| PhytoCAT-ID | Phytochemical name or plant extracts | Source of phytochemicals or plant Extracts | Target gene or protein | Cell line/ mice model |
|---|---|---|---|---|
| PhytoCAT-27 | D Rhamnose β-hederin (DRβ-H) | Clematis ganpiniana | Apaf-1, cyt-c, Caspase 3, Caspase 9, miR-16, miR-23a, miR-24, miR-26a, miR-27a | MDA-MB-231, MCF-7/Doc, MCF-7/S |
| PhytoCAT-74 | Platycodin D (PD) | Platycodon grandiflorus | ASK1, PERK, eIF 2alpha, GRP78/Bip, CHOP/GADD153, Caspase 4 | MDA-MB-231, MCF-7 |
| PhytoCAT-138 | Raddeanoside R13 | Pulsatilla chinensis | Cyclin D1, Cyclin A, Cyclin B1, PARP, Caspase 3 | NA |
| PhytoCAT-197 | Gypenoside 5 | Gynostemma pentaphyllum | Tyrosine phosphatase 1B | MCF-7, MCF-7/ADR, MDA-MB-231 |
| PhytoCAT-198 | Gypenoside LI | Gynostemma pentaphyllum | ERCC6L | MCF-7, MDA-MB-231 |
| PhytoCAT-246 | 3-O-α-L-arabinosyl oleanolic acid (3-O-L-AO) | Schumacheria castaneifolia | Bax, p53, Survivin, HIF-1α, HIF-2α | NA |
| PhytoCAT-247 | Methyl protogracillin (NSC-698792) | Dioscorea collettii | NA | MDA-MB-231 , MCF-7, NCI-ADR-RES, BT-549, MALME-3M, M14, KM12, SF-539, U251MDA-MB-435, |
| PhytoCAT-248 | Methyl protoneodioscin (NSC-698791) | Dioscorea collettii | NA | A549, HCT-116, SF-539, SNB-75, M14, CAKI-1, DU-145, HS 578T, MDA-MB-435 |
| PhytoCAT-427 | Fraction 35 (F035) | Acacia victoriae | AKT | MDA-MB-453, MDA-MB-435 |
| PhytoCAT-440 | Glycyrrhizin | Glycyrrhiza glabra | NA | MDA-MB-231, HeLa, MCF-7 |
| PhytoCAT-527 | β-sitosterol-glucoside | Vicia monantha | NA | MCF-7, HCT-116, HepG2 |
| PhytoCAT-542 | Gracillin (NSC-698787) | Dioscorea collettii | NA | CCRF-CEM, RPMT-8226, KM12, SF-539, U251, M14, 786-0, DU-145, MDA-MB-435 |
| PhytoCAT-552 | Polyphyllin VI | Paris polyphylla Sm | Rell2, miR-18a | Mouse mammary carcinoma 4T1, MDA-MB-231 |
| PhytoCAT-620 | Achyranthoside H methyl ester | Achyranthes fauriei | PARP | MCF-7, MDA-MB-453 |
| PhytoCAT-627 | AG36 | Ardisia gigantifolia | Cyclin B1, Cyclin D1, FAK, AKT, VEGF, VEGFR2, Caspase 3, Caspase 8, Bax, Bcl-2, Fas, FasL, TNFR1, DR5, cyt-c | MCF-7, MDA-MB-231, SKBR-3, BALB/c nude mice |
| PhytoCAT-679 | Formosanin C | Trachycarpus fortunei | NA | MCF-7, MDA-MB-231 |
| PhytoCAT-687 | Esculentoside A | Phytolacca acinosa | ALDH1A1, Sox2, Oct4, Bax, Caspase 3, Bcl-2, STAT3 | BALB/c mice, MCF-7 |
| PhytoCAT-719 | Saxifragifolin C | Androsace umbellata | p38 MAPK, ERK 1/2, JNK | MCF-7, MDA-MB-231 |
| PhytoCAT-770 | Ziyuglycoside II | Sanguisorba officinalis | Bax, Fas/FasL, Bcl-2, EMT | MCF-7 and MDA-MB-231 |
| PhytoCAT-823 | Escin Ia | Aesculus chinensis | LOXL2 | Female athymic nude mice, MCF-7, MDA-MB-231 |
| PhytoCAT-892 | Saikosaponin A | Bupleurum chinense | VEGFR2, PLCγ1, FAK, Src, AKT | 4T1, MCF-7, HCT-15, AGS, HepG2 |
| PhytoCAT-1006 | Julibroside (J29) | Albizia julibrissin | NA | MDA-MB-435, PC-3M-1E8, HeLa |
| PhytoCAT-1007 | Julibroside (J30) | Albizia julibrissin | NA | MDA-MB-435, PC-3M-1E8, HeLa |
| PhytoCAT-1008 | Julibroside (J31) | Albizia julibrissin | NA | MDA-MB-435, PC-3M-1E8, HeLa |
| PhytoCAT-1041 | Ziyuglycoside I | Sanguisorba officinalis | p53, p21WAF1, Bax, Bcl-2 | MDA-MB-231 |
| PhytoCAT-1077 | Chestnoside B | Castanea sativa | NA | MCF-7, PC3 |
| PhytoCAT-1094 | Dioscin | Dioscorea villosa | GATA3, DNMT3A, TET2, TET3, ZFPM2 , E-cad, TET1, VIM, MMP9, Bcl-2, cIAP-1, Mcl-1 | MCF-7, MDA-MB-231, T47D |
| PhytoCAT-1151 | Pennogenin 3-O-α-L-rhamnopyranosyl-(1→4)-[α-L-rhamnopyranosyl-(1→2)]-β-D-glucopyranoside | Paris quadrifolia | NA | HL-60, HeLa and MCF-7 |
| PhytoCAT-1152 | Pennogenin 3-O-α-L-rhamnopyranosyl-(1→4)-α-L-rhamnopyranosyl-(1→4)-[α-L-rhamnopyranosyl-(1→2)]-β-D-glucopyranoside | Paris quadrifolia | NA | HL-60, HeLa and MCF-7 |
| PhytoCAT-1176 | Bigelovii A | Salicornia bigelovii | Bcl-2, Cyclin D1, NF‑κB‑regulated gene products, Cyclin D1, COX‑2 | MDA‑MB‑231, MDA‑MB‑468HL-60, MCF-7, HepG2, A549 |
| PhytoCAT-1263 | Urs-12-ene-3beta,6beta,16beta-triol-3-O-beta-galactopyranosyl-(1-->2)-beta-glucopyranoside | Silphium radula Nutt | NA | MDA-MB-231 |
| PhytoCAT-1287 | Ardisiacrispins B | Ardisia Crenata | NA | MDA-MB-231 |
| PhytoCAT-1417 | Lobatoside N | Actinostemma lobatum | NA | HCT-116, HT-29, MCF-7, A549 |
| PhytoCAT-1448 | Polyphyllin V | Paris polyohylla var chinensis | NA | MDA-MB-231, HeLa |
| PhytoCAT-1470 | Hederagenin 3-O-β-D-glucopyranosyl-(1→4)-β-D-glucopyranosyl-(1→3)-α-L-rhamnopyranosyl-(1→2)-α-L-arabinopyranoside | Lonicera similis Hemsl | NA | HepG2, MCF-7, A-549 |
| PhytoCAT-1504 | Panaxadiol | Panax ginseng | MMP9, CDK2, CDK4, p21, p27, Cyclin D1, CDK6, EGFR,HER2 | MCF-7, A549 |
| PhytoCAT-1513 | Julibroside J19 | Albizzia julibrissin Durazz | NA | HeLa, Bel-7402 and MDA-MB-435 |
| PhytoCAT-1514 | Julibroside J18 | Albizzia julibrissin Durazz | NA | HeLa, Bel-7402 and MDA-MB-435 |
| PhytoCAT-1580 | Ginsenoside Rg1 | Panax ginseng | NA | MCF-7, HEK293 |
| PhytoCAT-1583 | Diosgenin | Trigonella foenum-graecum Paris polyphylla | XIAP, Survivin, Bcl-2, AKT, JNK, mTOR, Cyclin D1, CDK-2, CDK-4, FAS | MCF-7, T47D, MDA-MB-231, C6, T98G, MCF-7 and MDA-231 xenografts in nude mice |
| PhytoCAT-1688 | Saikosaponin b2 (SSb2) | Radix Bupleuri | STAT-3, VASP, MMP2, MMP9, c-myc, Cyclin D1 | MCF-7 |
| PhytoCAT-1731 | Saikosaponin-d (SSd) | Bupleurum falcatum | NA | MCF-7, HeLa, MDA-MB-231 |
| PhytoCAT-1922 | Clematis hederagenin saponin (CHS) | Clematis ganpiniana | NA | MCF-7 and MDA-MB-231 |
| PhytoCAT-1936 | Ginsenoside Rg5 | Black ginseng | p53, p21(WAF1/CIP1), p15(INK4B), Cyclin D1, Cyclin E2, CDK4 | BALB/c nude mouse model of human breast cancer, MCF-7 |
| PhytoCAT-2065 | Tubeimoside-1 | Bolbostemma paniculatum (Maxim) Franquet | Mcl-1, Bcl-xL, Bcl-2 | MDA-MB-231, T47D |
| PhytoCAT-2124 | Polyphylloside A | Paris polyohylla | NA | MCF-7, MDA-MB-231, A549, HeLa, HCT-116 |
| PhytoCAT-2125 | Polyphylloside B | Paris polyohylla | NA | MCF-7, MDA-MB-231, A549, HeLa, HCT-116 |
| PhytoCAT-2126 | Polyphylloside C | Paris polyohylla | NA | MCF-7, MDA-MB-231, A549, HeLa, HCT-116 |
| PhytoCAT-2127 | Polyphylloside D | Paris polyohylla | NA | MCF-7, MDA-MB-231, A549, HeLa, HCT-116 |
| PhytoCAT-2128 | Polyphylloside E | Paris polyohylla | NA | MCF-7, MDA-MB-231, A549, HeLa, HCT-116 |
| PhytoCAT-2129 | Polyphylloside F | Paris polyohylla | NA | MCF-7, MDA-MB-231, A549, HeLa, HCT-116 |
| PhytoCAT-2130 | 7-oxodioscin | Paris polyohylla | NA | MCF-7, MDA-MB-231, A549, HeLa, HCT-116 |
| PhytoCAT-2131 | Isonarthogenin 3-O-α-L-rhamnopyranosyl-(1 → 2)-[α-L-rhamnopyranosyl-(1 → 4)]-β-D-glucopyranoside | Paris polyohylla | NA | MCF-7, MDA-MB-231, A549, HeLa, HCT-116 |
| PhytoCAT-2132 | Trinervuloside C | Paris polyohylla | NA | MCF-7, MDA-MB-231, A549, HeLa, HCT-116 |
| PhytoCAT-2160 | Paris saponin VII | Trillium tschonoskii | NFR1, TRAIL R1/DR4, TRAIL R2/DR5, FADD, PARP, Caspase 8, Caspase 3, P-gp | MCF-7/ADR |