| PhytoCAT-ID | Phytochemical name or plant extracts | Source of phytochemicals or plant Extracts | Target gene or protein | Cell line/ mice model |
|---|---|---|---|---|
| PhytoCAT-12 | Kaempferol 3-O-α-l-rhamnopyranosyl-(1→6)-β-d-glucopyranoside | Calotropis procera | NA | MCF-7, HCT-116, HepG-2, A-549, SK-LU-1, KB |
| PhytoCAT-13 | Kudonol A | Sophora alopecuroides | NA | HeLa, Hep3B, MCF-7, H1299 |
| PhytoCAT-14 | Kudonol B | Sophora alopecuroides | NA | HeLa, Hep3B, MCF-7, H1299 |
| PhytoCAT-15 | Kudonol C | Sophora alopecuroides | NA | HeLa, Hep3B, MCF-7, H1299 |
| PhytoCAT-30 | Rhodoeosein | Fallopia convolvulus | ERβ | SKBR-3 |
| PhytoCAT-35 | Icariin | Alseodaphne semecarpifolia | ERK1/2 | SKBR-3, MCF-7, MCF-7/TAM |
| PhytoCAT-44 | Cajanol | Cajanus cajan | Bcl-2, Bax, cyt-c, Caspase 3, caspase 9, PARP | MCF-7 |
| PhytoCAT-48 | Rhamnazin | Retama sphaerocarpa | VEGFR2 | MDA-MB-231/xenograft, TK-10, MCF-7, UACC-62 |
| PhytoCAT-51 | 5,3′-dihydroxy-6,7,8,4′-tetramethoxyflavanone (HLBT-100) | Tillandsia recurvata | Caspase 3, Caspase 7 | U87 MG, MDA-MB-231, MV4-11, A375, IMR-32 |
| PhytoCAT-54 | Kaempferide | Azadirachta indica | ER | HL60, A549, AZ521, SKBR-3, MCF-7,PC-3, T-47D |
| PhytoCAT-56 | 4'-O-methyl-8-prenylnaringenin | Azadirachta indica | NA | HL60, A549, AZ521, SKBR-3 |
| PhytoCAT-57 | Euchrestaflavanone A | Azadirachta indica | NA | HL60, A549, AZ521, SKBR-3 |
| PhytoCAT-58 | 9, and 3-methoxy-3'-prenylnaringenin | Azadirachta indica | NA | HL60, A549, AZ521, SKBR-3 |
| PhytoCAT-85 | Betavulgarin | Beta vulgaris | NA | MDA-MB-231, MCF-7 |
| PhytoCAT-109 | Ugonin J | Helminthostachys zeylanica | p53, NANOG | MCF-7, MDA-MB-231 |
| PhytoCAT-111 | 5,7-Dimethoxyflavone | Anaphalis busua | NA | MDCK/Bcrp1 |
| PhytoCAT-112 | Capillarisin | Artemisia capillaris | MMP9 | MCF-7 |
| PhytoCAT-120 | Acacetin | Calea urticifolia | STAT-3, CYP1A1, CYP1B1 | MDA-MB-231, MCF-7, T47D |
| PhytoCAT-127 | Jaceosidin | Centaurea diluta Artemisia artica | NA | MCF-7 |
| PhytoCAT-134 | Pectolinarigenin | Cirsium chanroenicum | MMP2, MMP9, TIMP-2, STAT-3 | 4T1, MDA-MB-231, MCF-7 |
| PhytoCAT-135 | Cirsimaritin | Cirsium japonicum | VEGF, AKT, ERK | MDA-MB-231 |
| PhytoCAT-142 | Hispidulin | Dittrichia viscosa | Vimentin , E-cadherin, occludin | MCF-7, HCC38 |
| PhytoCAT-151 | Cyanidin-3-glucoside (Cy-3-gluc) | Puya laxa | ErbB2, Sirt1, KLF4, HER2, AKT, EMT | MCF-7, BT-474, HCC1569, MDA-MB-453, 6–7-week-old female nude mice |
| PhytoCAT-154 | Nepetin | Inula britannica | NA | MCF-7, Hep-2, Vero cell |
| PhytoCAT-155 | 3,3'-di-O-methylquercetin | Inula viscosa | NA | MCF-7, Hep-2, Vero cell |
| PhytoCAT-156 | 3-O-methylquercetin | Inula viscosa | NA | MCF-7, Hep-2, Vero cell |
| PhytoCAT-162 | Silymarin | Silybum marianum | P-gp, VEGF | DU145, MCF-7, MDA-MB-468 |
| PhytoCAT-163 | Silibinin | Silybum marianum | p21, STAT-3, AKT, ERK, EGFR, CD44, MMP2, BRCA1, LRP6, BNIP3, p53, Bak, Bcl-xL, VEGF, MMP9, RAC1, BNIP3 | HEK293, PC-3, DU-145, T-47D, MCF-7, MDA-MB-231, 4T1, MDA-MB-435/WT, MDA-MB-435/DOX, MCF-7/PAC |
| PhytoCAT-166 | Isorhamnetin | Tephroseris kirilowii | MMP2, MMP9, p38 MAPK, STAT-3 | B16F10, MCF-7, MDA-MB-231 |
| PhytoCAT-172 | Quercetin-3-methyl ether | Wollastonia biflora | Caspase 3, Caspase 7, PARP | SKBR-3 |
| PhytoCAT-240 | Peonidin-3-glucoside | Oryza sativa | HER2, AKT | BT-474, HCC1569, MDA-MB-453, 6–7-week-old female nude mice |
| PhytoCAT-241 | Vitexin | Oryza sativa | Bax, Caspase 7, Caspase 8, Caspase 9, p53, mdm2, Caspase 3 | MCF-7 |
| PhytoCAT-242 | Orientin | Oryza sativa | MMP9, IL-8 | MCF-7 |
| PhytoCAT-253 | Hibifolin | Helicteres isora | NA | MCF-7 |
| PhytoCAT-265 | Flavonoid extract of wheat germ | Triticum aestivum | NA | BCap-37 |
| PhytoCAT-294 | Paratocarpin E | Euphorbia humifusa | NA | MCF-7 |
| PhytoCAT-338 | Herbacetin | Ephedra sinica | TNF-α , IL-1β, JNK, NF-κB, c-met, AKT | MDA-MB-231, HepG2, RAW 264.7 |
| PhytoCAT-347 | Naringenin | Garcinia atroviridis | Bax, Bcl-2, MAPK, PI3K, IL-6, Caspase 3, Caspase 9 | T-47D, BT-474, MDA-MB-231, SKBR-3,A549, MDA-MB-435, HepG2 |
| PhytoCAT-348 | Epunctanone | Garcinia epunctata | NA | MDA-MB-231, HCT116CEM/ADR5000, MDA-MB-231-BCRP,HCT116 (p53-/-),U87MG |
| PhytoCAT-354 | 5,7-dihydroxy-3-(3'-hydroxy-4',5'-dimethoxyphenyl)-6-methoxy-4H-chromen-4-one | Garcinia nervosa | NA | MCF-7, MDA-MB 231 |
| PhytoCAT-378 | Juglanin | Juglans mandshurica | Caspase 3, Caspase 8, Caspase 9, LC3B-II, JNK | SKBR-3, MCF-7, MDA-MB-231, BT-474, mouse xenograft model |
| PhytoCAT-394 | Isothymusin | Ocimum tenuiflorum | COX- 2, 5-LOX, CatD, DHFR, hyaluronidase, ODC1 | NA |
| PhytoCAT-414 | 6-Hydroxyflavone | Scutellaria baicalensis | NA | ZR-75-1 |
| PhytoCAT-416 | Wogonoside | Scutellaria baicalensis | MST1 | TNBC cell xenograft model, HEC1A, BALB/c-nu mice |
| PhytoCAT-417 | Xanthomicrol | Sideritis leucantha | TNF-α, VEGF, MMP9, Ki67, Bax, Caspase 3, Caspase 9, miR21, miR27, miR125, miR29, miR34 | 4T1, Mouse fibroblast cells |
| PhytoCAT-425 | Fisetin | Acacia carneorum Acacia buxifolia | PTEN | MDA-MB-231, MCF-7, BT-549 |
| PhytoCAT-428 | 5,7,3',4'-tetrahydroxyisoflavone (THIF) | Ammopiptanthus mongolicus | cdc2, Chk1, p53 | T47D |
| PhytoCAT-436 | Isoneorautenol | Erythrina excelsa | NA | MDA-MB-231, CCRF-CEM, HCT116, U87MG |
| PhytoCAT-437 | Derrone | Erythrina orientalis | Aurora kinases | MCF-7, HeLa, KPL4, H1299 |
| PhytoCAT-442 | Pinocembrin | Glycyrrhiza glabra | Cyclin B1, Cdc2, PARP-1, Bcl-2, Survivin, PARP-1, Caspase 3, Caspase 9, Bax, ABCG2 | MDA-MB-231, MCF-7, HeLa |
| PhytoCAT-454 | Kanzonol W | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-455 | 3′-hydroxy-4′-O-methylglabridin | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-456 | Glabrene | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-457 | Hispaglabridin A (16) | Glycyrrhiza glabra | PTP1B | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-458 | Hispaglabridin B | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-460 | 8-prenyl-phaseollinisoflavan | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-461 | 3,4-didehydroglabridin | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-463 | 2′-O-demethybidwillol | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-466 | Glabrone (35) | Glycyrrhiza glabra | PTP1B | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-467 | Lupiwighteone | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-468 | 2,3-dehydrokievitone | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-469 | Parvisoflavones-A | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-470 | Isoglabrone | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-471 | 1″,2″-dehydrocyclokievitone | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-472 | 7,2′-dihydroxy-4′-methoxy-8-(3-methyl-2-butenyl) isoflavanone | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-473 | Glabrol | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-475 | Shinflavanone | Glycyrrhiza glabra | PTP1B | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-476 | (2S)-abyssinone I | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-478 | Kanzonol Z | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-479 | (2R,3R)-3,4′,7-trihydroxy-3′-prenylflavane | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-480 | 3-hydroxyglabrol | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-481 | Liquiritigenin | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-482 | Abyssinone II | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-487 | Paratocarpins B | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-492 | Shinpterocarpin | Glycyrrhiza glabra | NA | HepG2, SW480, A549, MCF-7 |
| PhytoCAT-501 | 2,3,9-Trimethoxypterocarpan | Pisum sativum | NA | MCF-7, T47D, HS578T |
| PhytoCAT-502 | Hyperoside | Lotus ucrainicus | Bcl-2, Bax, IL-6 | MDA-MB-231 |
| PhytoCAT-503 | Barbigerone | Millettia ferruginea | P-gp ATPase | MCF-7/ADR |
| PhytoCAT-511 | Ebenosin | Onobrychis ebenoides | NA | MCF-7, MDA-MB-231 |
| PhytoCAT-512 | Kievitone | Phaseolus vulgaris | EGFR kinase | MCF-7, T47D, SKBR-3 |
| PhytoCAT-513 | 7-O-beta-D-glucopyranosylchrysin | Podocytisus caramanicus | NA | MCF-7 |
| PhytoCAT-516 | Sophopterocarpan A | Sophora flavescens | NA | MCF-7 |
| PhytoCAT-521 | Tephrosin | Tephrosia uniflora | ABCG2, P-gp | MCF-7/MX, EPG85.257RDB |
| PhytoCAT-522 | Trigonella berythea extract | Trigonella berythea | NA | MCF-7, U937 |
| PhytoCAT-555 | (+)-Dihydrokaempferol | Manilkara zapota. | NA | BT-474, Chago-K1, HepG2, KATO-III, SW620 |
| PhytoCAT-560 | Kaempferol-7 glucoside | Strychnos nux-vomica | NA | MCF-7, Hep-2, HCT |
| PhytoCAT-562 | Quercetin-3-rhamnoside | Strychnos nux-vomica | NA | MCF-7, Hep-2, HCT |
| PhytoCAT-563 | Kaempferol 3-rutinoside | Strychnos nux-vomica | NA | MCF-7, Hep-2, HCT |
| PhytoCAT-566 | Delphinidin | Punica granatum | Cyclin B1, CDK-1, NF-κB, NF-κB/p65, PKCalpha, IKKalpha/beta, IkappaBalpha, STAT-3, MMP9, HER2, PARP, Caspase 3, Bcl-2, BAX, EGFR, AKT, MAPK, PI3K | MDA-MB-453, AU-565, MCF-10A, MCF-7, BT-474 |
| PhytoCAT-568 | Tricetin | Punica granatum | Bax, Bak, p21, cdc2, cdc25C, Cyclin B, Bcl-2, Bcl-xL, ABCG2 | MCF-7 |
| PhytoCAT-629 | Polymethoxyflavones | Citrus sinensis | NA | MCF-7 |
| PhytoCAT-632 | Glycitein | Glycine max | Bcl-2, Bax, MAPK, STAT-3 | SKBR-3, MCF-7 |
| PhytoCAT-633 | Morin | Psidium guajava Cudranaia tricuspidata | RAD51, H2AA.X, Caspase 3, Caspase 7, p38, JNK, PARP | SKBR‑3 |
| PhytoCAT-640 | Genistein | Genista tinctoria | miR-155, BRCA1 , PI3K/AKT, CDK2, Cyclin D1, VEGF, MMP2, MMP9, uPA, Cyclin B1, mir-23b, NF-κB, p53, Chk2, GPR30-Akt, pRb105, FOXO3, PTEN, casein kinase, p27, UPR, GRP78, IRE1α, ATF4, Beclin-1, TGFβ, Foxp3, CD8a, PI, PIPK, Aromatase, ATRX, SUV39H1/H2, HP1BP3, KLf4, hTERT, CDK1, ER-beta, BRCA1, TNF, BARD1, p53, pS2, jun, BAX, BAP1, BARD1, BRCA2 | MCF-7, MDA-MB-231, SK-N-SH, MDA-MB-468, T47D, MCF-12A, HepG2, PC12, BT-549, MDA-MB-435, G-292, SKBR-3, MMTV-Wnt-1 , BT-20, MDA468, GLC4/ADR, SW-1573/2R120, HT1080/DR4, MCF-7/Mitox, HL60/ADR, UACC-3199, MCF-10F, MDA-MB-435, Hs578t, |
| PhytoCAT-641 | Daidzein | Glycine max | BRCA1 ,BRCA2, VEGF-A, CXCL16, CDK1 , Cyclins A, Cyclin B, Cyclin D, CDK2, CDK4, p21(Cip1), p57(Kip2), caspase 9, ERα, c‑erbB‑2, AKR1BI, HRAS, GSTP1, p53, pS2, jun, GADD45, BAX, TNF, Rb1, p300 | MCF-7, MDA MB-231, PC12, MCF10a, T47D, G-292, SKBR-3, HS578T, ZR‑75‑1 , MMTV-neu, MDA-MB-453 |
| PhytoCAT-642 | Glyceollin | Glycine max | NGFR | HEK 293, MCF-7,nu/nu immune-compromised female ovariectomized mice, BG-1 |
| PhytoCAT-646 | (2S)-5,7,2',6'-tetrahydroxy-6,8-di (gamma,gamma-dimethylallyl) flavanone | Patrinia villosa | NA | MCF-7, BEL-7402, HT-29, SGC-7901, K562, A498, A549 |
| PhytoCAT-647 | (2S)-5,7,2',6'-tetrahydroxy-6-lavandulylated flavanone | Patrinia villosa | NA | MCF-7, BEL-7402, HT-29, SGC-7901, K562, A498, A549 |
| PhytoCAT-648 | (2S)-5,7,2',6'-tetrahydroxy-4'-lavandulylated flavanone | Patrinia villosa | NA | MCF-7, BEL-7402, HT-29, SGC-7901, K562, A498, A549 |
| PhytoCAT-649 | (2S)-5,2',6'-trihydroxy-2'',2''-dimethylpyrano [5'', 6'': 6, 7] flavanone | Patrinia villosa | NA | MCF-7, BEL-7402, HT-29, SGC-7901, K562, A498, A549 |
| PhytoCAT-650 | (2S, 3''S)-5,2',6'-trihydroxy-3''-gamma,gamma-dimethylallyl-2'',2''-dimethyl-3'',4''-dihydropyrano [5'', 6'': 6, 7] flavanone | Patrinia villosa | NA | MCF-7, BEL-7402, HT-29, SGC-7901, K562, A498, A549 |
| PhytoCAT-654 | Kaempferol-3-O-rhamnoside | Schima wallichii | Caspase 9, Caspase 3, PARP | MCF-7, HC-04 |
| PhytoCAT-672 | (2S)-5,2',6'-trihydroxy-6-lavandulyl-4''-(gamma,gamma-dimethylallyl)-2'',2''-dimethylpyrano-[5'',6'' : 7,8]-flavanone | Spiranthes australis | NA | MCF-7, BEL-7402, HT-29, SGC-7901, K562, A498 |
| PhytoCAT-698 | Kaempferol-3-O-β-D-(6″-n-butyl glucuronide) | Calligonum polygonoides | NA | MCF-7, HepG2 |
| PhytoCAT-699 | Quercetin 3-O-β-D-(6″-n-butyl glucuronide) | Calligonum polygonoides | NA | MCF-7, HepG2 |
| PhytoCAT-700 | Kaempferol-3-O-β-D-(6″-methyl glucuronide) | Calligonum polygonoides | NA | MCF-7, HepG2 |
| PhytoCAT-701 | Dehydrodicatechin A | Calligonum polygonoides | NA | MCF-7, HepG2 |
| PhytoCAT-702 | Catechin | Calligonum polygonoides | NA | MCF-7, HepG2 |
| PhytoCAT-703 | Taxifolin | Calligonum polygonoides | SOS1, Grb2, CCL2 | MCF-7, HepG2 |
| PhytoCAT-704 | Astragalin | Calligonum polygonoides | AKT, ZEB1, VEGF, and MMP9 | MCF-7, HepG2 |
| PhytoCAT-705 | Quercetin-3-O-β-D-(6″-methyl glucuronide) | Calligonum polygonoides | NA | MCF-7, HepG2 |
| PhytoCAT-706 | Quercetin-3-O-glucuronide | Calligonum polygonoides | NA | MCF-7, HepG2 |
| PhytoCAT-707 | Kaempferol-3-O-glucuronide | Calligonum polygonoides | NA | MCF-7, HepG2 |
| PhytoCAT-739 | Trollius chinensis flavonoids | Trollius chinensis | Bcl-2, NF-κB, Caspase 9, Caspase 3 | MCF-7 |
| PhytoCAT-741 | Rutoside | Frangula alnus | NA | Jurkat, MCF-7, HeLa, and HT-30 |
| PhytoCAT-742 | Trifolin | Frangula alnus | NA | Jurkat, MCF-7, HeLa, HT-31 |
| PhytoCAT-749 | Chamanetin | Cleistochlamys kirkii | NA | MDA-MB-231 |
| PhytoCAT-750 | Isochamanetin | Cleistochlamys kirkii | NA | MDA-MB-231 |
| PhytoCAT-753 | Dichamanetin | Cleistochlamys kirkii | PARP1 | MDA-MB-231, HT-29, DU145, |
| PhytoCAT-773 | Calycopterin | Dracocephalum kotschyi | Bax, Bcl-2 | MDA-MB-231, MCF-7 |
| PhytoCAT-774 | 7, 3', 5'-trihydroxyflavanone | Hydnophytum formicarum | Bcl-2, Bax | MCF-7 |
| PhytoCAT-785 | Isoquercitrin | Tetrastigma hemsleyanum | LSD1 | MDA-MB-231 |
| PhytoCAT-797 | Ampelopsin | Ampelopsis grossedentata | p21, Cyclin A, CDK2, IκBα, NF-κB p65 , CD44, MRP1, β-catenin, KLF4 | MDA-MB-231, MDA-MB-231/IR |
| PhytoCAT-806 | Robustaflavone A | Selaginella trichoclada | VDAC2 channel, Nedd4 E3 ubiquitin ligase | MCF-7 |
| PhytoCAT-807 | Didymin | Citrus latipes | NA | MDA-MB-231 |
| PhytoCAT-809 | Diosmetin | Dictamnus dasycarpus | Bcl-2, Cyclin D1, p53, Bax, Caspase 3, Caspase 9, Caspase 3 | MDA-MB-468, MCF-7, MDA-MB-231 |
| PhytoCAT-819 | Cynaroside | Peganum harmala | NA | MCF-7, Jurkat, HeLa, and HT-29 |
| PhytoCAT-881 | Theaflavins | Black tea | p53, Bax | MCF-7, MDA-MB-231, ZR-75-1 |
| PhytoCAT-884 | Camellianin A | Adinandra nitida | NA | MCF-7, HepG2 |
| PhytoCAT-887 | Chamaejasmenin B | Stellera chamaejasme | β3 integrin-TβRII, TGF-beta | MDA-MB-231, ZR75-1 and 4T1 |
| PhytoCAT-908 | Artelastin | Artocarpus elasticus | NA | MCF-7 |
| PhytoCAT-909 | Artonin E | Artocarpus elasticus | p21, Cyclin D, cyt-c, Bax, Caspase 7, Caspase 9, MAPK | MCF-7, MDA-MB-231, 1A9, HCT-8 |
| PhytoCAT-910 | Artocarpin | Artocarpus heterophyllus | Caspase 8, Caspase 10 | T47D |
| PhytoCAT-913 | Broussoflavonol B | Broussonetia papyrifera | c-Myc , p16(INK4a), p19(INK4D), p21(WAF1/CIP1), Cyclin B1, cdc2, cdc25C, ER-α36, Epidermal growth factor receptor | MDA-MB-231 |
| PhytoCAT-924 | Rhoifolin (RFL) | Callicarpa nudiflora | NA | MDA-MB-231 |
| PhytoCAT-925 | Apigenin | Clerodendrum viscosum | Cyclin D1, Cyclin D3, CDK4, HER2/neu , AKT, CTSS, C3, LAMC2, TLR2, GPRC5B, CNTNAP1, CLDN1, NFATC2, CXCL10, CXCL11, IRAK3, NR3C2, IL32, IL-24, SLIT2, TMEM132A, TMEM171, STAP2, MLKL, KDR, BMPER, KLHL36, STAT-3, YAP/TAZ, CTGF, CYR61, Caspase 3, VEGF, Progestrone receptor, PI3K, JAK3, PLD2, CYP1A1,CYP1B1 | MDA-MB-453, T47D, ZR-75-1, PC-3, MCF-7, HT-29, HeLa, A549, MDA-MB-231, ChaGo-I , NIH/3T3, A431, MDA-MB-468, Hs578T, SKBR-3 |
| PhytoCAT-931 | Ampelopsin A | Vitis thunbergii | AKT | MDA-MB-231 |
| PhytoCAT-932 | Ampelopsin C | Vitis thunbergii | AXL, Dtk (TYRO3), EphA2, EphA6, Fyn, Hck, SRMS | MDA-MB-231 |
| PhytoCAT-978 | Cyanidin-3-O-(6''-O-α-rhamnopyranosyl- β-glucopyranoside | Acer palmatum | NA | T47D, LLC |
| PhytoCAT-979 | Cyanidin-3-O- β- glucopyranoside | Acer palmatum | NA | T47D, LLC |
| PhytoCAT-980 | Cyanidin-3-O-[2''-O-(galloyl)-6''-O-(rhamnosyl)-β-glucoside] | Acer palmatum | NA | T47D, LLC |
| PhytoCAT-981 | Cyanidin-3-O-[2''-O-(galloyl)- β-glucopyranoside] | Acer palmatum | NA | T47D, LLC |
| PhytoCAT-1001 | Eupafolin | Eupatorium album | Bax, Caspase 3, Bcl-2, PI3K, AKT, mTOR | EO771 |
| PhytoCAT-1022 | Formononetin | Astragalus membranaceus | hTERT,c-MYC,Bcl-2, Ha-ras, QR, C3, COX7RP, SULT1A3, ERα, miR-375, AKT, Bcl-2, MMP2, MMP9, TIMP-1, TIMP-2, TNF-α, IL-6 and IL-1β, nitrite, PGE2, iNOS, COX-2 | MCF-7, MDA-MB-231, 4T1, ER-positive MCF-7, T47D, Caco-2, SKBR-3, HUVEC, LNCaP, PC-3 |
| PhytoCAT-1023 | Quercetin | Melia azedarach | PTEN, CYP1B1, EGFR, AKR1C3, PIP, SULT1E1, CDK6, STAT-3,UCA1, CAT, Bcl-2, EGFR, RRM2B, CYP3A4, POTEE, Bax, FAS, MMP2, MMP9, MYC, CASP3, CCND1, CD34, CDK2, CXCL10, CXCL11, DVL2, HSF2, RRM2B, PIG8, CD95, PIDD, Tp53INP, Noxa, p21, PUMA, AMPK, COX-2, PI, HER-2, VEGFR-2, PI3K, AKT, PKB, CYP1A1, CYP1B1 | HeLa, MDA-MB-231, HEP-2, RD, MCF-7, HepG-2, HCT-116, HeLa, CYP1B1, T47D, 143B, HT - 29, MDA-MB-231 - estrogen-negative breast cancer, MDA-MB-435, MDA-MB-468, HCC-38, BT-474, SK-Br3, TAMR-MCF-7, C6 and COLO-205,KBCHR8-5, DLD-1, DLD-1 human colorectal cancer xenograft model in nude mice, NUDE MICE created from green fluorescent protein-tagged MDA-MB-435 bone metastatic variant |
| PhytoCAT-1038 | Luteolin | Avicennia marina | Cyclin E2, Bcl-2, Caspase 3, Bax, VEGF, YAP/TAZ, ABCG2, CD44, EMT, VEGF, MPA, Aromatase, CYP1A1, CYP1B1 | MDA-MB-468, MCF-7, MDA-MB-453, MDA-MB-231, Hs578T, Progestin-dependent xenograft, LNM35, HT29, HepG2 |
| PhytoCAT-1039 | 6-prenylnaringenin (6-PN) | Humulus lupulus | NA | MDA-MB-231, T-47D, PC-3, HT-29, A-2780 |
| PhytoCAT-1040 | 8-prenylnaringenin (8-PN) | Humulus lupulus | NA | MDA-MB-231, T-47D, PC-3, HT-29, A-2780 |
| PhytoCAT-1042 | Quercitrin | Mangifera pajang | ABCG2 | MCF-7, HeLa, HT-29 |
| PhytoCAT-1052 | 3-hydroxyflavone | Acacia retinodes | NA | MCF-7/BUS |
| PhytoCAT-1058 | Kaempferol | Justicia gendarussa | IQGAP3, CYP1A1, CYP1B1, Survivin, PR, AHR, ERα, GREB1, Aromatase | MCF-7, HCT-15, T47D, C-6, BT-549, A549, HEK293,MDA-MB-231, MDA-MB-468 |
| PhytoCAT-1069 | Brazilin | Caesalpinia sappan | p38, p53, DNMT1, p21 | SiHa, MDA-MB-231, A549, NCI- H1299 |
| PhytoCAT-1073 | Epicatechin | Garcinia mangostana | DR4/DR5, Bad, Bax | MCF-7, T47D, MDA-MB-231, HCT116 |
| PhytoCAT-1074 | Epicatechin gallate | Garcinia mangostana | HIF-1, GLUT-1, VEGF, CDKN1A | T47D, MCF-7 |
| PhytoCAT-1078 | Luteolin-7-O-glucoside | Celosia argentea | NA | MCF-7, SiHa, HCT |
| PhytoCAT-1119 | Tectochrysin | Hedychium spicatum | ABCG2 | MDA-MB-231 |
| PhytoCAT-1125 | 5,7- dihydroxy-3,4'-dimethoxyflavone | Juglans regia | NA | MCF-7, BHY |
| PhytoCAT-1135 | Pomiferin | Maclura pomifera | NA | MCF-7, MDA-MB-231 |
| PhytoCAT-1164 | Neohesperidin | Poncirus trifoliata | p53, Bax, Bcl-2 | MDA-MB-231, MCF-7 |
| PhytoCAT-1182 | Scutellarein | Erigeron breviscapus | CYP1A1, CYP1B1 | MDA-MB-468, MCF-7, MCF10A |
| PhytoCAT-1183 | Baicalin | Scutellaria baicalensis | miR-338-3p, MORC4, ALPP, DUSP1, CYR61, ALPPL2, SPP1, TLR4, EMT | T-47D, MCF-7, MDA-MB-231 |
| PhytoCAT-1184 | Baicalein-8-sodium sulfonate (BcS) | Scutellaria baicalensis | NA | MCF-7 |
| PhytoCAT-1203 | Proanthocyanidin | Uncaria rhynchophylla | NA | MCF-7, A549, HS578T and HEK293 |
| PhytoCAT-1208 | Anthocyanin | Vitis coignetiae Pulliat | TNF-α, NF-kappaB, COX-2, C-myc, MMP2, MMP9, ICAM-1, VEGF | MDA-MB-435, HCT-116, MCF-7, NCI-H460, SF-268, AGS |
| PhytoCAT-1245 | Icaritin | Epimedium diphyllum | EGFR, GPER1 | MDA-MB-231, MCF-7, MDA-MB-453 , 4T1,SKBR-3 |
| PhytoCAT-1246 | Xanthohumol | Humulus lupulus (Common hop) | EGFR, STAT-3, PHB2, NIS | MDA-MB-231, SKBR-3, MCF-7, HT-29, A-2780 |
| PhytoCAT-1247 | quercetin 3-O-β-d-xylopyranosyl-(1‴→2″)-O-β-d-glucopyranoside | Callistemon viminalis | NA | MCF-7, HepG2 |
| PhytoCAT-1248 | Kaempferol 3-O-β-d-mannuronopyranoside | Callistemon viminalis | NA | MCF-7, HepG2 |
| PhytoCAT-1249 | Kaempferol 3-O-β-d-mannopyranoside | Callistemon viminalis | NA | MCF-7, HepG2 |
| PhytoCAT-1250 | Quercetin 3-O-β-d-mannuronopyranoside | Callistemon viminalis | NA | NA |
| PhytoCAT-1270 | 2'-Hydroxyflavanone | Citrus sinensis | Ki67, CD31, Vimentin, Survivin, Bcl-2, Bax, E-cadherin, PARP, RLIP76 | MCF-7 or SKBR-3 BC cells, MDA-MB-231, TMD231, MCF10a and T47D cells. |
| PhytoCAT-1275 | Pink Lady apples' peel-flavonoids (Peel-F) | Malus domestica 'Cripps Pink' | NA | LoVo, MCF-7 |
| PhytoCAT-1276 | Pink Lady apples' flesh-flavonoids (Flesh-F) | Malus domestica 'Cripps Pink' | NA | LoVo, MCF-7 |
| PhytoCAT-1284 | Biochanin A | Trifolium pratense | hTERT, c-MYC, Bcl-2, Ha-ras, QR, C3, COX7RP, p18, MSH2, NF2, WT1, ER?, miR-375, Aromatase | MCF-7, MDA435/LCC6 , MCF-7/ADR, T47-D, MDA-MB-468, MCF-7 MX100,SK-BR3,MCF12A HeLa, NCI-H460, HMEC |
| PhytoCAT-1291 | 5,4'-dihydroxy-3'-methoxyflavanone-7-(6''-O-α-L-rhamnopyranosyl)-β-D-glucopyranoside | Satureja spicigera | NA | T47D |
| PhytoCAT-1309 | Baicalein | Scutelleria baicalensis | PTEN, STAT-3, CYP1A1 , CDKN1A, CXCL9, CXCL10, FKBP5, ZBTB4, GILZ, EMT | HT-29, Caco-2, HepG2, SW480, MCF-7, MDA-MB-231, MCF10A., SKBR-3, MDA-MB-468 , MMTV-PyMT |
| PhytoCAT-1310 | Wogonin | Scutelleria baicalensis | H2AX, Cyclin D1, p21, Cdc25A | MCF-7, MDA?MB?231, MCF-7/DOX,SKBR-3, HepG2, SW480 and MCF-7 |
| PhytoCAT-1318 | Oroxylin A | Scutellaria baicalensis | NA | HepG2, SW480, MCF-7 |
| PhytoCAT-1321 | Apigenin 4'-geranyl-8-glucopyranosyl-7-O-α-glucopyranoside | Cupressus sempervirens | NA | HepG2, MCF-7, HCT116 and A549 |
| PhytoCAT-1322 | Apigenin 7-O-β-d-glucopyranoside | Cupressus sempervirens | NA | HepG2, MCF-7, HCT116 and A549 |
| PhytoCAT-1323 | Querctine-3-O-glucoside | Cupressus sempervirens | NA | HepG2, MCF-7, HCT116 and A549 |
| PhytoCAT-1324 | Apigenin 4'-pernyl-8-glucopyranosyl -7-O-α-glucopyranoside | Cupressus sempervirens | NA | HepG2, MCF-7, HCT116 and A549 |
| PhytoCAT-1330 | Bavachin | Psoralea corylifolia | ABCG2 | MCF-7/MX, EPG85.257RDB, HT-29, Caco-2, LLC-PK1, MCF-7 |
| PhytoCAT-1339 | Daidzin | Glycine max | ER | ZR-75-1, MDA-MB-231, MCF-7 |
| PhytoCAT-1351 | Isoflavones extracted from chickpea sprouts (ICS) | Cicer arietinum | Bax, Bcl-2, Caspase 7, Caspase 9, p53, P21 | SKBR-3, MCF-7 |
| PhytoCAT-1481 | Chrysin | Scutellaria baicalensis | BRCA1, FTO, H2AX, MMP2, MMP9, RAD51, STAT-3, Aromatase | MCF-7, BT-474, HeLa, HepG-2, MDA-MB-468, BCRP-MDCKII, Caco-2, 518A2, HCT-116 colon, KB-V1/Vbl cervix, MCF-7/Topo, MDA-MB-231, A549 , T47D, MV4-11, LoVo |
| PhytoCAT-1484 | 5,7,8,4'-tetramethoxyflavone | Citrus hystrix | NA | U87, A549, MCF-7 |
| PhytoCAT-1491 | Nobiletin | Arisaema franchetianum Engl , citrus fruits (lemons, oranges, tangerines, and grapefruits) | CXCR4, MMP9, CYP1A1, CYP1B1 | MCF-7, MDA-MB-231, H-29, Hs578T, BT-549 |
| PhytoCAT-1497 | Hesperetin | Citrus plant | CDK4, P21, Caspase 9, caspace-3, Bax, Bcl-2, eNOS, aromatase, p53, PPARG, NOTCH1, CDK2, Cyclin D, Mir-486-5p And H19 Lncrna, ICAM-1, HER2 | MCF-7, MDA-MB-435 |
| PhytoCAT-1510 | Glabridin | Glycyrrhiza glabra(licorine) | GLUT1, miR-148a, FAK/Src complex, AKT, ERK1/2 | MDA-MB-231, HEK-293, K562, MCF-7, HeLa, HepG2 and WRL-68 |
| PhytoCAT-1520 | Nitidulin | Dalbergia velutina | NA | KB, HeLa-S3, MCF-7, HepG-2, and HT-29 |
| PhytoCAT-1521 | Dalvelutinane B | Dalbergia velutina | NA | KB, HeLa-S3, MCF-7, HepG-2, and HT-29 |
| PhytoCAT-1533 | 4-O-methylbalanophonin | Mappianthus iodoies | NA | HL-60, SMMC-7721, A-549, MCF-7 and SW-480 |
| PhytoCAT-1535 | (3S)-7-hydroxy-8,2′-dimethoxy-4′,5′-methylenedioxyisoflavane | Spatholobus suberectus | NA | MCF-7, MDA-MB-231 |
| PhytoCAT-1536 | (S)-sativan | Spatholobus suberectus | NA | MCF-7, MDA-MB-231 |
| PhytoCAT-1541 | Balanophonin | Mappianthus iodoies, Cornus kousa, Eria bambusifolia | NA | HL-60, SMMC-7721, A-549, MCF-7 and SW-480 |
| PhytoCAT-1542 | (-)-maackiain | Spatholobus suberectus | NA | MDA-MB-231, MCF-7, Hep3B, H1299, HeLa, MCF-7, BHY, Miapaca‑2, Colo‑205, A-549 |
| PhytoCAT-1543 | (3S)-7,2'-Dihydroxy-8,4'-dimethoxyisoflavane | Spatholobus suberectus | NA | MDA-MB-231, MCF-7 |
| PhytoCAT-1559 | 6-Prenylchrysin | NA | ABCG2 | HEK-293, MDA-MB-231 |
| PhytoCAT-1562 | Putranjivain A | Euphorbia jolkini | p21, WAF1 | MCF-7 |
| PhytoCAT-1567 | 3,5,7,3',4'-pentahydroxyflavonol-3-O-beta-D-glucopyranoside | Cranberry | NA | HepG2, MCF-7 |
| PhytoCAT-1574 | Tricin | Sasa borealis | NA | MDA MB 468, MCF-7, SW480 |
| PhytoCAT-1575 | Kaempferol-3-O-methyl ether | Zingiber zerumbet | NA | MCF-7 |
| PhytoCAT-1576 | Kaempferol-3,4' -O-dimethyl ether | Zingiber zerumbet | NA | MCF-7 |
| PhytoCAT-1579 | Epimedonin L | Epimedium brevicornum | NA | HL-60, SMMC-7721, A-549, MCF-7, and SW-480 |
| PhytoCAT-1590 | Quercetin-3-O-beta-D-arabinofuranoside | Malus domestica | NA | HepG2, MCF-7 |
| PhytoCAT-1593 | 3-(4-methoxyphenyl) quinolin-4(1H)-one | NA | SerRS mRNA, VEGFA | MDA-MB-231, 4T1 / BALB/c mice |
| PhytoCAT-1596 | Naringin | Rhizoma drynariae | p21, Survivin | MCF-7, MDA-MB-231 xenograft mice |
| PhytoCAT-1597 | Phenylacetaldehyde | NA | STAT-3, IL-6 | MCF-7, MDA-MB-231 |
| PhytoCAT-1601 | Hesperidin | Yucca aloifolia variegata | p21, Cyclin D1, p53 | MCF-7, HepG2, MDA-MB-231 |
| PhytoCAT-1613 | Jacein | Centaurea schmidii | XBP1, sXBP1, ATF-4, ChoP | MCF-7 and MDA-MB 231 |
| PhytoCAT-1614 | 3-demethyljacein | Centaurea schmidii | XBP1, sXBP1, ATF-4, ChoP | MCF-7, MDA-MB 231 |
| PhytoCAT-1615 | Diosmin | NA | AURKA, CDK1, KIF11. | MCF-7, MDA-MB-231, SKBR-3 |
| PhytoCAT-1616 | Eriocitrin | NA | STAT-3, Bcl-2 | MCF-7 |
| PhytoCAT-1634 | Tocotrienol-alpha + Genistein | Palm oil and Soybean respectively | NA | MDA-MB-435, MCF-7 |
| PhytoCAT-1635 | Tocotrienol-alpha + Narigenin | Palm oil and Grapefruit respectively | NA | MDA-MB-435, MCF-7 |
| PhytoCAT-1636 | Tocotrienol-alpha + Hesperetin | Palm oil and Oranges respectively | NA | MDA-MB-435, MCF-7 |
| PhytoCAT-1637 | Tocotrienol-alpha + Tangeretin | Palm oil and Tangerine respectively | NA | MDA-MB-435, MCF-7 |
| PhytoCAT-1638 | Tocotrienol-alpha + Nobiletin | Palm oil and Tangerine respectively | NA | MDA-MB-435, MCF-7 |
| PhytoCAT-1639 | Tocotrienol-alpha + Quercetin | Palm oil and various plants respectively | NA | MDA-MB-435, MCF-7 |
| PhytoCAT-1640 | Tocotrienol-alpha + Apigenin | Palm oil and various plants respectively | NA | MDA-MB-435, MCF-7 |
| PhytoCAT-1641 | Tocotrienol-gamma + Genistein | Palm oil and Soybean respectively | NA | MDA-MB-435, MCF-7 |
| PhytoCAT-1642 | Tocotrienol-gamma + Narigenin | Palm oil and Grapefruit respectively | NA | MDA-MB-435, MCF-7 |
| PhytoCAT-1643 | Tocotrienol-gamma + Hesperetin | Palm oil and Oranges respectively | NA | MDA-MB-435, MCF-7 |
| PhytoCAT-1644 | Tocotrienol-gamma + Tangeretin | Palm oil and Tangerine respectively | NA | MDA-MB-435, MCF-7 |
| PhytoCAT-1645 | Tocotrienol-gamma + Nobiletin | Palm oil and Tangerine respectively | NA | MDA-MB-435, MCF-7 |
| PhytoCAT-1646 | Tocotrienol-gamma + Quercetin | Palm oil and various plants respectively | NA | MDA-MB-435, MCF-7 |
| PhytoCAT-1647 | Tocotrienol-gamma + Apigenin | Palm oil and various plants respectively | NA | MDA-MB-435, MCF-7 |
| PhytoCAT-1648 | Tocotrienol-delta + Genistein | Palm oil and Soybean respectively | NA | MDA-MB-435, MCF-7 |
| PhytoCAT-1649 | Tocotrienol-delta + Narigenin | Palm oil and Grapefruit respectively | NA | MDA-MB-435, MCF-7 |
| PhytoCAT-1650 | Tocotrienol-delta + Hesperetin | Palm oil and Oranges respectively | NA | MDA-MB-435, MCF-7 |
| PhytoCAT-1651 | Tocotrienol-delta + Tangeretin | Palm oil and Tangerine respectively | NA | MDA-MB-435, MCF-7 |
| PhytoCAT-1652 | Tocotrienol-delta + Nobiletin | Palm oil and Tangerine respectively | NA | MDA-MB-435, MCF-7 |
| PhytoCAT-1653 | Tocotrienol-delta + Quercetin | Palm oil and various plants respectively | NA | MDA-MB-435, MCF-7 |
| PhytoCAT-1654 | Tocotrienol-delta + Apigenin | Palm oil and various plants respectively | NA | MDA-MB-435, MCF-7 |
| PhytoCAT-1679 | Kuwanon C | Morus nigra | NA | MCF-7, HepG2 |
| PhytoCAT-1693 | (3S)-7-hydroxy-8,2′,4′-trimethoxyisoflavane | Spatholobus suberectus | NA | MCF-7, MD-MB-231 |
| PhytoCAT-1695 | Sinoflavonoidgs A | Sinopodophyllum hexandrum | NA | MCF-7, HepG2, HeLa, KB |
| PhytoCAT-1696 | Sinoflavonoidgs B | Sinopodophyllum hexandrum | NA | MCF-7, HepG2, HeLa, KB |
| PhytoCAT-1697 | 3-methoxyquercetin | Sinopodophyllum hexandrum | NA | HeLa |
| PhytoCAT-1705 | Candidone | Tephrosia candida, Pongamia pinnata,onchocarpus costaricensis | ABCG2 | MCF-7/MX, EPG85.257RDB |
| PhytoCAT-1709 | Tangeretin | Citrus tankan | Caspase 3,Caspase 8, Caspase 9, Bax, Bid, tBid, p53, p21/cip1, Fas, FasL, PIK3CA, MMP9, PTGS2, IKK, PCNA | MDA-MB-435, MCF-7, HT-29, MDA-MB-231 |
| PhytoCAT-1711 | Celastrus hindsii extract | Celastrus hindsii | NA | MCF-7, A549, HeLa, HK2. |
| PhytoCAT-1717 | Pashanone | Persicaria maculosa | NA | 4T1 |
| PhytoCAT-1724 | Quercetin-3-O-beta-D-arabinofuranoside | Malus domestica | NA | HepG2, MCF-7 |
| PhytoCAT-1729 | Sumadain C | Alpinia katsumadai | NA | HepG2, MCF-7 and BT-549 |
| PhytoCAT-1736 | Delphinidin-3-glucoside (Dp-3-gluc) | NA | NA | MCF-7 |
| PhytoCAT-1742 | Phaseollin | Phaseolus vulgaris | NA | MCF-7 |
| PhytoCAT-1787 | Protoapigenone | Macrothelypteris torresiana | (MAPK) ERK, JNK, p38, Bcl-2, Bcl-xL | HepG2, Hep3B, A549, MDA-MB-231,MCF-7 |
| PhytoCAT-1788 | Puerarin | Pueraria lobata | NA | MCF-7 |
| PhytoCAT-1792 | Sulfuretin | Calanticaria bicolor | MMP9 | MCF-7 |
| PhytoCAT-1798 | Calycosin | Radix astragali | RASD1, Bax, Bcl-2 | MCF-7 |
| PhytoCAT-1802 | Genkwanin | Daphne genkwa | NA | MCF-7, MDA-MB-231, Huh7, AGS, HT-29, B 16, Colo 205, A549, A2058 |
| PhytoCAT-1803 | Tiliroside | Daphne genkwa | NA | MCF-7, MDA-MB-231, Huh7, AGS, HT-29, B 16, Colo 205, A549, A2058 |
| PhytoCAT-1822 | Quercetin-4'-O-sulphate | NA | NA | MCF-7, Caco-2, BxPC-3 |
| PhytoCAT-1839 | Isoxanthohumol | Humulus lupulus | NA | MDA-MB-231, T-47D, PC-3, HT-29, A-2780 |
| PhytoCAT-1840 | 6,8-diprenylnarigenin (6,8-diPN) | Humulus lupulus | NA | MDA-MB-231 |
| PhytoCAT-1860 | Flavokawain A | Piper methsyticum | IFN-γ, IL-2, NO, iNOS, NF-κB, ICAM, COX-2 | Breast cancer murine model |
| PhytoCAT-1875 | Cinnamaldehyde | Cinnamomum cassia | BRCA1, TOPO1, ERCC1 | HT-29, LoVo, T47D, NCI-H322 |
| PhytoCAT-1876 | Myricetin | Withania coagulans | p53, BRCA1, GADD45, Bax, Bcl-2 | MCF-7, T47D, MDA-MB-231 |
| PhytoCAT-1892 | 5, 7, 4′-trihydroxy-3′-(3-methylbut-2-enyl)-3-methoxy flavone | Sinopodophyllum hexandrum | NA | T47D, MCF-7, MDA-MB-231 |
| PhytoCAT-1893 | Sinopodophylline B | Sinopodophyllum hexandrum | NA | T47D, MCF-7, MDA-MB-231 |
| PhytoCAT-1894 | Citrusinol | Sinopodophyllum hexandrum | NA | T47D, MCF-7, MDA-MB-231 |
| PhytoCAT-1895 | 6-prenylquercetin 3-methyl ether | Sinopodophyllum hexandrum | NA | T47D, MCF-7, MDA-MB-231 |
| PhytoCAT-1899 | Comophoroside A | Commiphora opobalsamum | NA | HepG-2, MCF-7 |
| PhytoCAT-1917 | Phloridzin | Malus pumila | NA | MDA-MB-231, MCF-7 |
| PhytoCAT-1953 | Theaflavin-3-gallate | Camellia sinensis | HSP90, MMP9, VEGFA, SPP1 | MCF-7, Caco-2 |
| PhytoCAT-1963 | Wikstrol B | Wikstroemia scytophylla | NA | HL-60, SMMC-7721, A549, MCF-7, and SW480 |
| PhytoCAT-1978 | 5-hydroxy-3,7,3'-trimethoxyflavone-4'-O-beta-D-glucoside | Viscum coloratum | NA | HeLa, SGC-7901, MCF-7, and U251 |
| PhytoCAT-2007 | Amplexicaule A | Polygonum amplexicaule D. Don var. sinense Forb | Caspase 3,-8,-9, PARP, MCL-1, Bcl-2 | MCF-7, MDA-MB-435, Female Kunming nude mice |
| PhytoCAT-2024 | Mammea A/AA | Marila pluricostata | NA | MCF-7, H-460, SF-268 |
| PhytoCAT-2025 | Mammea A/BA | Marila pluricostata | NA | MCF-7, H-460, SF-268 |
| PhytoCAT-2026 | Mammea A/AA cyclo D | Marila pluricostata | NA | MCF-7, H-460, SF-268 |
| PhytoCAT-2027 | Mammea A/AB cyclo D | Marila pluricostata | NA | MCF-7, H-460, SF-268 |
| PhytoCAT-2028 | Mammea A/AD cyclo D | Marila pluricostata | NA | MCF-7, H-460, SF-268 |
| PhytoCAT-2030 | Mammea A/AB | Marila pluricostata | NA | MCF-7, H-460, SF-268 |
| PhytoCAT-2031 | Mammea A/AD | Marila pluricostata | NA | MCF-7, H-460, SF-268 |
| PhytoCAT-2032 | Mammea A/BB | Marila pluricostata | NA | MCF-7, H-460, SF-268 |
| PhytoCAT-2034 | Mammea A/AA cyclo F | Marila pluricostata | NA | MCF-7, H-460, SF-268 |
| PhytoCAT-2036 | Mammea A/AB cyclo F | Marila pluricostata | NA | MCF-7, H-460, SF-268 |
| PhytoCAT-2068 | Brazilin A | Caesalpinia sappan. | NA | MCF-7, A549 |
| PhytoCAT-2089 | Morusin | Morus alba | E-cadherin, Vimentin, α2-, α6-, β1- integrin, MMP2, MMP9, iNOX, COX | MCF-7, A549, HepG2, MDA-MB-231 |
| PhytoCAT-2091 | Norartocarpetin | Morus nigra. | NA | MCF-7, HepG2 |
| PhytoCAT-2092 | Cudraflavone A | Morus nigra. | NA | MCF-7, HepG2 |
| PhytoCAT-2093 | Kuwanon G | Morus nigra. | NA | MCF-7, HepG2 |
| PhytoCAT-2095 | Mulberrofuran G | Morus nigra. | NA | MCF-7, HepG2 |
| PhytoCAT-2147 | Sinopodophylline C | Sinopodophyllum hexandrum | NA | MCF-7, MDA-MB-231, T47D |
| PhytoCAT-2148 | Sinopodophylline A | Sinopodophyllum hexandrum | NA | MCF-7, MDA-MB-231, T47D |
| PhytoCAT-2149 | Sinopodophylline D | Sinopodophyllum hexandrum | NA | MCF-7, MDA-MB-231, T47D |
| PhytoCAT-2150 | Topazolin | Sinopodophyllum hexandrum | NA | MCF-7, MDA-MB-231, T47D |
| PhytoCAT-2151 | Sinopodophylliside A | Sinopodophyllum hexandrum | NA | MCF-7, MDA-MB-231, T47D |
| PhytoCAT-2152 | Quercetin-3-O-β-Dglucopyranoside | Sinopodophyllum hexandrum | NA | MCF-7, MDA-MB-231, T47D |
| PhytoCAT-2153 | Quercetin-3-O-β-D-glucopyranoside5-methly ether | Sinopodophyllum hexandrum | NA | MCF-7, MDA-MB-231, T47D |
| PhytoCAT-2154 | Quercetin-3-O-β-D-glucopyranoside7-methly ether | Sinopodophyllum hexandrum | NA | MCF-7, MDA-MB-231, T47D |
| PhytoCAT-2155 | Kaempferol-3-O-β-D-glucopyranoside4′-methly ether | Sinopodophyllum hexandrum | NA | MCF-7, MDA-MB-231, T47D |
| PhytoCAT-2161 | Sophoflavescenol | Sophora flavescens | NA | MCF-7, HL-60, LLC, A549 |
| PhytoCAT-2163 | 3'-hydroxygenkwanin | Daphne genkwa | NA | MCF-7, MDA-MB-231, Huh7, AGS, HT-29, B 16, Colo 205, A549, A2058 |