| PhytoCAT-ID | Phytochemical name or plant extracts | Source of phytochemicals or plant Extracts | Target gene or protein | Cell line/ mice model |
|---|---|---|---|---|
| PhytoCAT-81 | Mangiferin | Mangifera indica | MMP7, MMP9, Vimentin, E-cadherin, β-catenin, NF-κB, P-gp | MDA-MB-231 xenograft mice, MCF-7 |
| PhytoCAT-349 | Gambogic acid | Garcinia hanburyi | Bid | T47D |
| PhytoCAT-351 | Garcinol | Garcinia indica | miR-200s, let-7s, NF-κB, E-cadherin, Vimentin, ZEB-1, ZEB-2, STAT-3 | MDA-MB-231, BT-549/xenograft mouse model |
| PhytoCAT-353 | α-mangostin | Garcinia mangostana | MMP2, MMP9, MARK4 | MCF-7, HepG2 |
| PhytoCAT-357 | Wightiic acid | Garcinia wightii | NA | MCF-7, SKBR-3, A-375 |
| PhytoCAT-608 | Cudraticusxanthone A | Cudrania tricuspidata | MMP9, IκBα | MCF-7 cells, MDA-MB-231 |
| PhytoCAT-1016 | Pyranocycloartobiloxanthone A (PA) | Artocarpus obtusus | Bax, Bcl-2 | MCF-7, K562, HL-60 |
| PhytoCAT-1111 | Gambogenic acid | Garcinia hanburyi | Fas, Caspase 3,-8,-9, Bax, Bcl-2 | MDA-MB-231 |
| PhytoCAT-1300 | Garcimangostanol | Garcinia mangostana | NA | MCF-7, A549, Hep-G2, CNE |
| PhytoCAT-1301 | 8-deoxygartanin | Garcinia mangostana | NA | MCF-7, A549, Hep-G2, CNE and HT-29 |
| PhytoCAT-1302 | 1-isomangostin | Garcinia mangostana | NA | MCF-7, A549, Hep-G2 and CNE |
| PhytoCAT-1303 | Garcinone C | Garcinia mangostana | CDK2 | MCF-7, A549, Hep-G2, CNE, 22Rν1and MDA-MB-231 |
| PhytoCAT-1445 | Isocowanin | Garcinia tetrandra | NA | Hep G2, HeLa S3, MCF-7, HT-29, KB |
| PhytoCAT-1446 | Parvifolixanthone C | Garcinia tetrandra | NA | Hep G2, HeLa S3, MCF-7, HT-29, KB |
| PhytoCAT-1460 | 9 - hydroxycalabaxanthone | Garcinia tetrandra | NA | MCF-7, HT-29, KB, Hep G2, and HeLa S3 |
| PhytoCAT-1537 | Cratochinone B | Cratoxylum cochinchinense | NA | KB, HeLa S-3, HT-29, MCF-7 and Hep G2 |
| PhytoCAT-1538 | Macluraxanthone | Cratoxylum cochinchinense | NA | KB, HeLa S-3, HT-29, MCF-7 and Hep G2 |
| PhytoCAT-1539 | Pruniflorone G | Cratoxylum cochinchinense | NA | KB, HeLa S-3, HT-29, MCF-7 and Hep G2 |
| PhytoCAT-1896 | 1, 3, 7, 8-tetrahydroxyxanthone | Sinopodophyllum hexandrum | NA | T47D, MCF-7, MDA-MB-231 |
| PhytoCAT-1918 | Mangostanaxanthone VII | Garcinia mangostana | NA | A549, MCF-7 |
| PhytoCAT-1991 | Xanthone V | Vismia laurentii | Caspase 3, Caspase 7 | CCRF-CEM, CEM/ADR5000, PF-382, HL-60, MiaPaCa-2, Capan-1, MCF-7, SW-680, 786-0, U87MG, A549, Colo-38, HeLa, Caski |
| PhytoCAT-2000 | 1,5,8-trihydroxy-3-methoxyxanthone (XD) | Swertia chirata | Bax, Bcl-2 | MCF-7, MDA-MB-231, Ehrlich ascites carcinoma (EAC), a mouse transplantable breast carcinoma cell line |