| PhytoCAT-ID | Phytochemical name or plant extracts | Source of phytochemicals or plant Extracts | Target gene or protein | Cell line/ mice model |
|---|---|---|---|---|
| PhytoCAT-1 | Limonin | Citrus limetta | VEGF, VEGFR2, STAT3, MMP9, miR-216a-3p, ABCG2 | MCF-7-Adr, MDA-MB-231, MCF-7 |
| PhytoCAT-3 | 25-O-acetylcimigenol-3-O-β-D-xylopyranoside | Cimicifuga yunnanensis | p53, Bax, Caspase 7 | MCF-7 , R-MCF-7 |
| PhytoCAT-4 | 23-O-acetylcimigenol-3-O-β-D-xylopyranoside | Cimicifuga yunnanensis | p53, Bax, Caspase 7 | MCF-7, R-MCF-7 |
| PhytoCAT-5 | 25-chlorodeoxycimigenol-3-O-β-D-xylopyranoside | Cimicifuga yunnanensis | p53, Bax, Caspase 7 | MCF-7, R-MCF-7 |
| PhytoCAT-6 | 25-O-acetylcimigenol-3-O-α-L-arabinopyranoside | Cimicifuga yunnanensis | p53, Bax, Caspase 7 | MCF-7, R-MCF-7 |
| PhytoCAT-27 | D Rhamnose β-hederin (DRβ-H) | Clematis ganpiniana | Apaf-1, cyt-c, Caspase 3, Caspase 9, miR-16, miR-23a, miR-24, miR-26a, miR-27a | MDA-MB-231, MCF-7/Doc, MCF-7/S |
| PhytoCAT-59 | Gedunin | Azadirachta indica | Hsp90 | MCF-7, SKBR-3 |
| PhytoCAT-60 | Nimbolide | Azadirachta indica | p21, Bax, Bad, Fas-L, TRAIL, FADDR, cyt-c, Bcl-2, Bcl-xL, Mcl-1, XIAP-1, pro-caspase 8, pro-caspase 3, integrin αV, integrin β3, ILK, FAK, PAK, DNMT-1, HDAC-6, miR-21, HOTAIR, H19, miR-148a/miR-152, PTEN, ABCB1/MDR1 mRNA, P-gp, HIF1α, FoxO1, MYC | MDA-MB-231, HCC38, HEK293T, MCF-7, HL-60, SMMC7721, A549, SW-480 |
| PhytoCAT-74 | Platycodin D (PD) | Platycodon grandiflorus | ASK1, PERK, eIF 2alpha, GRP78/Bip, CHOP/GADD153, Caspase 4 | MDA-MB-231, MCF-7 |
| PhytoCAT-75 | 18-hydroxydollabela-8(17)-ene | Cleome droserifolia | NA | MCF-7, HCT116 |
| PhytoCAT-79 | Demethylzeylasterone | Kokoona zeylanica | Topo II alpha | MCF-7 |
| PhytoCAT-82 | Triptolide | Tripterygium wilfordii | ADAM10, ATM, PARP-1, XRC1, RAD51, miR-146a, Bcl-2 family, RhoA, Rac1, PD-L1, CD206, Arginase 1, CD204, NF-κB, AP-1, MMP9, Notch-1, HES-1, HEY-1, DCLK1, ALDH1, CD133 | MCF-7, BT-20,MKN-45, MKN-7, KATO-III, HL-60 , MDA-MB-231, BT-474 |
| PhytoCAT-83 | Triptonide | Tripterygium wilfordii | SNAI1 | HCC1806, BT-549, MDA-MB-231 |
| PhytoCAT-86 | Coriolic acid | Salicornia herbacea | Nanog,Oct4, CD44, c-Myc | MDA-MB-231, MCF-7 |
| PhytoCAT-118 | Shionone | Aster poliothamnus | Caspase 3, Caspase 9, Bcl-2, Bax | SKBR-3, MB-157 |
| PhytoCAT-143 | Lupeol | Elephantopus scaber | Caspase 3, MMP9, MMP2, COX-2, NF-κB p65, Bcl-2, | MDA-MB-231, MCF-7, K 562, SW620, KATO-III, A-549, Hep-G2, Hep3B |
| PhytoCAT-164 | Paclitaxel | Taxus brevifolia | EF1a ,FOXO3a, Bcl-2 | MCF-7 |
| PhytoCAT-177 | Hinokitiol | Chamaecyparis obtusa | EGFR | AS-B244, MDA-MB-231 |
| PhytoCAT-181 | Casearin G | Casearia sylvestris | NA | PC-3, MCF-7 |
| PhytoCAT-197 | Gypenoside 5 | Gynostemma pentaphyllum | Tyrosine phosphatase 1B | MCF-7, MCF-7/ADR, MDA-MB-231 |
| PhytoCAT-198 | Gypenoside LI | Gynostemma pentaphyllum | ERCC6L | MCF-7, MDA-MB-231 |
| PhytoCAT-200 | Cucurbitacin B | Trichosanthes cucumerina | Cyclin D1, C-myc, β-catenin, F-actin, Vimentin, FAK, vinculin | SKBR-3, MCF-7 |
| PhytoCAT-202 | Bryonolic acid | Trichosanthes cucumerina | NA | SKBR-3, MCF-7, T47D, MDA-MB-435, A549, SK-LU1, Caco-2 |
| PhytoCAT-206 | Alisol A | Alisma plantago-aquatica | Cyclin D1, MMP2, MMP9 | MDA-MB-231 |
| PhytoCAT-224 | 3β,13β-dihydroxy-12,13-dihydrooleanolic acid (1) | Vitis vinifera | NA | MCF-7/DOX |
| PhytoCAT-226 | 3β,12β,13β-trihydroxy-12,13-dihydrooleanolic acid (2, TOA) | Vitis vinifera | NA | MCF-7/DOX |
| PhytoCAT-227 | 3β,13β-dihydroxy-12,13-dihydroursolic acid (7) | Vitis vinifera | NA | MCF-7/DOX |
| PhytoCAT-229 | 2-deacetoxytaxinine J (2-DAT-J) | Taxus baccata | NA | MCF-7, MDA-MB-231 |
| PhytoCAT-238 | Cimiracemoside A | Black cohosh | NA | MCF-7 |
| PhytoCAT-245 | Lycopene | Solanum lycopersicum | BRCA1, BRCA2 | MDA-MB-231, MCF-7, HT-29, T84 |
| PhytoCAT-246 | 3-O-α-L-arabinosyl oleanolic acid (3-O-L-AO) | Schumacheria castaneifolia | Bax, p53, Survivin, HIF-1α, HIF-2α | NA |
| PhytoCAT-257 | Hyperforin | Hypericum undulatum | ER1 | A431 ,SB1 ,SB3 ,MV3 ,1F6 ,HT144 ,Jurkat ,MCF-7 ,MDA-MB-468 ,SK-OV-3 |
| PhytoCAT-268 | Kongensin D (6) | Croton kongensis | AKT, p21, Cyclin B1, CDK1, Bcl-2, Bax, Caspase 3, PARP, β-catenin, MMP2, MMP9 | MDA-MB-231, MDA-MB-468, MCF-7, TNBC xenograft mouse model |
| PhytoCAT-269 | Euphoranginone D (3) | Croton kongensis | NA | MDA-MB-231, MDA-MB-468, MCF-7 |
| PhytoCAT-270 | Ent-kaurane-3-oxo-16β,17-diol (4) | Croton kongensis | NA | MDA-MB-231, MDA-MB-468, MCF-7 |
| PhytoCAT-271 | Ent-16β-H-3-oxokauran-17-ol (5) | Croton kongensis | NA | MDA-MB-231, MDA-MB-468, MCF-7 |
| PhytoCAT-272 | Kongeniod B (7) | Croton kongensis | NA | MDA-MB-231, MDA-MB-468, MCF-7 |
| PhytoCAT-273 | Kongensin A (8) | Croton kongensis | NA | MDA-MB-231, MDA-MB-468, MCF-7 |
| PhytoCAT-274 | Kongensin F (9) | Croton kongensis | NA | MDA-MB-231, MDA-MB-468, MCF-7 |
| PhytoCAT-275 | Crokongendin A (1) | Croton kongensis | NA | MDA-MB-231, MDA-MB-468, MCF-7 |
| PhytoCAT-276 | Crokongendin B (2) | Croton kongensis | NA | MDA-MB-231, MDA-MB-468, MCF-7 |
| PhytoCAT-277 | Laevifins A | Croton oblongus | NA | MCF-7 |
| PhytoCAT-278 | Laevifins B | Croton oblongus | NA | MCF-7 |
| PhytoCAT-279 | Laevifins G | Croton oblongus | NA | MCF-7 |
| PhytoCAT-281 | Resiniferatoxin | Euphorbia bicolor | NA | MDA-MB-231, MDA-MB-469 |
| PhytoCAT-282 | Ebracteolatain A | Euphorbia ebracteolata | NA | NA |
| PhytoCAT-283 | Jolkinolide B | Euphorbia fischeriana | Cyclin D1, Cyclin E, mTOR, PI3K, AKT, PTEN, eIF4E, β1-integrin, FAK, U0126, ERK | Female Balb/c nude mice, MCF-7, BT-474, MDA-MB-231 |
| PhytoCAT-284 | Euphorin C | Euphorbia fischeriana | NA | MCF-7 |
| PhytoCAT-285 | Euphorin E | Euphorbia fischeriana | NA | MCF-7 |
| PhytoCAT-286 | Euphorin H | Euphorbia fischeriana | NA | MCF-7 |
| PhytoCAT-287 | Ebractenoid C | Euphorbia fischeriana | NA | MCF-7 |
| PhytoCAT-288 | Ebractenoid F | Euphorbia fischeriana | NA | MCF-7 |
| PhytoCAT-289 | Yuexiandajisu E | Euphorbia fischeriana | NA | MCF-7 |
| PhytoCAT-290 | Ingenol-3-palmitate | Euphorbia fischeriana | NA | MCF-7 |
| PhytoCAT-291 | Ingenol-3- myristinate | Euphorbia fischeriana | NA | MCF-7 |
| PhytoCAT-292 | Ingenol-20-myristinate | Euphorbia fischeriana | NA | MCF-7 |
| PhytoCAT-293 | Jolkinol A | Euphorbia fischeriana | NA | MCF-7 |
| PhytoCAT-295 | Kopetdaghinane A | Euphorbia kopetdaghi | Bcl-2, Bax | MCF-7, OVCAR-3 |
| PhytoCAT-297 | Euphopubescenol | Euphorbia pubescens | NA | MCF-7, NCI-H460, SF-268 |
| PhytoCAT-298 | Euphopubescene | Euphorbia pubescens | NA | MCF-7, NCI-H460, SF-268 |
| PhytoCAT-299 | Euphosorophane A | Euphorbia sororia | NA | MCF-7/ADR |
| PhytoCAT-333 | Secofriedelanophyllemblicine | Phyllanthus emblica | NA | MCF-7 |
| PhytoCAT-355 | Friedelin | Garcinia penangiana | CDKN1a, pRb2, p53, Nrf2, Caspase 3, Bcl-2, mdm2, PCNA | MCF-7 |
| PhytoCAT-367 | Pristimerin | Reissantia buchananii | FASN | MDA-MB-231 |
| PhytoCAT-370 | Hyperelodiones A | Hypericum elodeoides | NA | HeLa, MCF-7 |
| PhytoCAT-371 | Hyperelodiones B | Hypericum elodeoides | NA | HeLa, MCF-7 |
| PhytoCAT-372 | Hyperelodiones C | Hypericum elodeoides | NA | HeLa, MCF-7 |
| PhytoCAT-375 | Crocin | Crocus sativus | ERα, HDAC2 | MKN-28, MCF-7, MDA-MB-231, Caco-2, BALB/c mice |
| PhytoCAT-376 | Ursolic acid | Prinsepia utilis | Fas receptor, Caspase 8, Caspase 3, Caspase 9, PARP, Bax, Bcl-2, cyt-c, Nrf2, NQO1, Keap1, miR-499a-5p, mTOR, AKT, MMP2, u-PA, NF-κB, Cyclin D, Cyclin E, CDK4, CDK2, PI3K, AKT, ERK, FoxO1/FoxO3a, DR4, DR5, Cyclin D1, PCNA, p21Waf1/Cip1, PLK1, CCNB1, ABCC1, MiR-186-5p, MAPK1/3, ABCG2 | A549, HCT116, MDA-MB-231, and CCRF-CEM, 4T1, ,MCF-7, BEL-7402, SPC-A-1, SGC-7901, HeLa, HT-29 , Caco-2, HepG2, HT-29, HDFn, SKBR-3, HeLa S3, KB, HL60, MDA-MB-468, Hep3B |
| PhytoCAT-381 | Ovatodiolide | Anisomeles indica | Oct4, Nanog, Hsp27, SMURF2 | AS-B145, BT-474 |
| PhytoCAT-382 | 2alpha-hydroxyursolic acid | Cunila lythrifolia | NF-κB | HepG2, MCF-7, Caco-2 |
| PhytoCAT-384 | Eriocalyxin B | Isodon eriocalyx | NF-κBp65, STAT-3 , Bax, Bcl-2, MMP, Caspase 3 | MCF-7, MDA-MB-231 / MDA-MB-231 xenograft model |
| PhytoCAT-391 | 14-Deoxy-11,12-didehydroandrographolide | Andrographis paniculata | GADD45A/p38 MAPK/DDIT3 | T-47D |
| PhytoCAT-392 | 1,8-cineole | Nepeta menthoides | NA | MCF-7, T47D, MDA-MB-231, A2780 |
| PhytoCAT-397 | Salvibuchanic acid | Salvia buchananii | NA | Jurkat, HeLa, MCF-7 |
| PhytoCAT-398 | Hyptadienic acid | Salvia buchananii | NA | Jurkat, HeLa, MCF-7 |
| PhytoCAT-399 | 7β-acetoxy-20-hydroxy-19,20-epoxyroyleanone (compound 1) | Salvia corrugata | ERK1/2 kinase | MCF-10A, SKBR-3, BT-474 |
| PhytoCAT-400 | 6,7-dehydroroyleanone (3) | Salvia deserta | NA | A549, MDA-MB-231, KB, KB-VIN, and MCF-7 |
| PhytoCAT-401 | 7-O-methylhorminone (5) | Salvia deserta | NA | A549, MDA-MB-231, KB, KB-VIN, and MCF-7 |
| PhytoCAT-402 | 14-deoxycoleon U (8) | Salvia deserta | NA | A549, MDA-MB-231, KB, KB-VIN, and MCF-7 |
| PhytoCAT-403 | Neotanshinlactone | Salvia digitaloides | NA | HL-60, SMMC-7721, A-549, SKBR-3, PANC-1 |
| PhytoCAT-405 | Tanshinone IIA | Salvia miltiorrhiza | LC3-II | MDA-MB-468, PC9, MCF-7, SKBR-3 |
| PhytoCAT-406 | 15,16-Dihydrotanshinone I | Salvia miltiorrhiza | ERp57 | MDA-MB-231 |
| PhytoCAT-409 | Cryptotanshinone | Salvia miltiorrhiza | p38/JNK, Erk1/2 | HepG2 , MCF-7, HA22T |
| PhytoCAT-411 | Sclareol | Salvia sclarea | IL-4, IFN-γ | MCF-7, breast-cancer-bearing Balb/c mice, HeLa |
| PhytoCAT-413 | Maslinic acid | Salvia tomentosa | NA | MDA-MB-231 |
| PhytoCAT-427 | Fraction 35 (F035) | Acacia victoriae | AKT | MDA-MB-453, MDA-MB-435 |
| PhytoCAT-440 | Glycyrrhizin | Glycyrrhiza glabra | NA | MDA-MB-231, HeLa, MCF-7 |
| PhytoCAT-441 | Glycyrrhetinic acid | Glycyrrhiza glabra | TOPO 2A | MDA-MB-231 |
| PhytoCAT-499 | erythrodiol-3-acetate (HU-1) | Humboldtia unijuga | Caspase 7 | MCF-7, A431 |
| PhytoCAT-504 | Cucurbitacin E | Hemsleya delavayi | Cyclin D1, Survivin, XIAP, Bcl-2, Mcl-1, JNK, AKT, ERK | MDA-MB-231, MDA-MB-468, SW527, MCF-7 |
| PhytoCAT-526 | β-amyrin | Vicia monantha | NA | MCF-7, HCT-116, HepG2 |
| PhytoCAT-565 | Corosolic acid | Lagerstroemia speciosa | NA | ACHN , A498, MDA-MB-231, SK-Hep1, Huh7, T47D, HT-29, K-562, MCF-7 |
| PhytoCAT-574 | Schisanol | Schisandra viridis | NA | MCF-7, CAL27, HEK293 |
| PhytoCAT-576 | Betulin | Hibiscus Syriacus | Bax, NOXA, PUMA, PERP, Bcl-x, TAp63, p21, Caspase 3, Bak, Caspase 7, Caspase 9, PARP | HBL-100, MDA-MB-231, H184B5F5/M10, MCF-7, K562, HeLa, HepG2, A549, SK-HEP-1, PC-3, NCI-H460 |
| PhytoCAT-579 | Angustifolianin | Aglaia angustifolia | NA | MCF-7 |
| PhytoCAT-581 | Aglaiabbreviatin E (AA-5) | Aglaia abbreviata | Caspase 9 | MCF-7, MCF-7/ADM |
| PhytoCAT-582 | Aglaiabbreviatin F (AA-6) | Aglaia abbreviata | Caspase 9, P-gp | MCF-7, MCF-7/ADM |
| PhytoCAT-584 | Amooranin | Amoora rohituka | Caspase 8 | MCF-7, MCF-7/TH, MCF-10A |
| PhytoCAT-587 | Toosendanin (TSN) | Melia azedarach | ABCB1, PI3K P110α, P110β, Procaspase 3, Procaspase 9, Bcl-xL, LC3B, Beclin-1, PI3K | MDA-MB-231, BT-549, 4T1 xenograft tumor |
| PhytoCAT-588 | Isotoosendanin (ITSN) | Melia azedarach | Procaspase 3, Procaspase 10, Bcl-xL, Beclin-1, LC3B | MDA-MB-231, BT-549, 4T1 xenograft tumor |
| PhytoCAT-593 | Azadirone | Turraea nilotica Turraea robusta | NA | 4T1, HEp2, Vero |
| PhytoCAT-594 | 12α-acetoxy-7-deacetylazadirone | Turraea nilotica Turraea robusta | NA | 4T1, HEp2, Vero |
| PhytoCAT-595 | Mzikonone | Turraea nilotica Turraea robusta | NA | 4T1, HEp2, Vero |
| PhytoCAT-596 | Azadironolide | Turraea robusta | NA | 4T1, HEp2, Vero |
| PhytoCAT-597 | 11-epi-Toonacilin | Turraea robusta | NA | 4T1, HEp2, Vero |
| PhytoCAT-627 | AG36 | Ardisia gigantifolia | Cyclin B1, Cyclin D1, FAK, AKT, VEGF, VEGFR2, Caspase 3, Caspase 8, Bax, Bcl-2, Fas, FasL, TNFR1, DR5, cyt-c | MCF-7, MDA-MB-231, SKBR-3, BALB/c nude mice |
| PhytoCAT-655 | Pseudolaric acid B | Pseudolarix kaempferi | HIF-1α, Caspase 8, Caspase 9, Cyclin B1 | MDA-MB-468, MDA-MB-435, L929, MRC5, SW579, MCF-7 |
| PhytoCAT-687 | Esculentoside A | Phytolacca acinosa | ALDH1A1, Sox2, Oct4, Bax, Caspase 3, Bcl-2, STAT3 | BALB/c mice, MCF-7 |
| PhytoCAT-719 | Saxifragifolin C | Androsace umbellata | p38 MAPK, ERK 1/2, JNK | MCF-7, MDA-MB-231 |
| PhytoCAT-721 | Delcosine | Aconitum barbatum Aconitum napellus Aconitum yesoense | NA | MCF-7, MDA-MB-231, A549, DU145,KB |
| PhytoCAT-722 | Sinchiangensine A | Aconitum sinchiangense | NA | HL-60, A-549, SMCC-7721, MCF-7 and SW480 cell line. |
| PhytoCAT-723 | Actein | Cimicifuga foetida | VEGFR1, pJNK, pERK | MCF-7, MDA-MB-361,SKBR-3, HT29, HepG2 and MKN28 / mouse xenograft model |
| PhytoCAT-724 | Cimicifoetiside A | Cimicifuga foetida | NA | MDA-MB-A231 |
| PhytoCAT-725 | Cimicifoetiside B | Cimicifuga foetida | NA | MDA-MB-A231 |
| PhytoCAT-726 | 23-epi-26-deoxyactein | Cimicifuga yunnanensis | NA | MCF-7, MDA-MB 231, SK-BR3 |
| PhytoCAT-727 | Cimigenol | Cimicifuga yunnanensis | NA | MCF-7, MDA-MB 231, SK-BR3 |
| PhytoCAT-747 | Ent-Kaur-16- en-19-oic acid | Annona senegalensis | NA | MCF-7 |
| PhytoCAT-756 | 3β-trans-cinnamoyloxy-2α-hydroxy-urs-12-en-28-oic acid (CHUA) | Malus pumila | Bax, Bcl-2, cyt-c, Bcl-xL | MDA-MB-231, MCF-7, HepG2, Caco-2, HeLa, A549/ old female nude mice (Balb/c-nu/nu) |
| PhytoCAT-758 | 13-methoxy-15-oxozoapatlin | Parinari curatellifolia | NA | ZR-75-1, Athymic mice carrying KB cells |
| PhytoCAT-770 | Ziyuglycoside II | Sanguisorba officinalis | Bax, Fas/FasL, Bcl-2, EMT | MCF-7 and MDA-MB-231 |
| PhytoCAT-775 | 3β, 6β, 19α, 24-tetrahydroxy-urs-12-en-28-oic acid | Mitragyna diversifolia | NA | MCF-7, HT-29 |
| PhytoCAT-776 | Rotundic acid | Mitragyna diversifolia | NA | MCF-7, HT-29 |
| PhytoCAT-777 | 23-nor-24-exomethylene- 3β, 6β, 19α-trihydroxy-urs-12-en-28-oic acid | Mitragyna diversifolia | NA | MCF-7, HT-29 |
| PhytoCAT-805 | Quinovic acid | Fagonia indica | Caspase 3, Caspase 8, PARP | NA |
| PhytoCAT-810 | Lanostane | Lyonia ovalifolia | Bax, Bcl-2 | SKBR-3, MB-157 |
| PhytoCAT-822 | Alpha-Santalol | Santalum album | NA | MDA-MB 231, MCF-7 |
| PhytoCAT-841 | Xanthorrhizol | Curcuma xanthorrhiza | Bcl-2, p53, PARP-1, pS2 | MDA-MB-231 and MCF-7 |
| PhytoCAT-845 | 6-methoxy-2E,9E-humuladien-8-one | Zingiber zerumbet | NA | MDA-MB-231 |
| PhytoCAT-846 | Zerumbone | Zingiber zerumbet | Bax, Caspase 7, Caspase 9, Bcl-2 | MCF-7 |
| PhytoCAT-847 | Melognine | Melodinus fusiformis | Caspase 3, p53, Bcl-2 | BT-549 |
| PhytoCAT-849 | 2,3-seco-taraxer-14-en-2,3-lactone (pycanocarpine) | Pleiocarpa pycnantha | NA | MCF-7 |
| PhytoCAT-852 | Bruceantin | Brucea javanica | NA | MCF-7, Lu1, LNCaP |
| PhytoCAT-868 | Pomolic acid | Euscaphis japonica | NA | Human breast cancer cells, MCF-7 and MDA-MB-231, and human umbilical vascular endothelial cells (HUVEC). |
| PhytoCAT-880 | Oleiferoside B | Camellia oleifera | NA | MCF-7, SMMC-7721 |
| PhytoCAT-892 | Saikosaponin A | Bupleurum chinense | VEGFR2, PLCγ1, FAK, Src, AKT | 4T1, MCF-7, HCT-15, AGS, HepG2 |
| PhytoCAT-899 | Conferone | Ferula gummosa | NA | MCF-7/Dox |
| PhytoCAT-900 | Feselol | Ferula gummosa | NA | MCF-7/Dox |
| PhytoCAT-903 | Galbanic acid | Ferula szowitsiana | NA | MCF-7 |
| PhytoCAT-928 | Icetexane-1 | Premna tomentosa | NA | MCF-7, HT-29, Hep-G2, A-431, and A-549 |
| PhytoCAT-929 | Icetexatriene-3 | Premna tomentosa | NA | MCF-7, HT-29, Hep-G2, A-431, and A-549 |
| PhytoCAT-952 | Panaxydol | Panax ginseng | EGFR | MCF-7 , PC3 and Renca mouse renal cancer cells |
| PhytoCAT-953 | Micranthin B | Isodon lophanthoides | NA | MCF-7, A549, HeLa |
| PhytoCAT-955 | Oridonin | Isodon rubescens | Bcl-2, Caspase 3, PARP, AKT | MDA-MB-231 , MCF-7, A375-S2 |
| PhytoCAT-963 | Solajiangxin I | Solanum lyratum | NA | MCF-7, HCT-8, A-549, SGC-7901 and BEL-7402 |
| PhytoCAT-964 | 7-Hydroxylsolajiangxin I | Solanum lyratum | NA | MCF-7, HCT-8, A-549, SGC-7901 and BEL-7402 |
| PhytoCAT-965 | Solajiangxin H | Solanum lyratum | Bcl-2, Survivin, Bcl-2-like 4, Caspase 3, c-Caspase 9 | MCF-7, HCT-8, A-549, SGC-7901 and BEL-7402 |
| PhytoCAT-966 | Lyratol D | Solanum lyratum | B-cell lymphoma (Bcl)-2, Survivin, Bcl-2-like protein 4, (c)-Caspase 3, c-Caspase 9 | MCF-7, HCT-8, A-549, SGC-7901 and BEL-7402 |
| PhytoCAT-967 | Dehydrovomifoliol | Solanum lyratum | NA | MCF-7, HCT-8, A-549, SGC-7901 and BEL-7402 |
| PhytoCAT-968 | Blumenol A | Solanum lyratum | NA | MCF-7, HCT-8, A-549, SGC-7901 and BEL-7402 |
| PhytoCAT-969 | Solajiangxin A | Solanum lyratum | NA | MCF-7, HCT-8, A-549, SGC-7901 and BEL-7402 |
| PhytoCAT-970 | Solajiangxin B | Solanum lyratum | NA | MCF-7, HCT-8, A-549, SGC-7901 and BEL-7402 |
| PhytoCAT-971 | Solajiangxin C | Solanum lyratum | NA | MCF-7, HCT-8, A-549, SGC-7901 and BEL-7402 |
| PhytoCAT-972 | Solajiangxin D | Solanum lyratum | NA | MCF-7, HCT-8, A-549, SGC-7901 and BEL-7402 |
| PhytoCAT-973 | Solajiangxin E | Solanum lyratum | NA | MCF-7, HCT-8, A-549, SGC-7901 and BEL-7402 |
| PhytoCAT-974 | 2-Hydroxysolajiangxin E | Solanum lyratum | NA | MCF-7, HCT-8, A-549, SGC-7901 and BEL-7402 |
| PhytoCAT-975 | Lyratol A | Solanum lyratum | NA | MCF-7, HCT-8, A-549, SGC-7901 and BEL-7402 |
| PhytoCAT-976 | Lyratol B | Solanum lyratum | NA | MCF-7, HCT-8, A-549, SGC-7901 and BEL-7402 |
| PhytoCAT-977 | Lyratol C | Solanum lyratum | NA | MCF-7, HCT-8, A-549, SGC-7901 and BEL-7402 |
| PhytoCAT-995 | Methyl angolensate | Soymida febrifuga | KU70, KU80 | T47D |
| PhytoCAT-1006 | Julibroside (J29) | Albizia julibrissin | NA | MDA-MB-435, PC-3M-1E8, HeLa |
| PhytoCAT-1007 | Julibroside (J30) | Albizia julibrissin | NA | MDA-MB-435, PC-3M-1E8, HeLa |
| PhytoCAT-1008 | Julibroside (J31) | Albizia julibrissin | NA | MDA-MB-435, PC-3M-1E8, HeLa |
| PhytoCAT-1009 | Voacamine | Voacanga africana | NA | MDA-MB-231, HEPG-2, A375, SH-SY5Y, CT26 |
| PhytoCAT-1010 | 19-epi-voacristine | Voacanga africana | NA | MDA-MB-231, HEPG-2, A375, SH-SY5Y, CT26 |
| PhytoCAT-1011 | Vobasine | Voacanga africana | NA | MDA-MB-231, HEPG-2, A375, SH-SY5Y, CT26 |
| PhytoCAT-1012 | Voacristine | Voacanga africana | NA | MDA-MB-231, HEPG-2, A375, SH-SY5Y, CT26 |
| PhytoCAT-1013 | Galanal A | Boesenbergia rotunda | NA | MCF-7, LK-2, A549, ECC4, HeLa, DU145 |
| PhytoCAT-1014 | Galanal B | Boesenbergia rotunda | NA | MCF-7, LK-2, A549, ECC4,HeLa, DU145 |
| PhytoCAT-1015 | Voacangine | Voacanga africana | NA | MDA-MB-231, HEPG-2, A375, SH-SY5Y, CT27 |
| PhytoCAT-1021 | Ginsenoside Rg3 | Panax ginseng | CXCR4, STXBP5-AS1, RFX3-AS1 , EEF2, MYCBP2, STXBP5, GRM1, RFX3, SLC1A1, WT1 | MDA-MB-231, MCF-7, MCF-10A |
| PhytoCAT-1035 | Grifolin | Albatrellus confluens | Bax, Bcl-2, Caspase 8, Caspase 9, Caspase 3, DAPK1 | MCF-7, HL-60, SMMC-7721, A-549 |
| PhytoCAT-1041 | Ziyuglycoside I | Sanguisorba officinalis | p53, p21WAF1, Bax, Bcl-2 | MDA-MB-231 |
| PhytoCAT-1045 | Camphoratin F | Taiwanofungus camphoratus | NA | MCF-7, Hep2, Hela |
| PhytoCAT-1046 | Camphoratin E | Taiwanofungus camphoratus | NA | MCF-7, Hep2, Hela |
| PhytoCAT-1048 | Antcin A | Taiwanofungus camphoratus | NA | MCF-7, Hep2, Hela |
| PhytoCAT-1050 | (6S,9S)-roseoside | Abutilon theophrasti | NA | MCF-7 |
| PhytoCAT-1072 | Sasanquasaponin (SQS) | Camellia oleifera | p21, Cyclin D1 | MCF-7, HepG2 |
| PhytoCAT-1075 | Δ9-tetrahydrocannabinolic acid | Cannabis sativa | NA | MDA-MB-231, HCT-116 |
| PhytoCAT-1077 | Chestnoside B | Castanea sativa | NA | MCF-7, PC3 |
| PhytoCAT-1081 | 25-O-acetyl-7,8-didehydrocimigenol-3-O-β-d-(2-acetyl)xylopyranoside (ADHC-AXpn) | Cimicifuga foetida | ERK1, ERK2, Raf,AKT | MCF-7, HepG2, HepG2/ADM, HeLa,PC3 |
| PhytoCAT-1085 | Kahweol | Coffea arabica | PEA3, AP-2, FASN, SREBP-1c, mTOR | SKBR-3 |
| PhytoCAT-1088 | Cucumol B | Cucumis melo | NA | SKOV-3, MCF-7, and HCT-116 |
| PhytoCAT-1108 | Farnesiferol A | Ferula persica | NA | MCF-7 |
| PhytoCAT-1120 | Phytoene | Hibiscus syriacus | NA | T47D, MCF-7, ECC-1 |
| PhytoCAT-1159 | Aucubin | Plantago media | NA | MCF-7, MDA-MB-231, HeLaS3, A549, and KB |
| PhytoCAT-1167 | Betulinic acid | Prunus dulcis | GRP78, NOP2, p120, WDR12, S6 ribisomal protein, p21 | MCF-7, HepG2, A549, HL-60,HCT-116, PC-3, HeLa |
| PhytoCAT-1169 | 3beta-trans-p-coumaroyloxy-2alpha-hydroxyolean-12-en-28-oic acid | Psidium guajava | NA | MCF-7, HepG2, Caco-2 |
| PhytoCAT-1174 | Carnosic acid | Rosmarinus officinalis | AKR1C2, TNXRD1, HMOX1, GDF15, PHLDA1, DDIT3, ID3, CDKN2C, Cyclin B1 | MDA-MB-453, NCI-H82 , DU-145 , Hep-3B , K-562 , MCF-7, PC-3, MDA-MB-231 |
| PhytoCAT-1175 | Carnosol | Rosmarinus officinalis | STAT-3, MMP9, Cyclin B1 | MDA-MB-231, Hs578T, MCF-7,T47D |
| PhytoCAT-1176 | Bigelovii A | Salicornia bigelovii | Bcl-2, Cyclin D1, NF‑κB‑regulated gene products, Cyclin D1, COX‑2 | MDA‑MB‑231, MDA‑MB‑468HL-60, MCF-7, HepG2, A549 |
| PhytoCAT-1177 | 3β-[(α-L-arabinopyranosyl)oxy]-19α,23-dihydroxyolean-12-en-28-oic acid 28-[6-O-acetyl-β-D-glucopyranosyl] ester | Sanguisorba officinalis | NA | MCF-7, HeLa, HepG2, SGC-7901, NCI-H460, and BGC-823 |
| PhytoCAT-1178 | 2α,3β,19α,23-tetrahydroxyurs-12-en-28-oic acid 28-[6-O-acetyl-β-D-glucopyranosyl] ester | Sanguisorba officinalis | NA | MCF-7, HeLa, HepG2, SGC-7901, NCI-H460, and BGC-823 |
| PhytoCAT-1179 | 3β-[(α-L-arabinopyranosyl)oxy]-19α-hydroxyurs-12,20(30)-dien-28-oic acid 28-[6-O-acetyl-β-D-glucopyranosyl] ester | Sanguisorba officinalis | NA | MCF-7, HeLa, HepG2, SGC-7901, NCI-H460, and BGC-823 |
| PhytoCAT-1185 | Scutebata A | Scutellaria barbata | NA | MCF-7, LoVo, SMMC-7721, HCT-116 |
| PhytoCAT-1191 | Tagetone A | Tagetes minuta | NA | MCF-7 and A549 |
| PhytoCAT-1193 | Arjunolic acid (AA) | Terminalia arjuna | NA | MCF-7, HeLa |
| PhytoCAT-1195 | Epoxy clerodane diterpene (ECD) | Tinospora cordifolia | Bax, Caspase 3, Caspase 8, Caspase 9, p21, Bcl-2, mdm2, PCNA | MCF-7 |
| PhytoCAT-1199 | Cucurbitacin D | Trichosanthes kirilowli | STAT-3 | MDA-MB-231 |
| PhytoCAT-1201 | Celastrol | Tripterygium wilfordii Hook F | CXCR4, NF- kB, MMP9, DCLK1, ALDH1, CD133 | MDA-MB-231, MCF-7 |
| PhytoCAT-1214 | Jujuboside B | Zizyphus jujuba | PARP, Caspase 3, LC3-II | MDA-MB-231 and MCF-7 xenografts |
| PhytoCAT-1226 | Genipin | Rothmannia wittii | UCP2 | MCF-7, MDA-MB-231, NCI-H187, T47D |
| PhytoCAT-1237 | Salvisertin A | Salvia deserta | NA | A549, MDA-MB-231, KB, KB-VIN, and MCF-7 |
| PhytoCAT-1238 | Horminone | Salvia deserta | NA | A549, MDA-MB-231, KB, KB-VIN, and MCF-7 |
| PhytoCAT-1239 | Sugiol | Salvia deserta | NA | A549, MDA-MB-231, KB, KB-VIN, and MCF-7 |
| PhytoCAT-1240 | Demethylcryptojaponol | Salvia deserta | NA | A549, MDA-MB-231, KB, KB-VIN, and MCF-7 |
| PhytoCAT-1242 | Zantholic acid | Zanthoxylum zanthoxyloides | NA | WRL-68, CaCO2, MCF-7, PC-3 |
| PhytoCAT-1251 | Scutestrigillosins A | Scutellaria strigillosa | NA | HONE-1, P-388, MCF-7 and HT29 |
| PhytoCAT-1252 | Scutestrigillosins B | Scutellaria strigillosa | NA | HONE-1, P-388, MCF-7 and HT29 |
| PhytoCAT-1253 | Scutestrigillosins C | Scutellaria strigillosa | NA | HONE-1, P-388, MCF-7 and HT29 |
| PhytoCAT-1254 | Scutestrigillosins D | Scutellaria strigillosa | NA | HONE-1, P-388, MCF-7 and HT29 |
| PhytoCAT-1255 | Scutestrigillosins E | Scutellaria strigillosa | NA | HONE-1, P-388, MCF-7 and HT29 |
| PhytoCAT-1263 | Urs-12-ene-3beta,6beta,16beta-triol-3-O-beta-galactopyranosyl-(1-->2)-beta-glucopyranoside | Silphium radula Nutt | NA | MDA-MB-231 |
| PhytoCAT-1277 | Adonioside A | Adonis multiflora Nishikawa & Koki Ito | NA | HCT-116, HepG2, HeLa, SK-OV-3, and SK-MEL-5, and SKBR-3 |
| PhytoCAT-1278 | Adonioside B | Adonis multiflora Nishikawa & Koki Ito | NA | HCT-116, HepG2, HeLa, SK-OV-3, and SK-MEL-5, and SKBR-3 |
| PhytoCAT-1279 | Cymarin | Adonis multiflora Nishikawa & Koki Ito | NA | HCT-116, HepG2, HeLa, SK-OV-3, and SK-MEL-5, and SKBR-3 |
| PhytoCAT-1287 | Ardisiacrispins B | Ardisia Crenata | NA | MDA-MB-231 |
| PhytoCAT-1288 | Toonayunnanin B | Toona ciliata var yunnanensis | NA | HL-60, SMMC-7721, A-549, MCF-7 and SW480 |
| PhytoCAT-1290 | Glaucocalyxin H | Isodon japonica Hara var glaucocalyx | NA | CE-1, U87, A-549, MCF-7, Hela, K-562, HepG-2 |
| PhytoCAT-1292 | 2α-O-trans-p-coumaroyl-3β,19α-dihydroxy-urs-12-en-28-oic acid | Prinsepia utilis Royle | NA | A549, HCT116, MDA-MB-231, CCRF-CEM |
| PhytoCAT-1293 | 3-O-trans-p-coumaroyltormentic acid | Prinsepia utilis Royle | NA | A549, HCT116, MDA-MB-231, CCRF-CEM |
| PhytoCAT-1294 | 3-O-cis-p-coumaroyltormentic acid | Prinsepia utilis Royle | NA | A549, HCT116, MDA-MB-231, CCRF-CEM |
| PhytoCAT-1295 | 3-O-trans-p-coumaroyl-2α-hydroxyursolic acid | Prinsepia utilis Royle | NA | A549, HCT116, MDA-MB-231, CCRF-CEM |
| PhytoCAT-1296 | 3-O‑cis-p-coumaroyl-2α-hydroxyursolic acid | Prinsepia utilis Royle | NA | A549, HCT116, MDA-MB-231, CCRF-CEM |
| PhytoCAT-1297 | 3-O-trans-p-coumaroylmaslinic acid | Prinsepia utilis Royle | NA | A549, HCT116, MDA-MB-231, CCRF-CEM |
| PhytoCAT-1298 | 3-O-cis-p-coumaroylmaslinic acid | Prinsepia utilis Royle | NA | A549, HCT116, MDA-MB-231, CCRF-CEM |
| PhytoCAT-1327 | 3-O-methylchangnanic acid | Schisandra chinensis | NA | MCF-7, A549, HeLa and RPMI8226 |
| PhytoCAT-1335 | Oleanolic acid | Gleditsia sinensis | ABCB1, CDK2, CDK4, CD34, Cyclin E, Cyclin D1, p-JNK, p-ERK, p21, p27, p53, cyt-c, Bax, PARP-1, VEGF-B, AMPK, VEGFR-2, Caspase 3, mTOR/FRAP1, RAPTOR, RICTOR, VEGF | A549, MDA-MB-231, PC-3, MCF-7, DU145, U87, HT-29, HDFn, HepG-2, Bel-7402, HeLa, MDA-MB-468, HCT-116, T-47D, HL-60/HAR, K562, A354-S2 |
| PhytoCAT-1337 | Dysobinin | Toona ciliata Chisocheton siamensis | NA | HL-60, SMMC-7721, A-549, MCF-7, SW480, NCI-H187, KB |
| PhytoCAT-1338 | Epoxyazadiradione | Toona ciliata, Neem | MMP9 | HL-60, SMMC-7721, A-549, MCF-7, SW480, MDA-MB-231 |
| PhytoCAT-1371 | Isocryptotanshinone | Salvia miltiorrhiza | JNK, ERK, p38 MAPK | MCF-7, MDA-MB-231, HepG2, A459 |
| PhytoCAT-1381 | Isoadenolin I | Isodon adenolomus | NA | HL-60, SMMC-7721, A-549, MCF-7, and SW-480 |
| PhytoCAT-1382 | lasiokaurin | Isodon adenolomus | NA | HL-60, SMMC-7721, A-549, MCF-7, and SW-480 |
| PhytoCAT-1383 | Xerophilusin N | Isodon adenolomus | NA | HL-60, SMMC-7721, A-549, MCF-7, and SW-480 |
| PhytoCAT-1384 | Effusanin B | Isodon adenolomus | NA | HL-60, SMMC-7721, A-549, MCF-7, and SW-480 |
| PhytoCAT-1385 | Longikaurin E | Isodon adenolomus | NA | HL-60, SMMC-7721, A-549, MCF-7, and SW-480 |
| PhytoCAT-1386 | Xerophilusin B | Isodon adenolomus | NA | HL-60, SMMC-7721, A-549, MCF-7, and SW-480 |
| PhytoCAT-1391 | Antiaroside A | Antiaris toxicaria | NA | KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9 and S-KMEL-2 |
| PhytoCAT-1392 | Convallatoxal | Antiaris toxicaria | NA | KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9 and S-KMEL-2 |
| PhytoCAT-1393 | Convallatoxin | Antiaris toxicaria | NA | KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2, HCT-116, SF-268, HL-60, BT-474, MDA-MB-231 |
| PhytoCAT-1394 | Desglucocheirotoxin | Antiaris toxicaria | NA | KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9 and S-KMEL-2 |
| PhytoCAT-1395 | α-antiarin | Antiaris toxicaria | NA | KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
| PhytoCAT-1397 | Cheiranthoside | Antiaris toxicaria | NA | KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
| PhytoCAT-1404 | Antiaroside C | Antiaris toxicaria | NA | KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
| PhytoCAT-1405 | Antiaroside D | Antiaris toxicaria | NA | KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
| PhytoCAT-1409 | β-antiarin | Antiaris toxicaria | NA | KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
| PhytoCAT-1410 | Antiaroside E | Antiaris toxicaria | NA | KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
| PhytoCAT-1411 | Antiaroside F | Antiaris toxicaria | NA | KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
| PhytoCAT-1412 | Antiaroside G | Antiaris toxicaria | NA | KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
| PhytoCAT-1413 | Antiaroside H | Antiaris toxicaria | NA | KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
| PhytoCAT-1414 | Antiaroside I | Antiaris toxicaria | NA | KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
| PhytoCAT-1415 | Antiarotoxinin A | Antiaris toxicaria | NA | KB, KB-VIN, A549, MCF-7, U-87-MG, PC-3, 1A9, CAKI-1, HCT-9, S-KMEL-2 |
| PhytoCAT-1417 | Lobatoside N | Actinostemma lobatum | NA | HCT-116, HT-29, MCF-7, A549 |
| PhytoCAT-1418 | Tupichinolide | Adonis multiflora, Tupistra chinensis | NA | HCT-116, HepG2, HeLa, SK-OV-3, SK-MEL-5, SKBR-3, HL-60, SMMC-7721,A-549,MCF-7,SW480 |
| PhytoCAT-1419 | Cryptojaponol | Clerodendrum kiangsiense | NA | HL-60, SMMC-7721, A-549 and MCF-7 |
| PhytoCAT-1420 | Fortunin E | Clerodendrum kiangsiense | NA | HL-60, SMMC-7721, A-549 and MCF-7 |
| PhytoCAT-1421 | 12-methoxy-6,11,14,16-tetrahydroxy-17(15→16)-abeo-5,8,11,13-abietatetraen-3,7-dione | Clerodendrum kiangsiense | NA | HL-60, SMMC-7721, A-549 and MCF-7 |
| PhytoCAT-1437 | Tripterregeline A | Tripterygium regelii | NA | HL-60, SMMC-7721, A-549, MCF-7, SW480 |
| PhytoCAT-1438 | Triptobenzene H | Tripterygium regelii | NA | HL-60, SMMC-7721, A-549, MCF-7, SW480 |
| PhytoCAT-1439 | Triptinin A | Tripterygium regelii | NA | HL-60, SMMC-7721, A-549, MCF-7, SW480 |
| PhytoCAT-1440 | Triptinin B | Tripterygium regelii | NA | HL-60, SMMC-7721, A-549, MCF-7, SW480 |
| PhytoCAT-1441 | Triptobenzene D | Tripterygium regelii | NA | HL-60, SMMC-7721, A-549, MCF-7, SW480 |
| PhytoCAT-1442 | Triptoquinone A | Tripterygium regelii | NA | HL-60, SMMC-7721, A-549, MCF-7, SW480 |
| PhytoCAT-1443 | Triptobenzene S | Tripterygium regelii | NA | HL-60, SMMC-7721, A-549, MCF-7, SW480 |
| PhytoCAT-1458 | Curcumol | Curcuma wenyujin | Bcl-2, Bak, IDH1, PUMA, p73 | MDA-MB-231, MDA-MB-468, MGC-803 |
| PhytoCAT-1463 | Abifadine E | Abies fargesii | NA | B16, MCF-7, HepG2 |
| PhytoCAT-1464 | 15-hydroxydehydroabietic acid | Abies fargesii | NA | B16, MCF-7, and HepG2 |
| PhytoCAT-1465 | Isojiangrubesin B | Isodon rubescens | NA | HL-60, SMMC-7721, A-549, MCF-7, RAW264.7 SW480 |
| PhytoCAT-1466 | Isojiangrubesin E | Isodon rubescens | NA | HL-60, SMMC-7721, A-549, MCF-7, RAW264.7 SW481 |
| PhytoCAT-1467 | Effusanin A | Isodon rubescens | NA | HL-60, SMMC-7721, A-549, MCF-7, RAW264.7 SW482 |
| PhytoCAT-1468 | Longikaurin A | Isodon rubescens | NA | HL-60, SMMC-7721, A-549, MCF-7, RAW264.7 SW483 |
| PhytoCAT-1469 | 7,14- O-(1-methylethylidene)oridonin | Isodon rubescens | NA | HL-60, SMMC-7721, A-549, MCF-7, RAW264.7 SW484 |
| PhytoCAT-1470 | Hederagenin 3-O-β-D-glucopyranosyl-(1→4)-β-D-glucopyranosyl-(1→3)-α-L-rhamnopyranosyl-(1→2)-α-L-arabinopyranoside | Lonicera similis Hemsl | NA | HepG2, MCF-7, A-549 |
| PhytoCAT-1486 | Citronellol | Citrus hystrix | Bcl-2 | MDA-MB-231 |
| PhytoCAT-1487 | Citronellal | Citrus hystrix | Bcl-2 | MDA-MB-231 |
| PhytoCAT-1493 | Glycyrrhizic acid | Glycyrrhiza glabra | p62, Beclin-1-associated protein | MDA-MB-231 |
| PhytoCAT-1504 | Panaxadiol | Panax ginseng | MMP9, CDK2, CDK4, p21, p27, Cyclin D1, CDK6, EGFR,HER2 | MCF-7, A549 |
| PhytoCAT-1512 | Tanshinone IIA (Tan IIA) and andrographolide (Andro) combination | Tanshinone IIA - Salvia miltiorrhiza Andrographolide - Andrographis paniculata | p53 | MCF-7, BGC823, SMMC7721 |
| PhytoCAT-1517 | Eichlerianic acid | Aglaia odorata | NA | HL-60, SMMC-7721, A-549, MCF-7 and SW480 |
| PhytoCAT-1518 | Vibsanol C | Viburnum odoratissimum | NA | HL-60, SMMC-7721, A-549, MCF-7, and SW-480 |
| PhytoCAT-1519 | Eucalrobusone C | Eucalyptus robusta | NA | HepG2, MCF-7, and U2OS |
| PhytoCAT-1544 | Achyranthes bidentata Blume extract | Achyranthes bidentata Blume | TNF-α | MCF-7 |
| PhytoCAT-1551 | Dehydrothyrsiferol | Laurencia viridis sp nov | NA | T47D, ZR-75-1, and Hs578T |
| PhytoCAT-1552 | Acetoxyscirpendiol | Paecilomyces tenuipes | Cyclin C, Mad-1 | MCF-7 |
| PhytoCAT-1554 | Farnesylthiosalicylic acid (FTS) | NA | s6k1, mTOR | MCF-7 |
| PhytoCAT-1555 | Laurenditerpenol | Laurenciaintricata | HIF-1, VEGF | T47D |
| PhytoCAT-1560 | Salvicine | Chinese herb | topo II, mdr-1, Bcl-2, p38 MAPK, ERK, DNA-dependent kinase (DNA-PK(CS)) | MCF-7, MDA-MB-435, MDR K562/A02, K562/A02, KB/VCR and MCF-7/ADR, K562, KB |
| PhytoCAT-1571 | Phytofluene | Hibiscus syriacus | NA | T47D, MCF-7, ECC-1 |
| PhytoCAT-1577 | 2a,3ß-dihydroxylup-20(29)-ene-27,28-dioic acid | Ampelozizyphus amazonicus Ducke | NA | SKBR-3, C-8161 |
| PhytoCAT-1580 | Ginsenoside Rg1 | Panax ginseng | NA | MCF-7, HEK293 |
| PhytoCAT-1595 | Mycoleptodiscin B | Endophytic fungus Mycoleptodiscus sp | NA | In silico |
| PhytoCAT-1603 | Tricholopardin C | Mushroom Tricholoma pardinum | NA | MCF-7. HeLa |
| PhytoCAT-1622 | (+)-Torreyol | Lignosus rhinocerotis | NA | MCF-7 |
| PhytoCAT-1623 | α-cadinol | Lignosus rhinocerotis | NA | MCF-7 |
| PhytoCAT-1658 | Fucoxanthin | Undaria pinnatifida | TIMP‐1, MMP2, MMP9 | MDA-MB-231 |
| PhytoCAT-1676 | 4-desoxynivalenol | Zea mays | NA | HCT-116, MDA-MB-23, SK-HEP-1 and SNU-639 |
| PhytoCAT-1681 | Isoforrethin-D | Isodon forrestii var forrestii | NA | SMMC-7721, A-549, MCF-7, SW-480 |
| PhytoCAT-1688 | Saikosaponin b2 (SSb2) | Radix Bupleuri | STAT-3, VASP, MMP2, MMP9, c-myc, Cyclin D1 | MCF-7 |
| PhytoCAT-1706 | Antcamphorol H | Antrodia camphorata | NA | MCF-7, U251, SW480 |
| PhytoCAT-1741 | Camphoratin J | Taiwanofungus camphoratus | NA | Hep2, MCF-7, Hela |
| PhytoCAT-1743 | Euphorbia factor L1 | Euphorbia lathyris | ABCB1 | C6, MCF-7, KBv200 |
| PhytoCAT-1754 | Asperuloside acid | Ardisia Crenata | NA | NA |
| PhytoCAT-1758 | Brusatol | Brucea javanica | NA | HL-60, SMMC-7721, A-549, MCF -7, SW480 |
| PhytoCAT-1759 | Bruceine B | Brucea javanica | NA | HL-60, SMMC-7721, A-549, MCF -7, SW480 |
| PhytoCAT-1765 | Ophiobolin O | Aspergillus ustus 094102 | JNK, p38 MAPK, ERK, Bcl-2 phosphorylation (Ser70) | MCF-7 |
| PhytoCAT-1767 | Ganoderiol E | Ganoderma sinense | NA | MCF-7 |
| PhytoCAT-1769 | Toxicarioside M | Antiaris toxicaria | NA | KB, HCT-116, SF-268, MCF-7, HL-60, PC-3, MRC-5 |
| PhytoCAT-1770 | Brevione A | Penicillium sp | NA | MCF-7 |
| PhytoCAT-1771 | Brevione I | Penicillium sp | NA | MCF-7 |
| PhytoCAT-1777 | Neocaesalpin AA | Caesalpinia minax | NA | Hela, HCT-8, HepG-2, MCF-7 and A549 |
| PhytoCAT-1778 | Neocaesalpin AB | Caesalpinia minax | NA | Hela, HCT-8, HepG-2, MCF-7 and A549 |
| PhytoCAT-1779 | Neocaesalpin AC | Caesalpinia minax | NA | Hela, HCT-8, HepG-2, MCF-7 and A549 |
| PhytoCAT-1780 | Neocaesalpin AD | Caesalpinia minax | NA | Hela, HCT-8, HepG-2, MCF-7 and A549 |
| PhytoCAT-1781 | Neocaesalpin AE | Caesalpinia minax | NA | Hela, HCT-8, HepG-2, MCF-7 and A549 |
| PhytoCAT-1782 | 12α-methoxyl,5α,14β-dihydroxy-1α,6α,7β-triacetoxycass-13(15)-en-16,12-olide | Caesalpinia minax | NA | Hela, HCT-8, HepG-2, MCF-7 and A549 |
| PhytoCAT-1784 | Methyl antcinate A | Antrodia camphorata, Antrodia cinnamomea | Bax, Bak, PUMA. | KB, TSCCa, GNM, OC-2, and OEC-M1 , Panc-1 , BT-474, PC-3, OVCAR-3, HeLa, and U2OS, ER+ T47D |
| PhytoCAT-1785 | Methyl antcinate B | Antrodia camphorata, Antrodia cinnamomea | NA | KB, TSCCa, GNM, OC-2, and OEC-M1 , Panc-1 , BT-474, PC-3, OVCAR-3, HeLa, U2OS, ER+ T47D |
| PhytoCAT-1786 | Dehydroeburicoic acid | Antrodia camphorata | NA | KB, TSCCa, GNM, OC-2, and OEC-M1 , Panc-1 , BT-474, PC-3, OVCAR-3, HeLa, and U2OS, ER+ T47D |
| PhytoCAT-1799 | Timosaponin AIII | Anemarrhena asphodeloidea Bunge | COX2, c-met, MMP9, ERK | MDA-MB-231 |
| PhytoCAT-1800 | Yuanhuacine | Daphne genkwa | NA | MCF-7, MDA-MB-231, Huh7, AGS, HT-29, B 16, Colo 205, A549, A2058 |
| PhytoCAT-1804 | Yuanhuadine | Daphne genkwa | NA | MCF-7, MDA-MB-231, Huh7, AGS, HT-29, B 16, Colo 205, A549, A2058 |
| PhytoCAT-1805 | Genkwanin III | Daphne genkwa | NA | MCF-7, MDA-MB-231, Huh7, AGS, HT-29, B 16, Colo 205, A549, A2058 |
| PhytoCAT-1806 | Genkwanin VIII | Daphne genkwa, Daphne mezereum | NA | MCF-7, MDA-MB-231, Huh7, AGS, HT-29, B 16, Colo 205, A549, A2058 |
| PhytoCAT-1809 | 18β-glycyrrhetinic acid | NA | NA | MCF-7 |
| PhytoCAT-1813 | 3alpha-O-acetyl-8,24-dien-tirucallic acid | Boswellia carteri | NA | Hep-G2, MCF-7, RAW 264.7 |
| PhytoCAT-1814 | Verticilla-4(20),7,11-triene | Boswellia carteri | COX-1, COX-2 | Hep-G2, MCF-7, RAW 264.7 |
| PhytoCAT-1826 | Furanodiene | Curcuma wenyujin | integrin αV , β-catenin, FAK, AKT, PI3 kinase p85 | MDA-MB-231 |
| PhytoCAT-1828 | Hawaiinolide A | Paraconiothyrium hawaiiense | NA | A549, T24, HeLa, HCT116, and MCF-7 |
| PhytoCAT-1832 | 11α-hydroxy-lup-20(29)-ene-3β-palmitate | Saussurea phyllocephala | NA | MCF-7, HeLa, HepG2, SGC-7901, NCI-H460 and BGC-823 |
| PhytoCAT-1833 | 28-hydroxy-20-oxo-30-norlupane-3β-palmitate | Saussurea phyllocephala | NA | (MCF-7, HeLa, HepG2, SGC-7901, NCI-H460 and BGC-824 |
| PhytoCAT-1834 | 1β,11α,28-tyrihydroxy oleana-9(11),12-dien-3β-palmitate | Saussurea phyllocephala | NA | MCF-7, HeLa, HepG2, SGC-7901, NCI-H460 and BGC-825 |
| PhytoCAT-1836 | Elaeodendroside B | Elaeodendron orientale | NA | HeLa, A-549, MCF-7 and HL-60, normal Vero cells |
| PhytoCAT-1837 | Elaeodendroside C | Elaeodendron orientale | NA | HeLa, A-549, MCF-7 and HL-60, normal Vero cells |
| PhytoCAT-1838 | Affinoside T | Elaeodendron orientale | NA | HeLa, A-549, MCF-7 and HL-60, normal Vero cells |
| PhytoCAT-1843 | 2α,3β-dihydroxy-urs-20(30)-en-28-oic acid | Sour jujube | NA | HepG2, MCF-7 |
| PhytoCAT-1844 | 2α,3β,28-trihydroxy-urs-20(30)-ene | Sour jujube | NA | HepG2, MCF-7 |
| PhytoCAT-1851 | Panepoxydone | Penicillium griseum | LDH-B, LDH-A, NF-κB | MDA-MB-231, MDA-MB-468, MDA-MB-453 |
| PhytoCAT-1852 | Trichothecinol A | Engleromyces goetzii | NA | HL-60, SMMC-7721, A549, MCF-7, SW-480 |
| PhytoCAT-1854 | Icacinlactone F | Icacina trichantha | NA | MDA-MB-435, MDA-MB-231, OVCAR3 |
| PhytoCAT-1862 | Dahliane B | Verticillium dahliae | NA | MCF-7 |
| PhytoCAT-1863 | Dahliane C | Verticillium dahliae | NA | MCF-7 |
| PhytoCAT-1882 | Germacrone | Curcuma wenyujin | TFF1, GREB1, CCND1, ERG3, PKIB, CTSD, CXCL12, PGR, MYC | MCF-7 |
| PhytoCAT-1897 | Tanshinones | Radix Salviae Miltiorrhizae | Caspase3, Caspase 9, ATF-4 , PARP, p-eIF2 α, P-JNK, Caspase 12 | MCF-7, A549, MKN-45, HGC-27, PC9, QGY-7703, HCT116, U266/ RPMI8226 |
| PhytoCAT-1900 | 3β-hydroxy-30-(4-phenyl-1-piperazinyl)olean-12-ene-11,30-dione | NA | NA | MCF-7, HeLa, HepG2,A549 |
| PhytoCAT-1908 | Artemisinic acid | Artemisia herba alba | NA | MCF-7, HeLa |
| PhytoCAT-1922 | Clematis hederagenin saponin (CHS) | Clematis ganpiniana | NA | MCF-7 and MDA-MB-231 |
| PhytoCAT-1925 | Trigohowimine A | Trigonostemon howii | NA | HL-60, SMMC-7721, A-549, MCF-7 and SW480. |
| PhytoCAT-1926 | Hebecarposide C | Lyonia ovalifolia var hebecarpa | NA | SMMC-7721, HL-60, SW480, MCF-7, and A-549 |
| PhytoCAT-1927 | Hebecarposide H | Lyonia ovalifolia var hebecarpa | NA | SMMC-7721, HL-60, SW480, MCF-7, and A-549 |
| PhytoCAT-1931 | Tebesinone B | Salvia tebesana Bunge | NA | MCF-7, B16F10, PC-3, C26 |
| PhytoCAT-1932 | Aegyptinone A | Salvia tebesana Bunge | NA | MCF-7, B16F10, PC-3, C27 |
| PhytoCAT-1936 | Ginsenoside Rg5 | Black ginseng | p53, p21(WAF1/CIP1), p15(INK4B), Cyclin D1, Cyclin E2, CDK4 | BALB/c nude mouse model of human breast cancer, MCF-7 |
| PhytoCAT-1938 | Astragaloside IV | Astragali radix | P-gp, BCRP, Nrf2 | Wild-type C57BL/6 mice |
| PhytoCAT-1944 | Ganoderic acid A (GA-A) | Ganoderma lucidum | STAT-3 | MDA-MB-231 |
| PhytoCAT-1954 | Ent-17-acetoxy-16β-hydroxykauran-3-one | Chloranthus anhuiensis | NA | MDA-MB-231, 4T1, HepG2, PC12 |
| PhytoCAT-1955 | (5R, 10S)-5,6,7,8-tetrahydro-8-mehtyl-5-(1-methylethyl)-2-naphthalenol | Chloranthus anhuiensis | NA | MDA-MB-231, 4T1, HepG2, and PC12 |
| PhytoCAT-1957 | Triregelin K | Tripterygium regelii | NA | MCF-7, A2780, HepG2 |
| PhytoCAT-1958 | Neotriptonoterpene | Tripterygium regelii | NA | MCF-7, A2780, HepG2 |
| PhytoCAT-1959 | Triregelin I | Tripterygium regelii | NA | MCF-7, A2780, HepG2 |
| PhytoCAT-1986 | Andrographolide | Andrographis paniculata | Heme oxygenase-1, MMP9, COX-2 | MCF-7 |
| PhytoCAT-2001 | Crassin (C4) | Croton crassifolius | pAKT, pERK | MDA-MB-231 |
| PhytoCAT-2013 | Ardisianone | Ardisia virens | NA | MCF-7, NCI-H460, SF-268 |
| PhytoCAT-2014 | Cornudentanone | Ardisia virens | NA | MCF-7, NCI-H460, SF-268 |
| PhytoCAT-2015 | Ardisianol | Ardisia virens | NA | MCF-7, NCI-H460, SF-268 |
| PhytoCAT-2019 | β-elemene | Zanthoxylum setulosum | SNAI1, SNAI2, TWIST, SIP1, TGF-β1, Smad3, EGFR, GLUT1, LDHA, PKM-2, importin α5, PTEN, Pgp, PKM2, EMT | MCF-7/Adr, MCF-7/Doc, MCF-7 |
| PhytoCAT-2029 | Isomesuol | Marila pluricostata | NA | MCF-7, H-460, SF-268 |
| PhytoCAT-2033 | Isodispar B | Marila pluricostata | NA | MCF-7, H-460, SF-268 |
| PhytoCAT-2035 | Disparinol A | Marila pluricostata | NA | MCF-7, H-460, SF-268 |
| PhytoCAT-2038 | 3b,16b,23,28-tetrahydroxy-11a-methoxy-olean-12-ene 3-O-b-Dfucopyranoside | Bupleurum chinense | NA | A549, HepG2, Hep3B, BCap-37, MCF-7 |
| PhytoCAT-2039 | 3b,16b, 28-trihydroxyl-11a-methoxy-olean-12-ene-O-b-D-fucopyranoside | Bupleurum chinense | NA | A549, HepG2, Hep3B, BCap-37, MCF-7 |
| PhytoCAT-2040 | 3b,16b-dihydroxy-23-O-acetyl-13b,28b-epoxyolean-11-ene 3-O-b-D-fucopyranoside. | Bupleurum chinense | NA | A549, HepG2, Hep3B, BCap-37, MCF-7 |
| PhytoCAT-2041 | 3b, 23, 28-trihydroxy-11, 13(18)-diene-16-one 3-O-b-D-glucopyranosyl-(1→3)-b-Dfucopyranoside. | Bupleurum chinense | NA | A549, HepG2, Hep3B, BCap-37, MCF-7 |
| PhytoCAT-2042 | Saikosaponin-b4 | Bupleurum chinense | NA | A549, HepG2, Hep3B, BCap-37, MCF-7 |
| PhytoCAT-2043 | Saikogenin G | Bupleurum chinense | NA | A549, HepG2, Hep3B, BCap-37, MCF-7 |
| PhytoCAT-2044 | Prosaikogenin F | Bupleurum chinense | NA | A549, HepG2, Hep3B, BCap-37, MCF-7 |
| PhytoCAT-2045 | Saikosaponin-A | Bupleurum chinense | NA | A549, HepG2, Hep3B, BCap-37, MCF-7 |
| PhytoCAT-2046 | Saikosaponin-D | Bupleurum chinense | NA | A549, HepG2, Hep3B, BCap-37, MCF-7 |
| PhytoCAT-2047 | Saikosaponin-E | Bupleurum chinense | NA | A549, HepG2, Hep3B, BCap-37, MCF-7 |
| PhytoCAT-2048 | 2''-O-Acetylsaikosaponin A | Bupleurum chinense | NA | A549, HepG2, Hep3B, BCap-37, MCF-7 |
| PhytoCAT-2049 | 3''-O-Acetylsaikosaponin A | Bupleurum chinense | NA | A549, HepG2, Hep3B, BCap-37, MCF-7 |
| PhytoCAT-2050 | 6''-O-Acetylsaikosaponin A | Bupleurum chinense | NA | A549, HepG2, Hep3B, BCap-37, MCF-7 |
| PhytoCAT-2051 | 23-O-Acetylsaikosaponin-a | Bupleurum chinense | NA | A549, HepG2, Hep3B, BCap-37, MCF-7 |
| PhytoCAT-2052 | Saikosaponin C | Bupleurum chinense | NA | A549, HepG2, Hep3B, BCap-37, MCF-7 |
| PhytoCAT-2053 | 6''-O-Acetylsaikosaponin D | Bupleurum chinense | NA | A549, HepG2, Hep3B, BCap-37, MCF-7 |
| PhytoCAT-2054 | Prosaikogenin D | Bupleurum chinense | NA | A549, HepG2, Hep3B, BCap-37, MCF-7 |
| PhytoCAT-2055 | Prosaikogenin A | Bupleurum chinense | NA | A549, HepG2, Hep3B, BCap-37, MCF-7 |
| PhytoCAT-2056 | Saikosaponin-b1 | Bupleurum chinense | NA | A549, HepG2, Hep3B, BCap-37, MCF-7 |
| PhytoCAT-2057 | 23- hydroxy-13b,28b-epoxy-olean-11-ene-16-one 3-O-b-D-glu-copyranosyl-(1 → 3)-b-D-fucopyranoside | Bupleurum chinense | NA | A549, HepG2, Hep3B, BCap-37, MCF-7 |
| PhytoCAT-2065 | Tubeimoside-1 | Bolbostemma paniculatum (Maxim) Franquet | Mcl-1, Bcl-xL, Bcl-2 | MDA-MB-231, T47D |
| PhytoCAT-2071 | Picraviane A | Picramnia glazioviana Engl. | NA | MDA-MB-231 |
| PhytoCAT-2076 | Jatrophone (JA) | Jatropha gossypiifolia | AXIN2, HMGA2, MYC, PCNA, CCND1, EMT | MDA-MB-231, MDA-MB-157, HCC-38, MDA-MB-468 |
| PhytoCAT-2078 | 7,15-isopimaradien-3β,19-diol | Aeollanthus rydingianus | NA | MDA-MB-231 |
| PhytoCAT-2096 | Ursolic acid-3-O-acetate | Morus nigra. | NA | MCF-7, HepG2 |
| PhytoCAT-2097 | Uvaol | Morus nigra. | NA | MCF-7, HepG2 |
| PhytoCAT-2098 | Heteroclitalactone A | Kadsura heteroclita () Craib (Schizandraceae) | NA | Bel-7402, BGC-823, MCF-7, HL-60 |
| PhytoCAT-2099 | Heteroclitalactone C | Kadsura heteroclita () Craib (Schizandraceae) | NA | Bel-7402, BGC-823, MCF-7, HL-60 |
| PhytoCAT-2100 | Heteroclitalactone D | Kadsura heteroclita () Craib (Schizandraceae) | NA | Bel-7402, BGC-823, MCF-7, HL-60 |
| PhytoCAT-2101 | Heteroclitalactone E | Kadsura heteroclita () Craib (Schizandraceae) | NA | Bel-7402, BGC-823, MCF-7, HL-60 |
| PhytoCAT-2102 | Schisandronic acid | Kadsura heteroclita () Craib (Schizandraceae) | NA | Bel-7402, BGC-823, MCF-7, HL-60 |
| PhytoCAT-2103 | Nigranoic acid | Kadsura heteroclita () Craib (Schizandraceae) | NA | Bel-7402, BGC-823, MCF-7, HL-60 |
| PhytoCAT-2104 | Changnanic acid | Kadsura heteroclita () Craib (Schizandraceae) | NA | Bel-7402, BGC-823, MCF-7, HL-60 |
| PhytoCAT-2106 | Saprorthoquinone + Aethiopinone | Salvia atropatana | NA | PC3, MCF-7, MDA-MB-231 |
| PhytoCAT-2107 | Atropatanene | Salvia atropatana | NA | PC3, MCF-7, MDA-MB-231 |
| PhytoCAT-2114 | Pachymic acid | Poria cocos | Cyclin D1, Cyclin E, CDK2, CDK4, p53, p21, Bcl-2, Bax, Cyt-c, Caspase 3, Caspase 8, Caspase 9, MMP9, PKM2 | SKBR-3, BALB/c nude mice/MDA-MB-231 |
| PhytoCAT-2142 | 14α-hydroxy-15-chlorosclareol | Salvia reuterana | NA | MCF-7, HeLa |
| PhytoCAT-2143 | 14α-hydroxy-15-acetoxysclareol | Salvia reuterana | NA | MCF-7, HeLa |
| PhytoCAT-2144 | 6β-hydroxy-14α-epoxysclareol | Salvia reuterana | NA | MCF-7, HeLa |
| PhytoCAT-2145 | 6β-hydroxysclareol | Salvia reuterana | NA | MCF-7, HeLa |
| PhytoCAT-2146 | 14α-epoxysclareol | Salvia reuterana | NA | MCF-7, HeLa |
| PhytoCAT-2164 | Rigidusol | Haplopappus rigidus phil. | NA | ED50 = 3.8 μg/mL against MCF-7 |
| PhytoCAT-2179 | 3β,6β,16β-trihydroxy-lup-20(29)-ene | Combretum leprosum | NA | MRC5, MCF-7, HepG2, T24, HCT116, HT29, CACO-2 |
| PhytoCAT-2189 | Parvifloron D | Plectranthus ecklonii | NA | MDA-MB-231 |
| PhytoCAT-2190 | Forskolin | Coleus barbatus | ERK1/2 | MDA-MB-231, MDA-MB-468, MCF7, HeLa |
| PhytoCAT-2191 | Gelomulide K | Suregada aequorea | PARP-1 | Xenograft model |