imperata cylindrica | NA | BT-549, HT-29 |
| PhytoCAT-1123 | 11, 16-Dihydroxypregn-4-ene-3, 20-dione | Imperata cylindrica | NA | BT-549, HT-29 |
| PhytoCAT-1124 | Daucosterol linolenate (DLA) | Ipomoea batatas | Caspase 3, Caspase 9, PARP-1 , Ki67, VEGF, Bcl-2,Bax, Bcl-xL | MCF-7 xenograft in nude mice, MDA-MB-231, 4T1 |
| PhytoCAT-1126 | Regiolone | Juglans regia | NA | MCF-7, BHY |
| PhytoCAT-1128 | Effususin B | Juncus effusus | NA | SHSY-5Y, SMMC-7721, HepG2, Hela, and MCF-7 |
| PhytoCAT-1132 | Methyl jasmonate | Lonicera japonica | Caspase 3, PAL | MDA-MB-435, MCF-7, A549 |
| PhytoCAT-1133 | Cudraxanthone I | Maclura cochinchinensis | Caspase 3, Caspase 7, Caspase 8, Caspase 9 | MDA-MB-231 BCRP |
| PhytoCAT-1134 | Tetramethoxystilbene | Maclura pomifera | CYP1A1 , CYP1B1, Nqo1 , IL-8 | MCF-7 |
| PhytoCAT-1139 | Mango polyphenolics | Mangifera indica | PI3K, AKT, HIF-1α, VEGF mRNA, pAKT, AKT, pPI3K (p85), VEGF, NF-κB , NF-κB (p65), PARP | BT-474, xenografts in mice |
| PhytoCAT-1142 | Phenethyl Isothiocyanate | Nasturtium officinale | MTDH , CDH1, TSC2, sfRON | MCF-7, MDA-MB-231, PC-3, DU145, U87, HCT116, HepG2, SKBR-3 |
| PhytoCAT-1147 | Oleuropein | Olea europaea | CASP1, CASP14, FADD, TNFRSF21, GADD45A, CYCS, BNIP2, BNIP3, BID, BCL10, CFLAR, BFAR, BRAF, IAP, BIRC3, RIPK2, TNFRSF10A, CASP4, CASP6, PYD, PAYCARD, BIRC5, TNFRSF11B, HDAC2, HDAC3 | MDA-MB-468, MDA-MB-231, SKBR-3 |
| PhytoCAT-1148 | Ophiopogonin D | Ophiopogon japonicus | TGF-β1, ITGB1, MMP9, FAK, Src, AKT | MDA-MB-231, Hs 578Bst |
| PhytoCAT-1150 | Rh2 | Panax ginseng | Cyclin D3, CIP1, RNF217, RNA STXBP5-AS1 | MCF-7 |
| PhytoCAT-1155 | Pinolenic acid | Pinus koraiensis | COX-2 | MDA-MB-231 |
| PhytoCAT-1157 | Baneh gum | Pistacia atlantica | p53, Caspase 3 | MCF-7 |
| PhytoCAT-1168 | Amygdalin | Prunus spinosa | Bcl-2, PARP, Bax, Caspase 3, Survivin, XIAP, GAS5, MALAT1 | MDA-MB-231, Hs578T, MCF-7, HepG2 |
| PhytoCAT-1170 | Eleostearic acid (alpha-ESA) | Momordica charantia | HER2/HER3, PTEN | MDA-MB-231, SKBR-3, T47D |
| PhytoCAT-1173 | Rhus verniciflua Stokes extract (PPEF) | Rhus verniciflua | NA | MCF-7, MDA-MB-231, SKBR-3, AGS, SNU-668, SNU-638, A549, NCI-H157, HCT116, HepG2 |
| PhytoCAT-1190 | Eugenol | Syzygium aromaticum | LC3, NUp62, E2F1/survivin | MCF-7, HeLa, MDA-MB-231 |
| PhytoCAT-1194 | Chebulinic acid (CA) | Terminalia chebula | SOD1 | MDA-MB-231, MCF-7, S115, HOS-1, PC-3 |
| PhytoCAT-1198 | 23,24-Dihydrocucurbitacin B | Trichosanthes kirilowli | NA | Bcap37, HeLa, SW620, SMMC-7721, K562, MCF-7 |
| PhytoCAT-1204 | Prodelphinidin B-2 3,3'-di-O-gallate | Myrica rubra | p53, p21/WAF1 | MCF-7 |
| PhytoCAT-1205 | Jatamanvaltrate P | Valeriana jatamansi Jones | PARP, Cyclin B1, Cyclin D1, Cdc-2 | MCF-7, MDA-MB-231, MDA-MB-453, MDA-MB-468, MCF-10A |
| PhytoCAT-1207 | Linoleic acid | Vitex agnus-castus | BRCA1, ER | MDA-MB-231, MCF-7, mouse mammary tumor, T47D, Ishikawa cells |
| PhytoCAT-1210 | Withaferin A | Withania somnifera | STAT-3, Notch2, Notch 4, ATR, CHK1 | MCF-7, SUM159, MDA-MB-231 |
| PhytoCAT-1212 | 6-shogaol | Zingiber officinale (Ginger) | MT1-MMP, c-Src kinase, cortactin, JNK, NF-κB, STAT-3, CCL2, Aromatase | MDA-MB-231, A549 |
| PhytoCAT-1215 | Indole-3-carbinol | Brassica oleracea | BRCA1, EGFR , MUC1, BRCA1, BRCA2, p53, MDM2, GATA3, ERalpha | MDA-MB-231, T47D, MCF-7, MDA-MB-468, PC3, LNCaP, DU-145, 10AT-Her2, tumor xenograft |
| PhytoCAT-1216 | Daucosterol Linoleate | Ipomoea batatas | Ki67, VEGF, Bcl-2, PI3K/AKT/NF-kB, XIAP, Bax, Bad | MDA-MB-231, MCF-7, 4T1, MCF-7 xenograft nude mice |
| PhytoCAT-1227 | 10-O-acetylmacrophyllide | Rothmannia wittii | NA | MCF-7, NCI-H187 |
| PhytoCAT-1228 | Garjasmine | Rothmannia wittii | NA | MCF-7, NCI-H187 |
| PhytoCAT-1229 | 1,2,3,4,6-Penta-O-galloyl-β-d-glucose | Macaranga tanarins | Skp2, FoxO1, p27 | MDA-MB-231, BT-474 |
| PhytoCAT-1230 | Mimusops zeyheri seed oil | Mimusops zeyheri | CD62P, CD63 | MCF-7, MDA-MB-231 |
| PhytoCAT-1234 | Pinostilbene | Commiphora africana | NA | MCF-7, A549, PC3, HepG2 |
| PhytoCAT-1235 | 5-methoxy-(E)-resveratrol 3-O-rutinoside | Commiphora africana | NA | MCF-7, A549, PC3, HepG2 |
| PhytoCAT-1241 | Ximenia caffra seed oil | Ximenia caffra | CD62P, CD63 | MCF-7, MDA-MB-231 |
| PhytoCAT-1256 | Artahongkongene A | Artabotrys hongkongensis | NA | HL-60, SMMC-7721, A-549, MCF-7 and SW480 |
| PhytoCAT-1257 | Artahongkongene B | Artabotrys hongkongensis | NA | HL-60, SMMC-7721, A-549, MCF-7 and SW480 |
| PhytoCAT-1258 | Artahongkongene C | Artabotrys hongkongensis | NA | HL-60, SMMC-7721, A-549, MCF-7 and SW480 |
| PhytoCAT-1259 | Artahongkongene D | Artabotrys hongkongensis | NA | HL-60, SMMC-7721, A-549, MCF-7 and SW480 |
| PhytoCAT-1260 | Artahongkongene E | Artabotrys hongkongensis | NA | HL-60, SMMC-7721, A-549, MCF-7 and SW480 |
| PhytoCAT-1261 | Artahongkongene F | Artabotrys hongkongensis | NA | HL-60, SMMC-7721, A-549, MCF-7 and SW480 |
| PhytoCAT-1264 | Wedebicoside A | Wedelia biflora | NA | HeLa, MCF-7 and NCI-H460 |
| PhytoCAT-1265 | Wedebicoside B | Wedelia biflora | NA | HeLa, MCF-7 and NCI-H460 |
| PhytoCAT-1266 | Wedebicoside C | Wedelia biflora | NA | HeLa, MCF-7 and NCI-H460 |
| PhytoCAT-1267 | Wedebicoside E | Wedelia biflora | NA | HeLa, MCF-7 and NCI-H460 |
| PhytoCAT-1280 | Phaitanthrin A | Cephalantheropsis gracilis | NA | MCF-7, NCI-H460, and SF-268 |
| PhytoCAT-1282 | Condensed tannins | Phaseolus vulgaris | MMP2, MMP9, VEGF | HEL 299, Caco-2, MCF-7, Hs578T, DU 145 |
| PhytoCAT-1283 | Guggulsterone | Commiphora mukul | NA | MCF-7, MDA-MB-231, HMEC |
| PhytoCAT-1285 | 5-hydroxymethyl-2-furalclehyde | Ardisia Crenata | NA | MDA-MB-231 |
| PhytoCAT-1286 | n-butyl-alpha-D-fructofuranoside | Ardisia Crenata | NA | MDA-MB-231 |
| PhytoCAT-1311 | Khz (fusion of Ganoderma lucidum and Polyporus umbellatus) | Ganoderma lucidum and Polyporus umbellatus | Caspase 7, Caspase 8, Caspase 9 | MCF?7 |
| PhytoCAT-1317 | Phaleria macrocarpa extract (PMEAF) | Phaleria macrocarpa (Scheff) Boerl | Bax, Bid, Caspase 3, Caspase 8, cyt-c, p21, p27, p53, SMAC, Bcl-2, Bcl-w, XIAP, Survivin | MDA-MB-231 |
| PhytoCAT-1328 | PH-1 (4-methyl-5-oxo-tetrahydrofuran-3-yl acetate) | Polygonum hydropiper | NA | MCF-7, HeLA, NIH/3T3 |
| PhytoCAT-1329 | ChalcEA (2',4'-dihydroxy-6-methoxy-3,5-dimethylchalcone) | Eugenia aquea | ERα , Caspase 3 | T47D, A549, MCF-7. |
| PhytoCAT-1334 | Benzyl isothiocyanate | Cruciferous vegetables | STAT-3, XIAP, Caspase 9, Caspase 3, Caspase 8, Bax, Bcl-2, Bcl-xL, Bak, sfRON, MFN2, MAPK, JNK, p38, E-cadherin, Vimentin, Fibronectin, Notch2, FocO1, PUMA, Ron, AKT | MDA-MB-231, MCF-7, MCF-10A, MDA-MB-453, MDA-MB-361, Female athymic mice, SUM159, HCT-1, MCF-12A |
| PhytoCAT-1336 | Cedrelone | Toona ciliata, Trichilia catigua | EGFR, MMP9, MMP | HL-60, SMMC-7721, A-549, MCF-7, SW480, MDA-MB-231 |
| PhytoCAT-1349 | Gugulipid | Commiphora mukul | TCF-4, Cyclin D1, C-myc, Survivin | MCF-7, MDA-MB-231 |
| PhytoCAT-1357 | Purple-fleshed sweet potato (PFSP) Tainung 73 | Ipomoea batatas | NF-κβ, TNF-α, Caspase 3, IL-6 | MCF-7, SNU-1, WiDr |
| PhytoCAT-1366 | Artemisia annua herbal preparation | Artemisia annua | Caspase 3 | MDA-MB-231, MCF-7,MIA PaCa-2, PC-3, A459, MDA-MB-231 xenografts grown on CAM as well as in nude mice. |
| PhytoCAT-1370 | Melaleuca Alternifolia Concentrate | Melaleuca Alternifolia | Caspase 3, Caspase 7 | MCF-7, LNCaP |
| PhytoCAT-1372 | Antcin-A | Antrodia cinnamomea | p53, E-cadherin, occludin, N-cadherin, Vimentin, ZEB1 | MCF-7 and MDA-MB-231 |
| PhytoCAT-1396 | Periplorhamnoside | Antiaris toxicaria | NA | KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
| PhytoCAT-1398 | Strophanthidol | Antiaris toxicaria | NA | KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
| PhytoCAT-1399 | Cannogenol | Antiaris toxicaria | NA | KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
| PhytoCAT-1400 | Strophathojavoside | Antiaris toxicaria | NA | KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
| PhytoCAT-1401 | Strophalloside | Antiaris toxicaria | NA | KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
| PhytoCAT-1402 | Convalloside | Antiaris toxicaria | NA | KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
| PhytoCAT-1403 | Glucostrophalloside | Antiaris toxicaria | NA | KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
| PhytoCAT-1406 | Malayoside | Antiaris toxicaria | NA | KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
| PhytoCAT-1407 | Antialloside | Antiaris toxicaria | NA | KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
| PhytoCAT-1408 | Toxicarioside B | Antiaris toxicaria | NA | KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
| PhytoCAT-1423 | Lansiumarin C | Clausena hainanensis | NA | HL-60, SMMC-7721, A-549, MCF-7, SW480 |
| PhytoCAT-1424 | Lansiumarin A | Clausena hainanensis | NA | HL-60, SMMC-7721, A-549, MCF-7, SW480 |
| PhytoCAT-1426 | Claucoumarin D | Clausena hainanensis | NA | HL-60, SMMC-7721, A-549, MCF-7, SW480 |
| PhytoCAT-1427 | Melicotriphyllin A | Clausena hainanensis | NA | HL-60, SMMC-7721, A-549, MCF-7, SW480 |
| PhytoCAT-1428 | Melicotriphyllin C | Clausena hainanensis | NA | HL-60, SMMC-7721, A-549, MCF-7, SW480 |
| PhytoCAT-1433 | Artahainanol A | Artabotrys hainanensis | NA | HL-60, SMMC-7721, A-549, MCF-7, SW480 |
| PhytoCAT-1434 | Flexuvarol B | Artabotrys hainanensis | NA | HL-60, SMMC-7721, A-549, MCF-7, SW480 |
| PhytoCAT-1435 | Uvamalol C | Artabotrys hainanensis | NA | HL-60, SMMC-7721, A-549, MCF-7, SW480 |
| PhytoCAT-1436 | Flexuvarol A | Artabotrys hainanensis | NA | HL-60, SMMC-7721, A-549, MCF-7, SW480 |
| PhytoCAT-1449 | Capsanthin | Capsicum annuum | p53, Bax, Bcl-2, p-gp | MCF-7, MDA-MB-231, MDR-1 gene-transfected L1210 mouse lymphoma cells |
| PhytoCAT-1450 | Cryptoyunnane D | Cryptocarya yunnanensis | NA | A549, HCT-116, MDA-MB-231, PC-3, HeLa |
| PhytoCAT-1451 | Obolactone | Cryptocarya yunnanensis | NA | A549, HCT-116, MDA-MB-231, PC-3, HeLa |
| PhytoCAT-1452 | Cryptoyunnane A | Cryptocarya yunnanensis | NA | HCT-116, MDA-MB-231 and PC-3 |
| PhytoCAT-1453 | Cryptoyunnane B | Cryptocarya yunnanensis | NA | HCT-116, MDA-MB-231, PC-3 |
| PhytoCAT-1454 | 7',8'-Dihydroobolactone | Cryptocarya yunnanensis | NA | HCT-116, MDA-MB-231, PC-3 |
| PhytoCAT-1457 | Lupinalbin D | Ficus altissima | NA | HepG2, MCF-7, MDA-MB-231 |
| PhytoCAT-1461 | 20-O-salicyl-kidjoranin | Cynanchum wilfordii | NA | HL-60, MCF-7 |
| PhytoCAT-1462 | Rostratamin | Cynanchum wilfordii | NA | MCF-7 |
| PhytoCAT-1482 | Sulforaphane | Cruciferous vegetables (Brassica oleracea) | MMP7, MMP14, p38, Caspase 7, Bax, EMT, CR1, CRIPTO-3/TDGF1P3 (CR3, a homologue of CR1), Nanog, ALDH1A1, Wnt3, Notch4, KLF4, hTERT, CDKN2A, PTEN, RARbeta2, DNMT1, p53, p21, PBR, vimentin, Twist1, POU5F1, IL-1beta, IL-6, TNF-alpha, IFN-gamma,IL-4, PDGF, VEGF. | MCF-7, MDA-MB-231, SKBR-3, MCF-12A, HeLa |
| PhytoCAT-1483 | Antrodin C | Antrodia cinnamomea | E-cadherin, occludin, N-cadherin, Vimentin, MMP2, MMP9 | MCF-7 |
| PhytoCAT-1485 | Citracridone I | Citrus hystrix | NA | U87, A549, MCF-7 |
| PhytoCAT-1488 | Fresh Yellow Onion | Allium cepa | CEA, CA125 | NA |
| PhytoCAT-1489 | Ellagic acid | Rubus idaeus | CDK6, ACTN4, AKT/mTOR | MCF-7, HeLa, HUVEC, HEL 299, Caco-2, Hs 578T, DU 145, C32, A375 |
| PhytoCAT-1490 | Fucoidan | Brown algae | TGFRI and TGFRII proteins, Smad2/3, Smad4 , TGF?, Bid, Caspase 7, Caspase 8, Caspase 9, PARP | MDA-MB-231, MCF-7, T47D, 4T1 xenograft female Balb/c mice |
| PhytoCAT-1492 | α-linolenic acid | Linum usitatissimum (Flaxseed) | FAS, liver X receptor (LXR), and farnesoid X receptor (FXR) | TM2H, MCF-7, BT-474, MDA-MB-231, MDA-MB-468 |
| PhytoCAT-1495 | Nemorosone | Clusia rosea | ESR2, GRB7, MAPK3, MLH1, MYC, Notch1, PRDM2, THBS1, Tp53, VEGFA, APC, CCND1, CCNE1, ESR1, IGFBP3, KRT19, MKI6, MUC1, PG | MCF-7 BUS, MCF-7, MDA-MB-231 |
| PhytoCAT-1498 | Punicic acid | Punica granatum | NA | MDA-MB-231, MDA-ERalpha7, HepG2, Huh7, HT29 , HCT116, DU145 |
| PhytoCAT-1501 | Isolate f6l | Cassia alata | NA | MCF-7,a breast carcinoma, SKBR-3, another breast carcinoma, T24 a bladder carcinoma, Col 2, a colorectal carcinoma, and A549, a non- small cell lung adenocarcinoma. |
| PhytoCAT-1503 | Rosmarinic acid | Melissa officinalis, Rosemary plant Salvia officinalis | MDM2, ZEB1, ABCB1, PTEN, TWIST1, COX-2, Tyrosinase | MDA-MB-231, MCF-7, HCT116, NCI-H460, NCI-H460/R , MCR-5, NCI-H82, DU-145, Hep-3B, K-562, PC-3 |
| PhytoCAT-1505 | Sesamol | Sesamum indicum | pS2, GREB1, DNMT3A, DNMT3B, miR-370-3p | MDA-MB-231, HUVEC and Hs-578T cells. |
| PhytoCAT-1506 | Ergost-25-ene-3,6-dione,5,12-dihydroxy-,(5.alpha.,12.beta.) | Solanum torvum | BRCA1 | MCF-7 |
| PhytoCAT-1507 | Daucosterol | Pterospermum yunnanense | NA | MCF-7 and BHY |
| PhytoCAT-1508 | Oxyresveratrol | Artocarpus lakoocha Wall ex | Rad51 | MCF-7, HepG2, PC–3, RAW 264.7 and A–549 |
| PhytoCAT-1509 | Papain | Carica papaya | NA | MDA-MB-231, A2058, MCF-7 |
| PhytoCAT-1515 | Merulin C | Endophytic fungus of Xylocarpus granatum | NA | BT-474, SW621 |
| PhytoCAT-1516 | Rocaglamide | Aglaia odorata | NA | HL-60, SMMC-7721, A-549, MCF-7 and SW480 |
| PhytoCAT-1540 | Merulin A | Endophytic fungus of Xylocarpus granat | NA | BT-474, SW620 |
| PhytoCAT-1545 | Ouabain | Acokanthera oppositifolia, Acokanthera schimperi | NA | CasKi, SiHa and Hela, MDA-MB-321 and MCF-7, A549, SW480, HPAF-II |
| PhytoCAT-1546 | Oleamide | Moringa oleifera | Bcl-2 | MDA-MB-231 |
| PhytoCAT-1550 | Rhizoxin | Rhizopus chinensis | NA | B16 melanoma, M5076 sarcoma, LOX melanoma, MX-1 breast cancer, A549 |
| PhytoCAT-1553 | Beta-sitosteryl-3beta-glucopyranoside-6'-O-palmitate | Plumbago zeylanica | NA | MCF-7, Bowes |
| PhytoCAT-1558 | 11,11'-dideoxyverticillin | Shiraia bambusicola | EGFR, VEGFR-1/Flt-1, HER2/ErbB-2, Erk1/2, Flt-1, KDR/Flk-1 | MDA-MB-468, HUVEC, Mice |
| PhytoCAT-1561 | Glossogyne tenuifolia extract | Glossogyne tenuifolia | NA | MCF-7, MDA-MB-231, Hep G2, Hep 3B |
| PhytoCAT-1568 | Red grape wine extract (RWPF) | Vitis palmata | NA | MCF-7 |
| PhytoCAT-1570 | Salvianolic Acid B | Salvia miltiorrhizae Binge | Glutathione, TNF-?, MMP8, Cyclin D1, Ki67, Caspase 3, p53, COX-2 | MCF-7, ESC treated mice |
| PhytoCAT-1573 | White button mushroom | Agaricus bisporous | Bak-1 | MCF-7, MCF-10A, MDA-MB-231, BT-20 |
| PhytoCAT-1582 | Triphala | NA | p53 | HeLa, MCF-7, T47D, MD-MB-231 |
| PhytoCAT-1584 | Oleic acid | Olea europaea | Her-2/neu (erbB-2), BCRP, FAS | MCF-7, MDA-MB-231, SKBR-3, caco-2, A549 |
| PhytoCAT-1585 | Beta-Sitosterol | Styrax perkinsiae Gastrodia elata Blume Zanthoxylum nitidum Goniothalamus laoticus | Caspase 8, Caspase 9 | HT29, MCF-7, PC3, MDA-MB-231 and U-87 MG |
| PhytoCAT-1586 | 3,3',4,4',5,5'-hexahydroxystilbene (M8) | NA | p53, MnSOD | ZR-75-1, MDA-MB-231, T47D |
| PhytoCAT-1587 | Cotylenin A | NA | Cyclin G2, AKT, mTOR | MCF-7 and A549 |
| PhytoCAT-1588 | Rhodiola crenulata extract | Rhodiola crenulata | HIF1, MYCN | MDA-MB-231, mice bearing tumor graft, NB-1691 |
| PhytoCAT-1591 | Monosporasols A | Monosporascus eutypoides | NA | HeLa, HCT-8, A549, MCF-7 |
| PhytoCAT-1592 | Monosporasols B | Monosporascus eutypoides | NA | HeLa, HCT-8, A549, MCF-7 |
| PhytoCAT-1598 | Rukamtenol | Flacourtia rukam Zoll & Moritzi | NA | MDA-MB-231, HepG2, and RD |
| PhytoCAT-1599 | 7-octenoic acid | Moringa oleifera | Bcl-2 | MDA-MB-231 |
| PhytoCAT-1600 | 1-phenyl-2-pentanol | Moringa oleifera | Bcl-2 | MDA-MB-231 |
| PhytoCAT-1602 | 4-Acetylantroquinonol B (4-AAQB) | Antrodia camphorata | NA | MCF-7 |
| PhytoCAT-1604 | Novel cold-water-soluble polysaccharide (BEP) | Boletus edulis | Bax, Bcl-2, cyt-c, Caspase 3, Caspase 9 | MDA-MB-231 and Ca761 |
| PhytoCAT-1607 | Porphyridium cruentum sulfated polysaccharides | Porphyridium cruentum | IL-6, TNF-α | HTC-116, U-937, HL-60, MCF-7, NCI-H460, HGF-1/ male Balb/C mice |
| PhytoCAT-1608 | Hydroxyl safflower yellow B (HSYB) | NA | Caspase 9, Bax, Caspase 3 | MCF-7 |
| PhytoCAT-1609 | Quercetin 3-O-β-d-mannuronpyranoside | Callistemon viminalis | 5-LOX | MCF-7, HepG2 |
| PhytoCAT-1621 | Atraric acid (PF-2) | Pseudevernia furfuracea | NA | PA-1, MCF-7 |
| PhytoCAT-1624 | Sargassum angustifolium extract | Sargassum angustifolium | NA | HT-29, HeLa and MCF-7 |
| PhytoCAT-1625 | Sargassum oligocystum extract | Sargassum oligocystum | NA | HT-29, HeLa and MCF-7 |
| PhytoCAT-1626 | Sargassum boveanum extract | Sargassum boveanum | NA | HT-29, HeLa and MCF-7 |
| PhytoCAT-1628 | Indole[3,2-b] carbazole | Cruciferous vegetables | Vimentin, E-cadherin, MMP2, MMP9, FAK | MCF-7 and MDA-MB-231 |
| PhytoCAT-1630 | Violaxanthin | Dunaliella tertiolecta | NA | MCF-7, MDA-MB-231, A549 , LNCaP |
| PhytoCAT-1632 | 1-naphthyl isothiocyanate | Cruciferous vegetables | NA | MCF-7/Adr, MCF-7/wt |
| PhytoCAT-1633 | beta-phenethyl isothiocyanate | Cruciferous vegetables | NA | MCF-7/Adr, MCF-7/wt |
| PhytoCAT-1655 | Guizhi Fuling Decoction (GFD) | NA | HRAS, EGFR, PTK2, SOS1, ITGB1 | MDA-MB-231 |
| PhytoCAT-1656 | Matcha green tea (MGT) | NA | NA | MCF-7 |
| PhytoCAT-1657 | Pseurotin A | Aspergillus fumigatus | PCSK9 | BT-474, T47D |
| PhytoCAT-1659 | Qingdu granule (QDG) | QDG is composed of eleven herbs, such as Bupleuri Radix (Bupleurum chinense DC, root), Citri Reticulatae Pericarpium (Citrus reticulata Blanco, peel), Curcumae Radix (Curcuma wenyujin Y H Chen et Cing, root tuber), Sophorae Flos (Sophora japonica, flower), Moutan Cortex (Paeonia suffruticosa Andr, root bark), Arnebiae Radix (Arnebia euchroma (Royle) Johnst, root), Prunellae Spica (Prunella vulgaris, ear), Salviae Miltiorrhizae Radix et Rhizoma (Salvia miltiorrhiza Bge, root and rhizome), Curcumae Rhizoma (Curcuma phaeocaulis Val, root tuber), Astragali Radix (Astragalus membranaceus (Fisch) Bge var mongholicus (Bge) Hsiao, root), and Glycyrrhizae Radix et Rhizoma (Glycyrrhiza uralensis Fisch, root and rhizome) | VEGF, VEGFR2, NFATc3 | Breast cancer xenograft model |
| PhytoCAT-1661 | Antcamphin A | Antrodia camphorata | NA | MDA-MB-231, A549, HS68 |
| PhytoCAT-1662 | Antcamphin B | Antrodia camphorata | NA | MDA-MB-231, A549, HS68 |
| PhytoCAT-1663 | Antcamphin E | Antrodia camphorata | NA | MDA-MB-231, A549, HS68 |
| PhytoCAT-1664 | Antcamphin F | Antrodia camphorata | NA | MDA-MB-231, A549, HS68 |
| PhytoCAT-1665 | Antcamphin G | Antrodia camphorata | NA | MDA-MB-231, A549, HS68 |
| PhytoCAT-1666 | Antcamphin H | Antrodia camphorata | NA | MDA-MB-231, A549, HS68 |
| PhytoCAT-1667 | Antcamphin I | Antrodia camphorata | NA | MDA-MB-231, A549, HS68 |
| PhytoCAT-1668 | Antcamphin J | Antrodia camphorata | NA | MDA-MB-231, A549, HS68 |
| PhytoCAT-1669 | Antcamphin K | Antrodia camphorata | NA | MDA-MB-231, A549, HS68 |
| PhytoCAT-1670 | Antcamphin L | Antrodia camphorata | NA | MDA-MB-231, A549, HS68 |
| PhytoCAT-1671 | Pulveraven A | Pulveroboletus ravenelii | Caspase 8, Caspase 7, Bax, Bcl-2 | MCF-7 |
| PhytoCAT-1672 | Phoenix Dan Cong tea | Phoenix Dan Cong tea | NA | L02, WI38, MDA-MB-231, SW480, HepG2, HeLa |
| PhytoCAT-1673 | Luteolin and its oxidovanadium(IV) complex [VO(lut)(H2O)2]Na·3H2O (VOlut) | NA | NA | MDA-MB-231, CT26, A549, Balb/C mice |
| PhytoCAT-1675 | Maizediterpene B | Zea mays | NA | HCT-116, MDA-MB-23, SK-HEP-1 and SNU-638 |
| PhytoCAT-1677 | Icariol | Zea mays | NA | HCT-116, MDA-MB-23, SK-HEP-1 and SNU-640 |
| PhytoCAT-1678 | (-)-Oleocanthal (OC) | Olea europaea | EGFR | BT-474 and SKBR-3 |
| PhytoCAT-1680 | 2',3,4'-trimethoxy-5-hydroxy-trans-stilbene | Morus nigra | NA | MCF-7, HepG2 |
| PhytoCAT-1684 | Walnuts | NA | NA | NA |
| PhytoCAT-1689 | Scrophularia umbrosa Dumort extract | Scrophularia umbrosa Dumort | NA | MCF-7 |
| PhytoCAT-1691 | Evolvulin I | Evolvulus alsinoides | NA | MCF-7 |
| PhytoCAT-1692 | Cordycepin | Cordyceps militaris | NA | MCF-7 |
| PhytoCAT-1699 | Alysicarpus vaginalis extract | Alysicarpus vaginalis | Bax, Bcl-2, Bcl-xL, PARP-1 | Sprague-Dawley rats, MCF-7 and MDA-MB-453 |
| PhytoCAT-1701 | 4',6'-dihydroxy-2',4-dimethoxy-5'-(2″-hydroxybenzyl)dihydrochalcone | Cyathostemma argenteum | Caspase 3, Caspase 8, Caspase 9, ATM, ATR | MDA-MB-231 and MCF-7 |
| PhytoCAT-1703 | Unguinol | Aspergillus | Aromatase | MDA-MB-231 |
| PhytoCAT-1704 | Aspergillusidone D | Aspergillus | NA | MDA-MB-231 |
| PhytoCAT-1708 | Machilin D | Saururus chinensis | IL-6, IL-8, NF-κB | MCF-7, MDA-MB-231 |
| PhytoCAT-1716 | 2'-hydroxy-3',4',6'-trimethoxychalcone | Persicaria maculosa | NA | 4T1 |
| PhytoCAT-1718 | Pentadecanoic acid | Staphisagria macrosperma | Caspase 3, Caspase 7, caspase 8, caspase 9, β-catenin, MDR1, MRP1-and epithelial-mesenchymal transition (EMT) markers-snail, slug, MMP9, MMP2. | MCF-7, MDA-MB-231 |
| PhytoCAT-1719 | Aurovertin B | Calcarisporium arbuscular | DUSP1 | MDA-MB-231, MCF-7 |
| PhytoCAT-1721 | 4-hydroxyisophthalic acid (4-HIPA) | Decalepis hamiltonii | NA | MCF-7, MDA-MB-468, MCF-10 |
| PhytoCAT-1730 | Caffeic acid phenethyl ester (CAPE) | Propolis, Euonymus alatus (Winged Spindle Tree) | TLR4, MyD88, IRAK4, TRIF, NF-κB p65 | MDA-MB-231, MCF-7, Hs578T, HaCaT |
| PhytoCAT-1733 | Scutellaria litwinowii extract | Scutellaria litwinowii | NA | AGS, HeLa, MCF-7, PC12 and NIH 3T3 |
| PhytoCAT-1740 | Malabaricone C (mal C) | NA | NA | MCF-7 |
| PhytoCAT-1745 | Bromelain | Ananas comosus | NA | MCF-7 , KB, SK-MEL-28, GI-101A |
| PhytoCAT-1749 | Ethyl-beta-D-fructopyranoside | Ardisia Crenata | NA | NA |
| PhytoCAT-1750 | Syringic acid | Ardisia Crenata | NA | NA |
| PhytoCAT-1751 | n-butyl-beta-D-fructofuranoside | Ardisia Crenata | NA | NA |
| PhytoCAT-1752 | Methyl-alpha-D-fructofuranoside | Ardisia Crenata | NA | NA |
| PhytoCAT-1753 | (+)-Bergenin | Ardisia Crenata | NA | NA |
| PhytoCAT-1755 | Sartoryglabin B | Neosartorya glabra | NA | MCF-7, NCI-H460, A375-C5 |
| PhytoCAT-1756 | Androstan glycoside | Caralluma tuberculata | NA | MDA-MB-469 |
| PhytoCAT-1760 | (20R)-O-(3)-β-D-glucopyranosyl-(1→2)-α-L-arabinopyranosyl-pregn-5-en-3β,20-diol | Brucea javanica | NA | HL-60, SMMC-7721, A-549, MCF -7, SW480 |
| PhytoCAT-1762 | Longirostrerones A | Chaetomium longirostre | NA | MCF-7 |
| PhytoCAT-1763 | 1-benzyl-I3C | NA | CD40, CDK6 | MCF-7, MDA-MB-231 |
| PhytoCAT-1768 | Geranyl (3-GAP) | NA | p53, cyt-c, Bax, Caspase 3, Caspase 7, Caspase 9 | MCF-7, HT1080 |
| PhytoCAT-1773 | Strigolactones | NA | ATM, ATR, DNA-PKcs, PARP-1, RAD51 | NA |
| PhytoCAT-1774 | Schizophyllan | Schizophyllum commune | NA | Female adult swiss albino mice |
| PhytoCAT-1775 | 1-O-methyl-6-acetoxy-5-(pentadec-10Z-enyl)resorcinol | Labisia pumila | NA | PC3, HCT116 and MCF-7 |
| PhytoCAT-1776 | 1-O-methyl-6-acetoxy-5-pentadecylresorcinol | Labisia pumila | NA | PC3, HCT116 and MCF-7 |
| PhytoCAT-1783 | Tubeimu | Bolbostemma paniculatum | NA | MDA-MB-231, SKBR-3 |
| PhytoCAT-1794 | (-)-Gossypol-enriched cottonseed oil [(-)-GPCSO] | Gossypium herbaceum | Bcl-2 | MDA-MB-231, MCF-7 |
| PhytoCAT-1810 | Falcarindiol 3-acetate | Daucus carota | NA | HEK293 |
| PhytoCAT-1811 | Falcarindiol 3,8-diacetate | NA | NA | NA |
| PhytoCAT-1812 | Radix ranunculus ternati polysaccharides | Ranunculus ternatus Thunb | NA | MCF-7 |
| PhytoCAT-1815 | Desoxyrhaponticin | Rheum tanguticum Maxim ex Balf (rhubarb) | Fatty acid synthase (FAS) | MCF-7 |
| PhytoCAT-1816 | Rhaponticin | Rheum tanguticum Maxim ex Balf (rhubarb) | Fatty acid synthase (FAS) | MCF-7 |
| PhytoCAT-1818 | α-eleostearic acid (α-ESA) | Momordica charantia | Bcl-2, BAD, HER2, PTEN, HER3 | SKBR-3, T47D, MCF-7 |
| PhytoCAT-1823 | p-hydroxybenzoic acid | Tetrastigma hemsleyanum Honey | NA | MCF-7, HeLa |
| PhytoCAT-1827 | Tocopherols | Palm oil/Palm fruits | p21, p27, Caspase 3, peroxisome proliferator activated receptor-gamma, AKT, OCT4, CD44, SOX-2, trefoil factor (TFF)/pS2, cathepsin D, PR, SERPINA1 | MCF-7 and MDA-MB 231 |
| PhytoCAT-1831 | Ouregidione | Pseuduvaria trimera | NA | HepG2, MDA-MB-231 |
| PhytoCAT-1845 | Bisdemethylcurcumin | NA | NA | SKBR-3, MCF-7 |
| PhytoCAT-1846 | 3,5-bis((E)-3,4-dimethoxystyryl)isoxazole | NA | NA | SKBR-3, MCF-7 |
| PhytoCAT-1853 | Deacetyl-mycoepoxydiene | Plant endophytic fungi Phomosis sp | Caspase 3, Bax, Caspase 9, PARP, p21, Bcl-2 | MCF-7, nude mice with human breast carcinoma xenografts. |
| PhytoCAT-1855 | Indole diketopiperazines | Endophytic Chaetomium sp 88194 | NA | MCF-7 |
| PhytoCAT-1856 | (+)- altholactone | Goniothalamus elegants Ast | NA | KB, MCF-7 and NCI-H187 |
| PhytoCAT-1858 | Bruceine D | Brucea javanica | NA | MCF-7, MDA-MB-231, HS 578T |
| PhytoCAT-1859 | KTH-13-amine-monophenyl | Cordyceps bassiana | Caspase 3, Caspase 9, Caspase-3, Caspase 8, Caspase 9, Bcl-2 | MDA-MB-231,HeLa ,C6 glioma |
| PhytoCAT-1864 | Pelingo apple juice | Pelingo apple | p21, ERK1/2, LC3B | MCF-7 , MDA-MB-231 |
| PhytoCAT-1865 | Methyl caffeate | Solanum torvum | Bcl-2, Bid, Bax, cyt-c | MCF-7, A549, COLO320, HepG-2, Vero |
| PhytoCAT-1867 | Conjugated linoleic acid | Agaricus bisporous,Momordica charantia | LXR, PTPgamma, c-myc | MDA-MB-231, MCF-7, SG652, 639V, ADF, PC3, LNCaP, SK-HEP-1, HepG2, MCF-7aro, MDA-wt, MDA-ERalpha7, M21-HPB, HT-29 |
| PhytoCAT-1870 | Norstictic acid | Usnea strigosa | NA | MDA-MB-231 |
| PhytoCAT-1871 | Corilagin | Euphorbia fischeriana | Hes1, Notch1, mTOR | MCF-7, HepG2, CCA |
| PhytoCAT-1873 | Geraniin | Phyllanthus urinariainn Nephelium lappaceum | Bcl-2, PARP, Caspase 3 | MCF-7 |
| PhytoCAT-1874 | Cladosporium cladosporioides 2 | Vernonia amygdalina | NA | MCF-7 |
| PhytoCAT-1887 | 3,4-bis-3,4,5-trimethoxybenzylidene-dihydrofuran (BTMB) | Taiwania cryptomerioides | CDC2, Cyclin D1, Cyclin E | MDA-MB-468 |
| PhytoCAT-1889 | Polysaccharide SpaTA | Sparganii Rhizoma | ERα | ZR-75-1, MDA-MB-231 |
| PhytoCAT-1902 | Tetrandrine (Tet) | Radix stephaniae tetrandrae | NA | MDA-MB-231 |
| PhytoCAT-1903 | ω-Hydroxyundec-9-enoic acid (ω-HUA) | NA | p38 | MDA-MB-231, MDA-MB-435 |
| PhytoCAT-1904 | Pine honey | NA | NA | MCF-7, SKBR-3, MDA -MB - 231 |
| PhytoCAT-1905 | Cladosporol A | Cladosporium cladosporioides | p21 | MCF-7 |
| PhytoCAT-1910 | Isoschaftoside | Artemisia herba alba | NA | MCF-7, HeLa |
| PhytoCAT-1912 | 10-hydroxy camptothecin | Nothapodytes nimmoniana | p21 | MCF-7, BGC823 and HepG2 |
| PhytoCAT-1920 | Lentinan (LNT) | Lentinus edodes | p53, p-ERK1/2, cleaved-Caspase 3, PARP 1, MDM2, TERT, NF-κB (NF-κB) p65, Bcl-2, ERα, PI3K, p-AKT, mTOR | MCF-7 |
| PhytoCAT-1921 | Baker's yeast | Saccharomyces cerevisiae | NA | The metastatic murine 4T1 line, the murine Ehrlich ascites carcinoma (EAC) line, and the human breast cancer MCF-7 cell line. |
| PhytoCAT-1929 | Cis-khellactone | Angelica amurensis | VDAC1, Bax, Bak | MCF-7, MDA-MB-231, BT-20, BT-549, T47D, SKBR-3, MDA-MB-453, HS578T, MDA-MB-468, HCT116, HT-29, HeLa, SiHa, HEK293T, HEK293 |
| PhytoCAT-1934 | Vulpinic Acid | Candelaria concolor lichen | p53 | MCF-7, SKBR-3 |
| PhytoCAT-1942 | (E)-resveratrol 3-O-rutinoside | Commiphora africana | NA | MCF-7, A549, PC3, and HepG2 |
| PhytoCAT-1945 | Stigmasterol | Citrus hystrix Garcinia penangiana Decaschistia parviflora | NA | HT29, MCF-7, PC3, U-87 MG |
| PhytoCAT-1948 | 2'-Hydroxycinnamaldehyde | Cinnamomum cassia Blume | E-cadherin, KLF17, Id-1, EMT | MCF-7, T47D, MDA-MB-231, MDA-MB-435, mice model |
| PhytoCAT-1951 | Raspberry oil emulsion: cold pressed (ROCOP) | Rubus idaeus | NA | MCF-7, MCF-7/DX, A549, LoVo, LoVo/DX |
| PhytoCAT-1960 | 7-acetylaltholactone | Goniothalamus macrocalyx Ban | NA | KB, HepG2, Lu, MCF-7 |
| PhytoCAT-1961 | Pentagalloyl glucose | Quercus aliena | GRO-α/CXCL1, IƙBKE, MAPK, DR4, DR5, TNF | MDA-MB-468, MDA-MB-231 |
| PhytoCAT-1962 | Dihydrocapsaicin | Capsicum annuum. Zingiber officinale Roscoe | Caspase family CASP9, CASP3, Bax | MDA-MB-231 |
| PhytoCAT-1969 | Usnic Acid | Niebla homalea | hsa-miR-5006-5p, hsa-miR-892c-3p, hsa-miR-4430, hsa-miR-5194, hsa-miR-3198, hsa-miR-3171, hsa-miR-933, hsa-miR-185-3p | A2780, HeLa, MCF-7, SKBR-3, HT-29, HCT-116 p53(+/+), HCT-116 p53(-/-), HL-60 and Jurkat |
| PhytoCAT-1970 | Atranorin | Stereocaulon alpinum | NA | A2780, HeLa, MCF-7, SKBR-3, HT-29, HCT-116 p53(+/+), HCT-116 p53(-/-), HL-60 and Jurkat |
| PhytoCAT-1971 | Fumarprotocetraric acid | Cetraria islandica | NA | T-47D and Panc-1 |
| PhytoCAT-1972 | Gyrophoric acid | NA | NA | A2780, HeLa, MCF-7, SKBR-3, HT-29, HCT-116 p53(+/+), HCT-116 p53(-/-), HL-60 and Jurkat |
| PhytoCAT-1975 | Pheophorbide-a | Scutellaria barbata | JNK, ERK | MDA-MB-231 |
| PhytoCAT-1977 | 1,7-Bis(4-hydroxyphenyl)-1,4-heptadien-3-one | Viscum coloratum | NA | HeLa, SGC-7901, MCF-7, and U251 |
| PhytoCAT-1979 | Demethylzeylasteral (T-96) | Tripterygium wilfordii Hook F | Vimentin, fibronectin, α-SMA | MDA-MB-231, 4T1 mouse model |
| PhytoCAT-1980 | Maytansinoids | Putterlickia pyracantha | NA | NA |
| PhytoCAT-1985 | 2,3,5,4'-Tetrahydroxystilbene-2-O-β-d-glucoside (THSG) | Polygonum multiflorum Thunb. | Bax, Bcl-2, Caspase 3 | MCF-7, H1299 and LNC |
| PhytoCAT-1988 | Trans-anethole (TA) | Foeniculum vulgare | NA | NA |
| PhytoCAT-1989 | Macrooxazole C | Ethyl acetate (EtOAc) extracts of Phoma sp. JS0228 cultures, an endophytic fungus of Morus alba (M. alba) | NA | MCF-7, LNCaP |
| PhytoCAT-1990 | SANT, a novel Chinese herbal monomer combination | Astragaloside IV - Astragalus membranaceus, α-solanine - Solanum nigruminn, neferine - otus plumule, and 2,3,5,6-tetramethylpyrazine -igusticum | ATG16L1, ATG9B, ATG4D, HB-EGF, thrombospondin-2, amphiregulin, leptin, IGFBP-9, EGF, coagulation factor III, and MMP9, serpin E1, platelet factor 4 | MDA-MB-231 hpa (231-Hpa) and MDA-MB-231 mock (231-Mock), BALB/c nude mice |
| PhytoCAT-1994 | Pygenic acid A (PA) | Prunella vulgaris | cIAP1, cIAP2, Survivin, p21, Cyclin D1, p-STAT-3, HO-1, IRE1α, p-elF2α, LC3B I, LC3B II | MDA-MB-231 cells (human) and 4T1 cells (mouse) |
| PhytoCAT-1998 | Alternate C | Alternaria alternata, an endophyte isolated from Paeonia lactiflora. | NA | A-549, MDA-MB-231, MCF-7, KB, KB-VIN |
| PhytoCAT-1999 | 3-Deoxy-2β,16-dihydroxynagilactone E (B6) | Podocarpus nagi | JAK-2, IL-6, STAT-3 | MDA-MB-231, MDA-MB-468 |
| PhytoCAT-2002 | Phenyl glucuronide | Euclea crispa | Her2 | In-silico |
| PhytoCAT-2003 | Hydrocortisone acetate | Euclea crispa | Her2 | In-silico |
| PhytoCAT-2004 | 6-(4,6-dioxo-1,4,5,6-tetrahydropyrimidin-2-yl-amino)hexanoic acid trifluoroacetate | Euclea crispa | Her2 | In-silico |
| PhytoCAT-2006 | Artichoke Polyphenols | Cynara cardunculus | FEN1 | MCF-7, MDA-MB-231 |
| PhytoCAT-2008 | Bikaverin | Fusarium oxysporum EPH2RAA endophytic in Ephedra fasciculata | CK2 | MCF-7, A427, A431 |
| PhytoCAT-2020 | Physagulide P | Physalis angulate. | JNK | MDA-MB-231, MDA-MB-468 |
| PhytoCAT-2061 | 4-coumaric acid methyl ester | Punica granatum | ERα, ERβ, ERγ | In-silico |
| PhytoCAT-2062 | Ferutinin | Ferula ovina | NA | MCF-7, TCC, HFF3 |
| PhytoCAT-2063 | 7-hydroxy, 5-methoxy, methyl cinnamate (1) | Phyllostachys heterocycla var. pubescens | EGFR tyrosine kinase | MCF-7, HepG2 |
| PhytoCAT-2064 | Cercosporamide | Endophytic fungus Phoma species ZJWCF006 in Arisaema erubescens | NA | HT-29, SMMC-772, MCF-7, HL-60, MGC80-3, P388 |
| PhytoCAT-2067 | Senecio glaucus extract | Senecio glaucus. | NA | MCF-7, HepG2, A549 |
| PhytoCAT-2073 | Aspergillus nidulans extract | Endophytic fungus Aspergillus nidulans, associated with Nyctanthes arbor-tristisinn. | NA | MCF-7, NCI-H460, HeLa |
| PhytoCAT-2074 | Sterigmatocystin | Endophytic fungus Aspergillus nidulans, associated with Nyctanthes arbor-tristisinn. | NA | MCF-7, NCI-H460, HeLa |
| PhytoCAT-2079 | Polysaccharides from Taxus cuspidata | Taxus cuspidata | NA | MCF-7, HepG2 |
| PhytoCAT-2083 | Silvestrol | Aglaia foveolata | Cyclin B, Cyclin D | MDA-MB-435 |
| PhytoCAT-2085 | Polydatin (PD) | Polygonum cuspidatum | Creb, Cyclin D1 | MDA-MB-231, MCF-7 |
| PhytoCAT-2090 | 2',3,4',5,5'-pentahydroxy-cis-stilbene | Morus nigra. | NA | MCF-7, HepG2 |
| PhytoCAT-2094 | Albafuran C | Morus nigra. | NA | MCF-7, HepG2 |
| PhytoCAT-2109 | Ginsenoside Rp1 | Panax ginseng | IGF-1R | MDA-MB-231, MCF-7, T-47D |
| PhytoCAT-2158 | (+/-)-trans-3-(3,4-dimethoxyphenyl)-4-[(E)-3,4-dimethoxystyryl]cyclohex-1-ene | Zingiber cassumunar | P-gp | MCF-7/ADR |
| PhytoCAT-2165 | Scutellariae radix | Scutellaria baicalensis | BCRP, MRP2 | Rats |
| PhytoCAT-2168 | Extra-Virgin Olive Oil (EVOO) | Olea Europea | HER2, FASN | MCF-7, SKBR3 |
| PhytoCAT-2169 | Valtrate | Valeriana jatamansi Jones | p-Akt, Cyclin B1, Caspase 8, p21, p-cdc2, Caspase 3, Caspase 9, MMP-9, MMP-2, PARP | MCF-7, MDA-MB-231, MDA-MB-468, MDA-MB-453, MCF10A, SK-OV-3 |
| PhytoCAT-2170 | Spinasterol | Pueraria mirifica Pueraria lobata | ERα, ERβ | NA |
| PhytoCAT-2178 | (Z)-β-farnesene | Cedrelopsis grevei | NA | MCF-7 |
| PhytoCAT-2183 | Solanum indicum extract | Solanum indicum var. recurvatum | NA | NA |
| PhytoCAT-2188 | Pumpkin | Cucurbita maxima | NA | NA |