PhytoCAT-ID |
Phytochemical name or plant extracts |
Source of phytochemicals or plant Extracts |
Target gene or protein |
Cell line/ mice model |
PhytoCAT-12 |
Kaempferol 3-O-α-l-rhamnopyranosyl-(1→6)-β-d-glucopyranoside |
Calotropis procera |
NA |
MCF-7, HCT-116, HepG-2, A-549, SK-LU-1, KB |
PhytoCAT-13 |
Kudonol A |
Sophora alopecuroides |
NA |
HeLa, Hep3B, MCF-7, H1299 |
PhytoCAT-14 |
Kudonol B |
Sophora alopecuroides |
NA |
HeLa, Hep3B, MCF-7, H1299 |
PhytoCAT-15 |
Kudonol C |
Sophora alopecuroides |
NA |
HeLa, Hep3B, MCF-7, H1299 |
PhytoCAT-30 |
Rhodoeosein |
Fallopia convolvulus |
ERβ |
SKBR-3 |
PhytoCAT-35 |
Icariin |
Alseodaphne semecarpifolia |
ERK1/2 |
SKBR-3, MCF-7, MCF-7/TAM |
PhytoCAT-44 |
Cajanol |
Cajanus cajan |
Bcl-2, Bax, cyt-c, Caspase 3, caspase 9, PARP |
MCF-7 |
PhytoCAT-48 |
Rhamnazin |
Retama sphaerocarpa |
VEGFR2 |
MDA-MB-231/xenograft, TK-10, MCF-7, UACC-62 |
PhytoCAT-51 |
5,3′-dihydroxy-6,7,8,4′-tetramethoxyflavanone (HLBT-100) |
Tillandsia recurvata |
Caspase 3, Caspase 7 |
U87 MG, MDA-MB-231, MV4-11, A375, IMR-32 |
PhytoCAT-54 |
Kaempferide |
Azadirachta indica |
ER |
HL60, A549, AZ521, SKBR-3, MCF-7,PC-3, T-47D |
PhytoCAT-56 |
4'-O-methyl-8-prenylnaringenin |
Azadirachta indica |
NA |
HL60, A549, AZ521, SKBR-3 |
PhytoCAT-57 |
Euchrestaflavanone A |
Azadirachta indica |
NA |
HL60, A549, AZ521, SKBR-3 |
PhytoCAT-58 |
9, and 3-methoxy-3'-prenylnaringenin |
Azadirachta indica |
NA |
HL60, A549, AZ521, SKBR-3 |
PhytoCAT-85 |
Betavulgarin |
Beta vulgaris |
NA |
MDA-MB-231, MCF-7 |
PhytoCAT-109 |
Ugonin J |
Helminthostachys zeylanica |
p53, NANOG |
MCF-7, MDA-MB-231 |
PhytoCAT-111 |
5,7-Dimethoxyflavone |
Anaphalis busua |
NA |
MDCK/Bcrp1 |
PhytoCAT-112 |
Capillarisin |
Artemisia capillaris |
MMP9 |
MCF-7 |
PhytoCAT-120 |
Acacetin |
Calea urticifolia |
STAT-3, CYP1A1, CYP1B1 |
MDA-MB-231, MCF-7, T47D |
PhytoCAT-127 |
Jaceosidin |
Centaurea diluta
Artemisia artica |
NA |
MCF-7 |
PhytoCAT-134 |
Pectolinarigenin |
Cirsium chanroenicum |
MMP2, MMP9, TIMP-2, STAT-3 |
4T1, MDA-MB-231, MCF-7 |
PhytoCAT-135 |
Cirsimaritin |
Cirsium japonicum |
VEGF, AKT, ERK |
MDA-MB-231 |
PhytoCAT-142 |
Hispidulin |
Dittrichia viscosa |
Vimentin , E-cadherin, occludin |
MCF-7, HCC38 |
PhytoCAT-151 |
Cyanidin-3-glucoside (Cy-3-gluc) |
Puya laxa |
ErbB2, Sirt1, KLF4, HER2, AKT, EMT |
MCF-7, BT-474, HCC1569, MDA-MB-453, 6–7-week-old female nude mice |
PhytoCAT-154 |
Nepetin |
Inula britannica |
NA |
MCF-7, Hep-2, Vero cell |
PhytoCAT-155 |
3,3'-di-O-methylquercetin |
Inula viscosa |
NA |
MCF-7, Hep-2, Vero cell |
PhytoCAT-156 |
3-O-methylquercetin |
Inula viscosa |
NA |
MCF-7, Hep-2, Vero cell |
PhytoCAT-162 |
Silymarin |
Silybum marianum |
P-gp, VEGF |
DU145, MCF-7, MDA-MB-468 |
PhytoCAT-163 |
Silibinin |
Silybum marianum |
p21, STAT-3, AKT, ERK, EGFR, CD44, MMP2, BRCA1, LRP6, BNIP3, p53, Bak, Bcl-xL, VEGF, MMP9, RAC1, BNIP3 |
HEK293, PC-3, DU-145, T-47D, MCF-7, MDA-MB-231, 4T1, MDA-MB-435/WT, MDA-MB-435/DOX, MCF-7/PAC |
PhytoCAT-166 |
Isorhamnetin |
Tephroseris kirilowii |
MMP2, MMP9, p38 MAPK, STAT-3 |
B16F10, MCF-7, MDA-MB-231 |
PhytoCAT-172 |
Quercetin-3-methyl ether |
Wollastonia biflora |
Caspase 3, Caspase 7, PARP |
SKBR-3 |
PhytoCAT-240 |
Peonidin-3-glucoside |
Oryza sativa |
HER2, AKT |
BT-474, HCC1569, MDA-MB-453, 6–7-week-old female nude mice |
PhytoCAT-241 |
Vitexin |
Oryza sativa |
Bax, Caspase 7, Caspase 8, Caspase 9, p53, mdm2, Caspase 3 |
MCF-7 |
PhytoCAT-242 |
Orientin |
Oryza sativa |
MMP9, IL-8 |
MCF-7 |
PhytoCAT-253 |
Hibifolin |
Helicteres isora |
NA |
MCF-7 |
PhytoCAT-265 |
Flavonoid extract of wheat germ |
Triticum aestivum |
NA |
BCap-37 |
PhytoCAT-294 |
Paratocarpin E |
Euphorbia humifusa |
NA |
MCF-7 |
PhytoCAT-338 |
Herbacetin |
Ephedra sinica |
TNF-α , IL-1β, JNK, NF-κB, c-met, AKT |
MDA-MB-231, HepG2, RAW 264.7 |
PhytoCAT-347 |
Naringenin |
Garcinia atroviridis |
Bax, Bcl-2, MAPK, PI3K, IL-6, Caspase 3, Caspase 9 |
T-47D, BT-474, MDA-MB-231, SKBR-3,A549, MDA-MB-435, HepG2 |
PhytoCAT-348 |
Epunctanone |
Garcinia epunctata |
NA |
MDA-MB-231, HCT116CEM/ADR5000, MDA-MB-231-BCRP,HCT116 (p53-/-),U87MG |
PhytoCAT-354 |
5,7-dihydroxy-3-(3'-hydroxy-4',5'-dimethoxyphenyl)-6-methoxy-4H-chromen-4-one |
Garcinia nervosa |
NA |
MCF-7, MDA-MB 231 |
PhytoCAT-378 |
Juglanin |
Juglans mandshurica |
Caspase 3, Caspase 8, Caspase 9, LC3B-II, JNK |
SKBR-3, MCF-7, MDA-MB-231, BT-474, mouse xenograft model |
PhytoCAT-394 |
Isothymusin |
Ocimum tenuiflorum |
COX- 2, 5-LOX, CatD, DHFR, hyaluronidase, ODC1 |
NA |
PhytoCAT-414 |
6-Hydroxyflavone |
Scutellaria baicalensis |
NA |
ZR-75-1 |
PhytoCAT-416 |
Wogonoside |
Scutellaria baicalensis |
MST1 |
TNBC cell xenograft model, HEC1A, BALB/c-nu mice |
PhytoCAT-417 |
Xanthomicrol |
Sideritis leucantha |
TNF-α, VEGF, MMP9, Ki67, Bax, Caspase 3, Caspase 9, miR21, miR27, miR125, miR29, miR34 |
4T1, Mouse fibroblast cells |
PhytoCAT-425 |
Fisetin |
Acacia carneorum
Acacia buxifolia |
PTEN |
MDA-MB-231, MCF-7, BT-549 |
PhytoCAT-428 |
5,7,3',4'-tetrahydroxyisoflavone (THIF) |
Ammopiptanthus mongolicus |
cdc2, Chk1, p53 |
T47D |
PhytoCAT-436 |
Isoneorautenol |
Erythrina excelsa |
NA |
MDA-MB-231, CCRF-CEM, HCT116, U87MG |
PhytoCAT-437 |
Derrone |
Erythrina orientalis |
Aurora kinases |
MCF-7, HeLa, KPL4, H1299 |
PhytoCAT-442 |
Pinocembrin |
Glycyrrhiza glabra |
Cyclin B1, Cdc2, PARP-1, Bcl-2, Survivin, PARP-1, Caspase 3, Caspase 9, Bax, ABCG2 |
MDA-MB-231, MCF-7, HeLa |
PhytoCAT-454 |
Kanzonol W |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-455 |
3′-hydroxy-4′-O-methylglabridin |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-456 |
Glabrene |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-457 |
Hispaglabridin A (16) |
Glycyrrhiza glabra |
PTP1B |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-458 |
Hispaglabridin B |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-460 |
8-prenyl-phaseollinisoflavan |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-461 |
3,4-didehydroglabridin |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-463 |
2′-O-demethybidwillol |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-466 |
Glabrone (35) |
Glycyrrhiza glabra |
PTP1B |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-467 |
Lupiwighteone |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-468 |
2,3-dehydrokievitone |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-469 |
Parvisoflavones-A |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-470 |
Isoglabrone |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-471 |
1″,2″-dehydrocyclokievitone |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-472 |
7,2′-dihydroxy-4′-methoxy-8-(3-methyl-2-butenyl) isoflavanone |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-473 |
Glabrol |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-475 |
Shinflavanone |
Glycyrrhiza glabra |
PTP1B |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-476 |
(2S)-abyssinone I |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-478 |
Kanzonol Z |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-479 |
(2R,3R)-3,4′,7-trihydroxy-3′-prenylflavane |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-480 |
3-hydroxyglabrol |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-481 |
Liquiritigenin |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-482 |
Abyssinone II |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-487 |
Paratocarpins B |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-492 |
Shinpterocarpin |
Glycyrrhiza glabra |
NA |
HepG2, SW480, A549, MCF-7 |
PhytoCAT-501 |
2,3,9-Trimethoxypterocarpan |
Pisum sativum |
NA |
MCF-7, T47D, HS578T |
PhytoCAT-502 |
Hyperoside |
Lotus ucrainicus |
Bcl-2, Bax, IL-6 |
MDA-MB-231 |
PhytoCAT-503 |
Barbigerone |
Millettia ferruginea |
P-gp ATPase |
MCF-7/ADR |
PhytoCAT-511 |
Ebenosin |
Onobrychis ebenoides |
NA |
MCF-7, MDA-MB-231 |
PhytoCAT-512 |
Kievitone |
Phaseolus vulgaris |
EGFR kinase |
MCF-7, T47D, SKBR-3 |
PhytoCAT-513 |
7-O-beta-D-glucopyranosylchrysin |
Podocytisus caramanicus |
NA |
MCF-7 |
PhytoCAT-516 |
Sophopterocarpan A |
Sophora flavescens |
NA |
MCF-7 |
PhytoCAT-521 |
Tephrosin |
Tephrosia uniflora |
ABCG2, P-gp |
MCF-7/MX, EPG85.257RDB |
PhytoCAT-522 |
Trigonella berythea extract |
Trigonella berythea |
NA |
MCF-7, U937 |
PhytoCAT-555 |
(+)-Dihydrokaempferol |
Manilkara zapota. |
NA |
BT-474, Chago-K1, HepG2, KATO-III, SW620 |
PhytoCAT-560 |
Kaempferol-7 glucoside |
Strychnos nux-vomica |
NA |
MCF-7, Hep-2, HCT |
PhytoCAT-562 |
Quercetin-3-rhamnoside |
Strychnos nux-vomica |
NA |
MCF-7, Hep-2, HCT |
PhytoCAT-563 |
Kaempferol 3-rutinoside |
Strychnos nux-vomica |
NA |
MCF-7, Hep-2, HCT |
PhytoCAT-566 |
Delphinidin |
Punica granatum |
Cyclin B1, CDK-1, NF-κB, NF-κB/p65, PKCalpha, IKKalpha/beta, IkappaBalpha, STAT-3, MMP9, HER2, PARP, Caspase 3, Bcl-2, BAX, EGFR, AKT, MAPK, PI3K |
MDA-MB-453, AU-565, MCF-10A, MCF-7, BT-474 |
PhytoCAT-568 |
Tricetin |
Punica granatum |
Bax, Bak, p21, cdc2, cdc25C, Cyclin B, Bcl-2, Bcl-xL, ABCG2 |
MCF-7 |
PhytoCAT-629 |
Polymethoxyflavones |
Citrus sinensis |
NA |
MCF-7 |
PhytoCAT-632 |
Glycitein |
Glycine max |
Bcl-2, Bax, MAPK, STAT-3 |
SKBR-3, MCF-7 |
PhytoCAT-633 |
Morin |
Psidium guajava
Cudranaia tricuspidata |
RAD51, H2AA.X, Caspase 3, Caspase 7, p38, JNK, PARP |
SKBR‑3 |
PhytoCAT-640 |
Genistein |
Genista tinctoria |
miR-155, BRCA1 , PI3K/AKT, CDK2, Cyclin D1, VEGF, MMP2, MMP9, uPA, Cyclin B1, mir-23b, NF-κB, p53, Chk2, GPR30-Akt, pRb105, FOXO3, PTEN, casein kinase, p27, UPR, GRP78, IRE1α, ATF4, Beclin-1, TGFβ, Foxp3, CD8a, PI, PIPK, Aromatase, ATRX, SUV39H1/H2, HP1BP3, KLf4, hTERT, CDK1, ER-beta, BRCA1, TNF, BARD1, p53, pS2, jun, BAX, BAP1, BARD1, BRCA2 |
MCF-7, MDA-MB-231, SK-N-SH, MDA-MB-468, T47D, MCF-12A, HepG2, PC12, BT-549, MDA-MB-435, G-292, SKBR-3, MMTV-Wnt-1 , BT-20, MDA468, GLC4/ADR, SW-1573/2R120, HT1080/DR4, MCF-7/Mitox, HL60/ADR, UACC-3199, MCF-10F, MDA-MB-435, Hs578t, |
PhytoCAT-641 |
Daidzein |
Glycine max |
BRCA1 ,BRCA2, VEGF-A, CXCL16, CDK1 , Cyclins A, Cyclin B, Cyclin D, CDK2, CDK4, p21(Cip1), p57(Kip2), caspase 9, ERα, c‑erbB‑2, AKR1BI, HRAS, GSTP1, p53, pS2, jun, GADD45, BAX, TNF, Rb1, p300 |
MCF-7, MDA MB-231, PC12, MCF10a, T47D, G-292, SKBR-3, HS578T, ZR‑75‑1 , MMTV-neu, MDA-MB-453 |
PhytoCAT-642 |
Glyceollin |
Glycine max |
NGFR |
HEK 293, MCF-7,nu/nu immune-compromised female ovariectomized mice, BG-1 |
PhytoCAT-646 |
(2S)-5,7,2',6'-tetrahydroxy-6,8-di (gamma,gamma-dimethylallyl) flavanone |
Patrinia villosa |
NA |
MCF-7, BEL-7402, HT-29, SGC-7901, K562, A498, A549 |
PhytoCAT-647 |
(2S)-5,7,2',6'-tetrahydroxy-6-lavandulylated flavanone |
Patrinia villosa |
NA |
MCF-7, BEL-7402, HT-29, SGC-7901, K562, A498, A549 |
PhytoCAT-648 |
(2S)-5,7,2',6'-tetrahydroxy-4'-lavandulylated flavanone |
Patrinia villosa |
NA |
MCF-7, BEL-7402, HT-29, SGC-7901, K562, A498, A549 |
PhytoCAT-649 |
(2S)-5,2',6'-trihydroxy-2'',2''-dimethylpyrano [5'', 6'': 6, 7] flavanone |
Patrinia villosa |
NA |
MCF-7, BEL-7402, HT-29, SGC-7901, K562, A498, A549 |
PhytoCAT-650 |
(2S, 3''S)-5,2',6'-trihydroxy-3''-gamma,gamma-dimethylallyl-2'',2''-dimethyl-3'',4''-dihydropyrano [5'', 6'': 6, 7] flavanone |
Patrinia villosa |
NA |
MCF-7, BEL-7402, HT-29, SGC-7901, K562, A498, A549 |
PhytoCAT-654 |
Kaempferol-3-O-rhamnoside |
Schima wallichii |
Caspase 9, Caspase 3, PARP |
MCF-7, HC-04 |
PhytoCAT-672 |
(2S)-5,2',6'-trihydroxy-6-lavandulyl-4''-(gamma,gamma-dimethylallyl)-2'',2''-dimethylpyrano-[5'',6'' : 7,8]-flavanone |
Spiranthes australis |
NA |
MCF-7, BEL-7402, HT-29, SGC-7901, K562, A498 |
PhytoCAT-698 |
Kaempferol-3-O-β-D-(6″-n-butyl glucuronide) |
Calligonum polygonoides |
NA |
MCF-7, HepG2 |
PhytoCAT-699 |
Quercetin 3-O-β-D-(6″-n-butyl glucuronide) |
Calligonum polygonoides |
NA |
MCF-7, HepG2 |
PhytoCAT-700 |
Kaempferol-3-O-β-D-(6″-methyl glucuronide) |
Calligonum polygonoides |
NA |
MCF-7, HepG2 |
PhytoCAT-701 |
Dehydrodicatechin A |
Calligonum polygonoides |
NA |
MCF-7, HepG2 |
PhytoCAT-702 |
Catechin |
Calligonum polygonoides |
NA |
MCF-7, HepG2 |
PhytoCAT-703 |
Taxifolin |
Calligonum polygonoides |
SOS1, Grb2, CCL2 |
MCF-7, HepG2 |
PhytoCAT-704 |
Astragalin |
Calligonum polygonoides |
AKT, ZEB1, VEGF, and MMP9 |
MCF-7, HepG2 |
PhytoCAT-705 |
Quercetin-3-O-β-D-(6″-methyl glucuronide) |
Calligonum polygonoides |
NA |
MCF-7, HepG2 |
PhytoCAT-706 |
Quercetin-3-O-glucuronide |
Calligonum polygonoides |
NA |
MCF-7, HepG2 |
PhytoCAT-707 |
Kaempferol-3-O-glucuronide |
Calligonum polygonoides |
NA |
MCF-7, HepG2 |
PhytoCAT-739 |
Trollius chinensis flavonoids |
Trollius chinensis |
Bcl-2, NF-κB, Caspase 9, Caspase 3 |
MCF-7 |
PhytoCAT-741 |
Rutoside |
Frangula alnus |
NA |
Jurkat, MCF-7, HeLa, and HT-30 |
PhytoCAT-742 |
Trifolin |
Frangula alnus |
NA |
Jurkat, MCF-7, HeLa, HT-31 |
PhytoCAT-749 |
Chamanetin |
Cleistochlamys kirkii |
NA |
MDA-MB-231 |
PhytoCAT-750 |
Isochamanetin |
Cleistochlamys kirkii |
NA |
MDA-MB-231 |
PhytoCAT-753 |
Dichamanetin |
Cleistochlamys kirkii |
PARP1 |
MDA-MB-231, HT-29, DU145, |
PhytoCAT-773 |
Calycopterin |
Dracocephalum kotschyi |
Bax, Bcl-2 |
MDA-MB-231, MCF-7 |
PhytoCAT-774 |
7, 3', 5'-trihydroxyflavanone |
Hydnophytum formicarum |
Bcl-2, Bax |
MCF-7 |
PhytoCAT-785 |
Isoquercitrin |
Tetrastigma hemsleyanum |
LSD1 |
MDA-MB-231 |
PhytoCAT-797 |
Ampelopsin |
Ampelopsis grossedentata |
p21, Cyclin A, CDK2, IκBα, NF-κB p65 , CD44, MRP1, β-catenin, KLF4 |
MDA-MB-231, MDA-MB-231/IR |
PhytoCAT-806 |
Robustaflavone A |
Selaginella trichoclada |
VDAC2 channel, Nedd4 E3 ubiquitin ligase |
MCF-7 |
PhytoCAT-807 |
Didymin |
Citrus latipes |
NA |
MDA-MB-231 |
PhytoCAT-809 |
Diosmetin |
Dictamnus dasycarpus |
Bcl-2, Cyclin D1, p53, Bax, Caspase 3, Caspase 9, Caspase 3 |
MDA-MB-468, MCF-7, MDA-MB-231 |
PhytoCAT-819 |
Cynaroside |
Peganum harmala |
NA |
MCF-7, Jurkat, HeLa, and HT-29 |
PhytoCAT-881 |
Theaflavins |
Black tea |
p53, Bax |
MCF-7, MDA-MB-231, ZR-75-1 |
PhytoCAT-884 |
Camellianin A |
Adinandra nitida |
NA |
MCF-7, HepG2 |
PhytoCAT-887 |
Chamaejasmenin B |
Stellera chamaejasme |
β3 integrin-TβRII, TGF-beta |
MDA-MB-231, ZR75-1 and 4T1 |
PhytoCAT-908 |
Artelastin |
Artocarpus elasticus |
NA |
MCF-7 |
PhytoCAT-909 |
Artonin E |
Artocarpus elasticus |
p21, Cyclin D, cyt-c, Bax, Caspase 7, Caspase 9, MAPK |
MCF-7, MDA-MB-231, 1A9, HCT-8 |
PhytoCAT-910 |
Artocarpin |
Artocarpus heterophyllus |
Caspase 8, Caspase 10 |
T47D |
PhytoCAT-913 |
Broussoflavonol B |
Broussonetia papyrifera |
c-Myc , p16(INK4a), p19(INK4D), p21(WAF1/CIP1), Cyclin B1, cdc2, cdc25C, ER-α36, Epidermal growth factor receptor |
MDA-MB-231 |
PhytoCAT-924 |
Rhoifolin (RFL) |
Callicarpa nudiflora |
NA |
MDA-MB-231 |
PhytoCAT-925 |
Apigenin |
Clerodendrum viscosum |
Cyclin D1, Cyclin D3, CDK4, HER2/neu , AKT, CTSS, C3, LAMC2, TLR2, GPRC5B, CNTNAP1, CLDN1, NFATC2, CXCL10, CXCL11, IRAK3, NR3C2, IL32, IL-24, SLIT2, TMEM132A, TMEM171, STAP2, MLKL, KDR, BMPER, KLHL36, STAT-3, YAP/TAZ, CTGF, CYR61, Caspase 3, VEGF, Progestrone receptor, PI3K, JAK3, PLD2, CYP1A1,CYP1B1 |
MDA-MB-453, T47D, ZR-75-1, PC-3, MCF-7, HT-29, HeLa, A549, MDA-MB-231, ChaGo-I , NIH/3T3, A431, MDA-MB-468, Hs578T, SKBR-3 |
PhytoCAT-931 |
Ampelopsin A |
Vitis thunbergii |
AKT |
MDA-MB-231 |
PhytoCAT-932 |
Ampelopsin C |
Vitis thunbergii |
AXL, Dtk (TYRO3), EphA2, EphA6, Fyn, Hck, SRMS |
MDA-MB-231 |
PhytoCAT-978 |
Cyanidin-3-O-(6''-O-α-rhamnopyranosyl- β-glucopyranoside |
Acer palmatum |
NA |
T47D, LLC |
PhytoCAT-979 |
Cyanidin-3-O- β- glucopyranoside |
Acer palmatum |
NA |
T47D, LLC |
PhytoCAT-980 |
Cyanidin-3-O-[2''-O-(galloyl)-6''-O-(rhamnosyl)-β-glucoside] |
Acer palmatum |
NA |
T47D, LLC |
PhytoCAT-981 |
Cyanidin-3-O-[2''-O-(galloyl)- β-glucopyranoside] |
Acer palmatum |
NA |
T47D, LLC |
PhytoCAT-1001 |
Eupafolin |
Eupatorium album |
Bax, Caspase 3, Bcl-2, PI3K, AKT, mTOR |
EO771 |
PhytoCAT-1022 |
Formononetin |
Astragalus membranaceus |
hTERT,c-MYC,Bcl-2, Ha-ras, QR, C3, COX7RP, SULT1A3, ERα, miR-375, AKT, Bcl-2, MMP2, MMP9, TIMP-1, TIMP-2, TNF-α, IL-6 and IL-1β, nitrite, PGE2, iNOS, COX-2 |
MCF-7, MDA-MB-231, 4T1, ER-positive MCF-7, T47D, Caco-2, SKBR-3, HUVEC, LNCaP, PC-3 |
PhytoCAT-1023 |
Quercetin |
Melia azedarach |
PTEN, CYP1B1, EGFR, AKR1C3, PIP, SULT1E1, CDK6, STAT-3,UCA1, CAT, Bcl-2, EGFR, RRM2B, CYP3A4, POTEE, Bax, FAS, MMP2, MMP9, MYC, CASP3, CCND1, CD34, CDK2, CXCL10, CXCL11, DVL2, HSF2, RRM2B, PIG8, CD95, PIDD, Tp53INP, Noxa, p21, PUMA, AMPK, COX-2, PI, HER-2, VEGFR-2, PI3K, AKT, PKB, CYP1A1, CYP1B1 |
HeLa, MDA-MB-231, HEP-2, RD, MCF-7, HepG-2, HCT-116, HeLa, CYP1B1, T47D, 143B, HT - 29, MDA-MB-231 - estrogen-negative breast cancer, MDA-MB-435, MDA-MB-468, HCC-38, BT-474, SK-Br3, TAMR-MCF-7, C6 and COLO-205,KBCHR8-5, DLD-1, DLD-1 human colorectal cancer xenograft model in nude mice, NUDE MICE created from green fluorescent protein-tagged MDA-MB-435 bone metastatic variant |
PhytoCAT-1038 |
Luteolin |
Avicennia marina |
Cyclin E2, Bcl-2, Caspase 3, Bax, VEGF, YAP/TAZ, ABCG2, CD44, EMT, VEGF, MPA, Aromatase, CYP1A1, CYP1B1 |
MDA-MB-468, MCF-7, MDA-MB-453, MDA-MB-231, Hs578T, Progestin-dependent xenograft, LNM35, HT29, HepG2 |
PhytoCAT-1039 |
6-prenylnaringenin (6-PN) |
Humulus lupulus |
NA |
MDA-MB-231, T-47D, PC-3, HT-29, A-2780 |
PhytoCAT-1040 |
8-prenylnaringenin (8-PN) |
Humulus lupulus |
NA |
MDA-MB-231, T-47D, PC-3, HT-29, A-2780 |
PhytoCAT-1042 |
Quercitrin |
Mangifera pajang |
ABCG2 |
MCF-7, HeLa, HT-29 |
PhytoCAT-1052 |
3-hydroxyflavone |
Acacia retinodes |
NA |
MCF-7/BUS |
PhytoCAT-1058 |
Kaempferol |
Justicia gendarussa |
IQGAP3, CYP1A1, CYP1B1, Survivin, PR, AHR, ERα, GREB1, Aromatase |
MCF-7, HCT-15, T47D, C-6, BT-549, A549, HEK293,MDA-MB-231, MDA-MB-468 |
PhytoCAT-1069 |
Brazilin |
Caesalpinia sappan |
p38, p53, DNMT1, p21 |
SiHa, MDA-MB-231, A549, NCI- H1299 |
PhytoCAT-1073 |
Epicatechin |
Garcinia mangostana |
DR4/DR5, Bad, Bax |
MCF-7, T47D, MDA-MB-231, HCT116 |
PhytoCAT-1074 |
Epicatechin gallate |
Garcinia mangostana |
HIF-1, GLUT-1, VEGF, CDKN1A |
T47D, MCF-7 |
PhytoCAT-1078 |
Luteolin-7-O-glucoside |
Celosia argentea |
NA |
MCF-7, SiHa, HCT |
PhytoCAT-1119 |
Tectochrysin |
Hedychium spicatum |
ABCG2 |
MDA-MB-231 |
PhytoCAT-1125 |
5,7- dihydroxy-3,4'-dimethoxyflavone |
Juglans regia |
NA |
MCF-7, BHY |
PhytoCAT-1135 |
Pomiferin |
Maclura pomifera |
NA |
MCF-7, MDA-MB-231 |
PhytoCAT-1164 |
Neohesperidin |
Poncirus trifoliata |
p53, Bax, Bcl-2 |
MDA-MB-231, MCF-7 |
PhytoCAT-1182 |
Scutellarein |
Erigeron breviscapus |
CYP1A1, CYP1B1 |
MDA-MB-468, MCF-7, MCF10A |
PhytoCAT-1183 |
Baicalin |
Scutellaria baicalensis |
miR-338-3p, MORC4, ALPP, DUSP1, CYR61, ALPPL2, SPP1, TLR4, EMT |
T-47D, MCF-7, MDA-MB-231 |
PhytoCAT-1184 |
Baicalein-8-sodium sulfonate (BcS) |
Scutellaria baicalensis |
NA |
MCF-7 |
PhytoCAT-1203 |
Proanthocyanidin |
Uncaria rhynchophylla |
NA |
MCF-7, A549, HS578T and HEK293 |
PhytoCAT-1208 |
Anthocyanin |
Vitis coignetiae Pulliat |
TNF-α, NF-kappaB, COX-2, C-myc, MMP2, MMP9, ICAM-1, VEGF |
MDA-MB-435, HCT-116, MCF-7, NCI-H460, SF-268, AGS |
PhytoCAT-1245 |
Icaritin |
Epimedium diphyllum |
EGFR, GPER1 |
MDA-MB-231, MCF-7, MDA-MB-453 , 4T1,SKBR-3 |
PhytoCAT-1246 |
Xanthohumol |
Humulus lupulus (Common hop) |
EGFR, STAT-3, PHB2, NIS |
MDA-MB-231, SKBR-3, MCF-7, HT-29, A-2780 |
PhytoCAT-1247 |
quercetin 3-O-β-d-xylopyranosyl-(1‴→2″)-O-β-d-glucopyranoside |
Callistemon viminalis |
NA |
MCF-7, HepG2 |
PhytoCAT-1248 |
Kaempferol 3-O-β-d-mannuronopyranoside |
Callistemon viminalis |
NA |
MCF-7, HepG2 |
PhytoCAT-1249 |
Kaempferol 3-O-β-d-mannopyranoside |
Callistemon viminalis |
NA |
MCF-7, HepG2 |
PhytoCAT-1250 |
Quercetin 3-O-β-d-mannuronopyranoside |
Callistemon viminalis |
NA |
NA |
PhytoCAT-1270 |
2'-Hydroxyflavanone |
Citrus sinensis |
Ki67, CD31, Vimentin, Survivin, Bcl-2, Bax, E-cadherin, PARP, RLIP76 |
MCF-7 or SKBR-3 BC cells, MDA-MB-231, TMD231, MCF10a and T47D cells. |
PhytoCAT-1275 |
Pink Lady apples' peel-flavonoids (Peel-F) |
Malus domestica 'Cripps Pink' |
NA |
LoVo, MCF-7 |
PhytoCAT-1276 |
Pink Lady apples' flesh-flavonoids (Flesh-F) |
Malus domestica 'Cripps Pink' |
NA |
LoVo, MCF-7 |
PhytoCAT-1284 |
Biochanin A |
Trifolium pratense |
hTERT, c-MYC, Bcl-2, Ha-ras, QR, C3, COX7RP, p18, MSH2, NF2, WT1, ER?, miR-375, Aromatase |
MCF-7, MDA435/LCC6 , MCF-7/ADR, T47-D, MDA-MB-468, MCF-7 MX100,SK-BR3,MCF12A
HeLa, NCI-H460, HMEC |
PhytoCAT-1291 |
5,4'-dihydroxy-3'-methoxyflavanone-7-(6''-O-α-L-rhamnopyranosyl)-β-D-glucopyranoside |
Satureja spicigera |
NA |
T47D |
PhytoCAT-1309 |
Baicalein |
Scutelleria baicalensis |
PTEN, STAT-3, CYP1A1 , CDKN1A, CXCL9, CXCL10, FKBP5, ZBTB4, GILZ, EMT |
HT-29, Caco-2, HepG2, SW480, MCF-7, MDA-MB-231, MCF10A., SKBR-3, MDA-MB-468 , MMTV-PyMT |
PhytoCAT-1310 |
Wogonin |
Scutelleria baicalensis |
H2AX, Cyclin D1, p21, Cdc25A |
MCF-7, MDA?MB?231, MCF-7/DOX,SKBR-3, HepG2, SW480 and MCF-7 |
PhytoCAT-1318 |
Oroxylin A |
Scutellaria baicalensis |
NA |
HepG2, SW480, MCF-7 |
PhytoCAT-1321 |
Apigenin 4'-geranyl-8-glucopyranosyl-7-O-α-glucopyranoside |
Cupressus sempervirens |
NA |
HepG2, MCF-7, HCT116 and A549 |
PhytoCAT-1322 |
Apigenin 7-O-β-d-glucopyranoside |
Cupressus sempervirens |
NA |
HepG2, MCF-7, HCT116 and A549 |
PhytoCAT-1323 |
Querctine-3-O-glucoside |
Cupressus sempervirens |
NA |
HepG2, MCF-7, HCT116 and A549 |
PhytoCAT-1324 |
Apigenin 4'-pernyl-8-glucopyranosyl -7-O-α-glucopyranoside |
Cupressus sempervirens |
NA |
HepG2, MCF-7, HCT116 and A549 |
PhytoCAT-1330 |
Bavachin |
Psoralea corylifolia |
ABCG2 |
MCF-7/MX, EPG85.257RDB, HT-29, Caco-2, LLC-PK1, MCF-7 |
PhytoCAT-1339 |
Daidzin |
Glycine max |
ER |
ZR-75-1, MDA-MB-231, MCF-7 |
PhytoCAT-1351 |
Isoflavones extracted from chickpea sprouts (ICS) |
Cicer arietinum |
Bax, Bcl-2, Caspase 7, Caspase 9, p53, P21 |
SKBR-3, MCF-7 |
PhytoCAT-1481 |
Chrysin |
Scutellaria baicalensis |
BRCA1, FTO, H2AX, MMP2, MMP9, RAD51, STAT-3, Aromatase |
MCF-7, BT-474, HeLa, HepG-2, MDA-MB-468, BCRP-MDCKII, Caco-2, 518A2, HCT-116 colon, KB-V1/Vbl cervix, MCF-7/Topo, MDA-MB-231, A549 , T47D, MV4-11, LoVo |
PhytoCAT-1484 |
5,7,8,4'-tetramethoxyflavone |
Citrus hystrix |
NA |
U87, A549, MCF-7 |
PhytoCAT-1491 |
Nobiletin |
Arisaema franchetianum Engl , citrus fruits (lemons, oranges, tangerines, and grapefruits) |
CXCR4, MMP9, CYP1A1, CYP1B1 |
MCF-7, MDA-MB-231, H-29, Hs578T, BT-549 |
PhytoCAT-1497 |
Hesperetin |
Citrus plant |
CDK4, P21, Caspase 9, caspace-3, Bax, Bcl-2, eNOS, aromatase, p53, PPARG, NOTCH1, CDK2, Cyclin D, Mir-486-5p And H19 Lncrna, ICAM-1, HER2 |
MCF-7, MDA-MB-435 |
PhytoCAT-1510 |
Glabridin |
Glycyrrhiza glabra(licorine) |
GLUT1, miR-148a, FAK/Src complex, AKT, ERK1/2 |
MDA-MB-231, HEK-293, K562, MCF-7, HeLa, HepG2 and WRL-68 |
PhytoCAT-1520 |
Nitidulin |
Dalbergia velutina |
NA |
KB, HeLa-S3, MCF-7, HepG-2, and HT-29 |
PhytoCAT-1521 |
Dalvelutinane B |
Dalbergia velutina |
NA |
KB, HeLa-S3, MCF-7, HepG-2, and HT-29 |
PhytoCAT-1533 |
4-O-methylbalanophonin |
Mappianthus iodoies |
NA |
HL-60, SMMC-7721, A-549, MCF-7 and SW-480 |
PhytoCAT-1535 |
(3S)-7-hydroxy-8,2′-dimethoxy-4′,5′-methylenedioxyisoflavane |
Spatholobus suberectus |
NA |
MCF-7, MDA-MB-231 |
PhytoCAT-1536 |
(S)-sativan |
Spatholobus suberectus |
NA |
MCF-7, MDA-MB-231 |
PhytoCAT-1541 |
Balanophonin |
Mappianthus iodoies, Cornus kousa, Eria bambusifolia |
NA |
HL-60, SMMC-7721, A-549, MCF-7 and SW-480 |
PhytoCAT-1542 |
(-)-maackiain |
Spatholobus suberectus |
NA |
MDA-MB-231, MCF-7, Hep3B, H1299, HeLa, MCF-7, BHY, Miapaca‑2, Colo‑205, A-549 |
PhytoCAT-1543 |
(3S)-7,2'-Dihydroxy-8,4'-dimethoxyisoflavane |
Spatholobus suberectus |
NA |
MDA-MB-231, MCF-7 |
PhytoCAT-1559 |
6-Prenylchrysin |
NA |
ABCG2 |
HEK-293, MDA-MB-231 |
PhytoCAT-1562 |
Putranjivain A |
Euphorbia jolkini |
p21, WAF1 |
MCF-7 |
PhytoCAT-1567 |
3,5,7,3',4'-pentahydroxyflavonol-3-O-beta-D-glucopyranoside |
Cranberry |
NA |
HepG2, MCF-7 |
PhytoCAT-1574 |
Tricin |
Sasa borealis |
NA |
MDA MB 468, MCF-7, SW480 |
PhytoCAT-1575 |
Kaempferol-3-O-methyl ether |
Zingiber zerumbet |
NA |
MCF-7 |
PhytoCAT-1576 |
Kaempferol-3,4' -O-dimethyl ether |
Zingiber zerumbet |
NA |
MCF-7 |
PhytoCAT-1579 |
Epimedonin L |
Epimedium brevicornum |
NA |
HL-60, SMMC-7721, A-549, MCF-7, and SW-480 |
PhytoCAT-1590 |
Quercetin-3-O-beta-D-arabinofuranoside |
Malus domestica |
NA |
HepG2, MCF-7 |
PhytoCAT-1593 |
3-(4-methoxyphenyl) quinolin-4(1H)-one |
NA |
SerRS mRNA, VEGFA |
MDA-MB-231, 4T1 / BALB/c mice |
PhytoCAT-1596 |
Naringin |
Rhizoma drynariae |
p21, Survivin |
MCF-7, MDA-MB-231 xenograft mice |
PhytoCAT-1597 |
Phenylacetaldehyde |
NA |
STAT-3, IL-6 |
MCF-7, MDA-MB-231 |
PhytoCAT-1601 |
Hesperidin |
Yucca aloifolia variegata |
p21, Cyclin D1, p53 |
MCF-7, HepG2, MDA-MB-231 |
PhytoCAT-1613 |
Jacein |
Centaurea schmidii |
XBP1, sXBP1, ATF-4, ChoP |
MCF-7 and MDA-MB 231 |
PhytoCAT-1614 |
3-demethyljacein |
Centaurea schmidii |
XBP1, sXBP1, ATF-4, ChoP |
MCF-7, MDA-MB 231 |
PhytoCAT-1615 |
Diosmin |
NA |
AURKA, CDK1, KIF11. |
MCF-7, MDA-MB-231, SKBR-3 |
PhytoCAT-1616 |
Eriocitrin |
NA |
STAT-3, Bcl-2 |
MCF-7 |
PhytoCAT-1634 |
Tocotrienol-alpha + Genistein |
Palm oil and Soybean respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1635 |
Tocotrienol-alpha + Narigenin |
Palm oil and Grapefruit respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1636 |
Tocotrienol-alpha + Hesperetin |
Palm oil and Oranges respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1637 |
Tocotrienol-alpha + Tangeretin |
Palm oil and Tangerine respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1638 |
Tocotrienol-alpha + Nobiletin |
Palm oil and Tangerine respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1639 |
Tocotrienol-alpha + Quercetin |
Palm oil and various plants respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1640 |
Tocotrienol-alpha + Apigenin |
Palm oil and various plants respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1641 |
Tocotrienol-gamma + Genistein |
Palm oil and Soybean respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1642 |
Tocotrienol-gamma + Narigenin |
Palm oil and Grapefruit respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1643 |
Tocotrienol-gamma + Hesperetin |
Palm oil and Oranges respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1644 |
Tocotrienol-gamma + Tangeretin |
Palm oil and Tangerine respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1645 |
Tocotrienol-gamma + Nobiletin |
Palm oil and Tangerine respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1646 |
Tocotrienol-gamma + Quercetin |
Palm oil and various plants respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1647 |
Tocotrienol-gamma + Apigenin |
Palm oil and various plants respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1648 |
Tocotrienol-delta + Genistein |
Palm oil and Soybean respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1649 |
Tocotrienol-delta + Narigenin |
Palm oil and Grapefruit respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1650 |
Tocotrienol-delta + Hesperetin |
Palm oil and Oranges respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1651 |
Tocotrienol-delta + Tangeretin |
Palm oil and Tangerine respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1652 |
Tocotrienol-delta + Nobiletin |
Palm oil and Tangerine respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1653 |
Tocotrienol-delta + Quercetin |
Palm oil and various plants respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1654 |
Tocotrienol-delta + Apigenin |
Palm oil and various plants respectively |
NA |
MDA-MB-435, MCF-7 |
PhytoCAT-1679 |
Kuwanon C |
Morus nigra |
NA |
MCF-7, HepG2 |
PhytoCAT-1693 |
(3S)-7-hydroxy-8,2′,4′-trimethoxyisoflavane |
Spatholobus suberectus |
NA |
MCF-7, MD-MB-231 |
PhytoCAT-1695 |
Sinoflavonoidgs A |
Sinopodophyllum hexandrum |
NA |
MCF-7, HepG2, HeLa, KB |
PhytoCAT-1696 |
Sinoflavonoidgs B |
Sinopodophyllum hexandrum |
NA |
MCF-7, HepG2, HeLa, KB |
PhytoCAT-1697 |
3-methoxyquercetin |
Sinopodophyllum hexandrum |
NA |
HeLa |
PhytoCAT-1705 |
Candidone |
Tephrosia candida, Pongamia pinnata,onchocarpus costaricensis |
ABCG2 |
MCF-7/MX, EPG85.257RDB |
PhytoCAT-1709 |
Tangeretin |
Citrus tankan |
Caspase 3,Caspase 8, Caspase 9, Bax, Bid, tBid, p53, p21/cip1, Fas, FasL, PIK3CA, MMP9, PTGS2, IKK, PCNA |
MDA-MB-435, MCF-7, HT-29, MDA-MB-231 |
PhytoCAT-1711 |
Celastrus hindsii extract |
Celastrus hindsii |
NA |
MCF-7, A549, HeLa, HK2. |
PhytoCAT-1717 |
Pashanone |
Persicaria maculosa |
NA |
4T1 |
PhytoCAT-1724 |
Quercetin-3-O-beta-D-arabinofuranoside |
Malus domestica |
NA |
HepG2, MCF-7 |
PhytoCAT-1729 |
Sumadain C |
Alpinia katsumadai |
NA |
HepG2, MCF-7 and BT-549 |
PhytoCAT-1736 |
Delphinidin-3-glucoside (Dp-3-gluc) |
NA |
NA |
MCF-7 |
PhytoCAT-1742 |
Phaseollin |
Phaseolus vulgaris |
NA |
MCF-7 |
PhytoCAT-1787 |
Protoapigenone |
Macrothelypteris torresiana |
(MAPK) ERK, JNK, p38, Bcl-2, Bcl-xL |
HepG2, Hep3B, A549, MDA-MB-231,MCF-7 |
PhytoCAT-1788 |
Puerarin |
Pueraria lobata |
NA |
MCF-7 |
PhytoCAT-1792 |
Sulfuretin |
Calanticaria bicolor |
MMP9 |
MCF-7 |
PhytoCAT-1798 |
Calycosin |
Radix astragali |
RASD1, Bax, Bcl-2 |
MCF-7 |
PhytoCAT-1802 |
Genkwanin |
Daphne genkwa |
NA |
MCF-7, MDA-MB-231, Huh7, AGS, HT-29, B 16, Colo 205, A549, A2058 |
PhytoCAT-1803 |
Tiliroside |
Daphne genkwa |
NA |
MCF-7, MDA-MB-231, Huh7, AGS, HT-29, B 16, Colo 205, A549, A2058 |
PhytoCAT-1822 |
Quercetin-4'-O-sulphate |
NA |
NA |
MCF-7, Caco-2, BxPC-3 |
PhytoCAT-1839 |
Isoxanthohumol |
Humulus lupulus |
NA |
MDA-MB-231, T-47D, PC-3, HT-29, A-2780 |
PhytoCAT-1840 |
6,8-diprenylnarigenin (6,8-diPN) |
Humulus lupulus |
NA |
MDA-MB-231 |
PhytoCAT-1860 |
Flavokawain A |
Piper methsyticum |
IFN-γ, IL-2, NO, iNOS, NF-κB, ICAM, COX-2 |
Breast cancer murine model |
PhytoCAT-1875 |
Cinnamaldehyde |
Cinnamomum cassia |
BRCA1, TOPO1, ERCC1 |
HT-29, LoVo, T47D, NCI-H322 |
PhytoCAT-1876 |
Myricetin |
Withania coagulans |
p53, BRCA1, GADD45, Bax, Bcl-2 |
MCF-7, T47D, MDA-MB-231 |
PhytoCAT-1892 |
5, 7, 4′-trihydroxy-3′-(3-methylbut-2-enyl)-3-methoxy flavone |
Sinopodophyllum hexandrum |
NA |
T47D, MCF-7, MDA-MB-231 |
PhytoCAT-1893 |
Sinopodophylline B |
Sinopodophyllum hexandrum |
NA |
T47D, MCF-7, MDA-MB-231 |
PhytoCAT-1894 |
Citrusinol |
Sinopodophyllum hexandrum |
NA |
T47D, MCF-7, MDA-MB-231 |
PhytoCAT-1895 |
6-prenylquercetin 3-methyl ether |
Sinopodophyllum hexandrum |
NA |
T47D, MCF-7, MDA-MB-231 |
PhytoCAT-1899 |
Comophoroside A |
Commiphora opobalsamum |
NA |
HepG-2, MCF-7 |
PhytoCAT-1917 |
Phloridzin |
Malus pumila |
NA |
MDA-MB-231, MCF-7 |
PhytoCAT-1953 |
Theaflavin-3-gallate |
Camellia sinensis |
HSP90, MMP9, VEGFA, SPP1 |
MCF-7, Caco-2 |
PhytoCAT-1963 |
Wikstrol B |
Wikstroemia scytophylla |
NA |
HL-60, SMMC-7721, A549, MCF-7, and SW480 |
PhytoCAT-1978 |
5-hydroxy-3,7,3'-trimethoxyflavone-4'-O-beta-D-glucoside |
Viscum coloratum |
NA |
HeLa, SGC-7901, MCF-7, and U251 |
PhytoCAT-2007 |
Amplexicaule A |
Polygonum amplexicaule D. Don var. sinense Forb |
Caspase 3,-8,-9, PARP, MCL-1, Bcl-2 |
MCF-7, MDA-MB-435, Female Kunming nude mice |
PhytoCAT-2024 |
Mammea A/AA |
Marila pluricostata |
NA |
MCF-7, H-460, SF-268 |
PhytoCAT-2025 |
Mammea A/BA |
Marila pluricostata |
NA |
MCF-7, H-460, SF-268 |
PhytoCAT-2026 |
Mammea A/AA cyclo D |
Marila pluricostata |
NA |
MCF-7, H-460, SF-268 |
PhytoCAT-2027 |
Mammea A/AB cyclo D |
Marila pluricostata |
NA |
MCF-7, H-460, SF-268 |
PhytoCAT-2028 |
Mammea A/AD cyclo D |
Marila pluricostata |
NA |
MCF-7, H-460, SF-268 |
PhytoCAT-2030 |
Mammea A/AB |
Marila pluricostata |
NA |
MCF-7, H-460, SF-268 |
PhytoCAT-2031 |
Mammea A/AD |
Marila pluricostata |
NA |
MCF-7, H-460, SF-268 |
PhytoCAT-2032 |
Mammea A/BB |
Marila pluricostata |
NA |
MCF-7, H-460, SF-268 |
PhytoCAT-2034 |
Mammea A/AA cyclo F |
Marila pluricostata |
NA |
MCF-7, H-460, SF-268 |
PhytoCAT-2036 |
Mammea A/AB cyclo F |
Marila pluricostata |
NA |
MCF-7, H-460, SF-268 |
PhytoCAT-2068 |
Brazilin A |
Caesalpinia sappan. |
NA |
MCF-7, A549 |
PhytoCAT-2089 |
Morusin |
Morus alba |
E-cadherin, Vimentin, α2-, α6-, β1- integrin, MMP2, MMP9, iNOX, COX |
MCF-7, A549, HepG2, MDA-MB-231 |
PhytoCAT-2091 |
Norartocarpetin |
Morus nigra. |
NA |
MCF-7, HepG2 |
PhytoCAT-2092 |
Cudraflavone A |
Morus nigra. |
NA |
MCF-7, HepG2 |
PhytoCAT-2093 |
Kuwanon G |
Morus nigra. |
NA |
MCF-7, HepG2 |
PhytoCAT-2095 |
Mulberrofuran G |
Morus nigra. |
NA |
MCF-7, HepG2 |
PhytoCAT-2147 |
Sinopodophylline C |
Sinopodophyllum hexandrum |
NA |
MCF-7, MDA-MB-231, T47D |
PhytoCAT-2148 |
Sinopodophylline A |
Sinopodophyllum hexandrum |
NA |
MCF-7, MDA-MB-231, T47D |
PhytoCAT-2149 |
Sinopodophylline D |
Sinopodophyllum hexandrum |
NA |
MCF-7, MDA-MB-231, T47D |
PhytoCAT-2150 |
Topazolin |
Sinopodophyllum hexandrum |
NA |
MCF-7, MDA-MB-231, T47D |
PhytoCAT-2151 |
Sinopodophylliside A |
Sinopodophyllum hexandrum |
NA |
MCF-7, MDA-MB-231, T47D |
PhytoCAT-2152 |
Quercetin-3-O-β-Dglucopyranoside |
Sinopodophyllum hexandrum |
NA |
MCF-7, MDA-MB-231, T47D |
PhytoCAT-2153 |
Quercetin-3-O-β-D-glucopyranoside5-methly ether |
Sinopodophyllum hexandrum |
NA |
MCF-7, MDA-MB-231, T47D |
PhytoCAT-2154 |
Quercetin-3-O-β-D-glucopyranoside7-methly ether |
Sinopodophyllum hexandrum |
NA |
MCF-7, MDA-MB-231, T47D |
PhytoCAT-2155 |
Kaempferol-3-O-β-D-glucopyranoside4′-methly ether |
Sinopodophyllum hexandrum |
NA |
MCF-7, MDA-MB-231, T47D |
PhytoCAT-2161 |
Sophoflavescenol |
Sophora flavescens |
NA |
MCF-7, HL-60, LLC, A549 |
PhytoCAT-2163 |
3'-hydroxygenkwanin |
Daphne genkwa |
NA |
MCF-7, MDA-MB-231, Huh7, AGS, HT-29, B 16, Colo 205, A549, A2058 |