| PhytoCAT-ID | Phytochemical name or plant extracts | Source of phytochemicals or plant Extracts | Target gene or protein | Cell line/ mice model |
|---|---|---|---|---|
| PhytoCAT-25 | Flavopereirine | Geissospermum sericeum | p-ERK, p38 MAPK siRNA, p-Akt, mTOR, LC3-II | MCF-7, MDA-MB-231 |
| PhytoCAT-31 | Isotetrandrine | Triclisia sacleuxii | P-gp | MCF-7/DOX, HeLa, Hep3B |
| PhytoCAT-32 | Magnoflorine | Berberidaceae, Magnoliaceae, Menispermaceae, or Papaveraceae botanical families Berberis cretica | NA | NCI-H1299, MDA-MB-468, T98G , TE671 |
| PhytoCAT-40 | 5-hydroxy-skytanthine hydrochloride | Tecoma stans | NA | Hep-G2, MCF-7 |
| PhytoCAT-148 | Klugine | Psychotria klugii | HIF-1 | T47D |
| PhytoCAT-149 | Isocephaeline | Psychotria klugii | HIF-1 | T47D |
| PhytoCAT-150 | Emetine | Psychotria klugii | HIF-1 | T47D |
| PhytoCAT-173 | Homoharringtonine | Cephalotaxus harringtonia | Bcl-x, Caspase 9 | MCF-7, A549, UACC903 |
| PhytoCAT-220 | Chelidonine | Chelidonium majus | AKT, ERK1/2 | MDA-MB-231 |
| PhytoCAT-230 | Papaverine | Papaver rhoeas | NA | MCF-7, MDA-MB-231 |
| PhytoCAT-243 | Capsaicin | Capsicum annuum | NA | MCF-7 |
| PhytoCAT-244 | Tomatine | Solanum lycopersicum | MMP2, MMP9, MMP9\NGAL | MCF-7 |
| PhytoCAT-266 | Cyclovirobuxine D (CVB-D) | Buxus microphylla | LC3-I, LC3-II, ATG5 | MCF-7 |
| PhytoCAT-302 | Terminamines K | Pachysandra terminalis | NA | MDA-MB-231 |
| PhytoCAT-303 | Terminamines L | Pachysandra terminalis | NA | MDA-MB-231 |
| PhytoCAT-304 | Terminamines M | Pachysandra terminalis | NA | MDA-MB-231 |
| PhytoCAT-305 | Terminamines N | Pachysandra terminalis | NA | MDA-MB-231 |
| PhytoCAT-306 | Terminamines O | Pachysandra terminalis | NA | MDA-MB-231 |
| PhytoCAT-307 | Terminamines P | Pachysandra terminalis | NA | MDA-MB-231 |
| PhytoCAT-308 | Terminamines Q | Pachysandra terminalis | NA | MDA-MB-231 |
| PhytoCAT-309 | Terminamines R | Pachysandra terminalis | NA | MDA-MB-231 |
| PhytoCAT-310 | Terminamines S | Pachysandra terminalis | NA | MDA-MB-231 |
| PhytoCAT-311 | (+)-pachysandrine B | Pachysandra terminalis | NA | MDA-MB-231 |
| PhytoCAT-312 | Epipachysandrine-A | Pachysandra terminalis | NA | MDA-MB-231 |
| PhytoCAT-313 | 3β-methylamino 16-oxo 5,17(20) cis-pregnadiene | Pachysandra terminalis | NA | MDA-MB-231 |
| PhytoCAT-314 | Z-salignone | Pachysandra terminalis | NA | MDA-MB-231 |
| PhytoCAT-315 | Terminamine H | Pachysandra terminalis | NA | MDA-MB-231 |
| PhytoCAT-316 | 3β-methylamino 16-oxo 5,17(20) trans-pregnadiene | Pachysandra terminalis | NA | MDA-MB-231 |
| PhytoCAT-317 | E-salignone | Pachysandra terminalis | NA | MDA-MB-231 |
| PhytoCAT-318 | (+)-spiropachysine | Pachysandra terminalis | NA | MDA-MB-231 |
| PhytoCAT-319 | Terminamines A | Pachysandra terminalis | Epithelial growth factor, integrin β | MDA-MB-231 |
| PhytoCAT-320 | Terminamines B | Pachysandra terminalis | Epithelial growth factor | MDA-MB-231 |
| PhytoCAT-321 | Terminamines C | Pachysandra terminalis | Epithelial growth factor | MDA-MB-231 |
| PhytoCAT-322 | Terminamines D | Pachysandra terminalis | Epithelial growth factor | MDA-MB-231 |
| PhytoCAT-323 | Terminamines E | Pachysandra terminalis | Epithelial growth factor | MDA-MB-231 |
| PhytoCAT-324 | Terminamines F | Pachysandra terminalis | NA | MDA-MB-231 |
| PhytoCAT-325 | Terminamines G | Pachysandra terminalis | NA | MDA-MB-231 |
| PhytoCAT-326 | Pachystermine B | Pachysandra terminalis | Epithelial growth factor | MDA-MB-231 |
| PhytoCAT-327 | Pachystermine A | Pachysandra terminalis | Epithelial growth factor | MDA-MB-231 |
| PhytoCAT-328 | Epipachysamine E | Pachysandra terminalis | Epithelial growth factor | MDA-MB-231 |
| PhytoCAT-329 | Epipachysamine B | Pachysandra terminalis | Epithelial growth factor | MDA-MB-231 |
| PhytoCAT-330 | Terminaline | Pachysandra terminalis | Epithelial growth factor | MDA-MB-231 |
| PhytoCAT-331 | Terminamine I | Pachysandra terminalis | NA | MDA-MB-231 |
| PhytoCAT-332 | Terminamine J | Pachysandra terminalis | NA | MDA-MB-231 |
| PhytoCAT-340 | Avenanthramide-C | Avena sativa | NA | MDA-MB-231 |
| PhytoCAT-346 | Neobractatin | Garcinia bracteata | MBNL2 | MDA-MB-231 xenografts mouse model, A549, HepG2, T98, MCF-7 |
| PhytoCAT-500 | Benzo[b]tryptanthrin | Indigofera tinctoria | topo I, topo II, MDR1, Caspase 3, PARP | HCT15, MCF-7 |
| PhytoCAT-515 | Matrine | Sophora flavescens | PTEN, miR-21 , AKT, Bad, p21(/WAF1/CIP1), p27(/KIP1), Bcl-2, Bax, VEGF, VEGFR-2, Caspase 3, Caspase 9, P-gp, MRP1, IKKβ, GRP78, eIF2α, CHOP, p62, mTOR, Topo I, LIN28A/Let-7 | MCF-7, 4T1 Balb/c mice, MCF-7/ADR, MDA-MB-231, BT-474, MDA-MB-468 |
| PhytoCAT-519 | Tonkinensine B | Sophora tonkinensis | Bax, Bcl-2, Caspase 3, Caspase 9 | MDA-MB-231, 4T1 |
| PhytoCAT-543 | 5,6-anhydrohupehenine | Fritillaria hupehensis | NA | MCF-7, HepG2 |
| PhytoCAT-558 | Colchicine | Buddleja davidii | NA | Mgc-803, BCap-37, MDA-MB-435, MDA-MB-231, OVCAR3 |
| PhytoCAT-586 | Rohitukine | Dysoxylum binectariferum | NA | MCF-7, T47D, MDA-MB-273, SKOV3, NCI/ADR-RES |
| PhytoCAT-601 | Sinomenine | Sinomenium acutum | TRAP, OSCAR, c-Fos, NFATc1, hIL-8, IL-8/CXCR1, MMP2, MMP9 | Tumor-bearing mice, MDA-MB-231 |
| PhytoCAT-602 | 6,7-di-O-acetylsinococuline (FK-3000) | Stephania delavayi | NF-kB, COX-2, cyclin B, p-CDC2 | MDA-MB-231 xenografted mice, MCF-7, MDA-MB-231, PC-3, HT-29 |
| PhytoCAT-603 | Sinococuline | Stephania delavayi | NA | MDA-MB-231 xenografted mice, MCF-7, MDA-MB-231, PC-3, HT-29 |
| PhytoCAT-605 | Cepharanthine | Stephania epigaea | Atg7, AMPK | MDA-MB-231, HeLa, A549, MCF-7, PC3, HepG2, Hep3B, 50MT-1, HL-60, H1299, SMMC-7721, SW480 |
| PhytoCAT-606 | Isotrilobine | Stephania japonica | NA | MCF-7/ADR |
| PhytoCAT-607 | Trilobine | Stephania japonica | NA | MCF-7/ADR |
| PhytoCAT-639 | Yuehchukene | Murraya paniculata | NA | MCF-7, MDA-MB-231 |
| PhytoCAT-659 | Jerantinine A | Tabernaemontana corymbosa | SF3B1, SF3B3 | MCF-7, MDA-MB-468, T47D, MCF-10A |
| PhytoCAT-665 | Camptothecine | Miquelia dentata | NA | MDA-MB-273, NCI/ADR-RES, SKOV, HepG2, Hep3B, MDA-MB- 231, MCF-7, A549, Ca9-22, NCI/ADR-RES, Hela, HCT116, GI 101A, MDA-MB-157 |
| PhytoCAT-678 | Lycorine | Sternbergia clusiana | Mcl-1, Bcl-xL, MMP2, MMP9, SHP-1, STAT-3 | Nude mouse models, A549, HCT116, SK-OV-3, NCI-H460, K562, MCF-7 and HL-60 |
| PhytoCAT-681 | Govaniadine | Corydalis govaniana | Bax, p53, Survivin, Caspase 7 | MCF-7 |
| PhytoCAT-682 | Corydalis saxicola Bunting total alkaloids (CSBTA) | Corydalis saxicola | RANKL/OPG | MDA-MB-231 |
| PhytoCAT-683 | Glaucine | Corydalis turtschaninovii | MMP9, NF-κB | MDA-MB-231 |
| PhytoCAT-684 | Leptopidine | Hypecoum leptocarpum | FAS | NA |
| PhytoCAT-685 | Noscapine | Papaver somniferum | Bcl-xL, Bcl-2 | MCF-7 and MDA-MB-231 |
| PhytoCAT-686 | Sanguinarine | Sanguinaria canadensis | STAT-3 , XIAP, Caspase 3, Bcl-2, cIAP2, XIAP, c-FLIPs, p21, p27, Cyclin D1, Topoisomerase II | NA |
| PhytoCAT-689 | Piperlongumine | Piper longum | SETDB1, EGFR, STAT-3, ZBTB4, Sp1, Sp3, Sp4, Cyclin D1, Survivin, cMyc, EGFR | A549, 786-O, SKBR-3, Female athymic nu/nu mice |
| PhytoCAT-721 | Delcosine | Aconitum barbatum Aconitum napellus Aconitum yesoense | NA | MCF-7, MDA-MB-231, A549, DU145,KB |
| PhytoCAT-722 | Sinchiangensine A | Aconitum sinchiangense | NA | HL-60, A-549, SMCC-7721, MCF-7 and SW480 cell line. |
| PhytoCAT-729 | Protoberberine | Coptis chinensis | NA | MCF-7, MADB106, SGC7901 |
| PhytoCAT-730 | Jatrorrhizine | Coptis chinensis | TNIK | MDA-MB-231, MCF-7 and 4T1 |
| PhytoCAT-737 | Berberine | Coptis chinensis | EGFR, GPER1, ABCG2, CYP1A1, HMGB1, ABCG2, IL-1β, IL-6,TNF-α, NF-κB, Bax, Bcl-2, EGFR, AKT, P38, ERK1/2 | Cytotoxic effect on MCF-7 cells, inhibitory effect on the growth of breast, liver and colon cancer cell lines (MCF-7, HepG2 and CACO-2, respectively). MDA-MB-231, the human ductal breast epithelial tumor cell line (T47D cell line) |
| PhytoCAT-761 | 3,10,11-trimethoxy-1,2-methylenedioxy-7-oxoaporphine | Fissistigma oldhamii | NA | MCF-7 |
| PhytoCAT-787 | Mitraphylline | Uncaria tomentosa | NA | HAE, BEAS-2B, SK-N-SH, HepG2, HEK293, MKN45, DLD1, A549, MCF7, LNCaP |
| PhytoCAT-789 | 8-hydroxyartabonatine C | Pseuduvaria trimera | NA | HepG2, MDA-MB-231 |
| PhytoCAT-799 | Mukonal | Murraya koenigii | PARP, Caspase 3, Bcl-2, Beclin-1, LC3B-I, LC3B-II | MDA-MB-231, CAMA-1, MDA-MB-435, SKBR-3/ xenografted mice models |
| PhytoCAT-811 | Girinimbine | Murraya euchrestifolia | NA | MDA-MB-453 |
| PhytoCAT-812 | Mahanine | Bergera koenigii | NA | MDA‑MB‑157, MCF‑7, MDA-MB-231 |
| PhytoCAT-814 | Paratrimerin I | Paramignya trimera | NA | MCF-7, HepG2 |
| PhytoCAT-816 | Harmine | Peganum harmala | Twist1, TAZ, p‑Erk, p‑Akt, Bcl‑2, Bax | BT-549 |
| PhytoCAT-817 | Harmine hydrochloride | Peganum harmala | PI3K, AKT, mTOR, FOXO3a | MCF-7, MDA-MB-231 |
| PhytoCAT-820 | Nitidine chloride | Zanthoxylum nitidum | PARP, Bax, Caspase 9, Caspase 3, Bcl-2 | MCF-7, MDA-MB-231 |
| PhytoCAT-826 | Halofuginone | Dichroa febrifuga | MMP9 | MDA-MB-231, PC3 |
| PhytoCAT-847 | Melognine | Melodinus fusiformis | Caspase 3, p53, Bcl-2 | BT-549 |
| PhytoCAT-855 | 9-methoxycanthin-6-one | Eurycoma longifolia | PKM, ANXA2, LGAL3, HNRNP1A1, PRDX3, GAPDH, ACAA2, ALDH1A1, CAPG,MDH2, EEF1A1, TPI1 | MCF-7, A2780, SKOV-3, HT29, A375, HeLa, DU-145, RD, CaOV-3, MDBK, A-549 |
| PhytoCAT-856 | Canthin-6-one | Eurycoma longifolia | NA | HCC 1395, DU 145, Vero E6, A549, MCF-7, HL60 , AZ521, SKBR-3 |
| PhytoCAT-858 | Picrasidine G | Picrasma quassioides | Caspase 3, PARP, STAT-3, EGFR, Survivin | MDA-MB-468 |
| PhytoCAT-862 | Isopicrinine | Rhazya stricta | PUMA, Survivin | MCF-7 |
| PhytoCAT-863 | Rhazyaminine | Rhazya stricta | Bcl-2 | MCF-7 |
| PhytoCAT-865 | Affinisine | Tabernaemontana catharinensis | NA | MCF-7, U251, NCI-ADR/RES, 786-0, NCI-H460, HT-29, K562 , PC-3 |
| PhytoCAT-912 | Boehmeriasin A | Boehmeria siamensis | Cyclin E2, Cyclin D1 | MDA-MB-231 |
| PhytoCAT-982 | Dehydrocorydaline | Corydali syanhusuo | CDK1, CCND1, Bcl-2, MMP2, MMP9, Caspase 3, Caspase 8, Caspase 9, Bax, Bcl-2 | MDA‑MB‑231 , MCF-7 |
| PhytoCAT-983 | Protopine | Corydalis yanhusuo | EGFR, ICAM-1, αv-integrin, β1-integrin, β5-integrin | MCF-7, MDA-MB-231 |
| PhytoCAT-1002 | Evodiamine | Evodia rutaecarpa | MMP9, uPA, uPAR, ERK, p38 MAPK, topo I, Bax, Bcl-2, Caspase 3, Survivin | MDA-MB-231, MCF-7, A375-S2, HeLa, THP-1, L929 |
| PhytoCAT-1005 | Tryptanthrin | Cephalantheropsis gracilis | NA | MCF-7, NCI-H460, and SF-268, HCT-15 |
| PhytoCAT-1009 | Voacamine | Voacanga africana | NA | MDA-MB-231, HEPG-2, A375, SH-SY5Y, CT26 |
| PhytoCAT-1010 | 19-epi-voacristine | Voacanga africana | NA | MDA-MB-231, HEPG-2, A375, SH-SY5Y, CT26 |
| PhytoCAT-1011 | Vobasine | Voacanga africana | NA | MDA-MB-231, HEPG-2, A375, SH-SY5Y, CT26 |
| PhytoCAT-1012 | Voacristine | Voacanga africana | NA | MDA-MB-231, HEPG-2, A375, SH-SY5Y, CT26 |
| PhytoCAT-1015 | Voacangine | Voacanga africana | NA | MDA-MB-231, HEPG-2, A375, SH-SY5Y, CT27 |
| PhytoCAT-1017 | Curcumin and berberine combination | Curcumin - Curcuma longa Berberine - Thalictrum delavayi | Bcl-2, JNK, Beclin-1 | MCF-7, MDA-MB-231 |
| PhytoCAT-1080 | Ukrain | Chelidonium majus | NA | SKBR-3, 4T07, TUBO, MDA-MB-231, PA-TU-8902, CCL-221 , U-138MG |
| PhytoCAT-1089 | Cuscutamine | Cuscuta chinensis | NA | MCF-7, T47D |
| PhytoCAT-1137 | Hirsutine | Uncaria tomentosa | γH2AX, Caspase 3, Caspase 7 | MCF-7, MDA-MB-231, MDA-MB-468, MDA-MB-453, ZR-75-1, BT-474 |
| PhytoCAT-1143 | Isoliensinine | Nelumbo nucifera | p38 MAPK, JNK, CDK2, p21, AKT, GSK3α | MCF-7, MDA-MB-231, HeLa, A549, PC3, HepG2, Hep3B, H1299 |
| PhytoCAT-1144 | Neferine (NEF) | Nelumbo nucifera | miR-374a/FGFR-2 | MDA-MB-231, MCF-7 |
| PhytoCAT-1189 | Oxymatrine | Sophora flavescens | αⅤβ3 integrin, E-cadherin, FAK, PI3K, and Akt | MCF-7, MDA-MB-231 and 4T1 |
| PhytoCAT-1217 | Clausehainanines A | Clausena hainanensis | NA | HL-60, SMMC-7721, A-549, MCF-7, SW480 |
| PhytoCAT-1218 | Clausehainanines B | Clausena hainanensis | NA | HL-60, SMMC-7721, A-549, MCF-7, SW480 |
| PhytoCAT-1219 | Clausehainanines C | Clausena hainanensis | NA | HL-60, SMMC-7721, A-549, MCF-7, SW480 |
| PhytoCAT-1220 | Clausehainanines D | Clausena hainanensis | NA | HL-60, SMMC-7721, A-549, MCF-7, SW480 |
| PhytoCAT-1221 | Clausehainanines E | Clausena hainanensis | NA | HL-60, SMMC-7721, A-549, MCF-7, SW480 |
| PhytoCAT-1262 | Lucidimine B | Ganoderma lucidum | NA | MCF-7 |
| PhytoCAT-1307 | Cordatine | Macleaya cordata | NA | MCF-7 and SF-268 |
| PhytoCAT-1308 | 8-methoxydihydrochelerythrine | Macleaya cordata | NA | MCF-7, SF-269 |
| PhytoCAT-1377 | 9-methoxy-18,19-dehydrocamptothecin | Nothapodytes foetida | NA | HepG2, Hep3B, MDA-MB- 231, MCF-7, A549, and Ca9-22 |
| PhytoCAT-1378 | 9-methoxy-camptothecin | Nothapodytes foetida | NA | HepG2, Hep3B, MDA-MB- 231, MCF-7, A549, and Ca9-22 |
| PhytoCAT-1379 | 5-hydroxycamptothecin | Nothapodytes foetida | NA | HepG2, Hep3B, MDA-MB- 231, MCF-7, A549, and Ca9-22 |
| PhytoCAT-1380 | 5-hydroxy-9-methoxycamptothecin | Nothapodytes foetida | NA | HepG2, Hep3B, MDA-MB- 231, MCF-7, A549, and Ca9-22 |
| PhytoCAT-1388 | Conophylline | Tabernaemontana divaricata, Tabernaemontana corymbosa | NA | HL-60, SMMC-7721, A-549, MCF-7, SW480, KB, PC-3, LNCaP, MDA-MB-231, HT-29, and HCT 116 |
| PhytoCAT-1429 | Nauclorienine | Nauclea orientalis | NA | HL-60, SMMC-7721, A-549, MCF-7, SW480 |
| PhytoCAT-1430 | Antirhine | Nauclea orientalis | NA | HL-60, SMMC-7721, A-549, MCF-7, SW480 |
| PhytoCAT-1431 | Iso-antirhine | Nauclea orientalis | NA | HL-60, SMMC-7721, A-549, MCF-7, SW480 |
| PhytoCAT-1432 | Alangine | Nauclea orientalis | NA | HL-60, SMMC-7721, A-549, MCF-7, SW480 |
| PhytoCAT-1478 | Kopsifoline I | Kopsia fruticosa | NA | HS-1, HS-4, SCL-1, A431, BGC-823, MCF-7, and W480 |
| PhytoCAT-1479 | Kopsifoline J | Kopsia fruticosa | NA | HS-1, HS-4, SCL-1, A431, BGC-823, MCF-7, and W480 |
| PhytoCAT-1480 | Kopsifoline K | Kopsia fruticosa | NA | HS-1, HS-4, SCL-1, A431, BGC-823, MCF-7, and W480 |
| PhytoCAT-1494 | Ellipticine | Berrywood tree, Asparagus cochinchinensis | ALDH1A1, Bax, Bcl-2, XIAP, cyt-c, Caspase 3, Caspase 9, p53, KIP1/p27 | MCF-7, MDA-MB-231/ HCT116 xenograft mouse tumor |
| PhytoCAT-1502 | Piperine | Piper nigrum Piper longum | MMP2 and -9 mRNA, GLO1, SREBP-1, FAS, CXCL7, sICAM-1, L-selectin | A549, MDA-MB-231, HepG2, MCF-7 |
| PhytoCAT-1511 | Stachydrine hydrochloride | Leonurus cardiaca | Caspase 3, Bcl-2, AKT, ERK | MCF-7 , T47D |
| PhytoCAT-1547 | Sarchookloide A | Sarcococca hookeriana | NA | Hela, A549, MCF-7, SW480, and CEM |
| PhytoCAT-1548 | Sarchookloide B | Sarcococca hookeriana | NA | Hela, A549, MCF-7, SW480, and CEM |
| PhytoCAT-1549 | Sarchookloide C | Sarcococca hookeriana | NA | Hela, A549, MCF-7, SW480, and CEM |
| PhytoCAT-1556 | Vincristine | Catharanthus roseus | Tp53, Bax, Bcl-2 mRNA , miR-222-3p | BT-20, SKBR- 3, MCF-7 |
| PhytoCAT-1557 | Vinblastine | Catharanthus roseus | Tp53, Bax, Bcl-2 mRNA , miR-222-3p | BT-20, SKBR- 3 |
| PhytoCAT-1572 | Cephalinone-F | Cephalanceropsis gracilis | NA | MCF-7, NCI-H460, and SF-268 |
| PhytoCAT-1738 | Pterogynine (PGN) | Pterogyne nitens | NA | ZR-7530 |
| PhytoCAT-1739 | Pterogynidine (PGD) | Pterogyne nitens | NA | ZR-7530 |
| PhytoCAT-1746 | Taspine | Radix et Rhizomaeonticis | ER, PR | ZR-75-30 human breast cancer xenografts in athymic mice |
| PhytoCAT-1764 | Vinorelbine | NA | Caspase 3, Caspase 9, Caspase 8, cyt-c, Bid, HER2, Tp53, Bax, Bcl-2 mRNA , miR-222-3p | MX-1, MCF-7 |
| PhytoCAT-1841 | Coptisine | Coptidis rhizoma | NA | MDA-MB-231 |
| PhytoCAT-1883 | Boldine | Lindera umbellata | p38, ERK, JNK | MCF-7, MDA-MB-231, Tumor-bearing mice |
| PhytoCAT-1898 | Apomorphine | NA | NA | MCF-7 |
| PhytoCAT-1914 | (+)-Tengerensine | Ficus fistulosa | NA | MDA-MB-468, MDA-MB-231, and MCF-7 |
| PhytoCAT-1915 | Tengechlorenine | Ficus fistulosa | NA | MDA-MB-468, MDA-MB-231, and MCF-7 |
| PhytoCAT-1956 | Tetrahydropalmatine (THP) and Berberine (Ber) | Corydalis yanhusuo W. T. Wang | NA | MDA-MB-231 |
| PhytoCAT-1995 | (+)-baphicacanthcusines A | Baphicacanthus cusia | NA | MCF-7 |
| PhytoCAT-1996 | (-)-baphicacanthcusines A | Baphicacanthus cusia | NA | MCF-7 |
| PhytoCAT-1997 | (-)-baphicacanthcusines B | Baphicacanthus cusia | NA | MCF-7 |
| PhytoCAT-2005 | Flavensomycinoic acid | Culture filtrate of endophytic Streptomyces sp. YIM66017 from Alpinia oxyphylla | NA | MCF-7 |
| PhytoCAT-2016 | Berbamine | Berberis amurensis | SNAP29, VAMP8, BNIP3, VAMP8, Bcl-2, Bax, pro-MMP9/pro-MMP2, c-met , AKT, nuclear factor kappaB p-65, Bcl-2/Bax, osteopontin, VEGF, MMP9, MMP2 | MDA-MB-231, MDA-MB-435S |
| PhytoCAT-2017 | Tylophorine | Tylophora indica | Caspase 3, Caspase 9 | T47D |
| PhytoCAT-2110 | 6, 7-dimethoxy-1-(α-hydroxy-4-methoxybenzyl)-2-methyl-1, 2, 3, 4-tetrahydroisoquinoline | Annona squamosa | NA | HepG-2, MCF-7, HCT-116 |
| PhytoCAT-2111 | Coclaurine | Annona squamosa | NA | HepG-2, MCF-7, HCT-116 |
| PhytoCAT-2115 | Luotonin A | Peganum nigellastrum | NA | MCF-7, HeLa |
| PhytoCAT-2157 | Lobeline | Lobelia inflata | P-gp | Caco-2, CCRF-CEM, MDA-MB-231pcDNA3-BCRP-clone23 |
| PhytoCAT-2159 | Thaliblastine (TBL) | Thalictrum foliolosum | P-gp | MCF/AdR |