| PhytoCAT-ID | Phytochemical name or plant extracts | Source of phytochemicals or plant Extracts | Target gene or protein | Cell line/ mice model |
|---|---|---|---|---|
| PhytoCAT-92 | Esculetin | Dryopteris fragrans | NA | A549, MCF-7 , MDA-MB-435, MDA-MB-231, HepG2 |
| PhytoCAT-93 | Isoscopoletin | Dryopteris fragrans | NA | A549, MCF-7, HepG2 |
| PhytoCAT-96 | Dryofracoumarin A | Dryopteris fragrans | NA | A549, MCF-7, HepG2 |
| PhytoCAT-358 | Mammea F/BB | Mammea americana | VEGF, HIF-1 | T47D, PC-3 |
| PhytoCAT-359 | Mammea F/BA | Mammea americana | NA | T47D, PC-3 |
| PhytoCAT-360 | Mammea C/AA | Mammea americana | NA | T47D, PC-3 |
| PhytoCAT-361 | Mammea C/AB | Mammea americana | NA | T47D, PC-3 |
| PhytoCAT-362 | Mammea C/BB | Mammea americana | NA | T47D, PC-3 |
| PhytoCAT-363 | Mammea B/AB | Mammea americana | NA | T47D, PC-3 |
| PhytoCAT-364 | Mammea B/BB | Mammea americana | NA | T47D, PC-3 |
| PhytoCAT-365 | Mammea A/AB | Mammea americana | NA | T47D, PC-3 |
| PhytoCAT-366 | Mammea A/BB | Mammea americana | NA | T47D, PC-3 |
| PhytoCAT-514 | Psoralen | Psoralea corylifolia | Rh123, P-gp, Fra-1, Axin2, β-catenin | MCF-7/ADR, MCF-7, MDA-MB-231, BALB/c nude mice |
| PhytoCAT-561 | 7-Hydroxy coumarin | Strychnos nux-vomica | NA | MCF-7, Hep-2, HCT |
| PhytoCAT-611 | Dichlorodiaportinol A | Myoporum bontioides (endophytic fungus Trichoderma sp. 09) | NA | MCF-7, HepG2 |
| PhytoCAT-668 | Fraxetin (FXT) | Fraxinus bungeana | Fas, FasL, Bax, Bcl-2 | MCF-7, HCC827, H1650, A549, H460, PC-9, H1975 |
| PhytoCAT-791 | Marmin | Aegle marmelos | NA | T47D |
| PhytoCAT-792 | Auraptene | Aegle marmelos | VEGF, VEGFR2, VCAM-1, TNFR-1, COX-2, IFNγ | T47D, 4T, MDA-MB-231, HUVEC |
| PhytoCAT-869 | Mansorin-A | Mansonia gagei | NA | MCF-7, HepG2, HCT-116, HeLa |
| PhytoCAT-870 | Mansorin-B | Mansonia gagei | NA | MCF-7, HepG2, HCT-116, HeLa |
| PhytoCAT-871 | Mansorin-C | Mansonia gagei | NA | MCF-7, HepG2, HCT-116, HeLa |
| PhytoCAT-872 | Mansorin-I | Mansonia gagei | NA | MCF-7, HepG2, HCT-116, HeLa |
| PhytoCAT-873 | Mansorin-II | Mansonia gagei | NA | MCF-7, HepG2, HCT-116, HeLa |
| PhytoCAT-874 | Mansorin III | Mansonia gagei | NA | MCF-7, HepG2, HCT-116, HeLa |
| PhytoCAT-898 | Ferulin C | Ferula ferulaeoides | NA | MCF-7 and MDA-MB-231 |
| PhytoCAT-902 | Umbelliprenin | Ferula szowitsiana | NA | MCF-7, M4Beu, A549, PC3, PA1 |
| PhytoCAT-906 | Prim-O-glucosylcimifugin | Saposhnikovia divaricata | Arg-1, iNOS | B16-F10, (4 T1) mouse tumour models |
| PhytoCAT-1083 | Osthole | Cnidium monnieri | GPX1, SOD2, GCL-c, G6pdh, NOX2, ACOX, FASN, c-met, c-FLIP, Bax, Akt, mTOR, p53, p21, Cdk2, cyclin D1 Caspase 3, Caspase 9 | MDA-MB-231, MDA-MB-435, Caki, U251MG, |
| PhytoCAT-1209 | Bis(4-hydroxy-2H-chromen-2-one) coumarin (4HC) | NA | CYP19A1, Bcl-2, Bax, Caspase 3, | MCF-7 |
| PhytoCAT-1223 | Dentatin (DTN) | Clausena excavata Burm | Bcl-2, Bax, Caspase 9, Caspase 3, Caspase 7, cyt-c | MCF-7 |
| PhytoCAT-1243 | Bergapten (Bg) | Ficus carica | p53, PTEN | MDA-MB-231, MCF-7, ZR75 |
| PhytoCAT-1425 | 8-[(2E)-6-oxo-3,7-dimethyloct-2-enyloxylpsoralen | Clausena hainanensis | NA | HL-60, SMMC-7721, A-549, MCF-7, SW480 |
| PhytoCAT-1522 | Clauhainanin A | Clausena hainanensis | NA | HL-60, SMMC-7721, A-549, MCF-7 and SW480 |
| PhytoCAT-1523 | Clausenalansimin A | Clausena hainanensis | NA | HL-60, SMMC-7721, A-549, MCF-7 and SW480 |
| PhytoCAT-1683 | Triphenylethylene-Coumarin Hybrid 5c | NA | NA | SKBR-3 |
| PhytoCAT-1801 | Daphnoretin | Daphne genkwa | NA | MCF-7, MDA-MB-231, Huh7, AGS, HT-29, B 16, Colo 205, A549, A2058 |
| PhytoCAT-1909 | Scopolin | Artemisia herba alba | NA | MCF-7, HeLa |
| PhytoCAT-1928 | Clauselenisin A | Clausena lenis | NA | HL-60, SMMC-7721, A-549, MCF-7 and SW480 |
| PhytoCAT-2021 | 5-hydroxy-8,8-dimethyl-4-phenyl-9,10-dihydro-8H-pyrano-[2,3-f]chromen-2-one | Marila pluricostata | NA | MCF-7, H-460, SF-268 |
| PhytoCAT-2022 | 5-hydroxy-8,8-dimethyl-4-phenyl-6-propionyl-9,10-dihydro-8H-pyrano-[2,3-f]chromen-2-one | Marila pluricostata | NA | MCF-7, H-460, SF-268 |
| PhytoCAT-2023 | 5,7-dihydroxy-8-(3-methylbut-2-enyl)-4-phenylchromen-2-one | Marila pluricostata | NA | MCF-7, H-460, SF-268 |
| PhytoCAT-2037 | Mammea A/AD cyclo F | Marila pluricostata | NA | MCF-7, H-460, SF-268 |
| PhytoCAT-2066 | (Z)-ethylidene-4,6-dimethoxycoumaran-3-one (Compound 1) | Pogostemon quadrifolius (Benth.) | NA | Caco-2, HeLa, THP-1, MCF-7, Jurkat E6-1 |
| PhytoCAT-2167 | Xanthotoxol | Angelica japonica | ERα, PR, EGFR, mTOR | In-silico |